AR030045A1 - Composicion farmaceutica que contiene compuestos antibioticos de azalida , metodos para obtencion - Google Patents

Composicion farmaceutica que contiene compuestos antibioticos de azalida , metodos para obtencion

Info

Publication number
AR030045A1
AR030045A1 ARP010100319A ARP010100319A AR030045A1 AR 030045 A1 AR030045 A1 AR 030045A1 AR P010100319 A ARP010100319 A AR P010100319A AR P010100319 A ARP010100319 A AR P010100319A AR 030045 A1 AR030045 A1 AR 030045A1
Authority
AR
Argentina
Prior art keywords
azalida
obtaining
methods
pharmaceutical composition
composition containing
Prior art date
Application number
ARP010100319A
Other languages
English (en)
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22652702&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR030045(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of AR030045A1 publication Critical patent/AR030045A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Virology (AREA)
  • Pulmonology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

Composiciones antibioticas que comprende una mezcla de equilibrio de isomeros de azalida, agua y uno o más ácidos y método para preparar estas composiciones. Las composiciones antibioticas pueden estabilizarse de modo ventajoso mediante la adicion de uno o más codisolventes miscibles en agua. En una realizacion preferida. Dicho uno o más codisolventes es el propilenglicol. Una composicion que comprende: (a) el compuesto de formula 1; y el compuesto de formula 2 en una proporcion desde aproximadamente 90% + o - 4% a aproximadamente 10% + o - 4%, respectivamente, (b) agua; y (c) uno o más ácidos presentes a una concentracion total desde aproximadamente 0,2 mmol a aproximadamente 1,0 mmol por ml de la composicion.
ARP010100319A 2000-01-27 2001-01-25 Composicion farmaceutica que contiene compuestos antibioticos de azalida , metodos para obtencion AR030045A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US17848100P 2000-01-27 2000-01-27

Publications (1)

Publication Number Publication Date
AR030045A1 true AR030045A1 (es) 2003-08-13

Family

ID=22652702

Family Applications (2)

Application Number Title Priority Date Filing Date
ARP010100319A AR030045A1 (es) 2000-01-27 2001-01-25 Composicion farmaceutica que contiene compuestos antibioticos de azalida , metodos para obtencion
ARP030101210A AR039387A2 (es) 2000-01-27 2003-04-07 Compuestos antibioticos de azalida

Family Applications After (1)

Application Number Title Priority Date Filing Date
ARP030101210A AR039387A2 (es) 2000-01-27 2003-04-07 Compuestos antibioticos de azalida

Country Status (21)

Country Link
US (2) US6514945B1 (es)
EP (1) EP1250343B1 (es)
JP (2) JP3893059B2 (es)
AR (2) AR030045A1 (es)
AT (1) ATE243703T1 (es)
AU (1) AU779748C (es)
BR (2) BRPI0017013B1 (es)
CA (1) CA2398485C (es)
CO (1) CO5251404A1 (es)
DE (1) DE60003586T2 (es)
DK (1) DK1250343T3 (es)
ES (1) ES2199884T3 (es)
MX (1) MXPA02007305A (es)
NZ (1) NZ518665A (es)
PA (1) PA8509801A1 (es)
PE (1) PE20011050A1 (es)
PT (1) PT1250343E (es)
TN (1) TNSN01017A1 (es)
TW (2) TWI318880B (es)
WO (1) WO2001055158A1 (es)
ZA (1) ZA200205958B (es)

Families Citing this family (41)

