ATE394383T1 - Biphenylkarbonsäureamidderivate als p38 kinase- inhibitoren - Google Patents
Biphenylkarbonsäureamidderivate als p38 kinase- inhibitorenInfo
- Publication number
- ATE394383T1 ATE394383T1 AT02782928T AT02782928T ATE394383T1 AT E394383 T1 ATE394383 T1 AT E394383T1 AT 02782928 T AT02782928 T AT 02782928T AT 02782928 T AT02782928 T AT 02782928T AT E394383 T1 ATE394383 T1 AT E394383T1
- Authority
- AT
- Austria
- Prior art keywords
- kinase inhibitors
- biphenyl
- acid amide
- carbonic acid
- amide derivatives
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/81—Amides; Imides
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Physical Education & Sports Medicine (AREA)
- Immunology (AREA)
- Rheumatology (AREA)
- Pulmonology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Diabetes (AREA)
- Cardiology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
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- Urology & Nephrology (AREA)
- Heart & Thoracic Surgery (AREA)
- Psychology (AREA)
- Pain & Pain Management (AREA)
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- Dermatology (AREA)
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Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0124933.3A GB0124933D0 (en) | 2001-10-17 | 2001-10-17 | Chemical compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
ATE394383T1 true ATE394383T1 (de) | 2008-05-15 |
Family
ID=9924029
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT02782928T ATE394383T1 (de) | 2001-10-17 | 2002-10-16 | Biphenylkarbonsäureamidderivate als p38 kinase- inhibitoren |
Country Status (8)
Country | Link |
---|---|
US (2) | US7151118B2 (de) |
EP (1) | EP1436272B1 (de) |
JP (1) | JP2005508967A (de) |
AT (1) | ATE394383T1 (de) |
DE (1) | DE60226469D1 (de) |
ES (1) | ES2305317T3 (de) |
GB (1) | GB0124933D0 (de) |
WO (1) | WO2003033483A1 (de) |
Families Citing this family (35)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
PE20020506A1 (es) * | 2000-08-22 | 2002-07-09 | Glaxo Group Ltd | Derivados de pirazol fusionados como inhibidores de la proteina cinasa |
GB0124932D0 (en) * | 2001-10-17 | 2001-12-05 | Glaxo Group Ltd | Chemical compounds |
GB0124938D0 (en) * | 2001-10-17 | 2001-12-05 | Glaxo Group Ltd | Chemical compounds |
GB0124931D0 (en) * | 2001-10-17 | 2001-12-05 | Glaxo Group Ltd | Chemical compounds |
GB0124936D0 (en) * | 2001-10-17 | 2001-12-05 | Glaxo Group Ltd | Chemical compounds |
GB0124939D0 (en) * | 2001-10-17 | 2001-12-05 | Glaxo Group Ltd | Chemical compounds |
GB0124941D0 (en) * | 2001-10-17 | 2001-12-05 | Glaxo Group Ltd | Chemical compounds |
GB0124934D0 (en) * | 2001-10-17 | 2001-12-05 | Glaxo Group Ltd | Chemical compounds |
EP1474395B1 (de) * | 2002-02-12 | 2007-10-17 | Smithkline Beecham Corporation | Nicotinamide und deren verwendung als p38 inhibitoren |
GB0209891D0 (en) | 2002-04-30 | 2002-06-05 | Glaxo Group Ltd | Novel compounds |
GB0217757D0 (en) | 2002-07-31 | 2002-09-11 | Glaxo Group Ltd | Novel compounds |
US20040242572A1 (en) * | 2002-08-24 | 2004-12-02 | Boehringer Ingelheim International Gmbh | New carboxamide compounds having melanin concentrating hormone antagonistic activity, pharmaceutical preparations comprising these compounds and process for their manufacture |
GB0308186D0 (en) * | 2003-04-09 | 2003-05-14 | Smithkline Beecham Corp | Novel compounds |
GB0308201D0 (en) * | 2003-04-09 | 2003-05-14 | Smithkline Beecham Corp | Novel compounds |
GB0308185D0 (en) * | 2003-04-09 | 2003-05-14 | Smithkline Beecham Corp | Novel compounds |
EP1616862A4 (de) * | 2003-04-18 | 2008-07-16 | Ono Pharmaceutical Co | Stickstoffhaltige heterocyclische verbindung und deren verwendung |
PT1635824E (pt) | 2003-06-03 | 2009-11-24 | Novartis Ag | Inibidores de p-38 à base de heterociclos de 5 membros |
PT2298743E (pt) | 2003-06-26 | 2012-12-04 | Novartis Ag | Inibidores de p38 quinase a base de heterociclo de 5 elementos |
AU2004261589B2 (en) * | 2003-07-25 | 2008-05-22 | Novartis Ag | p-38 kinase inhibitors |
GB0318814D0 (en) * | 2003-08-11 | 2003-09-10 | Smithkline Beecham Corp | Novel compounds |
GB0402137D0 (en) * | 2004-01-30 | 2004-03-03 | Smithkline Beecham Corp | Novel compounds |
GB0402143D0 (en) * | 2004-01-30 | 2004-03-03 | Smithkline Beecham Corp | Novel compounds |
GB0402138D0 (en) * | 2004-01-30 | 2004-03-03 | Smithkline Beecham Corp | Novel compounds |
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-
2001
- 2001-10-17 GB GBGB0124933.3A patent/GB0124933D0/en not_active Ceased
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2002
- 2002-10-16 DE DE60226469T patent/DE60226469D1/de not_active Expired - Fee Related
- 2002-10-16 JP JP2003536223A patent/JP2005508967A/ja active Pending
- 2002-10-16 AT AT02782928T patent/ATE394383T1/de not_active IP Right Cessation
- 2002-10-16 WO PCT/EP2002/011572 patent/WO2003033483A1/en active IP Right Grant
- 2002-10-16 ES ES02782928T patent/ES2305317T3/es not_active Expired - Lifetime
- 2002-10-16 EP EP02782928A patent/EP1436272B1/de not_active Expired - Lifetime
- 2002-10-16 US US10/492,697 patent/US7151118B2/en not_active Expired - Fee Related
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2006
- 2006-11-03 US US11/556,285 patent/US7309800B2/en not_active Expired - Fee Related
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EP1436272B1 (de) | 2008-05-07 |
JP2005508967A (ja) | 2005-04-07 |
US7151118B2 (en) | 2006-12-19 |
EP1436272A1 (de) | 2004-07-14 |
US20070105860A1 (en) | 2007-05-10 |
US20050020540A1 (en) | 2005-01-27 |
US7309800B2 (en) | 2007-12-18 |
WO2003033483A1 (en) | 2003-04-24 |
ES2305317T3 (es) | 2008-11-01 |
DE60226469D1 (de) | 2008-06-19 |
GB0124933D0 (en) | 2001-12-05 |
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