UY28924A1 - Compuestos antibioticos particularmente conteniendo anillos de oxazolidinona y isoxazolina sustituidos, composiciones farmaceuticas, preparación, intermedios para ello y su uso terapeutico. - Google Patents
Compuestos antibioticos particularmente conteniendo anillos de oxazolidinona y isoxazolina sustituidos, composiciones farmaceuticas, preparación, intermedios para ello y su uso terapeutico.Info
- Publication number
- UY28924A1 UY28924A1 UY28924A UY28924A UY28924A1 UY 28924 A1 UY28924 A1 UY 28924A1 UY 28924 A UY28924 A UY 28924A UY 28924 A UY28924 A UY 28924A UY 28924 A1 UY28924 A1 UY 28924A1
- Authority
- UY
- Uruguay
- Prior art keywords
- intermediates
- preparation
- pharmaceutical compositions
- therapeutic use
- antibiotic compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
Compuestos de fórmula (I) o una sal o profarmaco farmacéuticamente aceptable del mismo R1, R2, R3, R4 y R5, - C(O)R6 o R4 y R5 son como se definieron en la memoria descriptiva y reivindicaciones. Métodos para lograr los compuestos de fórmula I, composiciones que los contienen y su uso como agentes antibacteriales.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB0411594A GB0411594D0 (en) | 2004-05-25 | 2004-05-25 | Chemical compounds |
GB0500055A GB0500055D0 (en) | 2005-01-05 | 2005-01-05 | Chemical compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
UY28924A1 true UY28924A1 (es) | 2005-12-30 |
Family
ID=34968779
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UY28924A UY28924A1 (es) | 2004-05-25 | 2005-05-25 | Compuestos antibioticos particularmente conteniendo anillos de oxazolidinona y isoxazolina sustituidos, composiciones farmaceuticas, preparación, intermedios para ello y su uso terapeutico. |
Country Status (14)
Country | Link |
---|---|
US (1) | US20080064689A1 (es) |
EP (1) | EP1753756A1 (es) |
JP (1) | JP2008500315A (es) |
KR (1) | KR20070027614A (es) |
AR (1) | AR049121A1 (es) |
AU (1) | AU2005247663A1 (es) |
BR (1) | BRPI0511554A (es) |
CA (1) | CA2567454A1 (es) |
IL (1) | IL179348A0 (es) |
MX (1) | MXPA06013539A (es) |
NO (1) | NO20065863L (es) |
TW (1) | TW200604185A (es) |
UY (1) | UY28924A1 (es) |
WO (1) | WO2005116021A1 (es) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR100854211B1 (ko) * | 2003-12-18 | 2008-08-26 | 동아제약주식회사 | 신규한 옥사졸리디논 유도체, 그의 제조방법 및 이를유효성분으로 하는 항생제용 약학 조성물 |
KR100848232B1 (ko) * | 2007-04-12 | 2008-07-24 | 일동제약주식회사 | 신규 헤테로 고리 또는 알콕시아미노메틸 옥사졸리디논 및그 제조방법 |
AU2009303301B2 (en) | 2008-10-10 | 2014-09-11 | Merck Sharp & Dohme Llc | Methods for preparing oxazolidinones and compositions containing them |
AU2009318783A1 (en) | 2008-11-20 | 2011-06-23 | Panacea Biotec Ltd. | Novel antimicrobials |
KR20170040371A (ko) | 2009-02-03 | 2017-04-12 | 머크 샤프 앤드 돔 코포레이션 | R)-3-(4-(2-(2-메틸테트라졸-5-일)피리딘-5-일)-3-플루오로페닐)-5-히드록시메틸 옥사졸리딘-2-온 디히드로겐 포스페이트의 결정형 |
US8580767B2 (en) * | 2009-05-28 | 2013-11-12 | Trius Therapeutics, Inc. | Oxazolidinone containing dimer compounds, compositions and methods to make and use |
CN102803224A (zh) | 2009-06-26 | 2012-11-28 | 万能药生物有限公司 | 新的氮杂双环己烷类化合物 |
US9139575B2 (en) | 2010-04-13 | 2015-09-22 | The Regents Of The University Of California | Broad spectrum antiviral and antiparasitic agents |
CN114874131A (zh) * | 2015-02-27 | 2022-08-09 | 海洋规划生物工厂株式会社 | Kakeromycin及其衍生物的制造方法 |
CN111471041B (zh) * | 2019-01-23 | 2022-09-20 | 中国科学院上海药物研究所 | 一种噁唑烷酮类抗菌药物中间体的合成方法 |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BR0212458A (pt) * | 2001-09-11 | 2004-10-19 | Astrazeneca Ab | Composto ou sal farmaceuticamente aceitável, ou um éster hidrolizável in vivo deste, pró-droga, método para a produção de um efeito antibacteriano em um animal de sangue quente, uso de um composto ou sal farmaceuticamente aceitável, ou um éster hidrolizável in vivo deste, composição farmacêutica, e, processo para a preparação de um composto ou sais farmaceuticamente aceitável, ou ésteres hidrolizáveis in vivo deste |
GB0227701D0 (en) * | 2002-11-28 | 2003-01-08 | Astrazeneca Ab | Chemical compounds |
AU2003302404B2 (en) * | 2002-11-28 | 2008-06-19 | Astrazeneca Ab | Oxazolidinone and / or isoxazoline derivatives as antibacterial agents |
TW200500360A (en) * | 2003-03-01 | 2005-01-01 | Astrazeneca Ab | Hydroxymethyl compounds |
-
2004
- 2004-05-24 US US11/569,148 patent/US20080064689A1/en not_active Abandoned
