BG63124B1 - Нови производни на еритромицин, метод за тяхнотополучаване и използването им като лекарствени средства - Google Patents

Нови производни на еритромицин, метод за тяхнотополучаване и използването им като лекарствени средства Download PDF

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Publication number
BG63124B1
BG63124B1 BG103398A BG10339899A BG63124B1 BG 63124 B1 BG63124 B1 BG 63124B1 BG 103398 A BG103398 A BG 103398A BG 10339899 A BG10339899 A BG 10339899A BG 63124 B1 BG63124 B1 BG 63124B1
Authority
BG
Bulgaria
Prior art keywords
formula
methyl
radical
compound
compounds
Prior art date
Application number
BG103398A
Other languages
Bulgarian (bg)
English (en)
Other versions
BG103398A (en
Inventor
Jean-Michel Auger
Constantin Agouridas
Jean-Francois Chantot
Alexis Denis
Original Assignee
Hoechst Marion Roussel
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Marion Roussel filed Critical Hoechst Marion Roussel
Publication of BG103398A publication Critical patent/BG103398A/xx
Publication of BG63124B1 publication Critical patent/BG63124B1/bg

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Medicinal Preparation (AREA)
BG103398A 1996-12-12 1999-05-12 Нови производни на еритромицин, метод за тяхнотополучаване и използването им като лекарствени средства BG63124B1 (bg)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9615271A FR2757168B1 (fr) 1996-12-12 1996-12-12 Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
PCT/FR1997/002254 WO1998025942A1 (fr) 1996-12-12 1997-12-10 Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments

Publications (2)

Publication Number Publication Date
BG103398A BG103398A (en) 2000-01-31
BG63124B1 true BG63124B1 (bg) 2001-04-30

Family

ID=9498593

Family Applications (1)

Application Number Title Priority Date Filing Date
BG103398A BG63124B1 (bg) 1996-12-12 1999-05-12 Нови производни на еритромицин, метод за тяхнотополучаване и използването им като лекарствени средства

Country Status (28)

Country Link
EP (1) EP0946579B1 (es)
JP (1) JP4363666B2 (es)
KR (1) KR100490074B1 (es)
CN (2) CN100363375C (es)
AP (1) AP997A (es)
AT (1) ATE217008T1 (es)
AU (1) AU721732B2 (es)
BG (1) BG63124B1 (es)
BR (1) BR9714007A (es)
CA (1) CA2273985C (es)
CZ (1) CZ292403B6 (es)
DE (1) DE69712361T2 (es)
DK (1) DK0946579T3 (es)
EA (1) EA001733B1 (es)
ES (1) ES2174323T3 (es)
FR (1) FR2757168B1 (es)
GE (1) GEP20012518B (es)
HU (1) HUP0001180A3 (es)
ID (1) ID21873A (es)
IL (1) IL130420A (es)
NO (1) NO314040B1 (es)
NZ (1) NZ335325A (es)
PT (1) PT946579E (es)
SK (1) SK283715B6 (es)
TR (1) TR199901301T2 (es)
WO (1) WO1998025942A1 (es)
YU (1) YU25699A (es)
ZA (1) ZA9711101B (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2771008B1 (fr) * 1997-11-17 2000-04-28 Hoechst Marion Roussel Inc Utilisation des ketolides pour la preparation de compositions pharmaceutiques destinees a prevenir les complications thrombotiques arterielles liees a l'atherosclerose
EP1137654A1 (en) * 1998-12-10 2001-10-04 Pfizer Products Inc. Carbamate and carbazate ketolide antibiotics
EP1147121B1 (en) 1999-01-27 2003-12-17 Pfizer Products Inc. Ketolide antibiotics
KR20020007374A (ko) * 1999-04-16 2002-01-26 추후제출 매크롤라이드 항감염제
WO2000071557A1 (en) 1999-05-24 2000-11-30 Pfizer Products Inc. 13-methyl-erythromycin derivatives
US6472372B1 (en) 2000-12-06 2002-10-29 Ortho-Mcneil Pharmaceuticals, Inc. 6-O-Carbamoyl ketolide antibacterials
DK200201957A (da) * 2002-12-20 2003-01-20 Alpharma Aps 10-substituted erythromycin ketolides and methods of making

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4742049A (en) * 1986-06-04 1988-05-03 Abbott Laboratories Semisynthetic erythromycin antibiotics
IL114589A (en) * 1990-11-21 1999-12-22 Roussel Uclaf Intermediates for the preparation of the history of erythromycin
KR0166996B1 (ko) * 1992-04-22 1999-01-15 우에하라 아키라 5-o-데소사미닐에리쓰로노라이드a 유도체
US5527780A (en) * 1992-11-05 1996-06-18 Roussel Uclaf Erythromycin derivatives
JP3709997B2 (ja) * 1994-03-29 2005-10-26 日東電工株式会社 耐熱性ネガ型フォトレジスト組成物および感光性基材、ならびにネガ型パターン形成方法
FR2718450B1 (fr) * 1994-04-08 1997-01-10 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.
FR2719587B1 (fr) * 1994-05-03 1996-07-12 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.

Also Published As

Publication number Publication date
CN100363375C (zh) 2008-01-23
EA001733B1 (ru) 2001-08-27
KR20000057517A (ko) 2000-09-15
EP0946579A1 (fr) 1999-10-06
EA199900528A1 (ru) 1999-12-29
ES2174323T3 (es) 2002-11-01
YU25699A (sh) 2002-06-19
CN1239966A (zh) 1999-12-29
AU721732B2 (en) 2000-07-13
GEP20012518B (en) 2001-08-27
CZ208299A3 (cs) 1999-09-15
JP4363666B2 (ja) 2009-11-11
CN1238364C (zh) 2006-01-25
IL130420A0 (en) 2000-06-01
TR199901301T2 (xx) 1999-08-23
CA2273985A1 (fr) 1998-06-18
EP0946579B1 (fr) 2002-05-02
HUP0001180A2 (hu) 2000-09-28
NZ335325A (en) 2000-08-25
BG103398A (en) 2000-01-31
BR9714007A (pt) 2000-05-09
ID21873A (id) 1999-08-05
AP9901513A0 (en) 1999-06-30
ATE217008T1 (de) 2002-05-15
NO314040B1 (no) 2003-01-20
FR2757168A1 (fr) 1998-06-19
JP2001506620A (ja) 2001-05-22
WO1998025942A1 (fr) 1998-06-18
FR2757168B1 (fr) 1999-06-11
DE69712361D1 (de) 2002-06-06
CA2273985C (fr) 2007-03-20
AP997A (en) 2001-08-09
DK0946579T3 (da) 2002-08-12
AU5487798A (en) 1998-07-03
DE69712361T2 (de) 2002-11-28
SK283715B6 (sk) 2003-12-02
KR100490074B1 (ko) 2005-05-17
PT946579E (pt) 2002-10-31
CZ292403B6 (cs) 2003-09-17
HUP0001180A3 (en) 2003-05-28
IL130420A (en) 2003-01-12
NO992859L (no) 1999-06-11
CN1721427A (zh) 2006-01-18
NO992859D0 (no) 1999-06-11
ZA9711101B (en) 1998-12-10
SK75099A3 (en) 2000-01-18

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