SV2010003567A - Derivados bis-(sulfonilamino) en terapia 066 - Google Patents

Derivados bis-(sulfonilamino) en terapia 066

Info

Publication number
SV2010003567A
SV2010003567A SV2010003567A SV2010003567A SV2010003567A SV 2010003567 A SV2010003567 A SV 2010003567A SV 2010003567 A SV2010003567 A SV 2010003567A SV 2010003567 A SV2010003567 A SV 2010003567A SV 2010003567 A SV2010003567 A SV 2010003567A
Authority
SV
El Salvador
Prior art keywords
therapy
sulfonylamine
bis
derivatives
same
Prior art date
Application number
SV2010003567A
Other languages
English (en)
Inventor
Johan Bylund
Maria Ek
Joerg Holenz
Martin H Johansson
Gunnar Nordvall
Daniel Sohn
Jenny Viklund
Berg Stefan Von
Annika Kers
Katja Naerhi
Liselotte Oehberg
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40638954&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SV2010003567(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of SV2010003567A publication Critical patent/SV2010003567A/es

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    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/16—Central respiratory analeptics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
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    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P25/04—Centrally acting analgesics, e.g. opioids
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    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
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Abstract

COMPUESTOS DE FORMULA: (VER FORMULA); DONDE R1, R3, L1, L2, G1, G2, A Y M SON COMO LOS DEFINIDOS EN LA ESPECIFICACIÓN E ISÓMEROS ÓPTICOS, RACEMATOS Y TAUTÓMEROS DE LOS MISMOS, Y SALES FARMACÉUTICAMENTE ACEPTABLES DE LOS MISMOS; JUNTO CON PROCESOS PARA SU PREPARACIÓN, COMPOSICIONES FARMACÉUTICAS QUE LAS CONTIENEN Y SU USO EN TERAPIA. LOS COMPUESTOS SON INHIBIDORES DE LA PROSTAGLANDINA E SINTASA-1 MICROSOMAL
SV2010003567A 2007-11-15 2010-05-14 Derivados bis-(sulfonilamino) en terapia 066 SV2010003567A (es)

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