AR037407A1 - Composiciones farmaceuticas para el tratamiento de la diabetes mellitus de tipo ii - Google Patents

Composiciones farmaceuticas para el tratamiento de la diabetes mellitus de tipo ii

Info

Publication number
AR037407A1
AR037407A1 ARP020104498A ARP020104498A AR037407A1 AR 037407 A1 AR037407 A1 AR 037407A1 AR P020104498 A ARP020104498 A AR P020104498A AR P020104498 A ARP020104498 A AR P020104498A AR 037407 A1 AR037407 A1 AR 037407A1
Authority
AR
Argentina
Prior art keywords
treatment
pharmaceutical compositions
diabetes
mellitus type
type
Prior art date
Application number
ARP020104498A
Other languages
English (en)
Inventor
Alessandro Tosetti
Mauro Guiducci
Giovanni Viti
Original Assignee
Menarini Int Operations Lu Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=11442301&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR037407(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Menarini Int Operations Lu Sa filed Critical Menarini Int Operations Lu Sa
Publication of AR037407A1 publication Critical patent/AR037407A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/155Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/64Sulfonylureas, e.g. glibenclamide, tolbutamide, chlorpropamide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A61K9/209Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Composiciones farmacéuticas suministrables por vía oral en forma de comprimidos para el tratamiento de la diabetes mellitus de tipo II, que comprenden glibenclamida y metformina, o sus sales farmacéuticamente aceptables, como principios activos, mantenidos en forma separada entre ellos en el interior de la misma composición.
ARP020104498A 2001-11-29 2002-11-22 Composiciones farmaceuticas para el tratamiento de la diabetes mellitus de tipo ii AR037407A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT2001FI000230A ITFI20010230A1 (it) 2001-11-29 2001-11-29 Composizioni farmaceutiche per il trattamento del diabete mellito di tipo ii

Publications (1)

Publication Number Publication Date
AR037407A1 true AR037407A1 (es) 2004-11-10

Family

ID=11442301

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP020104498A AR037407A1 (es) 2001-11-29 2002-11-22 Composiciones farmaceuticas para el tratamiento de la diabetes mellitus de tipo ii

Country Status (40)

Country Link
US (1) US20050053661A1 (es)
EP (1) EP1458364B1 (es)
JP (1) JP4474162B2 (es)
KR (1) KR20040079898A (es)
CN (1) CN1596103B (es)
AR (1) AR037407A1 (es)
AT (1) ATE387190T1 (es)
AU (1) AU2002358061B2 (es)
BR (1) BR0214403A (es)
CA (1) CA2466677A1 (es)
CO (1) CO5590906A2 (es)
CY (1) CY1107966T1 (es)
DE (1) DE60225331T2 (es)
DK (1) DK1458364T3 (es)
EA (1) EA006766B1 (es)
EG (1) EG24124A (es)
ES (1) ES2302862T3 (es)
HK (1) HK1069974A1 (es)
HN (1) HN2002000341A (es)
HR (1) HRP20040501A2 (es)
HU (1) HUP0402154A3 (es)
IL (1) IL162143A0 (es)
IT (1) ITFI20010230A1 (es)
MA (1) MA27087A1 (es)
MX (1) MXPA04004974A (es)
MY (1) MY141243A (es)
NO (1) NO20042713L (es)
NZ (1) NZ533779A (es)
PA (1) PA8559801A1 (es)
PE (1) PE20030580A1 (es)
PL (1) PL206016B1 (es)
PT (1) PT1458364E (es)
RS (1) RS50937B (es)
SI (1) SI1458364T1 (es)
SV (1) SV2004001415A (es)
TN (1) TNSN04095A1 (es)
UA (1) UA81615C2 (es)
UY (1) UY27549A1 (es)
WO (1) WO2003045355A1 (es)
ZA (1) ZA200404880B (es)