* Cited by examiner, † Cited by third party
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JP2003040782A (ja) * 2001-05-31 2003-02-13 Pfizer Prod Inc アザリド抗生物質組成物
AU2002317415A1 (en) * 2001-08-01 2003-02-17 Pfizer Products Inc. Azalide antibiotic compositions
US7312248B2 (en) 2004-09-23 2007-12-25 Schering-Plough Animal Health Corporation Control of parasites in animals by the use of novel trifluoromethanesulfonanilide oxime ether derivatives
ATE446677T1 (de) * 2004-11-19 2009-11-15 Schering Plough Ltd Kontrolle von parasiten bei tieren mittels verwendung von parasitiziden 2-phenyl-3-(1h- pyrrol-2-yl) acrylonitril-derivaten
EP1890547A2 (en) * 2005-06-09 2008-02-27 Schering-Plough Ltd. Control of parasites in animals by n-[(phenyloxy)phenyl]-1,1,1-trifluoromethanesulfonamide and n-[(phenylsulfanyl)phenyl]-1,1,1-trifluoromethanesulfonamide derivatives
US8119667B2 (en) * 2005-12-29 2012-02-21 Schering-Plough Animal Health Corporation Carbonates of fenicol antibiotics
US20070238700A1 (en) * 2006-04-10 2007-10-11 Winzenberg Kevin N N-phenyl-1,1,1-trifluoromethanesulfonamide hydrazone derivative compounds and their usage in controlling parasites
US20080044455A1 (en) * 2006-08-21 2008-02-21 Chaim Welczer Tonsillitus Treatment
US8044230B2 (en) * 2006-12-13 2011-10-25 Intervet Inc. Water-soluble prodrugs of chloramphenicol, thiamphenicol, and analogs thereof
EP2091909A1 (en) * 2006-12-13 2009-08-26 Schering-Plough Ltd. Water-soluble prodrugs of florfenicol and its analogs
TWI430995B (zh) 2007-06-26 2014-03-21 Du Pont 萘異唑啉無脊椎有害動物控制劑
MX2009013748A (es) 2007-06-27 2010-01-26 Du Pont Metodo de control de plagas en animales.
US7795231B2 (en) * 2007-10-04 2010-09-14 Insite Vision Incorporated Concentrated aqueous azalide formulations
TWI468407B (zh) 2008-02-06 2015-01-11 Du Pont 中離子農藥
EP2321269B1 (en) * 2008-07-30 2018-09-19 Intervet International B.V. Process for preparing oxazoline-protected aminodiol compounds useful as intermediates to florfenicol
EP2462125A2 (en) 2009-08-05 2012-06-13 E. I. du Pont de Nemours and Company Mesoionic pesticides
CN102686570A (zh) 2009-08-05 2012-09-19 杜邦公司 介离子杀虫剂
UA107804C2 (en) 2009-08-05 2015-02-25 Du Pont Mixtures of pesticides mezoionnyh
UA110924C2 (uk) 2009-08-05 2016-03-10 Е. І. Дю Пон Де Немур Енд Компані Мезоіонні пестициди
UA108881C2 (xx) 2010-05-27 2015-06-25 Кристалічна форма 4-$5-$3-хлор-5-(трифторметил)феніл]-4,5-дигідро-5-(трифторметил)-3-ізоксазоліл]-n-$2-оксо-2-$(2,2,2-трифторетил)аміно]етил]-1-нафталінкарбоксаміду
EP4324524A2 (en) 2010-07-01 2024-02-21 Elanco Tiergesundheit AG Antibiotic compositions
BR112013001557A2 (pt) * 2010-07-23 2016-06-14 Acea Biotech Inc composto, composição farmacêutica, métodos para produzir composto e para tratar ou inibir infecção fúngica e/ou parasítica em sujeito e usos de composto e de composição farmacêutica
WO2012087630A1 (en) 2010-12-20 2012-06-28 E.I. Du Pont De Nemours And Company Pyridine and pyrimidine compounds for controlling invertebrate
WO2012177668A1 (en) 2011-06-20 2012-12-27 E. I. Du Pont De Nemours And Company Heterocyclic compounds for treating helminth infections
EP2736915A1 (en) 2011-07-27 2014-06-04 Farma GRS, d.o.o. New crystalline forms of tulathromycin
EP2776667B1 (en) 2011-11-11 2022-03-02 ExxonMobil Upstream Research Company Method and system for reservoir surveillance utilizing clumped isotope and noble gas data
US10330659B2 (en) 2011-11-11 2019-06-25 Exxonmobil Upstream Research Company Method for determining the location, size, and fluid composition of a subsurface hydrocarbon accumulation
CA2855001A1 (en) 2011-11-28 2013-06-06 E.I. Du Pont De Nemours And Company N- (4 -quinolinylmethyl) sulfonamide derivatives and their use as anthelmintics
WO2013158422A1 (en) 2012-04-17 2013-10-24 E. I. Du Pont De Nemours And Company Heterocyclic compounds for controlling invertebrate pests
WO2014099837A1 (en) 2012-12-18 2014-06-26 E. I. Du Pont De Nemours And Company Sulfonamide anthelmintics
US9044508B2 (en) * 2013-03-15 2015-06-02 Insite Vision Corporation Concentrated aqueous azalide formulations
MX2015014026A (es) 2013-04-04 2016-08-03 Harvard College Macrolidos y metodos para su preparacion y uso.
CN103588833B (zh) * 2013-10-30 2016-08-17 北京科技大学 动物抗菌素泰拉霉素的制备方法
RU2634793C1 (ru) 2014-03-07 2017-11-03 Эксонмобил Апстрим Рисерч Компани Способ разведки и система для обнаружения углеводородов по водяному столбу
CN104119413B (zh) * 2014-07-29 2016-08-24 华中农业大学 一种土拉霉素残留标示物的合成方法
JP2017531663A (ja) 2014-10-08 2017-10-26 プレジデント アンド フェローズ オブ ハーバード カレッジ １４員ケトライドならびにそれらの調製および使用の方法
JP2018509452A (ja) 2015-03-25 2018-04-05 プレジデント アンド フェローズ オブ ハーバード カレッジ 修飾デソサミン糖をもつマクロライドおよびその使用
EP3406619B1 (en) * 2016-01-18 2020-11-25 Zhejiang Hisun Pharmaceutical Co., Ltd. Method and intermediate for preparing tulathromycin
JP2022507795A (ja) * 2018-11-19 2022-01-18 ジカニ セラピューティクス， インコーポレイテッド Ｃ１０環状置換１３員マクロライド及びそれらの使用
KR20220156570A (ko) 2020-03-12 2022-11-25 조에티스 서비시즈 엘엘씨 면역조절성 유레아 아잘라이드
KR20240056746A (ko) 2021-09-07 2024-04-30 조에티스 서비시즈 엘엘씨 면역조정성 아잘라이드

