UY32855A - BICYCLIC HETEROCYCLES, DRUGS CONTAINING THESE COMPOUNDS, THEIR EMPLOYMENT AND PROCEDURES FOR THEIR PREPARATION - Google Patents
BICYCLIC HETEROCYCLES, DRUGS CONTAINING THESE COMPOUNDS, THEIR EMPLOYMENT AND PROCEDURES FOR THEIR PREPARATIONInfo
- Publication number
- UY32855A UY32855A UY0001032855A UY32855A UY32855A UY 32855 A UY32855 A UY 32855A UY 0001032855 A UY0001032855 A UY 0001032855A UY 32855 A UY32855 A UY 32855A UY 32855 A UY32855 A UY 32855A
- Authority
- UY
- Uruguay
- Prior art keywords
- preparation
- bicyclic heterocycles
- employment
- procedures
- compounds
- Prior art date
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
La presente invención se refiere a heterociclos bicíclicos de la fórmula general en la que Ra a Rc, A a B y X están definidos como en la reivindicación 1, a sus tautómeros, sus estereoisomeros y sus sales, en particular sus sales fisiológicamente compatibles con ácidos o bases inorgánicos u orgánicos, que presentan valiosas propiedades farmacológicas, en particular un efecto inhibidor sobre la transducción de señales inducida por tirosinaquinasas, a su empleo para el tratamiento de enfermedades, en particular enfermedades tumorales, de enfermedades de los pulmones y de las vías respiratorias, y a su preparación.The present invention relates to bicyclic heterocycles of the general formula in which Ra to Rc, A to B and X are defined as in claim 1, their tautomers, their stereoisomers and their salts, in particular their physiologically compatible salts with acids or inorganic or organic bases, which have valuable pharmacological properties, in particular an inhibitory effect on tyrosine kinase-induced signal transduction, for use in the treatment of diseases, in particular tumor diseases, diseases of the lungs and respiratory tract , and its preparation.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE1999128281 DE19928281A1 (en) | 1999-06-21 | 1999-06-21 | Arylamino and aralkylamino substituted quinoline and quinazoline derivatives, useful for the treatment of e.g. tumors, pulmonary, respiratory and gastrointestinal disorders and psoriasis |
DE2000123085 DE10023085A1 (en) | 2000-05-11 | 2000-05-11 | Arylamino and aralkylamino substituted quinoline and quinazoline derivatives, useful for the treatment of e.g. tumors, pulmonary, respiratory and gastrointestinal disorders and psoriasis |
Publications (1)
Publication Number | Publication Date |
---|---|
UY32855A true UY32855A (en) | 2012-03-30 |
Family
ID=26005635
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UY0001032855A UY32855A (en) | 1999-06-21 | 2010-08-26 | BICYCLIC HETEROCYCLES, DRUGS CONTAINING THESE COMPOUNDS, THEIR EMPLOYMENT AND PROCEDURES FOR THEIR PREPARATION |
Country Status (7)
Country | Link |
---|---|
AR (1) | AR024418A1 (en) |
BR (1) | BRPI0011834C1 (en) |
CO (1) | CO5180636A1 (en) |
MY (1) | MY140484A (en) |
PL (1) | PL212659B1 (en) |
TW (1) | TWI230156B (en) |
UY (1) | UY32855A (en) |
-
2000
- 2000-06-16 PL PL352357A patent/PL212659B1/en unknown
- 2000-06-16 BR BRPI0011834A patent/BRPI0011834C1/en not_active IP Right Cessation
- 2000-06-20 TW TW89112051A patent/TWI230156B/en not_active IP Right Cessation
- 2000-06-20 CO CO00045906A patent/CO5180636A1/en active IP Right Grant
- 2000-06-21 MY MYPI20002798 patent/MY140484A/en unknown
- 2000-06-21 AR ARP000103072 patent/AR024418A1/en active Pending
-
2010
- 2010-08-26 UY UY0001032855A patent/UY32855A/en unknown
Also Published As
Publication number | Publication date |
---|---|
BRPI0011834C1 (en) | 2021-05-25 |
AR024418A1 (en) | 2002-10-02 |
TWI230156B (en) | 2005-04-01 |
BR0011834A (en) | 2002-03-12 |
MY140484A (en) | 2009-12-31 |
CO5180636A1 (en) | 2002-07-30 |
BRPI0011834B8 (en) | 2015-12-22 |
PL352357A1 (en) | 2003-08-11 |
BR0011834B1 (en) | 2014-08-12 |
PL212659B1 (en) | 2012-11-30 |
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