TW200524930A - Quinolone antibacterial agents - Google Patents

Quinolone antibacterial agents Download PDF

Info

Publication number
TW200524930A
TW200524930A TW093135213A TW93135213A TW200524930A TW 200524930 A TW200524930 A TW 200524930A TW 093135213 A TW093135213 A TW 093135213A TW 93135213 A TW93135213 A TW 93135213A TW 200524930 A TW200524930 A TW 200524930A
Authority
TW
Taiwan
Prior art keywords
ethyl
methyl
cyclopropyl
dihydro
cyano
Prior art date
Application number
TW093135213A
Other languages
English (en)
Chinese (zh)
Inventor
Edmund Lee Ellsworth
Clarke Bentley Taylor
Sean Timothy Murphy
Mark Ryan Rauckhorst
Jeremy Tyson Starr
Kim Marie Hutchings
Chris Limberakis
Denton Wade Hoyer
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of TW200524930A publication Critical patent/TW200524930A/zh

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
TW093135213A 2003-11-18 2004-11-17 Quinolone antibacterial agents TW200524930A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US52307103P 2003-11-18 2003-11-18
US60549604P 2004-08-31 2004-08-31

Publications (1)

Publication Number Publication Date
TW200524930A true TW200524930A (en) 2005-08-01

Family

ID=34623167

Family Applications (1)

Application Number Title Priority Date Filing Date
TW093135213A TW200524930A (en) 2003-11-18 2004-11-17 Quinolone antibacterial agents

Country Status (6)

Country Link
AR (1) AR046638A1 (es)
NL (1) NL1027545C2 (es)
PE (1) PE20050582A1 (es)
TW (1) TW200524930A (es)
UY (1) UY28622A1 (es)
WO (1) WO2005049602A1 (es)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI382980B (zh) * 2006-02-09 2013-01-21 Aicuris Gmbh & Co Kg 經取代之喹諾酮類iii

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1666477B1 (en) 2003-09-10 2013-07-03 Kyorin Pharmaceutical Co., Ltd. 7-(4-substituted 3- cyclopropylaminomethyl-1- pyrrolidinyl) q uinolonecarboxylic acid derivative
ES2431050T3 (es) 2005-08-04 2013-11-22 Sirtris Pharmaceuticals, Inc. Benzotiazoles y tiazolopiridinas como moduladores de la sirtuína
DK2097400T3 (da) * 2007-01-05 2013-10-14 Daiichi Sankyo Co Ltd Kondenseret, substitueret aminopyrrolidinderivat
CN101622240B (zh) * 2007-01-05 2014-07-23 第一三共株式会社 稠合取代氨基吡咯烷衍生物
WO2008143343A1 (ja) 2007-05-24 2008-11-27 Kyorin Pharmaceutical Co., Ltd. １４位置換基に複素芳香環カルボン酸構造を有するムチリン誘導体
DE102007036068A1 (de) 2007-08-01 2009-02-05 Wacker Chemie Ag Verfahren zur Herstellung von Alkyl-methoxymethyl-trimethylsilanylmethylaminen
JP5566288B2 (ja) 2008-05-30 2014-08-06 武田薬品工業株式会社 複素環化合物
PL2394999T3 (pl) 2009-02-06 2014-06-30 Nippon Shinyaku Co Ltd Pochodna aminopirazyny i lek
AR091858A1 (es) * 2012-07-25 2015-03-04 Sova Pharmaceuticals Inc INHIBIDORES DE CISTATIONIN-g-LIASA (CSE)
WO2016198342A1 (de) 2015-06-09 2016-12-15 Bayer Pharma Aktiengesellschaft Positiv allosterische modulatoren des muskarinergen m2 rezeptors
WO2018011017A1 (de) 2016-07-11 2018-01-18 Bayer Pharma Aktiengesellschaft 7-substituierte 1-pyridyl-naphthyridin-3-carbonsäureamide und ihre verwendung
EP3296298A1 (de) 2016-09-14 2018-03-21 Bayer Pharma Aktiengesellschaft 7-substituierte 1-aryl-naphthyridin-3-carbonsäureamide und ihre verwendung
JOP20190045A1 (ar) 2016-09-14 2019-03-14 Bayer Ag مركبات أميد حمض 1- أريل-نفثيريدين-3-كربوكسيليك مستبدلة في الموضع 7 واستخدامها.
US20190218188A1 (en) 2016-09-29 2019-07-18 Bayer Cropscience Aktiengesellschaft Novel 5-substituted imidazole derivatives

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI382980B (zh) * 2006-02-09 2013-01-21 Aicuris Gmbh & Co Kg 經取代之喹諾酮類iii

Also Published As

Publication number Publication date
AR046638A1 (es) 2005-12-14
NL1027545A1 (nl) 2005-05-23
WO2005049602A1 (en) 2005-06-02
NL1027545C2 (nl) 2006-01-17
PE20050582A1 (es) 2005-08-25
UY28622A1 (es) 2005-06-30

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