UA85505C2 - Kinase inhibitors - Google Patents

Kinase inhibitors

Info

Publication number
UA85505C2
UA85505C2 UAA200610433A UAA200610433A UA85505C2 UA 85505 C2 UA85505 C2 UA 85505C2 UA A200610433 A UAA200610433 A UA A200610433A UA A200610433 A UAA200610433 A UA A200610433A UA 85505 C2 UA85505 C2 UA 85505C2
Authority
UA
Ukraine
Prior art keywords
kinase inhibitors
formula
present
inhibitors
provides kinase
Prior art date
Application number
UAA200610433A
Other languages
English (en)
Ukrainian (uk)
Inventor
Розанн Бонжуклян
Чафик Хамдоучи Хамдоучи
Чан Ши
Диос Альфонсо де
Прадо Мириам Филадельфа Дель
Агадо Карлос Харамильо
Прамила Котиян
Мери Маргарет Мадер
Шейла Плейт Сельгас
Консепсьон Санчес-Мартинес
Original Assignee
Эли Лилли Энд Компани
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34837430&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UA85505(C2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Эли Лилли Энд Компани filed Critical Эли Лилли Энд Компани
Publication of UA85505C2 publication Critical patent/UA85505C2/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Abstract

Это изобретение предлагает ингибиторы киназы Формулы I.
UAA200610433A 2004-01-30 2005-01-25 Kinase inhibitors UA85505C2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US54083004P 2004-01-30 2004-01-30

Publications (1)

Publication Number Publication Date
UA85505C2 true UA85505C2 (en) 2009-01-26

Family

ID=34837430

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA200610433A UA85505C2 (en) 2004-01-30 2005-01-25 Kinase inhibitors

Country Status (26)

Country Link
US (2) US7582652B2 (ru)
EP (1) EP1713805B1 (ru)
CN (1) CN100516064C (ru)
AR (1) AR047466A1 (ru)
AT (1) ATE433449T1 (ru)
AU (1) AU2005210459B2 (ru)
CA (1) CA2559128C (ru)
CY (1) CY1109234T1 (ru)
DE (1) DE602005014848D1 (ru)
DK (1) DK1713805T3 (ru)
DO (1) DOP2005000010A (ru)
ES (1) ES2326819T3 (ru)
HK (1) HK1100141A1 (ru)
IL (1) IL178103A (ru)
MY (1) MY143516A (ru)
NZ (1) NZ549780A (ru)
PE (1) PE20050689A1 (ru)
PL (1) PL1713805T3 (ru)
PT (1) PT1713805E (ru)
RU (1) RU2348635C2 (ru)
SI (1) SI1713805T1 (ru)
SV (1) SV2006002001A (ru)
TW (1) TWI332003B (ru)
UA (1) UA85505C2 (ru)
WO (1) WO2005075478A1 (ru)
ZA (1) ZA200607648B (ru)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI332003B (en) * 2004-01-30 2010-10-21 Lilly Co Eli Kinase inhibitors
US7776869B2 (en) * 2004-10-18 2010-08-17 Amgen Inc. Heteroaryl-substituted alkyne compounds and method of use
EP1992344A1 (en) 2007-05-18 2008-11-19 Institut Curie P38 alpha as a therapeutic target in pathologies linked to FGFR3 mutation
NZ604306A (en) * 2010-05-17 2015-02-27 Incozen Therapeutics Pvt Ltd Novel 3,5-disubstitued-3h-imidazo[4,5-b]pyridine and 3,5- disubstitued -3h-[1,2,3]triazolo[4,5-b] pyridine compounds as modulators of protein kinases
TWI410425B (zh) * 2010-12-03 2013-10-01 Lilly Co Eli 唑并［５，４－ｂ］吡啶－５－基化合物
PT2780011T (pt) * 2011-11-11 2018-05-14 Lilly Co Eli Terapia de combinação para cancro do ovário
CN104640918A (zh) * 2012-07-23 2015-05-20 阿克伦大学 含有有机改性蒙脱石的基于聚异丁烯的聚氨酯
TWI731317B (zh) 2013-12-10 2021-06-21 美商健臻公司 原肌球蛋白相關之激酶（ｔｒｋ）抑制劑
TWI780438B (zh) 2014-12-18 2022-10-11 美商健臻公司 原肌球蛋白相關激酶（ｔｒｋ）抑制劑之醫藥調配物
MA41179A (fr) 2014-12-19 2017-10-24 Cancer Research Tech Ltd Composés inhibiteurs de parg
MX371167B (es) * 2015-03-02 2020-01-21 Rigel Pharmaceuticals Inc Inhibidores de inhibidores del factor beta de crecimiento de transformacion (tgf-beta).
PT3691620T (pt) 2017-10-05 2022-10-06 Fulcrum Therapeutics Inc Os inibidores da quinase p38 reduzem a expressão de dux4 e genes a jusante para o tratamento de fshd
US10342786B2 (en) 2017-10-05 2019-07-09 Fulcrum Therapeutics, Inc. P38 kinase inhibitors reduce DUX4 and downstream gene expression for the treatment of FSHD
US10899869B2 (en) 2019-01-24 2021-01-26 The University Of Akron Glycerol containing polyurethanes and polyurethane nanocomposites
TW202112368A (zh) 2019-06-13 2021-04-01 荷蘭商法西歐知識產權股份有限公司 用於治療有關dux4表現之疾病的抑制劑組合

