KE2824A - New penicillins, their production and their medicinal use - Google Patents

New penicillins, their production and their medicinal use

Info

Publication number: KE2824A
Authority: KE; Kenya
Prior art keywords: production; medicinal use; new penicillins; penicillins; new
Prior art date: 1971-10-23

Application number

KE2824A

Inventor

H B Koenig

K G Metzger

W Schroeck

Original Assignee

Bayer Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1971-10-23

Filing date

1978-03-14

Publication date

1978-04-07

1978-03-14 Application filed by Bayer Ag filed Critical Bayer Ag

1978-04-07 Publication of KE2824A publication Critical patent/KE2824A/en

Links

229930182555 Penicillin Natural products 0.000 title 1
150000002960 penicillins Chemical class 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/06—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D239/08—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms directly attached in position 2
- C07D239/10—Oxygen or sulfur atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/06—Anabolic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/30—Oxygen or sulfur atoms
- C07D233/32—One oxygen atom
- C07D233/38—One oxygen atom with acyl radicals or hetero atoms directly attached to ring nitrogen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
- C07D275/02—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/30—Hetero atoms other than halogen
- C07D333/34—Sulfur atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/10—Compounds having one or more C—Si linkages containing nitrogen having a Si-N linkage

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Oncology (AREA)
Communicable Diseases (AREA)
Endocrinology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Neurology (AREA)
Orthopedic Medicine & Surgery (AREA)
Physical Education & Sports Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Fodder In General (AREA)

KE2824A 1971-10-23 1978-03-14 New penicillins, their production and their medicinal use KE2824A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE2152967A DE2152967C3 (en)	1971-10-23	1971-10-23	Acylureidopenicillins

Publications (1)

Publication Number	Publication Date
KE2824A true KE2824A (en)	1978-04-07

Family

ID=5823251

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
KE2824A KE2824A (en)	1971-10-23	1978-03-14	New penicillins, their production and their medicinal use

Country Status (31)

Country	Link
JP (2)	JPS57843B2 (en)
AR (1)	AR195805A1 (en)
AT (1)	AT320152B (en)
BE (1)	BE790440A (en)
BG (2)	BG21609A3 (en)
CA (1)	CA1019323A (en)
CH (1)	CH579089A5 (en)
CS (1)	CS188883B2 (en)
CY (1)	CY947A (en)
DD (1)	DD106044B3 (en)
DE (1)	DE2152967C3 (en)
DK (1)	DK134992C (en)
EG (1)	EG10826A (en)
ES (1)	ES407851A1 (en)
FI (1)	FI56839C (en)
FR (1)	FR2157908B1 (en)
GB (1)	GB1392849A (en)
HK (1)	HK18578A (en)
HU (1)	HU167986B (en)
IE (1)	IE37123B1 (en)
IL (1)	IL40628A (en)
KE (1)	KE2824A (en)
LU (1)	LU66332A1 (en)
NO (1)	NO143909C (en)
PH (1)	PH9893A (en)
PL (2)	PL93574B1 (en)
RO (2)	RO63066A (en)
SE (1)	SE412236B (en)
SU (1)	SU527139A3 (en)
YU (1)	YU264072A (en)
ZA (1)	ZA727473B (en)

