BG105919A - Erythromycin derivatives - Google Patents

Erythromycin derivatives

Info

Publication number
BG105919A
BG105919A BG105919A BG10591901A BG105919A BG 105919 A BG105919 A BG 105919A BG 105919 A BG105919 A BG 105919A BG 10591901 A BG10591901 A BG 10591901A BG 105919 A BG105919 A BG 105919A
Authority
BG
Bulgaria
Prior art keywords
alkyl
aralkyl
erythromycin derivatives
cycloalkyl
aryl
Prior art date
Application number
BG105919A
Other languages
Bulgarian (bg)
English (en)
Inventor
Hideo Kato
Noriyuki Kado
Toshihiko Yoshida
Akemi Nishimoto
Ken Narita
Original Assignee
Hokuriku Seiyaku Co., Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hokuriku Seiyaku Co., Ltd filed Critical Hokuriku Seiyaku Co., Ltd
Publication of BG105919A publication Critical patent/BG105919A/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Molecular Biology (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
BG105919A 1999-04-08 2001-09-19 Erythromycin derivatives BG105919A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP10072699 1999-04-08
PCT/JP2000/002226 WO2000061593A1 (fr) 1999-04-08 2000-04-06 Derives d'erythromycine

Publications (1)

Publication Number Publication Date
BG105919A true BG105919A (en) 2002-06-28

Family

ID=14281635

Family Applications (1)

Application Number Title Priority Date Filing Date
BG105919A BG105919A (en) 1999-04-08 2001-09-19 Erythromycin derivatives

Country Status (19)

Country Link
EP (1) EP1167375A4 (tr)
KR (1) KR20020007333A (tr)
CN (1) CN1343216A (tr)
AR (1) AR023264A1 (tr)
AU (1) AU3671000A (tr)
BG (1) BG105919A (tr)
BR (1) BR0010518A (tr)
CA (1) CA2367319A1 (tr)
CZ (1) CZ20013497A3 (tr)
HK (1) HK1045697A1 (tr)
HU (1) HUP0201116A3 (tr)
IL (1) IL145256A0 (tr)
NO (1) NO20014362L (tr)
NZ (1) NZ513998A (tr)
PL (1) PL354409A1 (tr)
SK (1) SK13972001A3 (tr)
TR (1) TR200102572T2 (tr)
WO (1) WO2000061593A1 (tr)
ZA (1) ZA200107346B (tr)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6946446B2 (en) 2000-02-24 2005-09-20 Abbott Laboratories Anti-infective agents useful against multidrug-resistant strains of bacteria
EP1259923B1 (en) * 2000-02-24 2005-12-14 Abbott Laboratories Anti-infective agents useful against mulitidrug-resistant strains of bacteria
JP2002173498A (ja) * 2000-09-27 2002-06-21 Hokuriku Seiyaku Co Ltd エリスロマイシン誘導体
UY27429A1 (es) * 2001-09-05 2003-10-31 Hokuriku Pharmaceutical Medicamento para el tratamiento terapéutico o preventivo de la tuberculosis que comprende un derivado de eritromicina
CA2801100A1 (en) 2003-03-10 2004-09-23 Optimer Pharmaceuticals, Inc. Macrolides and processes for their preparation
WO2004108744A2 (en) * 2003-05-19 2004-12-16 Prasad K Deshpande Azalides and azaketolides having antimicrobial activity
WO2006120541A1 (en) 2005-05-10 2006-11-16 Glaxosmithkline Istrazivacki Centar Zagreb D.O.O. Ether linked macrolides useful for the treatment of microbial infections
CN105732745A (zh) 2007-10-25 2016-07-06 森普拉制药公司 大环内酯类抗菌剂的制备方法
CN107854477A (zh) 2008-10-24 2018-03-30 森普拉制药公司 使用含***的大环内酯治疗抗性疾病的方法
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
WO2011032052A1 (en) 2009-09-10 2011-03-17 Cempra Pharmaceuticals, Inc. Methods for treating malaria, tuberculosis and mac diseases
PL2571506T3 (pl) * 2010-05-20 2017-10-31 Cempra Pharmaceuticals Inc Sposoby sporządzania makrolidów i ketolidów oraz ich produktów pośrednich
KR20180110181A (ko) 2010-09-10 2018-10-08 셈프라 파마슈티컬스, 인크. 질환을 치료하기 위한 수소결합 형성 플루오로 케토라이드
IN2014DN08939A (tr) 2012-03-27 2015-05-22 Cempra Pharmaceuticals Inc
AU2014239959A1 (en) 2013-03-14 2015-10-01 Cempra Pharmaceuticals, Inc. Methods for treating respiratory diseases and formulations therefor
EP2968384A4 (en) 2013-03-15 2017-02-15 Cempra Pharmaceuticals, Inc. Convergent processes for preparing macrolide antibacterial agents
AU2014252462A1 (en) * 2013-04-10 2015-10-01 Probiotic Pharmaceuticals Aps Azithromycin antimicrobial derivatives with non-antibiotic pharmaceutical effect

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8506380D0 (en) * 1985-03-12 1985-04-11 Beecham Group Plc Chemical compounds
DE3668894D1 (en) * 1985-03-12 1990-03-15 Beecham Group Plc Erythromycin-derivate.
US5302705A (en) * 1989-10-07 1994-04-12 Taisho Pharmaceutical Co., Ltd. 6-O-methylerythromycin a oxime derivatives
US5719272A (en) * 1996-04-02 1998-02-17 Abbott Laboratories 2'-protected 3'-dimethylamine, 9-etheroxime erythromycin A derivatives
EP0895999A1 (en) * 1997-08-06 1999-02-10 Pfizer Products Inc. C-4" substituted macrolide antibiotics

Also Published As

Publication number Publication date
NO20014362D0 (no) 2001-09-07
HK1045697A1 (zh) 2002-12-06
NO20014362L (no) 2001-12-04
BR0010518A (pt) 2002-01-08
SK13972001A3 (sk) 2002-08-06
ZA200107346B (en) 2002-11-27
AU3671000A (en) 2000-11-14
HUP0201116A3 (en) 2003-03-28
IL145256A0 (en) 2002-06-30
CZ20013497A3 (cs) 2002-05-15
HUP0201116A2 (en) 2002-08-28
NZ513998A (en) 2001-09-28
TR200102572T2 (tr) 2002-02-21
EP1167375A4 (en) 2002-10-30
PL354409A1 (en) 2004-01-12
CA2367319A1 (en) 2000-10-19
KR20020007333A (ko) 2002-01-26
AR023264A1 (es) 2002-09-04
CN1343216A (zh) 2002-04-03
WO2000061593A1 (fr) 2000-10-19
EP1167375A1 (en) 2002-01-02

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