UA94065C2 - Dihydropseudoerythromycin derivatives - Google Patents

Dihydropseudoerythromycin derivatives

Info

Publication number
UA94065C2
UA94065C2 UAA200806366A UAA200806366A UA94065C2 UA 94065 C2 UA94065 C2 UA 94065C2 UA A200806366 A UAA200806366 A UA A200806366A UA A200806366 A UAA200806366 A UA A200806366A UA 94065 C2 UA94065 C2 UA 94065C2
Authority
UA
Ukraine
Prior art keywords
dihydropseudoerythromycin
derivatives
dihydropseudoerythromycin derivatives
compounds
salts
Prior art date
Application number
UAA200806366A
Other languages
English (en)
Ukrainian (uk)
Inventor
Сатоши Омура
Тошияки Суназука
Кеничиро Нагаи
Хидеаки Шима
Харуко Ямабе
Original Assignee
Зе Китасато Инститьют
Афиникс, Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Зе Китасато Инститьют, Афиникс, Инк. filed Critical Зе Китасато Инститьют
Publication of UA94065C2 publication Critical patent/UA94065C2/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/10—Drugs for disorders of the urinary system of the bladder
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/16—Otologicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Dermatology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Medical Preparation Storing Or Oral Administration Devices (AREA)

Abstract

Изобретение касается соединения, представленного формулой [I], где каждый радикал является таким, как определено в описании, или его фармацевтически приемлемой соли, а также фармацевтической композиции, которая содержит соединение как активный ингредиент.[I]
UAA200806366A 2005-10-14 2006-10-13 Dihydropseudoerythromycin derivatives UA94065C2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2005301070 2005-10-14

Publications (1)

Publication Number Publication Date
UA94065C2 true UA94065C2 (en) 2011-04-11

Family

ID=37942921

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA200806366A UA94065C2 (en) 2005-10-14 2006-10-13 Dihydropseudoerythromycin derivatives

Country Status (18)

Country Link
US (1) US8133871B2 (ru)
EP (1) EP1950219B1 (ru)
JP (1) JP5118973B2 (ru)
KR (1) KR101384927B1 (ru)
CN (1) CN101326192B (ru)
AT (1) ATE513842T1 (ru)
AU (1) AU2006300215B2 (ru)
BR (1) BRPI0617391A2 (ru)
CA (1) CA2625055C (ru)
EA (1) EA015737B1 (ru)
ES (1) ES2369898T3 (ru)
IL (1) IL190643A (ru)
MY (1) MY147211A (ru)
NZ (1) NZ567772A (ru)
PL (1) PL1950219T3 (ru)
UA (1) UA94065C2 (ru)
WO (1) WO2007043710A1 (ru)
ZA (1) ZA200803414B (ru)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7776314B2 (en) 2002-06-17 2010-08-17 Grunenthal Gmbh Abuse-proofed dosage system
DE10336400A1 (de) 2003-08-06 2005-03-24 Grünenthal GmbH Gegen Missbrauch gesicherte Darreichungsform
DE102005005446A1 (de) 2005-02-04 2006-08-10 Grünenthal GmbH Bruchfeste Darreichungsformen mit retardierter Freisetzung
DE10361596A1 (de) 2003-12-24 2005-09-29 Grünenthal GmbH Verfahren zur Herstellung einer gegen Missbrauch gesicherten Darreichungsform
US20070048228A1 (en) 2003-08-06 2007-03-01 Elisabeth Arkenau-Maric Abuse-proofed dosage form
DE102004032049A1 (de) 2004-07-01 2006-01-19 Grünenthal GmbH Gegen Missbrauch gesicherte, orale Darreichungsform
DE102005005449A1 (de) 2005-02-04 2006-08-10 Grünenthal GmbH Verfahren zur Herstellung einer gegen Missbrauch gesicherten Darreichungsform
DE102007011485A1 (de) 2007-03-07 2008-09-11 Grünenthal GmbH Darreichungsform mit erschwertem Missbrauch
US8383152B2 (en) 2008-01-25 2013-02-26 Gruenenthal Gmbh Pharmaceutical dosage form
SI2273983T1 (sl) 2008-05-09 2016-11-30 Gruenenthal Gmbh Postopek za pripravo intermediatne praškaste formulacije in končne trdne odmerne oblike z uporabo stopnje strjevanja z razprševanjem
TW201105316A (en) 2009-07-22 2011-02-16 Gruenenthal Gmbh Hot-melt extruded pharmaceutical dosage form
AU2010275755B2 (en) 2009-07-22 2014-04-24 Grünenthal GmbH Oxidation-stabilized tamper-resistant dosage form
MX2013002377A (es) 2010-09-02 2013-04-29 Gruenenthal Gmbh Forma de dosificacion resistente a manipulacion que comprende una sal inorganica.
CN103179954A (zh) 2010-09-02 2013-06-26 格吕伦塔尔有限公司 包含阴离子聚合物的抗破碎剂型
US10201502B2 (en) 2011-07-29 2019-02-12 Gruenenthal Gmbh Tamper-resistant tablet providing immediate drug release
RS56527B1 (sr) 2011-07-29 2018-02-28 Gruenenthal Gmbh Tableta za trenutno oslobađanje leka rezistentna na zloupotrebu
MX356421B (es) 2012-02-28 2018-05-29 Gruenenthal Gmbh Forma de dosificacion resistente a la manipulacion indebida que comprende un compuesto farmacologicamente activo y un polimero anionico.
EA201401139A1 (ru) 2012-04-18 2015-03-31 Грюненталь Гмбх Устойчивая к разрушению и к сбросу дозы фармацевтическая лекарственная форма
US10064945B2 (en) 2012-05-11 2018-09-04 Gruenenthal Gmbh Thermoformed, tamper-resistant pharmaceutical dosage form containing zinc
BR112015026549A2 (pt) 2013-05-29 2017-07-25 Gruenenthal Gmbh forma de dosagem à prova de violação contendo uma ou mais partículas
CA2913209A1 (en) 2013-05-29 2014-12-04 Grunenthal Gmbh Tamper resistant dosage form with bimodal release profile
CA2917136C (en) 2013-07-12 2022-05-31 Grunenthal Gmbh Tamper-resistant dosage form containing ethylene-vinyl acetate polymer
WO2015078891A1 (en) 2013-11-26 2015-06-04 Farmaceutici Formenti S.P.A. Preparation of a powdery pharmaceutical composition by means of cryo-milling
WO2015173195A1 (en) 2014-05-12 2015-11-19 Grünenthal GmbH Tamper resistant immediate release capsule formulation comprising tapentadol
MX2016015417A (es) 2014-05-26 2017-02-22 Gruenenthal Gmbh Multiparticulas protegidas contra vertido de dosis etanolico.
CN107531737A (zh) * 2015-03-25 2018-01-02 哈佛大学的校长及成员们 脱氧糖胺的合成
EP3285745A1 (en) 2015-04-24 2018-02-28 Grünenthal GmbH Tamper-resistant dosage form with immediate release and resistance against solvent extraction
JP2018526414A (ja) 2015-09-10 2018-09-13 グリュネンタール・ゲゼルシャフト・ミト・ベシュレンクテル・ハフツング 乱用抑止性の即放性製剤を用いた経口過剰摂取に対する保護