Families Citing this family (37)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3972870A (en) *	1971-10-23	1976-08-03	Bayer Aktiengesellschaft	Penicillins
NL175419C (en) *	1971-10-23	1984-11-01	Bayer Ag	METHOD FOR PREPARING OR MANUFACTURING ANTIBIOTIC ACTIVE PHARMACEUTICAL PREPARATIONS AND METHOD FOR PREPARING ANTIBIOTIC ACTIVE ALPHA-SUBSTITUTED 6- (ALFA- (3-ACYLUREIDO) -PETYL-ACIDYL-ACIDYL-ACIDYL)
US3978056A (en) *	1971-10-23	1976-08-31	Bayer Aktiengesellschaft	Penicillins
US4009272A (en) *	1971-10-23	1977-02-22	Bayer Aktiengesellschaft	Penicillins
US3974142A (en) *	1971-10-23	1976-08-10	Bayer Aktiengesellschaft	Penicillins
US3972869A (en) *	1971-10-23	1976-08-03	Bayer Aktiengesellschaft	Penicillins
US3974141A (en) *	1971-10-23	1976-08-10	Bayer Aktiengesellschaft	Penicillins
US3983105A (en) *	1971-10-23	1976-09-28	Bayer Aktiengesellschaft	Penicillins
DE2258973A1 (en) *	1972-12-01	1974-06-06	Bayer Ag	PENICILLIN, THE METHOD FOR MANUFACTURING IT AND THEIR USE AS A MEDICINAL PRODUCT
JPS587637B2 (en) *	1973-12-27	1983-02-10	住友化学工業株式会社	Shinkipenicillin no Seihou
DE2407715C2 (en) *	1974-02-18	1982-12-02	Bayer Ag, 5090 Leverkusen	Cephalosporins, processes for their production, as well as pharmaceuticals
IL47168A (en) *	1974-05-09	1979-07-25	Toyama Chemical Co Ltd	Mono or dioxo piperazino(thio)carbonylamino derivatives ofpenicillins and cephalosporins and process for producing the same
DE2525541C2 (en) *	1975-06-07	1984-01-12	Bayer Ag, 5090 Leverkusen	β-lactam antibiotics, processes for their preparation and pharmaceuticals containing them
DE2810083A1 (en)	1978-03-08	1979-09-20	Bayer Ag	BETA-LACTAM COMPOUNDS
GB0420722D0 (en)	2004-09-17	2004-10-20	Addex Pharmaceuticals Sa	Novel allosteric modulators
EP1780213A1 (en)	2005-10-27	2007-05-02	3M Innovative Properties Company	Silicon-urea-azolides, their preparation and use in the preparation of silicones with isocyanate terminal groups
AR059898A1 (en)	2006-03-15	2008-05-07	Janssen Pharmaceutica Nv	DERIVATIVES OF 3-CIANO-PIRIDONA 1,4-DISUSTITUTED AND ITS USE AS ALLOSTERIC MODULATORS OF MGLUR2 RECEIVERS
TW200845978A (en)	2007-03-07	2008-12-01	Janssen Pharmaceutica Nv	3-cyano-4-(4-tetrahydropyran-phenyl)-pyridin-2-one derivatives
TW200900065A (en)	2007-03-07	2009-01-01	Janssen Pharmaceutica Nv	3-cyano-4-(4-pyridinyloxy-phenyl)-pyridin-2-one derivatives
US8252937B2 (en)	2007-09-14	2012-08-28	Janssen Pharmaceuticals, Inc.	1,3-disubstituted 4-(aryl-X-phenyl)-1H-pyridin-2-ones
AU2008297877C1 (en)	2007-09-14	2013-11-07	Addex Pharma S.A.	1,3-disubstituted-4-phenyl-1 H-pyridin-2-ones
BRPI0816767B8 (en)	2007-09-14	2021-05-25	Addex Pharmaceuticals Sa	compound 4-phenyl-3,4,5,6-tetrahydro-2h,1'h-[1,4']bipyridinyl-2'-disubstituted 1',3'-ones, pharmaceutical composition and use of same
US8785486B2 (en)	2007-11-14	2014-07-22	Janssen Pharmaceuticals, Inc.	Imidazo[1,2-A]pyridine derivatives and their use as positive allosteric modulators of mGluR2 receptors
ES2439291T3 (en)	2008-09-02	2014-01-22	Janssen Pharmaceuticals, Inc.	3-Azabicyclo [3.1.0] hexyl derivatives as modulators of metabotropic glutamate receptors
EP2346505B1 (en)	2008-10-16	2014-04-23	Janssen Pharmaceuticals, Inc.	Indole and benzomorpholine derivatives as modulators of metabotropic glutamate receptors
WO2010060589A1 (en)	2008-11-28	2010-06-03	Ortho-Mcneil-Janssen Pharmaceuticals, Inc.	Indole and benzoxazine derivatives as modulators of metabotropic glutamate receptors
NZ596053A (en)	2009-05-12	2013-05-31	Janssen Pharmaceuticals Inc	1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mglur2 receptors
CN102439008B (en)	2009-05-12	2015-04-29	杨森制药有限公司	1,2,3-triazolo [4,3-a] pyridine derivatives and their use for the treatment or prevention of neurological and psychiatric disorders
MY153913A (en)	2009-05-12	2015-04-15	Janssen Pharmaceuticals Inc	7-aryl-1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mglur2 receptors
EP2440523A4 (en) *	2009-06-10	2014-03-19	Chongxi Yu	High penetration compositions or prodrugs of antimicrobials and antimicrobial-related compounds
US9271967B2 (en)	2010-11-08	2016-03-01	Janssen Pharmaceuticals, Inc.	1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mGluR2 receptors
ES2536433T3 (en)	2010-11-08	2015-05-25	Janssen Pharmaceuticals, Inc.	1,2,4-Triazolo [4,3-a] pyridine derivatives and their use as positive allosteric modulators of mGluR2 receptors
US8993591B2 (en)	2010-11-08	2015-03-31	Janssen Pharmaceuticals, Inc.	1,2,4-triazolo[4,3-a] pyridine derivatives and their use as positive allosteric modulators of MGLUR2 receptors
JO3368B1 (en)	2013-06-04	2019-03-13	Janssen Pharmaceutica Nv	6,7-DIHYDROPYRAZOLO[1,5-a]PYRAZIN-4(5H)-ONE COMPOUNDS AND THEIR USE AS NEGATIVE ALLOSTERIC MODULATORS OF MGLUR2 RECEPTORS
JO3367B1 (en)	2013-09-06	2019-03-13	Janssen Pharmaceutica Nv	1,2,4-TRIAZOLO[4,3-a]PYRIDINE COMPOUNDS AND THEIR USE AS POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 RECEPTORS
DK3096790T3 (en)	2014-01-21	2019-10-07	Janssen Pharmaceutica Nv	COMBINATIONS INCLUDING POSITIVE ALLOSTERIC MODULATORS OR ORTHOSTERIC AGONISTS OF METABOTROP GLUTAMATERG SUBTYPE 2 RECEPTOR AND APPLICATION OF THESE
DK3431106T3 (en)	2014-01-21	2021-03-15	Janssen Pharmaceutica Nv	COMBINATIONS INCLUDING POSITIVE ALLOSTERIC MODULATORS OR ORTHOSTERIC AGONISTS OF METABOTROP GLUTAMATERG SUBTYPE 2 RECEPTOR AND USE OF THESE