Families Citing this family (30)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL362687A1 (en) * 2001-01-12 2004-11-02 Sun Pharmaceutical Industries Limited Spaced drug delivery system
US8911781B2 (en) 2002-06-17 2014-12-16 Inventia Healthcare Private Limited Process of manufacture of novel drug delivery system: multilayer tablet composition of thiazolidinedione and biguanides
US9060941B2 (en) 2002-09-20 2015-06-23 Actavis, Inc. Pharmaceutical formulation containing a biguanide and a thiazolidinedione derivative
US7785627B2 (en) 2002-09-20 2010-08-31 Watson Pharmaceuticals, Inc. Pharmaceutical formulation containing a biguanide and a thiazolidinedione derivative
DK2316456T3 (en) 2003-04-29 2017-09-11 Orexigen Therapeutics Inc Compositions for affecting weight loss comprising an opioid antagonist and bupropion
UY29445A1 (es) * 2005-03-30 2006-10-02 Generex Pharm Inc Composiciones para la transmisión transmucosa oral de la metformina
TWI471145B (zh) * 2005-06-13 2015-02-01 Bristol Myers Squibb & Gilead Sciences Llc 單一式藥學劑量型
KR101735466B1 (ko) * 2006-11-09 2017-05-15 오렉시젠 세러퓨틱스 인크. 신속하게 용해되는 중간층을 포함하는 층상의 약제학적 제형
ITMI20062254A1 (it) * 2006-11-24 2008-05-25 Acraf Uso di un acido metossi-alcanoico dell'indazolo per preparare una composizione farmaceutca
JP2011521973A (ja) 2008-05-30 2011-07-28 オレキシジェン・セラピューティクス・インコーポレーテッド 内臓脂肪の状態を処置するための方法
CA2638240C (en) 2008-08-29 2010-02-02 Alexander Macgregor Method of treating dysglycemia and glucose excursions
CN102724878A (zh) 2010-01-11 2012-10-10 奥雷西根治疗公司 在重度抑郁症患者中提供体重减轻疗法的方法
RU2483717C2 (ru) * 2010-11-22 2013-06-10 Открытое акционерное общество "Химико-фармацевтический комбинат "АКРИХИН" (ОАО "АКРИХИН") Фармацевтическая композиция для лечения диабета (варианты)
US11974971B2 (en) 2011-01-07 2024-05-07 Anji Pharmaceuticals Inc. Compositions and methods for treating metabolic disorders
US11759441B2 (en) 2011-01-07 2023-09-19 Anji Pharmaceuticals Inc. Biguanide compositions and methods of treating metabolic disorders
US9572784B2 (en) 2011-01-07 2017-02-21 Elcelyx Therapeutics, Inc. Compositions comprising statins, biguanides and further agents for reducing cardiometabolic risk
WO2013103919A2 (en) 2012-01-06 2013-07-11 Elcelyx Therapeutics, Inc. Compositions and methods for treating metabolic disorders
US8796338B2 (en) 2011-01-07 2014-08-05 Elcelyx Therapeutics, Inc Biguanide compositions and methods of treating metabolic disorders
KR20140035331A (ko) 2011-01-07 2014-03-21 엘셀릭스 테라퓨틱스 인코포레이티드 화학감각 수용체 리간드-기반 요법
US9211263B2 (en) 2012-01-06 2015-12-15 Elcelyx Therapeutics, Inc. Compositions and methods of treating metabolic disorders
US9480663B2 (en) 2011-01-07 2016-11-01 Elcelyx Therapeutics, Inc. Biguanide compositions and methods of treating metabolic disorders
KR102035879B1 (ko) 2012-01-06 2019-10-23 엘셀릭스 테라퓨틱스 인코포레이티드 바이구아나이드 조성물 및 대사 장애를 치료하는 방법
LT3730132T (lt) 2012-06-06 2022-08-25 Nalpropion Pharmaceuticals Llc Kompozicija, skirta panaudoti pacientų su didele širdies ir kraujagyslių ligų rizika antsvorio ir nutukimo gydymo būde
WO2016076280A1 (ja) 2014-11-11 2016-05-19 塩野義製薬株式会社 光に対して不安定な薬物を含有する多層錠剤
KR101750690B1 (ko) * 2015-10-28 2017-06-27 주식회사 종근당 메트포르민 및 로베글리타존을 포함하는 약제학적 조성물
CN105596339A (zh) * 2015-12-23 2016-05-25 青岛海之源智能技术有限公司 一种二甲双胍阿昔莫司复方组合物及制备方法
CN110128305A (zh) * 2019-05-10 2019-08-16 天津大学 二甲双胍-甲苯磺丁脲新盐型、其制备方法及医药用途
JP2021120357A (ja) * 2020-01-30 2021-08-19 サンノーバ株式会社 錠剤
GB2599950A (en) * 2020-10-16 2022-04-20 Zentiva Ks Pharmaceutical compositions with low amounts of nitrosamine impurities and methods for producing the same
CN113143940A (zh) * 2020-12-30 2021-07-23 成都恒瑞制药有限公司 一种抗糖尿病药物组合物的制备方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2347531A1 (de) * 1973-09-21 1975-04-30 Hoechst Ag Arzneizubereitungen zur oralen diabetes-behandlung
IT1276130B1 (it) * 1995-11-14 1997-10-27 Gentili Ist Spa Associazione glibenclamide-metformina, composizioni farmaceutiche che la contengono e loro uso nel trattamento del diabete mellito di tipo
NZ506202A (en) * 1998-03-19 2003-10-31 Bristol Myers Squibb Co Biphasic controlled release delivery system for high solubility pharmaceuticals and method
DK0974356T3 (da) * 1998-07-15 2003-10-27 Merck Sante Sas Tabletter omfattende en kombination af metformin og glibenclamid
US6780432B1 (en) * 2000-05-01 2004-08-24 Aeropharm Technology, Inc. Core formulation
PL362687A1 (en) * 2001-01-12 2004-11-02 Sun Pharmaceutical Industries Limited Spaced drug delivery system

