ATE266012T1 - Thiazole derivate - Google Patents

Thiazole derivate

Info

Publication number: ATE266012T1
Authority: AT; Austria
Prior art keywords: thiazole derivatives; thiazole; derivatives
Prior art date: 1998-10-22

Application number

AT99970988T

Other languages

English (en)

Inventor

Leo Alig

Kurt Hilpert

Thomas Weller

Original Assignee

Hoffmann La Roche

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-10-22

Filing date

1999-10-15

Publication date

2004-05-15

1999-10-15 Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche

2004-05-15 Application granted granted Critical

2004-05-15 Publication of ATE266012T1 publication Critical patent/ATE266012T1/de

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/44—Acylated amino or imino radicals
- C07D277/48—Acylated amino or imino radicals by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof, e.g. carbonylguanidines
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

AT99970988T 1998-10-22 1999-10-15 Thiazole derivate ATE266012T1 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP98119985		1998-10-22
PCT/EP1999/007824 WO2000024724A1 (en)	1998-10-22	1999-10-15	Thiazole-derivatives

Publications (1)

Publication Number	Publication Date
ATE266012T1 true ATE266012T1 (de)	2004-05-15

Family

ID=8232838

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT99970988T ATE266012T1 (de)	1998-10-22	1999-10-15	Thiazole derivate

Country Status (31)

Country	Link
US (1)	US6297266B1 (de)
EP (1)	EP1123283B1 (de)
JP (1)	JP3530137B2 (de)
KR (1)	KR100469219B1 (de)
CN (1)	CN1211375C (de)
AR (1)	AR023058A1 (de)
AT (1)	ATE266012T1 (de)
AU (1)	AU760219B2 (de)
BR (1)	BR9914666A (de)
CA (1)	CA2347741C (de)
CO (1)	CO5150186A1 (de)
CZ (1)	CZ20011395A3 (de)
DE (1)	DE69917058T2 (de)
DK (1)	DK1123283T3 (de)
ES (1)	ES2221482T3 (de)
HK (1)	HK1047281A1 (de)
HR (1)	HRP20010275A2 (de)
HU (1)	HUP0104202A3 (de)
ID (1)	ID28356A (de)
IL (1)	IL142090A0 (de)
MA (1)	MA26756A1 (de)
NO (1)	NO20011908D0 (de)
NZ (1)	NZ510676A (de)
PE (1)	PE20001116A1 (de)
PL (1)	PL347427A1 (de)
PT (1)	PT1123283E (de)
RU (1)	RU2214404C2 (de)
TR (1)	TR200101115T2 (de)
WO (1)	WO2000024724A1 (de)
YU (1)	YU29201A (de)
ZA (1)	ZA200102653B (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
RU2312860C2 (ru)	1999-04-15	2007-12-20	Бристол-Маерс Сквибб Компани	Циклические ингибиторы протеинтирозинкиназ
US7125875B2 (en)	1999-04-15	2006-10-24	Bristol-Myers Squibb Company	Cyclic protein tyrosine kinase inhibitors
MXPA02007099A (es) *	2000-01-19	2004-08-23	Alteon Inc	Compuestos de tiazola, imidazola y oxazola y tratamientos de desordenes asociados con la maduracion de la proteina.
US6716995B2 (en)	2000-08-17	2004-04-06	Lumera Corporation	Design and synthesis of advanced NLO materials for electro-optic applications
ATE318812T1 (de)	2000-12-21	2006-03-15	Bristol Myers Squibb Co	Thiazolyl-inhibitoren von tyrosinkinasen der tec- familie
JP2008513386A (ja) *	2004-09-20	2008-05-01	４エスシーアーゲー	新規な複素環式ＮＦ−κＢ阻害剤
UA103319C2 (en)	2008-05-06	2013-10-10	Глаксосмитклайн Ллк	Thiazole- and oxazole-benzene sulfonamide compounds
WO2010012793A1 (en) *	2008-08-01	2010-02-04	Bayer Cropscience Sa	Fungicide aminothiazole derivatives

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IL95548A0 (en) *	1989-09-15	1991-06-30	Fujisawa Pharmaceutical Co	Thiazole derivatives,processes for the preparation thereof and pharmaceutical composition containing the same
US5273982A (en)	1990-03-09	1993-12-28	Hoffmann-La Roche Inc.	Acetic acid derivatives
CA2037153A1 (en) *	1990-03-09	1991-09-10	Leo Alig	Acetic acid derivatives
US6306840B1 (en) *	1995-01-23	2001-10-23	Biogen, Inc.	Cell adhesion inhibitors
JPH0987237A (ja) *	1995-09-21	1997-03-31	Kyowa Hakko Kogyo Co Ltd	芳香族誘導体
EP0928793B1 (de) *	1998-01-02	2002-05-15	F. Hoffmann-La Roche Ag	Thiazol-Derivate
EP0928790B1 (de) *	1998-01-02	2003-03-05	F. Hoffmann-La Roche Ag	Thiazole Derivate

