UY32415A - NUEVOS DERIVADOS DE TETRAHIDROPIRAZOLO[3,4-c]ISOQUINOLIN-5-AMINA - Google Patents

NUEVOS DERIVADOS DE TETRAHIDROPIRAZOLO[3,4-c]ISOQUINOLIN-5-AMINA

Info

Publication number
UY32415A
UY32415A UY0001032415A UY32415A UY32415A UY 32415 A UY32415 A UY 32415A UY 0001032415 A UY0001032415 A UY 0001032415A UY 32415 A UY32415 A UY 32415A UY 32415 A UY32415 A UY 32415A
Authority
UY
Uruguay
Prior art keywords
isoquinolin
tetrahydropirazolo
amina
new derivatives
new
Prior art date
Application number
UY0001032415A
Other languages
English (en)
Inventor
Joan Taltavull Moll
Jordi Gracia Ferrer
Lluis Miquel Pages Santacana
Original Assignee
Almirall Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Almirall Sa filed Critical Almirall Sa
Publication of UY32415A publication Critical patent/UY32415A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Abstract

Se describen nuevos derivados de tetrahidropirazolo[3,4-c]isoquinolin-5-amina que tienen la estructura química de fórmula (I); así como un procedimiento para su preparación, composiciones farmacéuticas que los comprenden y su uso como inhibidores de la fosfodiesterasa IV (PDE4)
UY0001032415A 2009-02-27 2010-02-03 NUEVOS DERIVADOS DE TETRAHIDROPIRAZOLO[3,4-c]ISOQUINOLIN-5-AMINA UY32415A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP09382025A EP2226323A1 (en) 2009-02-27 2009-02-27 New tetrahydropyrazolo[3,4-c]isoquinolin-5-amine derivatives

Publications (1)

Publication Number Publication Date
UY32415A true UY32415A (es) 2010-04-30

Family

ID=40527935

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001032415A UY32415A (es) 2009-02-27 2010-02-03 NUEVOS DERIVADOS DE TETRAHIDROPIRAZOLO[3,4-c]ISOQUINOLIN-5-AMINA

Country Status (5)

Country Link
EP (1) EP2226323A1 (es)
AR (1) AR075603A1 (es)
TW (1) TW201031663A (es)
UY (1) UY32415A (es)
WO (1) WO2010097172A1 (es)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2599774A1 (en) * 2010-07-29 2013-06-05 Astellas Pharma Inc. Condensed ring pyridine compound

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2014087208A2 (en) * 2012-12-06 2014-06-12 Enaltec Labs Pvt. Ltd. A process of preparing alcaftadine
WO2017089347A1 (en) 2015-11-25 2017-06-01 Inserm (Institut National De La Sante Et De La Recherche Medicale) Methods and pharmaceutical compositions for the treatment of braf inhibitor resistant melanomas

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Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2599774A1 (en) * 2010-07-29 2013-06-05 Astellas Pharma Inc. Condensed ring pyridine compound
EP2599774A4 (en) * 2010-07-29 2014-01-08 Astellas Pharma Inc PYRIDINE COMPOUND WITH CONDENSED CYCLE

Also Published As

Publication number Publication date
AR075603A1 (es) 2011-04-20
EP2226323A1 (en) 2010-09-08
WO2010097172A1 (en) 2010-09-02
TW201031663A (en) 2010-09-01

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Effective date: 20110414