Family Cites Families (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL104369A0 (en) 1992-01-13 1993-05-13 Smithkline Beecham Corp Novel compounds and compositions
DE19503806A1 (de) * 1994-02-11 1995-08-17 Bernhardt Apparatebau Gmbh Co Vorrichtung zum Aufblasen eines Behälters oder eines Schwimmkörpers, insbesondere einer Schwimmweste
US6426360B1 (en) 1994-07-28 2002-07-30 G D Searle & Co. 4,5-substituted imidazolyl compounds for the treatment of inflammation
US5620999A (en) 1994-07-28 1997-04-15 Weier; Richard M. Benzenesulfonamide subtituted imidazolyl compounds for the treatment of inflammation
US5717100A (en) 1995-10-06 1998-02-10 Merck & Co., Inc. Substituted imidazoles having anti-cancer and cytokine inhibitory activity
WO1998007425A1 (en) 1996-08-21 1998-02-26 Smithkline Beecham Corporation Imidazole compounds, compositions and use
US6087496A (en) 1998-05-22 2000-07-11 G. D. Searle & Co. Substituted pyrazoles suitable as p38 kinase inhibitors
US6180632B1 (en) 1997-05-28 2001-01-30 Aventis Pharmaceuticals Products Inc. Quinoline and quinoxaline compounds which inhibit platelet-derived growth factor and/or p56lck tyrosine kinases
WO1999000130A1 (en) 1997-06-30 1999-01-07 Temple University - Of The Commonwealth System Of Higher Education Method for treating vulvar vestibulitis
AR016294A1 (es) * 1997-07-02 2001-07-04 Smithkline Beecham Corp Compuesto de imidazol sustituido, composicion farmaceutica que la contiene, su uso en la fabricacion de un medicamento y procedimiento para supreparacion
AU1924699A (en) 1997-12-19 1999-07-12 Smithkline Beecham Corporation Compounds of heteroaryl substituted imidazole, their pharmaceutical compositionsand uses
US6207687B1 (en) 1998-07-31 2001-03-27 Merck & Co., Inc. Substituted imidazoles having cytokine inhibitory activity
US6291457B1 (en) 1999-07-01 2001-09-18 Merck & Co., Inc. Compounds having cytokine inhibitory activity
ATE311385T1 (de) * 1999-10-27 2005-12-15 Novartis Pharma Gmbh Thiazol und imidazo(4,5-b)pyridin verbindungen und ihre verwendung als pharmazeutika
GB0007405D0 (en) * 2000-03-27 2000-05-17 Smithkline Beecham Corp Compounds
NZ526528A (en) 2001-03-09 2005-02-25 Pfizer Prod Inc Triazolopyridines as anti-inflammatory agents
CN100540538C (zh) 2001-04-16 2009-09-16 田边三菱制药株式会社 高传导率钙-活化k通道开启剂
WO2003062215A1 (en) 2002-01-25 2003-07-31 Kylix Pharmaceuticals B.V. 4(hetero-) aryl substituted (thia-/oxa-/pyra) zoles for inhibition of tie-2
DE60304718T2 (de) 2002-08-06 2007-04-26 Astrazeneca Ab Kondensierte pyridine und pyrimidine mit tie2 (tek) aktivität
TWI332003B (en) * 2004-01-30 2010-10-21 Lilly Co Eli Kinase inhibitors

Also Published As

Publication number Publication date
US7582652B2 (en) 2009-09-01
US20090318443A1 (en) 2009-12-24
PT1713805E (pt) 2009-08-20
CA2559128A1 (en) 2005-08-18
US20090036445A1 (en) 2009-02-05
AR047466A1 (es) 2006-01-18
CA2559128C (en) 2013-04-16
SV2006002001A (es) 2006-02-15
CN100516064C (zh) 2009-07-22
TWI332003B (en) 2010-10-21
IL178103A (en) 2011-04-28
CN1938302A (zh) 2007-03-28
EP1713805A1 (en) 2006-10-25
ES2326819T3 (es) 2009-10-20
HK1100141A1 (en) 2007-09-07
RU2006138606A (ru) 2008-05-10
AU2005210459A1 (en) 2005-08-18
PL1713805T3 (pl) 2009-10-30
ATE433449T1 (de) 2009-06-15
DE602005014848D1 (de) 2009-07-23
NZ549780A (en) 2010-01-29
MY143516A (en) 2011-05-31
AU2005210459B2 (en) 2010-10-21
PE20050689A1 (es) 2005-09-27
TW200526660A (en) 2005-08-16
WO2005075478A1 (en) 2005-08-18
SI1713805T1 (sl) 2009-10-31
ZA200607648B (en) 2008-06-25
DK1713805T3 (da) 2009-08-17
RU2348635C2 (ru) 2009-03-10
CY1109234T1 (el) 2014-07-02
EP1713805B1 (en) 2009-06-10
DOP2005000010A (es) 2005-11-15

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