-
2005
- 2005-05-18 TW TW094116025A patent/TW200604185A/zh unknown
- 2005-05-24 EP EP05746731A patent/EP1753756A1/en not_active Withdrawn
- 2005-05-24 KR KR1020067027174A patent/KR20070027614A/ko not_active Application Discontinuation
- 2005-05-24 AU AU2005247663A patent/AU2005247663A1/en not_active Abandoned
- 2005-05-24 WO PCT/GB2005/002040 patent/WO2005116021A1/en not_active Application Discontinuation
- 2005-05-24 BR BRPI0511554-0A patent/BRPI0511554A/pt not_active Application Discontinuation
- 2005-05-24 AR ARP050102159A patent/AR049121A1/es unknown
- 2005-05-24 CA CA002567454A patent/CA2567454A1/en not_active Abandoned
- 2005-05-24 JP JP2007514084A patent/JP2008500315A/ja active Pending
- 2005-05-24 MX MXPA06013539A patent/MXPA06013539A/es not_active Application Discontinuation
- 2005-05-25 UY UY28924A patent/UY28924A1/es not_active Application Discontinuation
-
2006
- 2006-11-16 IL IL179348A patent/IL179348A0/en unknown
- 2006-12-19 NO NO20065863A patent/NO20065863L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
EP1753756A1 (en) | 2007-02-21 |
CA2567454A1 (en) | 2005-12-08 |
MXPA06013539A (es) | 2007-01-26 |
IL179348A0 (en) | 2007-03-08 |
KR20070027614A (ko) | 2007-03-09 |
JP2008500315A (ja) | 2008-01-10 |
WO2005116021A1 (en) | 2005-12-08 |
AR049121A1 (es) | 2006-06-28 |
BRPI0511554A (pt) | 2008-01-02 |
US20080064689A1 (en) | 2008-03-13 |
AU2005247663A1 (en) | 2005-12-08 |
TW200604185A (en) | 2006-02-01 |
NO20065863L (no) | 2007-02-20 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
UY28924A1 (es) | Compuestos antibioticos particularmente conteniendo anillos de oxazolidinona y isoxazolina sustituidos, composiciones farmaceuticas, preparación, intermedios para ello y su uso terapeutico. | |
UY32462A (es) | Derivados de bifenilo novedosos para el tratamiento de infección por virus de hepatitis c 644 | |
UY28885A1 (es) | 4-fenilamino-quinazolin-6-il-amidas referencia cruzada a solicitud(es) relacionada(s) | |
DOP2009000124A (es) | Derivados de benzamida como receptores agonista ep4 | |
UY29087A1 (es) | Derivados de adamantilo, composiciones farmaceuticas que los contienen, procesos para su preparacion y uso terapeutico | |
PA8591701A1 (es) | Derivados de pirrolopirimidina | |
UY30819A1 (es) | Derivados de pirazol, composiciones farmacéuticas conteniéndolos, procesos de preparacion y aplicaciones | |
UY29234A1 (es) | Derivados de adamantano, composiciones farmacéuticas que los contienen, procedimientos de preparación de ambos y aplicaciones. | |
UY31430A1 (es) | Derivados de piridina y pirazina -83 | |
GT200600518A (es) | Derivados de pirimidina | |
UY30310A1 (es) | Derivados 2-azetidinona, sales, solvatos, composiciones farmacéuticas conteniéndolos, procesos de preparacion y aplicaciones | |
CL2011002706A1 (es) | Compuestos derivados de 4-(1,3-oxazol-2-il)-1h-indazol; composicion farmaceutica que los comprende; y sus usos en el tratamiento de enfermedades tales como epoc, autoinmunes, asma, entre otras. | |
ECSP099371A (es) | INHIBIDORES ESPIRO CETONA DE ACETIL-CoA CARBOXILASA | |
AR054347A1 (es) | Combinaciones terapeuticas para el tratamiento o la prevencion de la depresion | |
UY30327A1 (es) | Nuevos compuestos ii | |
UY30183A1 (es) | Derivados de quinolina | |
UY28756A1 (es) | Compuestos | |
ECSP12012292A (es) | Ciertas amino-piridazinas, composicioines de las mismas y métodos de uso de los mismos | |
BRPI0518993A2 (pt) | composto ou um sal, solvato ou Éster farmaceuticamente aceitÁvel do mesmo, composiÇço farmacÊutica, e, uso de um composto | |
UY29198A1 (es) | Derivados sustituidos de quinazolinona y derivados sustituidos de quinazolina-2, 4-diona, composiciones conteniéndolos, procedimientos de preparación y aplicaciones | |
UY29370A1 (es) | Derivados de tiazol, composiciones que lo contienen, procedimientos de preparación y aplicaciones | |
CU20090058A7 (es) | Compuestos de pirazolina y su uso y composiciones farmacéuticas | |
UY31141A1 (es) | Compuestos de piperidina y sus usos | |
UY31071A1 (es) | Derivados heterociclicos sustituidos y su uso farmaceutico y composiciones | |
AR074604A1 (es) | Derivados de 5-amino-2-(1-hidroxi-etil)-tetrahidropirano. |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
109 | Application deemed to be withdrawn |
Effective date: 20160518 |