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5106961A (en) 1987-05-26 1992-04-21 Eli Lilly And Company Erythromycin ring-contracted derivatives
ATE321770T1 (de) 2000-08-17 2006-04-15 Kitasato Inst Pseudoerythromycin-derivate
CA2429709A1 (en) * 2000-12-01 2002-07-04 Gary Ashley Motilide compounds
US20020094962A1 (en) 2000-12-01 2002-07-18 Gary Ashley Motilide compounds
US20040067896A1 (en) 2002-07-25 2004-04-08 The Kitasato Institute Novel pseudoerythromycin derivatives
WO2004039823A1 (ja) * 2002-10-29 2004-05-13 The Kitasato Institute 抗真菌活性増強作用を有する新規マクロライド誘導体

Also Published As

Publication number Publication date
US20090131341A1 (en) 2009-05-21
US8133871B2 (en) 2012-03-13
NZ567772A (en) 2010-07-30
ZA200803414B (en) 2009-09-30
PL1950219T3 (pl) 2011-11-30
EP1950219A4 (en) 2010-02-03
ATE513842T1 (de) 2011-07-15
CN101326192B (zh) 2012-06-20
AU2006300215A1 (en) 2007-04-19
KR20080064861A (ko) 2008-07-09
WO2007043710A9 (ja) 2007-06-07
EA015737B1 (ru) 2011-10-31
BRPI0617391A2 (pt) 2011-07-26
MY147211A (en) 2012-11-14
IL190643A0 (en) 2008-11-03
CA2625055A1 (en) 2007-04-19
ES2369898T3 (es) 2011-12-07
IL190643A (en) 2012-03-29
EP1950219B1 (en) 2011-06-22
KR101384927B1 (ko) 2014-04-11
CA2625055C (en) 2013-12-24
EP1950219A1 (en) 2008-07-30
EA200801083A1 (ru) 2009-02-27
CN101326192A (zh) 2008-12-17
JP5118973B2 (ja) 2013-01-16
JPWO2007043710A1 (ja) 2009-07-16
WO2007043710A1 (ja) 2007-04-19
AU2006300215B2 (en) 2012-06-21

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