EG10826A - Process for preparation of new penicillins - Google Patents

Process for preparation of new penicillins

Info

Publication number: EG10826A
Authority: EG; Egypt
Prior art keywords: preparation; new penicillins; penicillins; new
Prior art date: 1971-10-23

Application number

EG437/72A

Original Assignee

Bayer Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1971-10-23

Filing date

1972-10-21

Publication date

1976-12-31

1972-10-21 Application filed by Bayer Ag filed Critical Bayer Ag

1976-12-31 Application granted granted Critical

1976-12-31 Publication of EG10826A publication Critical patent/EG10826A/en

Links

229930182555 Penicillin Natural products 0.000 title 1
150000002960 penicillins Chemical class 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/06—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D239/08—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms directly attached in position 2
- C07D239/10—Oxygen or sulfur atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/06—Anabolic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/30—Oxygen or sulfur atoms
- C07D233/32—One oxygen atom
- C07D233/38—One oxygen atom with acyl radicals or hetero atoms directly attached to ring nitrogen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
- C07D275/02—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/30—Hetero atoms other than halogen
- C07D333/34—Sulfur atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/10—Compounds having one or more C—Si linkages containing nitrogen having a Si-N linkage

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Oncology (AREA)
Communicable Diseases (AREA)
Endocrinology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Neurology (AREA)
Orthopedic Medicine & Surgery (AREA)
Physical Education & Sports Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Fodder In General (AREA)

EG437/72A 1971-10-23 1972-10-21 Process for preparation of new penicillins EG10826A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE2152967A DE2152967C3 (en)	1971-10-23	1971-10-23	Acylureidopenicillins

Publications (1)

Publication Number	Publication Date
EG10826A true EG10826A (en)	1976-12-31

Family

ID=5823251

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
EG437/72A EG10826A (en)	1971-10-23	1972-10-21	Process for preparation of new penicillins

Country Status (31)

Country	Link
JP (2)	JPS57843B2 (en)
AR (1)	AR195805A1 (en)
AT (1)	AT320152B (en)
BE (1)	BE790440A (en)
BG (2)	BG21609A3 (en)
CA (1)	CA1019323A (en)
CH (1)	CH579089A5 (en)
CS (1)	CS188883B2 (en)
CY (1)	CY947A (en)
DD (1)	DD106044B3 (en)
DE (1)	DE2152967C3 (en)
DK (1)	DK134992C (en)
EG (1)	EG10826A (en)
ES (1)	ES407851A1 (en)
FI (1)	FI56839C (en)
FR (1)	FR2157908B1 (en)
GB (1)	GB1392849A (en)
HK (1)	HK18578A (en)
HU (1)	HU167986B (en)
IE (1)	IE37123B1 (en)
IL (1)	IL40628A (en)
KE (1)	KE2824A (en)
LU (1)	LU66332A1 (en)
NO (1)	NO143909C (en)
PH (1)	PH9893A (en)
PL (2)	PL93574B1 (en)
RO (2)	RO63066A (en)
SE (1)	SE412236B (en)
SU (1)	SU527139A3 (en)
YU (1)	YU264072A (en)
ZA (1)	ZA727473B (en)

