UY32855A - BICYCLIC HETEROCYCLES, DRUGS CONTAINING THESE COMPOUNDS, THEIR EMPLOYMENT AND PROCEDURES FOR THEIR PREPARATION - Google Patents

BICYCLIC HETEROCYCLES, DRUGS CONTAINING THESE COMPOUNDS, THEIR EMPLOYMENT AND PROCEDURES FOR THEIR PREPARATION

Info

Publication number
UY32855A
UY32855A UY0001032855A UY32855A UY32855A UY 32855 A UY32855 A UY 32855A UY 0001032855 A UY0001032855 A UY 0001032855A UY 32855 A UY32855 A UY 32855A UY 32855 A UY32855 A UY 32855A
Authority
UY
Uruguay
Prior art keywords
preparation
bicyclic heterocycles
employment
procedures
compounds
Prior art date
Application number
UY0001032855A
Other languages
Spanish (es)
Inventor
Frank Dr Himmelsbach
Elke Dr Langkopf
Thomas Dr Metz
Flavio Dr Solca
Birgit Dr Jung
Anke Dr Baum
Original Assignee
Boehringer Ingelheim Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE1999128281 external-priority patent/DE19928281A1/en
Priority claimed from DE2000123085 external-priority patent/DE10023085A1/en
Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma
Publication of UY32855A publication Critical patent/UY32855A/en

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

La presente invención se refiere a heterociclos bicíclicos de la fórmula general en la que Ra a Rc, A a B y X están definidos como en la reivindicación 1, a sus tautómeros, sus estereoisomeros y sus sales, en particular sus sales fisiológicamente compatibles con ácidos o bases inorgánicos u orgánicos, que presentan valiosas propiedades farmacológicas, en particular un efecto inhibidor sobre la transducción de señales inducida por tirosinaquinasas, a su empleo para el tratamiento de enfermedades, en particular enfermedades tumorales, de enfermedades de los pulmones y de las vías respiratorias, y a su preparación.The present invention relates to bicyclic heterocycles of the general formula in which Ra to Rc, A to B and X are defined as in claim 1, their tautomers, their stereoisomers and their salts, in particular their physiologically compatible salts with acids or inorganic or organic bases, which have valuable pharmacological properties, in particular an inhibitory effect on tyrosine kinase-induced signal transduction, for use in the treatment of diseases, in particular tumor diseases, diseases of the lungs and respiratory tract , and its preparation.

UY0001032855A 1999-06-21 2010-08-26 BICYCLIC HETEROCYCLES, DRUGS CONTAINING THESE COMPOUNDS, THEIR EMPLOYMENT AND PROCEDURES FOR THEIR PREPARATION UY32855A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE1999128281 DE19928281A1 (en) 1999-06-21 1999-06-21 Arylamino and aralkylamino substituted quinoline and quinazoline derivatives, useful for the treatment of e.g. tumors, pulmonary, respiratory and gastrointestinal disorders and psoriasis
DE2000123085 DE10023085A1 (en) 2000-05-11 2000-05-11 Arylamino and aralkylamino substituted quinoline and quinazoline derivatives, useful for the treatment of e.g. tumors, pulmonary, respiratory and gastrointestinal disorders and psoriasis

Publications (1)

Publication Number Publication Date
UY32855A true UY32855A (en) 2012-03-30

Family

ID=26005635

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001032855A UY32855A (en) 1999-06-21 2010-08-26 BICYCLIC HETEROCYCLES, DRUGS CONTAINING THESE COMPOUNDS, THEIR EMPLOYMENT AND PROCEDURES FOR THEIR PREPARATION

Country Status (7)

Country Link
AR (1) AR024418A1 (en)
BR (1) BRPI0011834C1 (en)
CO (1) CO5180636A1 (en)
MY (1) MY140484A (en)
PL (1) PL212659B1 (en)
TW (1) TWI230156B (en)
UY (1) UY32855A (en)

Also Published As

Publication number Publication date
BRPI0011834C1 (en) 2021-05-25
AR024418A1 (en) 2002-10-02
TWI230156B (en) 2005-04-01
BR0011834A (en) 2002-03-12
MY140484A (en) 2009-12-31
CO5180636A1 (en) 2002-07-30
BRPI0011834B8 (en) 2015-12-22
PL352357A1 (en) 2003-08-11
BR0011834B1 (en) 2014-08-12
PL212659B1 (en) 2012-11-30

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