AU616706B2 - 5-ht3 receptor antagonists for treatment of cough and bronchoconstriction - Google Patents
5-ht3 receptor antagonists for treatment of cough and bronchoconstriction Download PDFInfo
- Publication number
- AU616706B2 AU616706B2 AU26264/88A AU2626488A AU616706B2 AU 616706 B2 AU616706 B2 AU 616706B2 AU 26264/88 A AU26264/88 A AU 26264/88A AU 2626488 A AU2626488 A AU 2626488A AU 616706 B2 AU616706 B2 AU 616706B2
- Authority
- AU
- Australia
- Prior art keywords
- international
- hydrogen
- formula
- document
- pct
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/46—8-Azabicyclo [3.2.1] octane; Derivatives thereof, e.g. atropine, ***e
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Emergency Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Electrotherapy Devices (AREA)
- Conductive Materials (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB878726717A GB8726717D0 (en) | 1987-11-14 | 1987-11-14 | Treatment |
GB878726716A GB8726716D0 (en) | 1987-11-14 | 1987-11-14 | Treatment |
GB8726717 | 1987-11-14 | ||
GB8726716 | 1987-11-14 |
Publications (2)
Publication Number | Publication Date |
---|---|
AU2626488A AU2626488A (en) | 1989-06-14 |
AU616706B2 true AU616706B2 (en) | 1991-11-07 |
Family
ID=26293045
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU26264/88A Ceased AU616706B2 (en) | 1987-11-14 | 1988-11-14 | 5-ht3 receptor antagonists for treatment of cough and bronchoconstriction |
Country Status (9)
Country | Link |
---|---|
US (1) | US5098909A (ja) |
EP (1) | EP0340270B1 (ja) |
JP (1) | JPH02502185A (ja) |
KR (1) | KR890701099A (ja) |
AT (1) | ATE78162T1 (ja) |
AU (1) | AU616706B2 (ja) |
DE (1) | DE3872872T2 (ja) |
DK (1) | DK345889D0 (ja) |
WO (1) | WO1989004660A1 (ja) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU8072691A (en) * | 1990-06-28 | 1992-01-23 | Beecham Group Plc | Pharmaceutical preparations |
HU211081B (en) * | 1990-12-18 | 1995-10-30 | Sandoz Ag | Process for producing indole derivatives as serotonin antagonists and pharmaceutical compositions containing the same |
CA2112487C (en) * | 1991-06-26 | 2003-04-15 | James W. Young | Method and compositions for treating emesis, nausea and other disorders using optically pure r(+) ondansetron |
JP2002538102A (ja) | 1999-03-01 | 2002-11-12 | セプラコア インコーポレーテッド | 光学的に純粋なr(+)オンダンセトロンを使用する無呼吸および無呼吸障害の治療方法 |
JP2003501462A (ja) * | 1999-06-15 | 2003-01-14 | レスピラトリウス アクチボラゲット | 受容体アゴニストおよびアンタゴニスト |
GB9918425D0 (en) * | 1999-08-04 | 1999-10-06 | Novartis Ag | Organic compounds |
AU2001225664A1 (en) * | 2000-06-15 | 2001-12-24 | Respiratorius Ab | 5-ht3 receptor antagonists for treatment of disorders involving airway constriction |
PL210065B1 (pl) | 2002-09-25 | 2011-11-30 | Memory Pharm Corp | Związki indazole, benzotiazole i benzoizotiazole, kompozycje farmaceutyczne je zawierające oraz zastosowanie związków |
WO2004091606A1 (en) * | 2003-04-16 | 2004-10-28 | Orchid Chemicals & Pharmaceuticals, Ltd. | Treatment of bronchial asthma using 5-ht3 receptor antagonists |
DE602004010299T2 (de) * | 2003-12-22 | 2008-09-18 | Memory Pharmaceuticals Corp. | Indole, 1h-indazole, 1,2-benzisoxazole und 1,2-benzisothiazole und deren herstellung und anwendungen |
AU2005227324A1 (en) | 2004-03-25 | 2005-10-06 | Memory Pharmaceuticals Corporation | Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, and preparation and uses thereof |
EP1742944B1 (en) * | 2004-04-22 | 2010-11-10 | Memory Pharmaceuticals Corporation | Indoles, 1h-indazoles, 1,2-benzisoxazoles, 1,2-benzoisothiazoles, and preparation and uses thereof |
