YU264072A - Process for preparing penicillins - Google Patents

Process for preparing penicillins

Info

Publication number: YU264072A
Authority: YU; Yugoslavia
Prior art keywords: penicillins; preparing; preparing penicillins
Prior art date: 1971-10-23

Application number

YU02640/72A

Inventor

Koenig Hans-Bodo

Hans-Bodo Koenig

Schroeck Wilfried

Wilfried Schroeck

Metzger Karl-Georg

Karl-Georg Metzger

Original Assignee

Bayer Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1971-10-23

Filing date

1972-10-23

Publication date

1982-06-18

1972-10-23 Application filed by Bayer Ag filed Critical Bayer Ag

1982-06-18 Publication of YU264072A publication Critical patent/YU264072A/en

Links

229930182555 Penicillin Natural products 0.000 title 1
238000004519 manufacturing process Methods 0.000 title 1
150000002960 penicillins Chemical class 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/06—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D239/08—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms directly attached in position 2
- C07D239/10—Oxygen or sulfur atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/06—Anabolic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/30—Oxygen or sulfur atoms
- C07D233/32—One oxygen atom
- C07D233/38—One oxygen atom with acyl radicals or hetero atoms directly attached to ring nitrogen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
- C07D275/02—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/30—Hetero atoms other than halogen
- C07D333/34—Sulfur atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/10—Compounds having one or more C—Si linkages containing nitrogen having a Si-N linkage

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Oncology (AREA)
Communicable Diseases (AREA)
Endocrinology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Neurology (AREA)
Orthopedic Medicine & Surgery (AREA)
Physical Education & Sports Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Fodder In General (AREA)

YU02640/72A 1971-10-23 1972-10-23 Process for preparing penicillins YU264072A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE2152967A DE2152967C3 (en)	1971-10-23	1971-10-23	Acylureidopenicillins

Publications (1)

Publication Number	Publication Date
YU264072A true YU264072A (en)	1982-06-18

Family

ID=5823251

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
YU02640/72A YU264072A (en)	1971-10-23	1972-10-23	Process for preparing penicillins

Country Status (31)

Country	Link
JP (2)	JPS57843B2 (en)
AR (1)	AR195805A1 (en)
AT (1)	AT320152B (en)
BE (1)	BE790440A (en)
BG (2)	BG21609A3 (en)
CA (1)	CA1019323A (en)
CH (1)	CH579089A5 (en)
CS (1)	CS188883B2 (en)
CY (1)	CY947A (en)
DD (1)	DD106044B3 (en)
DE (1)	DE2152967C3 (en)
DK (1)	DK134992C (en)
EG (1)	EG10826A (en)
ES (1)	ES407851A1 (en)
FI (1)	FI56839C (en)
FR (1)	FR2157908B1 (en)
GB (1)	GB1392849A (en)
HK (1)	HK18578A (en)
HU (1)	HU167986B (en)
IE (1)	IE37123B1 (en)
IL (1)	IL40628A (en)
KE (1)	KE2824A (en)
LU (1)	LU66332A1 (en)
NO (1)	NO143909C (en)
PH (1)	PH9893A (en)
PL (2)	PL93574B1 (en)
RO (2)	RO63066A (en)
SE (1)	SE412236B (en)
SU (1)	SU527139A3 (en)
YU (1)	YU264072A (en)
ZA (1)	ZA727473B (en)