Also Published As

Publication number Publication date
HUP0402154A3 (en) 2008-04-28
MY141243A (en) 2010-03-31
WO2003045355A1 (en) 2003-06-05
HUP0402154A2 (hu) 2005-02-28
PL206016B1 (pl) 2010-06-30
MA27087A1 (fr) 2004-12-20
ATE387190T1 (de) 2008-03-15
RS47304A (en) 2006-10-27
JP4474162B2 (ja) 2010-06-02
MXPA04004974A (es) 2004-08-11
HK1069974A1 (en) 2005-06-10
RS50937B (sr) 2010-08-31
SI1458364T1 (sl) 2008-08-31
PT1458364E (pt) 2008-05-26
JP2005518360A (ja) 2005-06-23
PE20030580A1 (es) 2003-09-05
PA8559801A1 (es) 2003-06-30
CY1107966T1 (el) 2013-09-04
ES2302862T3 (es) 2008-08-01
CO5590906A2 (es) 2005-12-30
EG24124A (en) 2008-07-07
AU2002358061A1 (en) 2003-06-10
CN1596103B (zh) 2010-06-16
DE60225331D1 (de) 2008-04-10
EA006766B1 (ru) 2006-04-28
AU2002358061B2 (en) 2007-01-11
DE60225331T2 (de) 2009-02-26
CA2466677A1 (en) 2003-06-05
NZ533779A (en) 2007-02-23
US20050053661A1 (en) 2005-03-10
IL162143A0 (en) 2005-11-20
DK1458364T3 (da) 2008-06-23
UY27549A1 (es) 2003-06-30
TNSN04095A1 (en) 2006-06-01
KR20040079898A (ko) 2004-09-16
EP1458364A1 (en) 2004-09-22
NO20042713L (no) 2004-07-16
EP1458364B1 (en) 2008-02-27
CN1596103A (zh) 2005-03-16
HRP20040501A2 (en) 2004-12-31
EA200400664A1 (ru) 2004-10-28
PL369851A1 (en) 2005-05-02
ITFI20010230A1 (it) 2003-05-29
ZA200404880B (en) 2005-07-29
HN2002000341A (es) 2009-12-07
SV2004001415A (es) 2004-05-07
UA81615C2 (ru) 2008-01-25
BR0214403A (pt) 2004-10-19

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