Families Citing this family (37)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3983105A (en) *	1971-10-23	1976-09-28	Bayer Aktiengesellschaft	Penicillins
US3972870A (en) *	1971-10-23	1976-08-03	Bayer Aktiengesellschaft	Penicillins
US3974142A (en) *	1971-10-23	1976-08-10	Bayer Aktiengesellschaft	Penicillins
NL175419C (en) *	1971-10-23	1984-11-01	Bayer Ag	METHOD FOR PREPARING OR MANUFACTURING ANTIBIOTIC ACTIVE PHARMACEUTICAL PREPARATIONS AND METHOD FOR PREPARING ANTIBIOTIC ACTIVE ALPHA-SUBSTITUTED 6- (ALFA- (3-ACYLUREIDO) -PETYL-ACIDYL-ACIDYL-ACIDYL)
US4009272A (en) *	1971-10-23	1977-02-22	Bayer Aktiengesellschaft	Penicillins
US3978056A (en) *	1971-10-23	1976-08-31	Bayer Aktiengesellschaft	Penicillins
US3974141A (en) *	1971-10-23	1976-08-10	Bayer Aktiengesellschaft	Penicillins
US3972869A (en) *	1971-10-23	1976-08-03	Bayer Aktiengesellschaft	Penicillins
DE2258973A1 (en) *	1972-12-01	1974-06-06	Bayer Ag	PENICILLIN, THE METHOD FOR MANUFACTURING IT AND THEIR USE AS A MEDICINAL PRODUCT
JPS587637B2 (en) *	1973-12-27	1983-02-10	住友化学工業株式会社	Shinkipenicillin no Seihou
DE2407715C2 (en) *	1974-02-18	1982-12-02	Bayer Ag, 5090 Leverkusen	Cephalosporins, processes for their production, as well as pharmaceuticals
IL47168A (en) *	1974-05-09	1979-07-25	Toyama Chemical Co Ltd	Mono or dioxo piperazino(thio)carbonylamino derivatives ofpenicillins and cephalosporins and process for producing the same
DE2525541C2 (en) *	1975-06-07	1984-01-12	Bayer Ag, 5090 Leverkusen	β-lactam antibiotics, processes for their preparation and pharmaceuticals containing them
DE2810083A1 (en)	1978-03-08	1979-09-20	Bayer Ag	BETA-LACTAM COMPOUNDS
GB0420722D0 (en)	2004-09-17	2004-10-20	Addex Pharmaceuticals Sa	Novel allosteric modulators
EP1780213A1 (en) *	2005-10-27	2007-05-02	3M Innovative Properties Company	Silicon-urea-azolides, their preparation and use in the preparation of silicones with isocyanate terminal groups
TWI417095B (en)	2006-03-15	2013-12-01	Janssen Pharmaceuticals Inc	1,4-disubstituted 3-cyano-pyridone derivatives and their use as positive allosteric modulators of mglur2-receptors
TW200900065A (en)	2007-03-07	2009-01-01	Janssen Pharmaceutica Nv	3-cyano-4-(4-pyridinyloxy-phenyl)-pyridin-2-one derivatives
TW200845978A (en)	2007-03-07	2008-12-01	Janssen Pharmaceutica Nv	3-cyano-4-(4-tetrahydropyran-phenyl)-pyridin-2-one derivatives
EA019085B1 (en)	2007-09-14	2014-01-30	Янссен Фармасьютикалз, Инк.	1,3-disubstituted 4-(aryl-x-phenyl)-1h-pyridin-2-ones
US9114138B2 (en)	2007-09-14	2015-08-25	Janssen Pharmaceuticals, Inc.	1′,3′-disubstituted-4-phenyl-3,4,5,6-tetrahydro-2H,1′H-[1,4′] bipyridinyl-2′-ones
TW200927731A (en)	2007-09-14	2009-07-01	Ortho Mcneil Janssen Pharm	1,3-disubstituted-4-phenyl-1H-pyridin-2-ones
JP5433582B2 (en)	2007-11-14	2014-03-05	ジャンセンファーマシューティカルズ，インコーポレイテッド．	Imidazo [1,2-a] pyridine derivatives and their use as positive allosteric modulators of the mGluR2 receptor
WO2010025890A1 (en)	2008-09-02	2010-03-11	Ortho-Mcneil-Janssen Pharmaceuticals, Inc	3-azabicyclo[3.1.0]hexyl derivatives as modulators of metabotropic glutamate receptors
AU2009304293B2 (en)	2008-10-16	2012-04-26	Addex Pharma S.A.	Indole and benzomorpholine derivatives as modulators of metabotropic glutamate receptors
AU2009319387B2 (en)	2008-11-28	2012-05-10	Addex Pharma S.A.	Indole and benzoxazine derivatives as modulators of metabotropic glutamate receptors
CA2760259C (en)	2009-05-12	2018-05-01	Janssen Pharmaceuticals, Inc.	1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mglur2 receptors
MY153913A (en)	2009-05-12	2015-04-15	Janssen Pharmaceuticals Inc	7-aryl-1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mglur2 receptors
JP5634506B2 (en)	2009-05-12	2014-12-03	ジャンセンファーマシューティカルズ，インコーポレイテッド	1,2,3-Triazolo [4,3-a] pyridine derivatives and their use for the treatment or prevention of neurological and psychiatric disorders
MX366035B (en) *	2009-06-10	2019-06-25	Techfields Biochem Co Ltd	High penetration compositions or prodrugs of antimicrobials and antimicrobial-related compounds.
ES2552455T3 (en)	2010-11-08	2015-11-30	Janssen Pharmaceuticals, Inc.	1,2,4-Triazolo [4,3-a] pyridine derivatives and their use as positive allosteric modulators of mGluR2 receptors
JP5852666B2 (en)	2010-11-08	2016-02-03	ジヤンセン・フアーマシユーチカルズ・インコーポレーテツド	1,2,4-Triazolo [4,3-a] pyridine derivatives and their use as positive allosteric modulators of the mGluR2 receptor
JP5852665B2 (en)	2010-11-08	2016-02-03	ジヤンセン・フアーマシユーチカルズ・インコーポレーテツド	1,2,4-Triazolo [4,3-a] pyridine derivatives and their use as positive allosteric modulators of the mGluR2 receptor
JO3368B1 (en)	2013-06-04	2019-03-13	Janssen Pharmaceutica Nv	6,7-DIHYDROPYRAZOLO[1,5-a]PYRAZIN-4(5H)-ONE COMPOUNDS AND THEIR USE AS NEGATIVE ALLOSTERIC MODULATORS OF MGLUR2 RECEPTORS
JO3367B1 (en)	2013-09-06	2019-03-13	Janssen Pharmaceutica Nv	1,2,4-TRIAZOLO[4,3-a]PYRIDINE COMPOUNDS AND THEIR USE AS POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 RECEPTORS
WO2015110435A1 (en)	2014-01-21	2015-07-30	Janssen Pharmaceutica Nv	Combinations comprising positive allosteric modulators or orthosteric agonists of metabotropic glutamatergic receptor subtype 2 and their use
LT3096790T (en)	2014-01-21	2019-10-10	Janssen Pharmaceutica, N.V.	Combinations comprising positive allosteric modulators or orthosteric agonists of metabotropic glutamatergic receptor subtype 2 and their use

