TN2009000551A1 - Nouveaux composes chimiques - Google Patents
Nouveaux composes chimiquesInfo
- Publication number
- TN2009000551A1 TN2009000551A1 TNP2009000551A TN2009000551A TN2009000551A1 TN 2009000551 A1 TN2009000551 A1 TN 2009000551A1 TN P2009000551 A TNP2009000551 A TN P2009000551A TN 2009000551 A TN2009000551 A TN 2009000551A TN 2009000551 A1 TN2009000551 A1 TN 2009000551A1
- Authority
- TN
- Tunisia
- Prior art keywords
- chemical compounds
- new chemical
- compounds
- drug
- excessive
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/08—Bridged systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Immunology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Peptides Or Proteins (AREA)
Abstract
La présente invention concerne des composés de formule générale (1), dans laquelle R1 à R3 et L sont définis dans la revendication 1, qui sont appropriés pour le traitement de maladies caractérisées par une prolifération cellulaire excessive ou anormale, et leur utilisation pour préparer un médicament possédant les propriétés mentionnées ci-dessus.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP07111566 | 2007-07-02 | ||
PCT/EP2008/058433 WO2009003999A2 (fr) | 2007-07-02 | 2008-07-01 | Nouveaux composés chimiques |
Publications (1)
Publication Number | Publication Date |
---|---|
TN2009000551A1 true TN2009000551A1 (fr) | 2011-03-31 |
Family
ID=38792475
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
TNP2009000551A TN2009000551A1 (fr) | 2007-07-02 | 2009-12-31 | Nouveaux composes chimiques |
Country Status (21)
Country | Link |
---|---|
US (1) | US8889665B2 (fr) |
EP (1) | EP2173734B1 (fr) |
JP (1) | JP5511658B2 (fr) |
KR (1) | KR20100039849A (fr) |
CN (1) | CN101796045A (fr) |
AR (1) | AR067397A1 (fr) |
AU (1) | AU2008270300A1 (fr) |
BR (1) | BRPI0814601A2 (fr) |
CA (1) | CA2692383A1 (fr) |
CL (1) | CL2008001943A1 (fr) |
CO (1) | CO6251316A2 (fr) |
EA (1) | EA201000105A1 (fr) |
EC (1) | ECSP099823A (fr) |
IL (1) | IL202625A0 (fr) |
MA (1) | MA32120B1 (fr) |
MX (1) | MX2009013935A (fr) |
PE (1) | PE20090837A1 (fr) |
TN (1) | TN2009000551A1 (fr) |
TW (1) | TW200911789A (fr) |
UY (1) | UY31198A1 (fr) |
WO (1) | WO2009003999A2 (fr) |
Families Citing this family (26)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP2041116A1 (fr) | 2006-07-07 | 2009-04-01 | Boehringer Ingelheim International GmbH | Dérivés d'hétéroaryle substitués par phényle et leur utilisation en tant qu'agents antitumoraux |
CA2692379A1 (fr) * | 2007-07-02 | 2009-01-08 | Boehringer Ingelheim International Gmbh | Nouveaux composes chimiques |
PE20090837A1 (es) | 2007-07-02 | 2009-07-24 | Boehringer Ingelheim Int | Nuevos compuestos quimicos |
TW201014860A (en) | 2008-09-08 | 2010-04-16 | Boehringer Ingelheim Int | New chemical compounds |
CN102227421A (zh) | 2008-09-29 | 2011-10-26 | 贝林格尔.英格海姆国际有限公司 | 抗增殖化合物 |
WO2010094695A1 (fr) | 2009-02-17 | 2010-08-26 | Boehringer Ingelheim International Gmbh | Dérivés pyrimido-[5,4-d]-pyrimidine pour l'inhibition des tyrosine-kinases |
JP2010235575A (ja) * | 2009-03-09 | 2010-10-21 | Konica Minolta Holdings Inc | 含窒素縮合複素環化合物の製造方法 |
DE102009019962A1 (de) * | 2009-05-05 | 2010-11-11 | Merck Patent Gmbh | 3-([1,2,3]Triazol-4-yl)-pyrrolo[2,3-b]pyridinderivate |
WO2011117382A1 (fr) | 2010-03-26 | 2011-09-29 | Boehringer Ingelheim International Gmbh | Pyridyltriazoles |