NZ551712A (en) * | 2004-05-07 | 2010-07-30 | Memory Pharm Corp | 1H-indazoles, benzothiazoles, 1,2-benzoisoxazoles, 1,2-benzoisothiazoles, and chromones and preparations and uses thereof |
AU2005319248A1 (en) * | 2004-12-22 | 2006-06-29 | Memory Pharmaceuticals Corporation | Nicotinic alpha-7 receptor ligands and preparation and uses thereof |
US8106066B2 (en) * | 2005-09-23 | 2012-01-31 | Memory Pharmaceuticals Corporation | Indazoles, benzothiazoles, benzoisothiazoles, benzisoxazoles, pyrazolopyridines, isothiazolopyridines, and preparation and uses thereof |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0200444B1 (en) * | 1985-04-27 | 1992-11-11 | Beecham Group Plc | Azabicyclononyl-indazole-carboxamide having 5-ht antagonist activity |
-
1988
- 1988-11-14 DE DE8888909596T patent/DE3872872T2/de not_active Expired - Fee Related
- 1988-11-14 EP EP88909596A patent/EP0340270B1/en not_active Expired - Lifetime
- 1988-11-14 WO PCT/GB1988/000994 patent/WO1989004660A1/en active IP Right Grant
- 1988-11-14 AT AT88909596T patent/ATE78162T1/de not_active IP Right Cessation
- 1988-11-14 AU AU26264/88A patent/AU616706B2/en not_active Ceased
- 1988-11-14 US US07/381,666 patent/US5098909A/en not_active Expired - Fee Related
- 1988-11-14 JP JP63508864A patent/JPH02502185A/ja active Pending
-
1989
- 1989-07-12 DK DK345889A patent/DK345889D0/da not_active Application Discontinuation
- 1989-07-13 KR KR1019890701320A patent/KR890701099A/ko not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
DE3872872D1 (de) | 1992-08-20 |
JPH02502185A (ja) | 1990-07-19 |
DK345889A (da) | 1989-07-12 |
WO1989004660A1 (en) | 1989-06-01 |
AU2626488A (en) | 1989-06-14 |
KR890701099A (ko) | 1989-12-19 |
DE3872872T2 (de) | 1993-02-04 |
US5098909A (en) | 1992-03-24 |
EP0340270B1 (en) | 1992-07-15 |
ATE78162T1 (de) | 1992-08-15 |
DK345889D0 (da) | 1989-07-12 |
EP0340270A1 (en) | 1989-11-08 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
AU616706B2 (en) | 5-ht3 receptor antagonists for treatment of cough and bronchoconstriction | |
Bohannon et al. | Vincristine in the treatment of lymphomas and leukemias | |
AU643075B2 (en) | 5HT-3 antagonists for the prevention or reduction of dependence | |
KR960008234B1 (ko) | 신경중독손상을 감소시키기 위한 약제 조성물 | |
RU2165760C2 (ru) | Применение антагонистов серотонина (5нт3) для лечения фибромиалгии | |
KR19990067527A (ko) | 동통의 치료를 위한 에피나스틴의 용도 | |
US5547964A (en) | Medical use for tachykinin antagonists | |
JPH10316567A (ja) | 過敏性腸症候群の症状の治療用のnk−1受容体アンタゴニスト | |
JPH08183735A (ja) | 不安症の治療 | |
EP0506813A1 (en) | 5-ht 3? antagonists for treatment of nausea, bradycardia of hypotension associated with myocardial instability | |
US5340826A (en) | Pharmaceutical agents for treatment of urinary incontinence | |
AU4043793A (en) | Agents for treating substance abuse disorders | |
NO315119B1 (no) | Heterocyklus-kondenserte morfin-derivater, anvendelse derav og farmasöytiske blandinger inneholdende dem | |
EP0421587A2 (en) | Xanthine derivatives used in asthma | |
JPS62424A (ja) | 医薬組成物 | |
AU758936B2 (en) | Method of treatment | |
AU657412B2 (en) | Agent for increasing somatostatin or for inhibiting decrease of somatostatin | |
AU626358B2 (en) | Antiemesis ergoline derivatives | |
CA2058258A1 (en) | Substituted benzene derivatives for use in the treatment of glaucoma | |
CA2296468A1 (en) | Treatment and prevention of cardiac disorders using selective serotonin re-uptake inhibitors (ssri) | |
US4904673A (en) | Agent for treating bradycardia and bradyarrhythmia | |
MXPA01000466A (en) | Method of treatment | |
CA2058249A1 (en) | Substituted pyridine derivatives for use in the treatment of glaucoma | |
JPH03502806A (ja) | ガンの処理 | |
JPH0881374A (ja) | 皮膚そう痒症の予防または治療薬 |