Families Citing this family (37)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3972870A (en) *	1971-10-23	1976-08-03	Bayer Aktiengesellschaft	Penicillins
NL175419C (en) *	1971-10-23	1984-11-01	Bayer Ag	METHOD FOR PREPARING OR MANUFACTURING ANTIBIOTIC ACTIVE PHARMACEUTICAL PREPARATIONS AND METHOD FOR PREPARING ANTIBIOTIC ACTIVE ALPHA-SUBSTITUTED 6- (ALFA- (3-ACYLUREIDO) -PETYL-ACIDYL-ACIDYL-ACIDYL)
US3978056A (en) *	1971-10-23	1976-08-31	Bayer Aktiengesellschaft	Penicillins
US4009272A (en) *	1971-10-23	1977-02-22	Bayer Aktiengesellschaft	Penicillins
US3974142A (en) *	1971-10-23	1976-08-10	Bayer Aktiengesellschaft	Penicillins
US3972869A (en) *	1971-10-23	1976-08-03	Bayer Aktiengesellschaft	Penicillins
US3974141A (en) *	1971-10-23	1976-08-10	Bayer Aktiengesellschaft	Penicillins
US3983105A (en) *	1971-10-23	1976-09-28	Bayer Aktiengesellschaft	Penicillins
DE2258973A1 (en) *	1972-12-01	1974-06-06	Bayer Ag	PENICILLIN, THE METHOD FOR MANUFACTURING IT AND THEIR USE AS A MEDICINAL PRODUCT
JPS587637B2 (en) *	1973-12-27	1983-02-10	住友化学工業株式会社	Shinkipenicillin no Seihou
DE2407715C2 (en) *	1974-02-18	1982-12-02	Bayer Ag, 5090 Leverkusen	Cephalosporins, processes for their production, as well as pharmaceuticals
IL47168A (en) *	1974-05-09	1979-07-25	Toyama Chemical Co Ltd	Mono or dioxo piperazino(thio)carbonylamino derivatives ofpenicillins and cephalosporins and process for producing the same
DE2525541C2 (en) *	1975-06-07	1984-01-12	Bayer Ag, 5090 Leverkusen	β-lactam antibiotics, processes for their preparation and pharmaceuticals containing them
DE2810083A1 (en)	1978-03-08	1979-09-20	Bayer Ag	BETA-LACTAM COMPOUNDS
GB0420722D0 (en)	2004-09-17	2004-10-20	Addex Pharmaceuticals Sa	Novel allosteric modulators
EP1780213A1 (en)	2005-10-27	2007-05-02	3M Innovative Properties Company	Silicon-urea-azolides, their preparation and use in the preparation of silicones with isocyanate terminal groups
AR059898A1 (en)	2006-03-15	2008-05-07	Janssen Pharmaceutica Nv	DERIVATIVES OF 3-CIANO-PIRIDONA 1,4-DISUSTITUTED AND ITS USE AS ALLOSTERIC MODULATORS OF MGLUR2 RECEIVERS
TW200845978A (en)	2007-03-07	2008-12-01	Janssen Pharmaceutica Nv	3-cyano-4-(4-tetrahydropyran-phenyl)-pyridin-2-one derivatives
TW200900065A (en)	2007-03-07	2009-01-01	Janssen Pharmaceutica Nv	3-cyano-4-(4-pyridinyloxy-phenyl)-pyridin-2-one derivatives
US8252937B2 (en)	2007-09-14	2012-08-28	Janssen Pharmaceuticals, Inc.	1,3-disubstituted 4-(aryl-X-phenyl)-1H-pyridin-2-ones
AU2008297877C1 (en)	2007-09-14	2013-11-07	Addex Pharma S.A.	1,3-disubstituted-4-phenyl-1 H-pyridin-2-ones
BRPI0816767B8 (en)	2007-09-14	2021-05-25	Addex Pharmaceuticals Sa	compound 4-phenyl-3,4,5,6-tetrahydro-2h,1'h-[1,4']bipyridinyl-2'-disubstituted 1',3'-ones, pharmaceutical composition and use of same
US8785486B2 (en)	2007-11-14	2014-07-22	Janssen Pharmaceuticals, Inc.	Imidazo[1,2-A]pyridine derivatives and their use as positive allosteric modulators of mGluR2 receptors
ES2439291T3 (en)	2008-09-02	2014-01-22	Janssen Pharmaceuticals, Inc.	3-Azabicyclo [3.1.0] hexyl derivatives as modulators of metabotropic glutamate receptors
EP2346505B1 (en)	2008-10-16	2014-04-23	Janssen Pharmaceuticals, Inc.	Indole and benzomorpholine derivatives as modulators of metabotropic glutamate receptors
WO2010060589A1 (en)	2008-11-28	2010-06-03	Ortho-Mcneil-Janssen Pharmaceuticals, Inc.	Indole and benzoxazine derivatives as modulators of metabotropic glutamate receptors
NZ596053A (en)	2009-05-12	2013-05-31	Janssen Pharmaceuticals Inc	1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mglur2 receptors
CN102439008B (en)	2009-05-12	2015-04-29	杨森制药有限公司	1,2,3-triazolo [4,3-a] pyridine derivatives and their use for the treatment or prevention of neurological and psychiatric disorders
MY153913A (en)	2009-05-12	2015-04-15	Janssen Pharmaceuticals Inc	7-aryl-1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mglur2 receptors
EP2440523A4 (en) *	2009-06-10	2014-03-19	Chongxi Yu	High penetration compositions or prodrugs of antimicrobials and antimicrobial-related compounds
US9271967B2 (en)	2010-11-08	2016-03-01	Janssen Pharmaceuticals, Inc.	1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mGluR2 receptors
ES2536433T3 (en)	2010-11-08	2015-05-25	Janssen Pharmaceuticals, Inc.	1,2,4-Triazolo [4,3-a] pyridine derivatives and their use as positive allosteric modulators of mGluR2 receptors
US8993591B2 (en)	2010-11-08	2015-03-31	Janssen Pharmaceuticals, Inc.	1,2,4-triazolo[4,3-a] pyridine derivatives and their use as positive allosteric modulators of MGLUR2 receptors
JO3368B1 (en)	2013-06-04	2019-03-13	Janssen Pharmaceutica Nv	6,7-DIHYDROPYRAZOLO[1,5-a]PYRAZIN-4(5H)-ONE COMPOUNDS AND THEIR USE AS NEGATIVE ALLOSTERIC MODULATORS OF MGLUR2 RECEPTORS
JO3367B1 (en)	2013-09-06	2019-03-13	Janssen Pharmaceutica Nv	1,2,4-TRIAZOLO[4,3-a]PYRIDINE COMPOUNDS AND THEIR USE AS POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 RECEPTORS
DK3096790T3 (en)	2014-01-21	2019-10-07	Janssen Pharmaceutica Nv	COMBINATIONS INCLUDING POSITIVE ALLOSTERIC MODULATORS OR ORTHOSTERIC AGONISTS OF METABOTROP GLUTAMATERG SUBTYPE 2 RECEPTOR AND APPLICATION OF THESE
DK3431106T3 (en)	2014-01-21	2021-03-15	Janssen Pharmaceutica Nv	COMBINATIONS INCLUDING POSITIVE ALLOSTERIC MODULATORS OR ORTHOSTERIC AGONISTS OF METABOTROP GLUTAMATERG SUBTYPE 2 RECEPTOR AND USE OF THESE