JP5871896B2 (ja) | 2010-03-26 | 2016-03-01 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | B−rafキナーゼインヒビター |
UY33817A (es) | 2010-12-21 | 2012-07-31 | Boehringer Ingelheim Int | ?nuevas oxindolpirimidinas bencílicas?. |
US8710055B2 (en) | 2010-12-21 | 2014-04-29 | Boehringer Ingelheim International Gmbh | Triazolylphenyl sulfonamides as serine/threonine kinase inhibitors |
US8889684B2 (en) | 2011-02-02 | 2014-11-18 | Boehringer Ingelheim International Gmbh | Azaindolylphenyl sulfonamides as serine/threonine kinase inhibitors |
US9156837B2 (en) | 2011-07-29 | 2015-10-13 | Takeda Pharmaceutical Company Limited | Heterocyclic compound |
CN103172617A (zh) * | 2011-12-20 | 2013-06-26 | 天津市国际生物医药联合研究院 | 1,5-二取代-1,2,3-三氮唑三氟甲基类化合物的应用 |
CN103539784B (zh) * | 2012-07-09 | 2016-08-17 | 中国科学院广州生物医药与健康研究院 | 杂环苯甲酰胺类化合物、药用组合物及其应用 |
WO2015143653A1 (fr) | 2014-03-26 | 2015-10-01 | Merck Sharp & Dohme Corp. | Inhibiteurs de la kinase trka, compositions et méthodes associées |
WO2015143654A1 (fr) | 2014-03-26 | 2015-10-01 | Merck Sharp & Dohme Corp. | Inhibiteurs de la kinase trka, compositions et méthodes associées |
WO2015143652A1 (fr) | 2014-03-26 | 2015-10-01 | Merck Sharp & Dohme Corp. | Inhibiteurs de la kinase trka, compositions et méthodes associées |
WO2016161572A1 (fr) | 2015-04-08 | 2016-10-13 | Merck Sharp & Dohme Corp. | Inhibiteurs de la kinase trka, compositions et procédés associés |
CA2986083A1 (fr) | 2015-06-11 | 2016-12-15 | Basilea Pharmaceutica International AG | Inhibiteurs de la pompe a efflux et utilisations therapeutiques correspondantes |
KR101723881B1 (ko) * | 2016-03-28 | 2017-04-07 | 이화여자대학교 산학협력단 | 신규한 트리아졸 유도체, 이의 제조방법 및 이를 유효성분으로 함유하는 오로라 키나제 관련 약학적 조성물 |
WO2020007729A1 (fr) * | 2018-07-04 | 2020-01-09 | Boehringer Ingelheim International Gmbh | Dérivés de triazole benzamide en tant qu'agonistes de gpr142 |
CN116761801A (zh) * | 2021-03-12 | 2023-09-15 | 四川科伦博泰生物医药股份有限公司 | 具有蛋白激酶抑制活性的杂环化合物、包含其的药物组合物及其制备方法和用途 |
WO2023205703A2 (fr) * | 2022-04-19 | 2023-10-26 | Watershed Medical, Inc. | Formulation pour le traitement de troubles du système urinaire |
CN114805334B (zh) * | 2022-05-24 | 2023-06-09 | 深圳大学 | 一种QC和GSK-3β多靶向抑制剂及其制备方法与应用 |
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JPH03174153A (ja) | 1989-09-20 | 1991-07-29 | Fuji Photo Film Co Ltd | カラー画像形成方法 |
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JP4824576B2 (ja) | 2003-12-03 | 2011-11-30 | ベーリンガー インゲルハイム ファーマシューティカルズ インコーポレイテッド | サイトカイン生成のインヒビターとしての1,2,3−トリアゾールアミド誘導体 |
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US7858804B2 (en) | 2006-04-18 | 2010-12-28 | Boehringer Ingelheim International Gmbh | Process for making cytokine inhibiting compounds containing 4- and 5-imidazolyl rings and the intermediates thereof |
PE20120006A1 (es) | 2006-05-15 | 2012-02-02 | Boehringer Ingelheim Int | Compuestos derivados de pirimidina como inhibidores de la quinasa aurora |
EP2041138B1 (fr) | 2006-07-07 | 2014-06-25 | Bristol-Myers Squibb Company | Inhibiteurs de pyrrolotriazine kinase |
EP2041116A1 (fr) | 2006-07-07 | 2009-04-01 | Boehringer Ingelheim International GmbH | Dérivés d'hétéroaryle substitués par phényle et leur utilisation en tant qu'agents antitumoraux |
WO2008008234A1 (fr) | 2006-07-07 | 2008-01-17 | Targegen, Inc. | Inhibiteurs de type 2-amino-5-substituant-pyrimidines |
TW200813033A (en) | 2006-07-07 | 2008-03-16 | Schering Corp | 3, 4-di-substituted cyclobutene-1, 2-diones as CXC-chemokine receptor ligands |