1999
- 1999-10-15 AU AU11519/00A patent/AU760219B2/en not_active Ceased
- 1999-10-15 ES ES99970988T patent/ES2221482T3/es not_active Expired - Lifetime
- 1999-10-15 EP EP99970988A patent/EP1123283B1/de not_active Expired - Lifetime
- 1999-10-15 YU YU29201A patent/YU29201A/sh unknown
- 1999-10-15 PT PT99970988T patent/PT1123283E/pt unknown
- 1999-10-15 CN CNB998124265A patent/CN1211375C/zh not_active Expired - Fee Related
- 1999-10-15 CA CA002347741A patent/CA2347741C/en not_active Expired - Fee Related
- 1999-10-15 DK DK99970988T patent/DK1123283T3/da active
- 1999-10-15 WO PCT/EP1999/007824 patent/WO2000024724A1/en active IP Right Grant
- 1999-10-15 KR KR10-2001-7004899A patent/KR100469219B1/ko not_active IP Right Cessation
- 1999-10-15 AT AT99970988T patent/ATE266012T1/de not_active IP Right Cessation
- 1999-10-15 NZ NZ510676A patent/NZ510676A/xx unknown
- 1999-10-15 ID IDW20010863A patent/ID28356A/id unknown
- 1999-10-15 JP JP2000578294A patent/JP3530137B2/ja not_active Expired - Fee Related
- 1999-10-15 CZ CZ20011395A patent/CZ20011395A3/cs unknown
- 1999-10-15 TR TR2001/01115T patent/TR200101115T2/xx unknown
- 1999-10-15 BR BR9914666-5A patent/BR9914666A/pt not_active IP Right Cessation
- 1999-10-15 HU HU0104202A patent/HUP0104202A3/hu unknown
- 1999-10-15 DE DE69917058T patent/DE69917058T2/de not_active Expired - Fee Related
- 1999-10-15 IL IL14209099A patent/IL142090A0/xx unknown
- 1999-10-15 PL PL99347427A patent/PL347427A1/xx not_active Application Discontinuation
- 1999-10-15 RU RU2001113285/04A patent/RU2214404C2/ru not_active IP Right Cessation
- 1999-10-18 PE PE1999001048A patent/PE20001116A1/es not_active Application Discontinuation
- 1999-10-19 US US09/420,387 patent/US6297266B1/en not_active Expired - Fee Related
- 1999-10-20 AR ARP990105306A patent/AR023058A1/es not_active Application Discontinuation
- 1999-10-20 CO CO99066263A patent/CO5150186A1/es unknown
2001
- 2001-03-30 ZA ZA200102653A patent/ZA200102653B/en unknown
- 2001-04-12 HR HR20010275A patent/HRP20010275A2/hr not_active Application Discontinuation
- 2001-04-18 NO NO20011908A patent/NO20011908D0/no not_active Application Discontinuation
- 2001-04-20 MA MA26171A patent/MA26756A1/fr unknown
2002
- 2002-12-09 HK HK02108922.4A patent/HK1047281A1/zh unknown

Also Published As

Publication number	Publication date
CZ20011395A3 (cs)	2001-08-15
MA26756A1 (fr)	2004-12-20
CN1359381A (zh)	2002-07-17
ES2221482T3 (es)	2004-12-16
PE20001116A1 (es)	2000-10-27
TR200101115T2 (tr)	2002-01-21
PL347427A1 (en)	2002-04-08
RU2214404C2 (ru)	2003-10-20
YU29201A (sh)	2005-06-10
HUP0104202A3 (en)	2003-12-29
CO5150186A1 (es)	2002-04-29
DE69917058T2 (de)	2005-04-07
WO2000024724A1 (en)	2000-05-04
AR023058A1 (es)	2002-09-04
JP2002528442A (ja)	2002-09-03
HUP0104202A2 (hu)	2002-03-28
US6297266B1 (en)	2001-10-02
JP3530137B2 (ja)	2004-05-24
CN1211375C (zh)	2005-07-20
KR100469219B1 (ko)	2005-02-07
PT1123283E (pt)	2004-09-30
BR9914666A (pt)	2001-07-17
HK1047281A1 (zh)	2003-02-14
DE69917058D1 (de)	2004-06-09
NO20011908L (no)	2001-04-18
DK1123283T3 (da)	2004-09-13
NO20011908D0 (no)	2001-04-18
KR20010080243A (ko)	2001-08-22
AU1151900A (en)	2000-05-15
EP1123283B1 (de)	2004-05-06
ZA200102653B (en)	2002-07-01
HRP20010275A2 (en)	2002-06-30
IL142090A0 (en)	2002-03-10
CA2347741A1 (en)	2000-05-04
NZ510676A (en)	2003-06-30
AU760219B2 (en)	2003-05-08
EP1123283A1 (de)	2001-08-16
ID28356A (id)	2001-05-17
CA2347741C (en)	2006-12-12

Legal Events

Date

Code

Title

Description

2005-01-15

UEP

Publication of translation of european patent specification

Ref document number: 1123283

Country of ref document: EP

2007-07-15

REN

Ceased due to non-payment of the annual fee

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