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE1770620A1 (en) *	1968-06-12	1971-11-11	Bayer Ag	New penicillins

0
- BE BE790440D patent/BE790440A/xx not_active IP Right Cessation
1971
- 1971-10-23 DE DE2152967A patent/DE2152967C3/en not_active Expired
1972
- 1972-10-12 SU SU1839113A patent/SU527139A3/en active
- 1972-10-17 RO RO197285500A patent/RO63066A/en unknown
- 1972-10-17 RO RO197272544A patent/RO60670A/ro unknown
- 1972-10-17 PH PH14018A patent/PH9893A/en unknown
- 1972-10-19 FI FI2897/72A patent/FI56839C/en active
- 1972-10-19 BG BG21665A patent/BG21609A3/xx unknown
- 1972-10-19 CS CS727048A patent/CS188883B2/en unknown
- 1972-10-19 HU HUBA2815A patent/HU167986B/hu not_active IP Right Cessation
- 1972-10-19 BG BG24757A patent/BG20813A3/xx unknown
- 1972-10-19 DD DD72166352A patent/DD106044B3/en unknown
- 1972-10-20 DK DK522172A patent/DK134992C/en active
- 1972-10-20 IL IL7240628A patent/IL40628A/en unknown
- 1972-10-20 AT AT901072A patent/AT320152B/en not_active IP Right Cessation
- 1972-10-20 LU LU66332A patent/LU66332A1/xx unknown
- 1972-10-20 SE SE7213592A patent/SE412236B/en unknown
- 1972-10-20 CA CA154,338A patent/CA1019323A/en not_active Expired
- 1972-10-20 IE IE1422/72A patent/IE37123B1/en unknown
- 1972-10-20 CH CH1531272A patent/CH579089A5/xx not_active IP Right Cessation
- 1972-10-20 ZA ZA727473A patent/ZA727473B/en unknown
- 1972-10-21 PL PL1972183057A patent/PL93574B1/pl unknown
- 1972-10-21 JP JP10490272A patent/JPS57843B2/ja not_active Expired
- 1972-10-21 EG EG437/72A patent/EG10826A/en active
- 1972-10-21 JP JP10490172A patent/JPS55391B2/ja not_active Expired
- 1972-10-21 ES ES407851A patent/ES407851A1/en not_active Expired
- 1972-10-21 PL PL1972158392A patent/PL89056B1/pl unknown
- 1972-10-23 GB GB4869972A patent/GB1392849A/en not_active Expired
- 1972-10-23 CY CY947A patent/CY947A/en unknown
- 1972-10-23 YU YU02640/72A patent/YU264072A/en unknown
- 1972-10-23 FR FR7237482A patent/FR2157908B1/fr not_active Expired
- 1972-10-23 NO NO723810A patent/NO143909C/en unknown
- 1972-10-23 AR AR244770A patent/AR195805A1/en active
1978
- 1978-03-14 KE KE2824A patent/KE2824A/en unknown
- 1978-04-04 HK HK185/78A patent/HK18578A/en unknown

