ZA200410102B - Use of nefopam for the treatment of nausea or emesis - Google Patents
Use of nefopam for the treatment of nausea or emesis Download PDFInfo
- Publication number
- ZA200410102B ZA200410102B ZA200410102A ZA200410102A ZA200410102B ZA 200410102 B ZA200410102 B ZA 200410102B ZA 200410102 A ZA200410102 A ZA 200410102A ZA 200410102 A ZA200410102 A ZA 200410102A ZA 200410102 B ZA200410102 B ZA 200410102B
- Authority
- ZA
- South Africa
- Prior art keywords
- use according
- condition
- nefopam
- induced
- emesis
- Prior art date
Links
- RGPDEAGGEXEMMM-UHFFFAOYSA-N Nefopam Chemical compound C12=CC=CC=C2CN(C)CCOC1C1=CC=CC=C1 RGPDEAGGEXEMMM-UHFFFAOYSA-N 0.000 title claims description 24
- 229960000751 nefopam Drugs 0.000 title claims description 23
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- 206010028813 Nausea Diseases 0.000 title claims description 4
- 230000008693 nausea Effects 0.000 title claims description 4
- LNEPOXFFQSENCJ-UHFFFAOYSA-N haloperidol Chemical compound C1CC(O)(C=2C=CC(Cl)=CC=2)CCN1CCCC(=O)C1=CC=C(F)C=C1 LNEPOXFFQSENCJ-UHFFFAOYSA-N 0.000 claims description 6
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- UUVWYPNAQBNQJQ-UHFFFAOYSA-N hexamethylmelamine Chemical compound CN(C)C1=NC(N(C)C)=NC(N(C)C)=N1 UUVWYPNAQBNQJQ-UHFFFAOYSA-N 0.000 description 1
- OROGSEYTTFOCAN-UHFFFAOYSA-N hydrocodone Natural products C1C(N(CCC234)C)C2C=CC(O)C3OC2=C4C1=CC=C2OC OROGSEYTTFOCAN-UHFFFAOYSA-N 0.000 description 1
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- SGDBTWWWUNNDEQ-LBPRGKRZSA-N melphalan Chemical compound OC(=O)[C@@H](N)CC1=CC=C(N(CCCl)CCCl)C=C1 SGDBTWWWUNNDEQ-LBPRGKRZSA-N 0.000 description 1
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- 238000012544 monitoring process Methods 0.000 description 1
- JCSREICEMHWFAY-HUUCEWRRSA-N naxagolide Chemical compound C1=C(O)C=C2[C@H]3OCCN(CCC)[C@@H]3CCC2=C1 JCSREICEMHWFAY-HUUCEWRRSA-N 0.000 description 1
- 229950005651 naxagolide Drugs 0.000 description 1
- 229960001800 nefazodone Drugs 0.000 description 1
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- 229960002340 pentostatin Drugs 0.000 description 1
- FPVKHBSQESCIEP-JQCXWYLXSA-N pentostatin Chemical compound C1[C@H](O)[C@@H](CO)O[C@H]1N1C(N=CNC[C@H]2O)=C2N=C1 FPVKHBSQESCIEP-JQCXWYLXSA-N 0.000 description 1
- 229960004851 pergolide Drugs 0.000 description 1
- YEHCICAEULNIGD-MZMPZRCHSA-N pergolide Chemical compound C1=CC([C@H]2C[C@@H](CSC)CN([C@@H]2C2)CCC)=C3C2=CNC3=C1 YEHCICAEULNIGD-MZMPZRCHSA-N 0.000 description 1
- 230000003389 potentiating effect Effects 0.000 description 1
- 238000002360 preparation method Methods 0.000 description 1
- 229960000624 procarbazine Drugs 0.000 description 1
- CPTBDICYNRMXFX-UHFFFAOYSA-N procarbazine Chemical compound CNNCC1=CC=C(C(=O)NC(C)C)C=C1 CPTBDICYNRMXFX-UHFFFAOYSA-N 0.000 description 1
- 229940002612 prodrug Drugs 0.000 description 1
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- 239000011780 sodium chloride Substances 0.000 description 1