PE20080906A1 (es) | 2006-08-17 | 2008-07-05 | Kemia Inc | Derivados heteroarilo como inhibidores de citocina |
WO2008079909A1 (fr) | 2006-12-21 | 2008-07-03 | Plexxikon, Inc. | Composés et méthodes de modulation des kinases, et indications connexes |
WO2008089034A2 (fr) | 2007-01-11 | 2008-07-24 | Kemia, Inc. | Inhibiteurs de cytokine |
CA2679659C (fr) | 2007-03-01 | 2016-01-19 | Novartis Ag | Inhibiteurs de pim kinase et procedes de leur utilisation |
CA2692379A1 (fr) | 2007-07-02 | 2009-01-08 | Boehringer Ingelheim International Gmbh | Nouveaux composes chimiques |
PE20090837A1 (es) | 2007-07-02 | 2009-07-24 | Boehringer Ingelheim Int | Nuevos compuestos quimicos |
US20100190777A1 (en) | 2007-07-17 | 2010-07-29 | Plexxikon Inc. | Compounds and methods for kinase modulation, and indications therefor |
BRPI0916356B1 (pt) | 2008-07-24 | 2022-08-23 | Nerviano Medical Sciences S.R.L | 3,4-diaril pirazois como inibidores da proteína quinase |
TW201014860A (en) | 2008-09-08 | 2010-04-16 | Boehringer Ingelheim Int | New chemical compounds |
CN102227421A (zh) | 2008-09-29 | 2011-10-26 | 贝林格尔.英格海姆国际有限公司 | 抗增殖化合物 |
WO2010094695A1 (fr) | 2009-02-17 | 2010-08-26 | Boehringer Ingelheim International Gmbh | Dérivés pyrimido-[5,4-d]-pyrimidine pour l'inhibition des tyrosine-kinases |
JP5871896B2 (ja) | 2010-03-26 | 2016-03-01 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | B−rafキナーゼインヒビター |
WO2011117382A1 (fr) | 2010-03-26 | 2011-09-29 | Boehringer Ingelheim International Gmbh | Pyridyltriazoles |
US8710055B2 (en) | 2010-12-21 | 2014-04-29 | Boehringer Ingelheim International Gmbh | Triazolylphenyl sulfonamides as serine/threonine kinase inhibitors |
US20130023531A1 (en) | 2011-01-27 | 2013-01-24 | Boehringer Ingelheim International Gmbh | Pyrimido[5,4-d]pyrimidylamino phenyl sulfonamides as serine/threonine kinase inhibitors |
US8889684B2 (en) | 2011-02-02 | 2014-11-18 | Boehringer Ingelheim International Gmbh | Azaindolylphenyl sulfonamides as serine/threonine kinase inhibitors |
-
2008
- 2008-06-30 PE PE2008001114A patent/PE20090837A1/es not_active Application Discontinuation
- 2008-06-30 CL CL2008001943A patent/CL2008001943A1/es unknown
- 2008-07-01 AU AU2008270300A patent/AU2008270300A1/en not_active Abandoned
- 2008-07-01 AR ARP080102852A patent/AR067397A1/es unknown
- 2008-07-01 BR BRPI0814601A patent/BRPI0814601A2/pt not_active IP Right Cessation
- 2008-07-01 TW TW097124780A patent/TW200911789A/zh unknown
- 2008-07-01 US US12/665,769 patent/US8889665B2/en active Active
- 2008-07-01 EP EP08774579.0A patent/EP2173734B1/fr active Active
- 2008-07-01 EA EA201000105A patent/EA201000105A1/ru unknown
- 2008-07-01 MX MX2009013935A patent/MX2009013935A/es not_active Application Discontinuation
- 2008-07-01 CA CA002692383A patent/CA2692383A1/fr not_active Abandoned
- 2008-07-01 JP JP2010513966A patent/JP5511658B2/ja active Active
- 2008-07-01 WO PCT/EP2008/058433 patent/WO2009003999A2/fr active Application Filing
- 2008-07-01 UY UY31198A patent/UY31198A1/es not_active Application Discontinuation
- 2008-07-01 KR KR1020107001120A patent/KR20100039849A/ko not_active Application Discontinuation
- 2008-07-01 CN CN200880105329A patent/CN101796045A/zh active Pending
-
2009
- 2009-12-09 IL IL202625A patent/IL202625A0/en unknown
- 2009-12-21 EC EC2009009823A patent/ECSP099823A/es unknown
- 2009-12-28 CO CO09148258A patent/CO6251316A2/es not_active Application Discontinuation