Also Published As

Publication number	Publication date
IL40628A0 (en)	1972-12-29
JPS57843B2 (en)	1982-01-08
NO143909C (en)	1981-05-06
ZA727473B (en)	1973-07-25
DK134992B (en)	1977-02-21
DK134992C (en)	1977-07-18
HK18578A (en)	1978-04-14
FI56839B (en)	1979-12-31
HU167986B (en)	1976-02-28
AT320152B (en)	1975-01-27
RO63066A (en)	1978-06-15
GB1392849A (en)	1975-04-30
BG21609A3 (en)	1976-07-20
PH9893A (en)	1976-06-08
CS188883B2 (en)	1979-03-30
CH579089A5 (en)	1976-08-31
LU66332A1 (en)	1973-01-23
BG20813A3 (en)	1975-12-20
PL89056B1 (en)	1976-10-30
NO143909B (en)	1981-01-26
CY947A (en)	1978-06-23
PL93574B1 (en)	1977-06-30
DE2152967B2 (en)	1981-02-19
AU4806472A (en)	1974-04-26
CA1019323A (en)	1977-10-18
FR2157908B1 (en)	1976-03-19
IE37123L (en)	1973-04-23
IL40628A (en)	1976-08-31
DD106044A5 (en)	1974-05-20
YU264072A (en)	1982-06-18
KE2824A (en)	1978-04-07
SE412236B (en)	1980-02-25
BE790440A (en)	1973-04-24
SU527139A3 (en)	1976-08-30
JPS55391B2 (en)	1980-01-08
IE37123B1 (en)	1977-05-11
AR195805A1 (en)	1973-11-09
DE2152967C3 (en)	1981-11-19
DE2152967A1 (en)	1973-05-03
RO60670A (en)	1976-10-15
ES407851A1 (en)	1975-10-01
JPS4849910A (en)	1973-07-14
FR2157908A1 (en)	1973-06-08
JPS4849787A (en)	1973-07-13
FI56839C (en)	1980-04-10
DD106044B3 (en)	1990-07-18

Publication	Publication Date	Title
EG10826A (en)	1976-12-31	Process for preparation of new penicillins
IL39225A (en)	1975-07-28	Process for the manufacture of methyl substituted p-benzoquinones
EG11092A (en)	1979-09-30	Process for preparing of new penicillin compounds
GB1399160A (en)	1975-06-25	Process for the manufacture of polylauryl-lactam
IL39382A0 (en)	1972-07-26	Process for the preparation of cephalosporin
JPS5246050A (en)	1977-04-12	Process for manufacture of 22nnpentyll33 22oxopropyl*11cyclopentanone
EG11037A (en)	1977-12-31	Process for the preparation of new phenylimino-3-aza-1-thia cycloalkanes
EG11021A (en)	1977-12-31	Process for preparing of new penicillins
EG10550A (en)	1976-06-30	Process for preparation of benzodiazepin derivatives
ZA727738B (en)	1973-09-26	Process for the preparation of 4-chloro-2-dimethoxy-aniline
CH609065A5 (en)	1979-02-15	Process for the preparation of 21-adamantoyloxysteroids
PH11915A (en)	1978-09-08	Process for the preparation of 2-amino-4-phenyl-imidazoline derivatives
EG11062A (en)	1977-08-15	Process for preparing of new penicillins
CA959853A (en)	1974-12-24	Process for preparation of 3-hydroxy-2-alkyl-4-pyrone
CS180600B2 (en)	1978-01-31	Process for preparing new derivatives of 2-formyl-3-carboxamidochinoxalin-di-n-oxides
CS186217B2 (en)	1978-11-30	Process for preparing derivatives of bycicloalkane
ZA727831B (en)	1973-07-25	Process for the preparation of methylcobalamine
ZA723748B (en)	1973-03-28	Process for the preparation of pivalolactone
EG10782A (en)	1976-12-31	Process for preparation of penicillin amin
ZA717402B (en)	1972-08-30	Process for the preparation of argininemalate
YU36533B (en)	1984-02-29	Process for obtaining derivatives of antibiotics
EG10570A (en)	1976-01-31	Process for the preparation of 7-chloro-benzodiazepine derivatives
ZA726400B (en)	1973-07-25	Process for the preparation of dea-steroids
ZA726125B (en)	1973-07-25	Process for the preparation of carboxyarylmethyl and carboaryloxyarylmethyl penicillins
CS179403B2 (en)	1977-10-31	Method for production of l-aralkyl-2-pyrryl-2-aminoethanols