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- ZSJLQEPLLKMAKR-GKHCUFPYSA-N streptozocin Chemical compound O=NN(C)C(=O)N[C@H]1[C@@H](O)O[C@H](CO)[C@@H](O)[C@@H]1O ZSJLQEPLLKMAKR-GKHCUFPYSA-N 0.000 description 1
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- PNVNVHUZROJLTJ-UHFFFAOYSA-N venlafaxine Chemical compound C1=CC(OC)=CC=C1C(CN(C)C)C1(O)CCCCC1 PNVNVHUZROJLTJ-UHFFFAOYSA-N 0.000 description 1
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/5545—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having eight-membered rings not containing additional condensed or non-condensed nitrogen-containing 3-7 membered rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
Landscapes
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pain & Pain Management (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Hospice & Palliative Care (AREA)
- Otolaryngology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0213869.1A GB0213869D0 (en) | 2002-06-17 | 2002-06-17 | The treatment of pain |
Publications (1)
Publication Number | Publication Date |
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ZA200410102B true ZA200410102B (en) | 2006-07-26 |
Family
ID=9938718
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ZA200410102A ZA200410102B (en) | 2002-06-17 | 2004-12-14 | Use of nefopam for the treatment of nausea or emesis |
Country Status (15)
Country | Link |
---|---|
US (2) | US20060040905A1 (fr) |
EP (2) | EP1513518A1 (fr) |
JP (2) | JP2005533784A (fr) |
CN (1) | CN100482221C (fr) |
AU (2) | AU2003240113B2 (fr) |
BR (1) | BR0311874A (fr) |
CA (2) | CA2489306A1 (fr) |
GB (1) | GB0213869D0 (fr) |
IL (1) | IL165773A0 (fr) |
MX (1) | MXPA04012826A (fr) |
NO (1) | NO20045496L (fr) |
NZ (1) | NZ537197A (fr) |
PL (1) | PL374418A1 (fr) |
WO (2) | WO2003105832A1 (fr) |
ZA (1) | ZA200410102B (fr) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0330049D0 (en) * | 2003-12-24 | 2004-02-04 | Arakis Ltd | The treatment of neuropathic pain conditions |
GB0408864D0 (en) * | 2004-04-21 | 2004-05-26 | Arakis Ltd | Novel benzoxazocines |
GB0515703D0 (en) * | 2005-07-29 | 2005-09-07 | Arakis Ltd | Therapeutic use of nefopam |
WO2009002933A1 (fr) * | 2007-06-22 | 2008-12-31 | Hydra Biosciences, Inc. | Procédés et compositions pour le traitement de troubles |
GB0721013D0 (en) | 2007-10-25 | 2007-12-05 | Sosei R & D Ltd | New Salts |
PT2293794E (pt) | 2008-05-27 | 2013-07-10 | Univ Melbourne | Métodos de tratamento de mamíferos com disfunções da trompa de eustáquio |
US20110092493A1 (en) * | 2008-09-24 | 2011-04-21 | Clark Levi | Dose-controlled transdermal promethazine compositions and methods of use |
CN102458400B (zh) | 2009-05-20 | 2014-10-08 | 国立健康与医学研究所 | 用于治疗病灶性前庭功能障碍的血清素5-ht3受体拮抗剂 |
US8957107B2 (en) * | 2009-12-15 | 2015-02-17 | The Hospital For Sick Children | Method of treating scars and β-catenin-mediated disorders using Nefopam compounds |
EP4335508A3 (fr) | 2016-04-14 | 2024-07-10 | Sensorion | (+)-azasetron destiné à être utilisé dans le traitement de troubles de l'oreille |
US10736905B1 (en) | 2016-09-09 | 2020-08-11 | Shahin Fatholahi | Nefopam dosage forms and methods of treatment |
