ATE246681T1 - Sulfonamide - Google Patents

Sulfonamide

Info

Publication number
ATE246681T1
ATE246681T1 AT95941706T AT95941706T ATE246681T1 AT E246681 T1 ATE246681 T1 AT E246681T1 AT 95941706 T AT95941706 T AT 95941706T AT 95941706 T AT95941706 T AT 95941706T AT E246681 T1 ATE246681 T1 AT E246681T1
Authority
AT
Austria
Prior art keywords
pct
sec
compounds
date
endothelin
Prior art date
Application number
AT95941706T
Other languages
English (en)
Inventor
Volker Breu
Kaspar Burri
Jean-Marie Cassal
Martine Clozel
Georges Hirth
Bernd-Michael Loeffler
Marcel Mueller
Werner Neidhart
Henri Ramuz
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Application granted granted Critical
Publication of ATE246681T1 publication Critical patent/ATE246681T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/69—Benzenesulfonamido-pyrimidines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Cardiology (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Bipolar Transistors (AREA)
  • Surgical Instruments (AREA)
  • Lubricants (AREA)
  • Steroid Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
AT95941706T 1994-12-20 1995-12-08 Sulfonamide ATE246681T1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CH383794 1994-12-20
CH241995 1995-08-24
PCT/EP1995/004843 WO1996019459A1 (en) 1994-12-20 1995-12-08 Novel sulfonamides

Publications (1)

Publication Number Publication Date
ATE246681T1 true ATE246681T1 (de) 2003-08-15

Family

ID=25690401

Family Applications (1)

Application Number Title Priority Date Filing Date
AT95941706T ATE246681T1 (de) 1994-12-20 1995-12-08 Sulfonamide

Country Status (26)

Country Link
US (1) US6004965A (de)
EP (1) EP0799209B1 (de)
JP (1) JP2989014B2 (de)
KR (1) KR100445085B1 (de)
CN (1) CN1098254C (de)
AT (1) ATE246681T1 (de)
AU (1) AU701767B2 (de)
BR (1) BR9510104A (de)
CA (1) CA2208018C (de)
CY (1) CY2495B1 (de)
CZ (1) CZ287916B6 (de)
DE (1) DE69531457T2 (de)
DK (1) DK0799209T3 (de)
ES (1) ES2203649T3 (de)
FI (1) FI120397B (de)
HK (1) HK1001973A1 (de)
HU (1) HU228619B1 (de)
IL (1) IL116385A (de)
MA (1) MA23744A1 (de)
MY (1) MY131126A (de)
NO (1) NO316645B1 (de)
NZ (1) NZ297797A (de)
PT (1) PT799209E (de)
SA (1) SA95160421B1 (de)
TW (1) TW313568B (de)
WO (1) WO1996019459A1 (de)

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Also Published As

Publication number Publication date
CN1170407A (zh) 1998-01-14
DE69531457D1 (en) 2003-09-11
KR100445085B1 (ko) 2004-10-14
US6004965A (en) 1999-12-21
HUT77884A (hu) 1998-09-28
FI972628A (fi) 1997-06-18
AU4304196A (en) 1996-07-10
HK1001973A1 (en) 1998-07-24
IL116385A0 (en) 1996-03-31
WO1996019459A1 (en) 1996-06-27
CZ187497A3 (en) 1997-10-15
MX9704587A (es) 1998-07-31
SA95160421B1 (ar) 2006-05-01
FI120397B (fi) 2009-10-15
PT799209E (pt) 2003-12-31
JP2989014B2 (ja) 1999-12-13
ES2203649T3 (es) 2004-04-16
NZ297797A (en) 1999-10-28
NO972538L (no) 1997-06-04
NO316645B1 (no) 2004-03-22
CN1098254C (zh) 2003-01-08
AU701767B2 (en) 1999-02-04
MA23744A1 (fr) 1996-07-01
BR9510104A (pt) 1997-11-25
HU228619B1 (en) 2013-04-29
TW313568B (de) 1997-08-21
CA2208018C (en) 2007-03-27
EP0799209A1 (de) 1997-10-08
CY2495B1 (en) 2005-09-02
EP0799209B1 (de) 2003-08-06
DE69531457T2 (de) 2004-06-24
DK0799209T3 (da) 2003-11-24
MY131126A (en) 2007-07-31
NO972538D0 (no) 1997-06-04
IL116385A (en) 2000-07-16
CA2208018A1 (en) 1996-06-27
JPH10509182A (ja) 1998-09-08
CZ287916B6 (cs) 2001-03-14
FI972628A0 (fi) 1997-06-18

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