TW200744598A - Process for the production of freeze-dried preparations containing quinolones - Google Patents
Process for the production of freeze-dried preparations containing quinolonesInfo
- Publication number
- TW200744598A TW200744598A TW095136062A TW95136062A TW200744598A TW 200744598 A TW200744598 A TW 200744598A TW 095136062 A TW095136062 A TW 095136062A TW 95136062 A TW95136062 A TW 95136062A TW 200744598 A TW200744598 A TW 200744598A
- Authority
- TW
- Taiwan
- Prior art keywords
- freeze
- production
- mixture
- preparations containing
- dried preparations
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/19—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles lyophilised, i.e. freeze-dried, solutions or dispersions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/4375—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having nitrogen as a ring heteroatom, e.g. quinolizines, naphthyridines, berberine, vincamine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5383—1,4-Oxazines, e.g. morpholine ortho- or peri-condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/02—Inorganic compounds
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2005282393 | 2005-09-28 |
Publications (1)
Publication Number | Publication Date |
---|---|
TW200744598A true TW200744598A (en) | 2007-12-16 |
Family
ID=37899754
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
TW095136062A TW200744598A (en) | 2005-09-28 | 2006-09-28 | Process for the production of freeze-dried preparations containing quinolones |
Country Status (5)
Country | Link |
---|---|
US (1) | US8129533B2 (zh) |
EP (1) | EP1930006A4 (zh) |
JP (1) | JPWO2007037330A1 (zh) |
TW (1) | TW200744598A (zh) |
WO (1) | WO2007037330A1 (zh) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN102961328A (zh) * | 2012-12-13 | 2013-03-13 | 鼎正动物药业(天津)有限公司 | 一种左氧氟沙星注射液及其制备方法 |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7928232B2 (en) * | 2005-05-20 | 2011-04-19 | Daiichi Sankyo Company, Limited | Method for producing asymmetric tetrasubstituted carbon atom-containing compound |
US7977346B2 (en) | 2006-01-17 | 2011-07-12 | Guoqing Paul Chen | Spiro compounds and methods of use |
TWI386401B (zh) * | 2006-03-27 | 2013-02-21 | Daiichi Seiyaku Co | 醫藥用水合物 |
JP2009079003A (ja) * | 2007-09-26 | 2009-04-16 | Daiichi Sankyo Co Ltd | 医薬用水和物を含有する医薬 |
JP5195655B2 (ja) * | 2009-06-11 | 2013-05-08 | 富士通株式会社 | 移動端末、通信システムおよび通信方法 |
CN103087042B (zh) * | 2012-03-09 | 2015-02-18 | 南京优科生物医药有限公司 | 西他沙星的盐及制药用途 |
CN103230372B (zh) * | 2013-01-17 | 2016-04-06 | 北京赛盟医药科技发展有限公司 | 注射用盐酸莫西沙星粉针及其制备方法 |
JP2016511273A (ja) * | 2013-03-08 | 2016-04-14 | メリンタ セラピューティクス、インク | D−グルシトール,1−デオキシ−1−(メチルアミノ)−,1−(6−アミノ−3,5−ジフルオロピリジン−2−イル)−8−クロロ−6−フルオロ−1,4−ジヒドロ−7−(3−ヒドロキシアゼチジン−1−イル)−4−オキソ−3−キノリンカルボン酸塩の結晶型 |
JP6487051B2 (ja) * | 2014-12-30 | 2019-03-20 | サムヤン バイオファーマシューティカルズ コーポレイションSamyang Biopharmaceuticals Corporation | ポリマーナノ粒子の凍結乾燥物、及びその製造方法 |
Family Cites Families (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS57127406A (en) * | 1981-01-29 | 1982-08-07 | Nippon Chemiphar Co Ltd | Production of crystalline freeze dried powder |
JPH06786B2 (ja) * | 1984-02-22 | 1994-01-05 | 塩野義製薬株式会社 | セフアロチンナトリウムの結晶性凍結乾燥製剤の製造法 |
US4839355A (en) * | 1987-09-09 | 1989-06-13 | Sterling Drug Inc. | Tricyclic-pyridinylquinoline compounds, their preparation and use |
JPH01175935A (ja) * | 1987-12-28 | 1989-07-12 | Kyorin Pharmaceut Co Ltd | 凍結乾燥注射剤 |
JPH02104527A (ja) * | 1988-10-11 | 1990-04-17 | Kayaku:Kk | 1−〔(4´‐ヒドロキシ‐2´‐ブテノキシ)メチル〕‐2‐ニトロイミダゾールの凍結乾燥製剤の製造法 |
US7176313B2 (en) * | 2000-02-09 | 2007-02-13 | Daiichi Pharmaceutical Co., Ltd. | Anti acid-fast bacterial agent containing pyridonecarboxylic acids as active ingredient |
IT1319664B1 (it) * | 2000-11-17 | 2003-10-23 | Pharma Biotech Ltd | Addotti di antibatterici chinolonici con polimeri polisaccaridicinaturali. |
DE60130359T2 (de) * | 2000-11-20 | 2008-06-26 | Daiichi Sankyo Co., Ltd. | Deshalogenverbindungen |
JP4384402B2 (ja) | 2001-11-30 | 2009-12-16 | 富山化学工業株式会社 | デスフルオロピリドンカルボン酸系化合物を含有する水溶液剤およびその粉末化物並びにそれら製造方法 |
DE10204792A1 (de) * | 2002-02-06 | 2003-08-14 | Merck Patent Gmbh | Lyophilisierte Zubereitung enthaltend Immuncytokine |
US7563805B2 (en) | 2005-05-19 | 2009-07-21 | Daiichi Pharmaceutical Co., Ltd. | Tri-, tetra-substituted-3-aminopyrrolidine derivative |
-
2006
- 2006-09-28 EP EP06810754A patent/EP1930006A4/en not_active Withdrawn
- 2006-09-28 JP JP2007537678A patent/JPWO2007037330A1/ja active Pending
- 2006-09-28 TW TW095136062A patent/TW200744598A/zh unknown
- 2006-09-28 WO PCT/JP2006/319307 patent/WO2007037330A1/ja active Application Filing
- 2006-09-28 US US12/067,826 patent/US8129533B2/en not_active Expired - Fee Related
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN102961328A (zh) * | 2012-12-13 | 2013-03-13 | 鼎正动物药业(天津)有限公司 | 一种左氧氟沙星注射液及其制备方法 |
CN102961328B (zh) * | 2012-12-13 | 2014-12-03 | 鼎正动物药业(天津)有限公司 | 一种左氧氟沙星注射液及其制备方法 |
Also Published As
Publication number | Publication date |
---|---|
EP1930006A1 (en) | 2008-06-11 |
EP1930006A4 (en) | 2010-10-13 |
US20080300403A1 (en) | 2008-12-04 |
WO2007037330A1 (ja) | 2007-04-05 |
US8129533B2 (en) | 2012-03-06 |
JPWO2007037330A1 (ja) | 2009-04-09 |
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