US10736874B1 (en) | 2017-09-08 | 2020-08-11 | Shahin Fatholahi | Methods for treating pain associated with sickle cell disease |
US11446311B2 (en) | 2017-09-08 | 2022-09-20 | Shahin Fatholahi | Methods for treating pain associated with sickle cell disease |
RS65140B1 (sr) * | 2019-05-06 | 2024-02-29 | Chemcom Sa | Upotreba kompozicije protiv neprijatnih mirisa i povezani postupak |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
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ES2234266T3 (es) * | 1998-07-24 | 2005-06-16 | Jago Research Ag | Formulaciones medicas para aerosoles. |
US20020013331A1 (en) * | 2000-06-26 | 2002-01-31 | Williams Robert O. | Methods and compositions for treating pain of the mucous membrane |
-
2002
- 2002-06-17 GB GBGB0213869.1A patent/GB0213869D0/en not_active Ceased
-
2003
- 2003-06-17 WO PCT/GB2003/002586 patent/WO2003105832A1/fr active Application Filing
- 2003-06-17 EP EP03740737A patent/EP1513518A1/fr not_active Withdrawn
- 2003-06-17 CA CA002489306A patent/CA2489306A1/fr not_active Abandoned
- 2003-06-17 CN CNB038167050A patent/CN100482221C/zh not_active Expired - Fee Related
- 2003-06-17 US US10/517,882 patent/US20060040905A1/en not_active Abandoned
- 2003-06-17 WO PCT/GB2003/002618 patent/WO2003105833A1/fr active Application Filing
- 2003-06-17 MX MXPA04012826A patent/MXPA04012826A/es unknown
- 2003-06-17 EP EP03732727A patent/EP1513517A1/fr not_active Withdrawn
- 2003-06-17 NZ NZ537197A patent/NZ537197A/en unknown
- 2003-06-17 US US10/517,881 patent/US20060063753A1/en not_active Abandoned
- 2003-06-17 AU AU2003240113A patent/AU2003240113B2/en not_active Ceased
- 2003-06-17 BR BR0311874-6A patent/BR0311874A/pt not_active IP Right Cessation
- 2003-06-17 JP JP2004512736A patent/JP2005533784A/ja active Pending
- 2003-06-17 CA CA002489315A patent/CA2489315A1/fr not_active Abandoned
- 2003-06-17 JP JP2004512737A patent/JP2005531612A/ja active Pending
- 2003-06-17 AU AU2003277077A patent/AU2003277077B2/en not_active Ceased
- 2003-06-17 PL PL03374418A patent/PL374418A1/xx not_active Application Discontinuation
-
2004
- 2004-12-14 IL IL16577304A patent/IL165773A0/xx unknown
- 2004-12-14 ZA ZA200410102A patent/ZA200410102B/en unknown
- 2004-12-16 NO NO20045496A patent/NO20045496L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
NZ537197A (en) | 2007-10-26 |
AU2003240113A1 (en) | 2003-12-31 |
PL374418A1 (en) | 2005-10-17 |
MXPA04012826A (es) | 2005-03-31 |
JP2005531612A (ja) | 2005-10-20 |
WO2003105833A1 (fr) | 2003-12-24 |
JP2005533784A (ja) | 2005-11-10 |
US20060040905A1 (en) | 2006-02-23 |
IL165773A0 (en) | 2006-01-15 |
AU2003277077A1 (en) | 2003-12-31 |
CA2489306A1 (fr) | 2003-12-24 |
EP1513517A1 (fr) | 2005-03-16 |
NO20045496L (no) | 2005-01-12 |
AU2003277077B2 (en) | 2006-11-02 |
CA2489315A1 (fr) | 2003-12-24 |
EP1513518A1 (fr) | 2005-03-16 |
CN1668294A (zh) | 2005-09-14 |
GB0213869D0 (en) | 2002-07-31 |
AU2003240113B2 (en) | 2006-11-16 |
BR0311874A (pt) | 2005-05-10 |
CN100482221C (zh) | 2009-04-29 |
US20060063753A1 (en) | 2006-03-23 |
WO2003105832A1 (fr) | 2003-12-24 |
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