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE1770620A1 (en) *	1968-06-12	1971-11-11	Bayer Ag	New penicillins

0
- BE BE790440D patent/BE790440A/xx not_active IP Right Cessation
1971
- 1971-10-23 DE DE2152967A patent/DE2152967C3/en not_active Expired
1972
- 1972-10-12 SU SU1839113A patent/SU527139A3/en active
- 1972-10-17 PH PH14018A patent/PH9893A/en unknown
- 1972-10-17 RO RO197285500A patent/RO63066A/en unknown
- 1972-10-17 RO RO197272544A patent/RO60670A/ro unknown
- 1972-10-19 HU HUBA2815A patent/HU167986B/hu not_active IP Right Cessation
- 1972-10-19 FI FI2897/72A patent/FI56839C/en active
- 1972-10-19 BG BG21665A patent/BG21609A3/xx unknown
- 1972-10-19 DD DD72166352A patent/DD106044B3/en unknown
- 1972-10-19 BG BG24757A patent/BG20813A3/xx unknown
- 1972-10-19 CS CS727048A patent/CS188883B2/en unknown
- 1972-10-20 IE IE1422/72A patent/IE37123B1/en unknown
- 1972-10-20 LU LU66332A patent/LU66332A1/xx unknown
- 1972-10-20 ZA ZA727473A patent/ZA727473B/en unknown
- 1972-10-20 IL IL7240628A patent/IL40628A/en unknown
- 1972-10-20 DK DK522172A patent/DK134992C/en active
- 1972-10-20 AT AT901072A patent/AT320152B/en not_active IP Right Cessation
- 1972-10-20 SE SE7213592A patent/SE412236B/en unknown
- 1972-10-20 CH CH1531272A patent/CH579089A5/xx not_active IP Right Cessation
- 1972-10-20 CA CA154,338A patent/CA1019323A/en not_active Expired
- 1972-10-21 JP JP10490272A patent/JPS57843B2/ja not_active Expired
- 1972-10-21 PL PL1972183057A patent/PL93574B1/pl unknown
- 1972-10-21 JP JP10490172A patent/JPS55391B2/ja not_active Expired
- 1972-10-21 ES ES407851A patent/ES407851A1/en not_active Expired
- 1972-10-21 PL PL1972158392A patent/PL89056B1/pl unknown
- 1972-10-21 EG EG437/72A patent/EG10826A/en active
- 1972-10-23 GB GB4869972A patent/GB1392849A/en not_active Expired
- 1972-10-23 AR AR244770A patent/AR195805A1/en active
- 1972-10-23 NO NO723810A patent/NO143909C/en unknown
- 1972-10-23 FR FR7237482A patent/FR2157908B1/fr not_active Expired
- 1972-10-23 YU YU02640/72A patent/YU264072A/en unknown
- 1972-10-23 CY CY947A patent/CY947A/en unknown
1978
- 1978-03-14 KE KE2824A patent/KE2824A/en unknown
- 1978-04-04 HK HK185/78A patent/HK18578A/en unknown