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE1770620A1 (en) *	1968-06-12	1971-11-11	Bayer Ag	New penicillins

0
- BE BE790440D patent/BE790440A/xx not_active IP Right Cessation
1971
- 1971-10-23 DE DE2152967A patent/DE2152967C3/en not_active Expired
1972
- 1972-10-12 SU SU1839113A patent/SU527139A3/en active
- 1972-10-17 PH PH14018A patent/PH9893A/en unknown
- 1972-10-17 RO RO197285500A patent/RO63066A/en unknown
- 1972-10-17 RO RO197272544A patent/RO60670A/ro unknown
- 1972-10-19 HU HUBA2815A patent/HU167986B/hu not_active IP Right Cessation
- 1972-10-19 FI FI2897/72A patent/FI56839C/en active
- 1972-10-19 BG BG21665A patent/BG21609A3/xx unknown
- 1972-10-19 DD DD72166352A patent/DD106044B3/en unknown
- 1972-10-19 BG BG24757A patent/BG20813A3/xx unknown
- 1972-10-19 CS CS727048A patent/CS188883B2/en unknown
- 1972-10-20 IE IE1422/72A patent/IE37123B1/en unknown
- 1972-10-20 LU LU66332A patent/LU66332A1/xx unknown
- 1972-10-20 ZA ZA727473A patent/ZA727473B/en unknown
- 1972-10-20 IL IL7240628A patent/IL40628A/en unknown
- 1972-10-20 DK DK522172A patent/DK134992C/en active
- 1972-10-20 AT AT901072A patent/AT320152B/en not_active IP Right Cessation
- 1972-10-20 SE SE7213592A patent/SE412236B/en unknown
- 1972-10-20 CH CH1531272A patent/CH579089A5/xx not_active IP Right Cessation
- 1972-10-20 CA CA154,338A patent/CA1019323A/en not_active Expired
- 1972-10-21 JP JP10490272A patent/JPS57843B2/ja not_active Expired
- 1972-10-21 PL PL1972183057A patent/PL93574B1/pl unknown
- 1972-10-21 JP JP10490172A patent/JPS55391B2/ja not_active Expired
- 1972-10-21 ES ES407851A patent/ES407851A1/en not_active Expired
- 1972-10-21 PL PL1972158392A patent/PL89056B1/pl unknown
- 1972-10-21 EG EG437/72A patent/EG10826A/en active
- 1972-10-23 GB GB4869972A patent/GB1392849A/en not_active Expired
- 1972-10-23 AR AR244770A patent/AR195805A1/en active
- 1972-10-23 NO NO723810A patent/NO143909C/en unknown
- 1972-10-23 FR FR7237482A patent/FR2157908B1/fr not_active Expired
- 1972-10-23 YU YU02640/72A patent/YU264072A/en unknown
- 1972-10-23 CY CY947A patent/CY947A/en unknown
1978
- 1978-03-14 KE KE2824A patent/KE2824A/en unknown
- 1978-04-04 HK HK185/78A patent/HK18578A/en unknown