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HN1998000074A (es) * 1997-06-11 1999-01-08 Pfizer Prod Inc Derivados de macrolidos c-4 sustituidos
HN1998000086A (es) * 1997-06-11 1999-03-08 Pfizer Prod Inc Derivados de 9 - desofo - 9 aza - 9a - homoeritromicina a - c - 4 sustituidos.
US6128174A (en) 1997-08-29 2000-10-03 Stereotaxis, Inc. Method and apparatus for rapidly changing a magnetic field produced by electromagnets
EP1011689B8 (en) * 1997-09-10 2007-05-09 Merial Ltd. USE OF 9a-AZALIDES AS VETERINARY ANTIMICROBIAL AGENTS
OA11876A (en) * 1999-05-18 2006-03-27 Pfizer Prod Inc Novel crystalline forms of a macrolide antibiotic.

Also Published As

Publication number Publication date
TWI318880B (en) 2010-01-01
AU1722801A (en) 2001-08-07
PA8509801A1 (es) 2002-02-21
ATE243703T1 (de) 2003-07-15
EP1250343A1 (en) 2002-10-23
NZ518665A (en) 2005-02-25
TNSN01017A1 (fr) 2005-11-10
DE60003586T2 (de) 2004-01-08
AU779748B2 (en) 2005-02-10
AU779748C (en) 2005-12-08
BRPI0017013B1 (pt) 2015-07-14
PE20011050A1 (es) 2001-10-19
BR0017013A2 (pt) 2010-07-13
BRPI0017013B8 (pt) 2022-11-16
EP1250343B1 (en) 2003-06-25
MXPA02007305A (es) 2002-11-29
TW201006476A (en) 2010-02-16
US6514945B1 (en) 2003-02-04
JP2006282676A (ja) 2006-10-19
WO2001055158A1 (en) 2001-08-02
CA2398485C (en) 2008-01-29
TWI331527B (en) 2010-10-11
AR039387A2 (es) 2005-02-16
PT1250343E (pt) 2003-11-28
DE60003586D1 (de) 2003-07-31
JP2004500384A (ja) 2004-01-08
ES2199884T3 (es) 2004-03-01
JP3893059B2 (ja) 2007-03-14
US20030073825A1 (en) 2003-04-17
DK1250343T3 (da) 2003-09-22
ZA200205958B (en) 2003-09-29
US6667393B2 (en) 2003-12-23
CO5251404A1 (es) 2003-02-28
BR0017013A (pt) 2002-10-22
US20030013860A1 (en) 2003-01-16
CA2398485A1 (en) 2001-08-02

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