- 2009-12-30 MA MA32465A patent/MA32120B1/fr unknown
- 2009-12-31 TN TNP2009000551A patent/TN2009000551A1/fr unknown
Also Published As
Publication number | Publication date |
---|---|
US8889665B2 (en) | 2014-11-18 |
WO2009003999A3 (fr) | 2009-07-16 |
CL2008001943A1 (es) | 2009-09-11 |
US20110183952A1 (en) | 2011-07-28 |
CO6251316A2 (es) | 2011-02-21 |
MA32120B1 (fr) | 2011-03-01 |
AU2008270300A1 (en) | 2009-01-08 |
IL202625A0 (en) | 2010-06-30 |
MX2009013935A (es) | 2010-01-28 |
UY31198A1 (es) | 2009-01-30 |
EA201000105A1 (ru) | 2010-06-30 |
TW200911789A (en) | 2009-03-16 |
JP5511658B2 (ja) | 2014-06-04 |
KR20100039849A (ko) | 2010-04-16 |
CA2692383A1 (fr) | 2009-01-08 |
EP2173734A2 (fr) | 2010-04-14 |
WO2009003999A2 (fr) | 2009-01-08 |
PE20090837A1 (es) | 2009-07-24 |
EP2173734B1 (fr) | 2016-03-23 |
CN101796045A (zh) | 2010-08-04 |
ECSP099823A (es) | 2010-01-29 |
AR067397A1 (es) | 2009-10-07 |
BRPI0814601A2 (pt) | 2019-09-24 |
JP2010531851A (ja) | 2010-09-30 |
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TN2009000551A1 (fr) | Nouveaux composes chimiques | |
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MA30514B1 (fr) | Nouveaux composes. | |
TN2015000547A1 (fr) | Composes heteroaromatiques et leur utilisation comme ligands de dopamine d1 | |
MA33302B1 (fr) | 2, 4-diaminopyrimidines pour le traitement de maladies caracterisees par une proliferation cellulaire excessive ou anormale | |
MA29692B1 (fr) | Derives de la xanthine en tant qu'agonistes selectifs du hm74a | |
MA41625A (fr) | Composés de benzazépine dicarboxamide | |
MA33450B1 (fr) | Dérivés d'oxazine et leur utilisation en tant qu'inhibiteurs de bace pour le traitement de troubles neurologiques | |
TNSN07070A1 (fr) | Composes aminoheteroaryliques enantiomeriquement purs servant d'inhibiteurs de proteine-kinases | |
TN2009000324A1 (fr) | Composes tricycliques et leur utilisation comme modulateurs du recepteur de glucocorticoides | |
MA27675A1 (fr) | Derives de piperazine et leur utilisation dans le traitement de maladies neurologiques et psychiatriques | |
MA38099B1 (fr) | Des nouveaux composes triazolopyrazines substitues inhibiteurs des brd4 | |
MA32506B1 (fr) | Nouveaux composes | |
MA30232B1 (fr) | Inhibiteurs de kinase bases sur l'hydantoine | |
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MY140187A (en) | Novel tricyclic compounds useful for the treatment of inflammatory and allergic disorders: process for their preparation and pharmaceutical compositions containing them | |
MA39219B1 (fr) | Nouveaux composés inhibiteurs de la kinase lrrk2 utilisés pour le traitement du parkinson, de l’alzheimer et de la sclérose latérale amyotrophique | |
MA38284A1 (fr) | Inhibiteurs de la phospholipase associée aux lipoprotéines a2 (lp-pla2) à base de 2,3-dihydro-imidazol[1,2-c]pyrimidin-5(1 h)-one | |
MA32158B1 (fr) | Thiazolyldihydroindazoles | |
MA33239B1 (fr) | 3h-imidazo [4,5-c] pyridine-6-carboxamides en tant qu'anti-inflammatoires | |
MA33737B1 (fr) | Dérivés de glycoside et utilisations de ceux-ci | |
TN2010000230A1 (fr) | Agonistes nouveaux des recepteurs de glucocorticoides | |
MA31167B1 (fr) | Inhibiteurs de l'activite de akt | |
MA31906B1 (fr) | Inhibiteurs de la replication du virus de limmunodeficience humaine | |
MA29652B1 (fr) | 7-aza-indazoles substitues, compositions les contenant, procede de fabrication et utilisation |