Also Published As

Publication number	Publication date
JPS57843B2 (en)	1982-01-08
DE2152967B2 (en)	1981-02-19
FI56839B (en)	1979-12-31
HU167986B (en)	1976-02-28
AU4806472A (en)	1974-04-26
CA1019323A (en)	1977-10-18
DK134992B (en)	1977-02-21
FI56839C (en)	1980-04-10
DE2152967C3 (en)	1981-11-19
CS188883B2 (en)	1979-03-30
DE2152967A1 (en)	1973-05-03
FR2157908B1 (en)	1976-03-19
IE37123L (en)	1973-04-23
JPS4849787A (en)	1973-07-13
CH579089A5 (en)	1976-08-31
LU66332A1 (en)	1973-01-23
AT320152B (en)	1975-01-27
IE37123B1 (en)	1977-05-11
SU527139A3 (en)	1976-08-30
FR2157908A1 (en)	1973-06-08
JPS55391B2 (en)	1980-01-08
GB1392849A (en)	1975-04-30
DD106044B3 (en)	1990-07-18
YU264072A (en)	1982-06-18
RO60670A (en)	1976-10-15
BG21609A3 (en)	1976-07-20
NO143909C (en)	1981-05-06
HK18578A (en)	1978-04-14
CY947A (en)	1978-06-23
PL93574B1 (en)	1977-06-30
BE790440A (en)	1973-04-24
DK134992C (en)	1977-07-18
ZA727473B (en)	1973-07-25
PL89056B1 (en)	1976-10-30
ES407851A1 (en)	1975-10-01
RO63066A (en)	1978-06-15
IL40628A0 (en)	1972-12-29
NO143909B (en)	1981-01-26
SE412236B (en)	1980-02-25
PH9893A (en)	1976-06-08
BG20813A3 (en)	1975-12-20
IL40628A (en)	1976-08-31
AR195805A1 (en)	1973-11-09
DD106044A5 (en)	1974-05-20
JPS4849910A (en)	1973-07-14
EG10826A (en)	1976-12-31

Publication	Publication Date	Title
KE2824A (en)	1978-04-07	New penicillins, their production and their medicinal use
ZA722348B (en)	1972-12-27	New esters,their production,and their medicinal use
ZA722355B (en)	1972-12-27	New esters,their production,and their medicinal use
ZA731504B (en)	1973-11-28	New bridgehead-heterocyclic compounds,their production and their medicinal use
HK15378A (en)	1978-03-23	New penicillin compounds, their production and their medicinal use
EG10637A (en)	1976-04-30	New aminophenylamidines,their production and their pharmaceutical use
ZA713765B (en)	1972-01-26	New aminophenylamidines,their production and their medicinal use
ZA713764B (en)	1972-01-26	New aminophenyl-cycloamidines,their production and their medicinal use
ZA735460B (en)	1974-07-31	New 2-alkylamino-dihydropyridines,their production and their medicinal use
ZA726484B (en)	1973-06-27	New triazene derivatives,their production and their medicinal use
HK38578A (en)	1978-07-21	New 1-ethyl-imidazoles, their production, and their medicinal use
IL40338A0 (en)	1972-11-28	New phenylimino-3-aza-1-thiacycloalkanes,their preparation,and their medicinal use
ZA739331B (en)	1974-10-30	New penicillins,their production and their pharmaceutical use
CY829A (en)	1976-03-19	New penicillins, their preparation and their pharmaceutical use
ZA734890B (en)	1974-06-26	New 2-amino-4 h-pyrane compounds,their production and their medicinal use
ZA742381B (en)	1975-04-30	New-1-substituted pyrazol-5-sones, their production and their medicinal use
IL39071A0 (en)	1972-05-30	New penicillins and their preparation
ZA713371B (en)	1972-01-26	New penicillins,their preparation and their pharmaceutical use
AU485089B2 (en)	1974-04-26	New penicillins, their production, and their medicinal use
ZA738075B (en)	1974-08-28	Phenylguanidin-derivatives,their production and their medicinal use
ZA738287B (en)	1974-09-25	New amidophenylisothioureas,their production and their medicinal use
ZA723065B (en)	1973-02-28	New heterocyclic n,n-dioxides and their salts,their production,and their medicinal use
AU485090B2 (en)	1974-04-26	New penicillin compounds, their production and their medicinal use
KE2657A (en)	1976-09-17	New benzoylphenylisothioureas, their production, and their medicinal use
AU448290B2 (en)	1973-01-25	New aminophenylamidines, their production and their medicinal use