WO2010079506A3 - Pharmaceutical composition of aripiprazole - Google Patents

Pharmaceutical composition of aripiprazole Download PDF

Info

Publication number
WO2010079506A3
WO2010079506A3 PCT/IN2009/000356 IN2009000356W WO2010079506A3 WO 2010079506 A3 WO2010079506 A3 WO 2010079506A3 IN 2009000356 W IN2009000356 W IN 2009000356W WO 2010079506 A3 WO2010079506 A3 WO 2010079506A3
Authority
WO
WIPO (PCT)
Prior art keywords
aripiprazole
pharmaceutical composition
present
solid oral
oral pharmaceutical
Prior art date
Application number
PCT/IN2009/000356
Other languages
French (fr)
Other versions
WO2010079506A2 (en
Inventor
Rakesh Sheth
Original Assignee
Torrent Pharmaceuticals Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Torrent Pharmaceuticals Ltd. filed Critical Torrent Pharmaceuticals Ltd.
Publication of WO2010079506A2 publication Critical patent/WO2010079506A2/en
Publication of WO2010079506A3 publication Critical patent/WO2010079506A3/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

The present invention relates to stable, solid oral pharmaceutical composition comprising aripiprazole manufactured by wet granulation, wherein intragranular stage is devoid of diluent. The present invention further relates to processes for the preparation of said solid oral pharmaceutical composition of aripiprazole.
PCT/IN2009/000356 2008-06-23 2009-06-22 Pharmaceutical composition of aripiprazole WO2010079506A2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN1302/MUM/2008 2008-06-23
IN1302MU2008 2008-06-23

Publications (2)

Publication Number Publication Date
WO2010079506A2 WO2010079506A2 (en) 2010-07-15
WO2010079506A3 true WO2010079506A3 (en) 2010-09-10

Family

ID=42272511

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/IN2009/000356 WO2010079506A2 (en) 2008-06-23 2009-06-22 Pharmaceutical composition of aripiprazole

Country Status (1)

Country Link
WO (1) WO2010079506A2 (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TR201000948A1 (en) * 2010-02-09 2011-08-22 Sanovel İlaç San.Ve Ti̇c.A.Ş. Aripiprazole formulations.
WO2013100878A1 (en) * 2011-12-27 2013-07-04 Mahmut Bilgic Pharmaceutical formulations comprising aripiprazole
WO2014104989A1 (en) * 2011-12-27 2014-07-03 Mahmut Bilgic Pharmaceutical compositions comprising aripiprazole
TW201343201A (en) * 2012-03-06 2013-11-01 Otsuka Pharma Co Ltd Sustained release oral solid preparation
WO2013175508A2 (en) * 2012-05-24 2013-11-28 Medreich Limited Stable pharmaceutical composition of aripiprazole

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20060257471A1 (en) * 2005-03-17 2006-11-16 Ettema Gerrit J Pharmaceutical tablets of crystalline Type II aripiprazole
WO2007081366A1 (en) * 2006-01-05 2007-07-19 Teva Pharmaceutical Industries Ltd. Wet granulation pharmaceutical compositions of aripiprazole
WO2007081367A1 (en) * 2006-01-05 2007-07-19 Teva Pharmaceutical Industries Ltd. Dry formulations of aripiprazole

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5006528A (en) 1988-10-31 1991-04-09 Otsuka Pharmaceutical Co., Ltd. Carbostyril derivatives
AR033485A1 (en) 2001-09-25 2003-12-26 Otsuka Pharma Co Ltd MEDICINAL SUBSTANCE OF ARIPIPRAZOL OF LOW HYGROSCOPICITY AND PROCESS FOR THE PREPARATION OF THE SAME

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20060257471A1 (en) * 2005-03-17 2006-11-16 Ettema Gerrit J Pharmaceutical tablets of crystalline Type II aripiprazole
WO2007081366A1 (en) * 2006-01-05 2007-07-19 Teva Pharmaceutical Industries Ltd. Wet granulation pharmaceutical compositions of aripiprazole
WO2007081367A1 (en) * 2006-01-05 2007-07-19 Teva Pharmaceutical Industries Ltd. Dry formulations of aripiprazole

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
AOKI S ET AL: "Study on Crystal Transformation of ARIPIPRAZOL", 19961006, 6 October 1996 (1996-10-06), pages 937 - 940, XP002970982 *

Also Published As

Publication number Publication date
WO2010079506A2 (en) 2010-07-15

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