Also Published As

Publication number	Publication date
JPS57843B2 (en)	1982-01-08
DE2152967B2 (en)	1981-02-19
FI56839B (en)	1979-12-31
HU167986B (en)	1976-02-28
AU4806472A (en)	1974-04-26
CA1019323A (en)	1977-10-18
DK134992B (en)	1977-02-21
FI56839C (en)	1980-04-10
DE2152967C3 (en)	1981-11-19
CS188883B2 (en)	1979-03-30
DE2152967A1 (en)	1973-05-03
FR2157908B1 (en)	1976-03-19
IE37123L (en)	1973-04-23
JPS4849787A (en)	1973-07-13
CH579089A5 (en)	1976-08-31
LU66332A1 (en)	1973-01-23
AT320152B (en)	1975-01-27
IE37123B1 (en)	1977-05-11
SU527139A3 (en)	1976-08-30
FR2157908A1 (en)	1973-06-08
JPS55391B2 (en)	1980-01-08
GB1392849A (en)	1975-04-30
DD106044B3 (en)	1990-07-18
RO60670A (en)	1976-10-15
BG21609A3 (en)	1976-07-20
NO143909C (en)	1981-05-06
HK18578A (en)	1978-04-14
CY947A (en)	1978-06-23
PL93574B1 (en)	1977-06-30
BE790440A (en)	1973-04-24
DK134992C (en)	1977-07-18
ZA727473B (en)	1973-07-25
PL89056B1 (en)	1976-10-30
ES407851A1 (en)	1975-10-01
RO63066A (en)	1978-06-15
IL40628A0 (en)	1972-12-29
NO143909B (en)	1981-01-26
KE2824A (en)	1978-04-07
SE412236B (en)	1980-02-25
PH9893A (en)	1976-06-08
BG20813A3 (en)	1975-12-20
IL40628A (en)	1976-08-31
AR195805A1 (en)	1973-11-09
DD106044A5 (en)	1974-05-20
JPS4849910A (en)	1973-07-14
EG10826A (en)	1976-12-31

Publication	Publication Date	Title
YU264072A (en)	1982-06-18	Process for preparing penicillins
YU298072A (en)	1982-06-18	Process for preparing isothiocyanobenzazoles
ZA725556B (en)	1973-05-30	Process for preparing an iron-saccharide complex
YU263872A (en)	1981-06-30	Process for preparing novel penicillins
YU216872A (en)	1980-09-25	Process for preparing cinnamoyl-5-benzofuran derivatives
YU34897B (en)	1980-04-30	Process for preparing 4-aza-benzimidazoles
CS180608B2 (en)	1978-01-31	Process for preparing dialkoxyxanthogendisulfines
CS190400B2 (en)	1979-05-31	Process for preparing hetacephalexine
YU142879A (en)	1982-10-31	Process for obtaining thiazoline-azetidinone
JPS53127458A (en)	1978-11-07	Process for preparing alphaaisopropylidenee11 azethidineacetate
YU194572A (en)	1980-04-30	Process for preparing tetramisoles
YU99179A (en)	1981-08-31	Process for obtaining novel hydroxy-pyrimidines
ZA724841B (en)	1974-02-27	Process for preparing cephalosporings
YU34999B (en)	1980-06-30	Process for preparing novel substituted n-methalyl-n-phenyl-amino-imidazolines
YU267272A (en)	1982-02-28	Process for obtaining benzyl-pyridyl-amino-ethanol
CS190382B2 (en)	1979-05-31	Process for preparing 3-alkylthiomethyl-7-acylamidocephalosporines
YU239672A (en)	1979-12-31	Process for preparing steroid-21-alcohols
YU115972A (en)	1980-04-30	Process for preparing 4-hydroxy-benzodioxides
CS190379B2 (en)	1979-05-31	Process for preparing penicilinamine
YU259972A (en)	1982-06-30	Process for producing penicillin
GB1400875A (en)	1975-07-16	Process for preparing cyclicdicarboximidophosphonothioates
ZA722397B (en)	1972-12-27	Process for preparing 5-hydroxy-1-tetralone
YU47272A (en)	1982-02-28	Improved process for preparing 1-dihydrocodeine
YU233572A (en)	1980-10-31	Process for obtaining delta-carboxyarylmethyl-1delta-carboaryloxyarylmethyl penicillins
YU99072A (en)	1979-04-30	Process for preparing 1-allyl-2-amino-methyl-pyrrolidines