SI2167502T1 - Derivati oskadizola in njihova uporaba kot ojačevalci -842 receptorja metabotropskega glutamata - Google Patents

Derivati oskadizola in njihova uporaba kot ojačevalci -842 receptorja metabotropskega glutamata

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Publication number
SI2167502T1
SI2167502T1 SI200830807T SI200830807T SI2167502T1 SI 2167502 T1 SI2167502 T1 SI 2167502T1 SI 200830807 T SI200830807 T SI 200830807T SI 200830807 T SI200830807 T SI 200830807T SI 2167502 T1 SI2167502 T1 SI 2167502T1
Authority
SI
Slovenia
Prior art keywords
glutamate receptor
metabotropic glutamate
oxadiazole derivatives
receptor potentiators
potentiators
Prior art date
Application number
SI200830807T
Other languages
English (en)
Inventor
Joshua Clayton
Ian Egle
James Empfield
James Folmer
Methvin Isaac
Fupeng Ma
Abdelmalik Slassi
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40093925&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SI2167502(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of SI2167502T1 publication Critical patent/SI2167502T1/sl

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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • A61P21/02Muscle relaxants, e.g. for tetanus or cramps
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P25/00Drugs for disorders of the nervous system
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    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
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    • A61P25/06Antimigraine agents
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    • A61P25/08Antiepileptics; Anticonvulsants
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    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
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    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
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    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/30Drugs for disorders of the nervous system for treating abuse or dependence
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    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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    • A61P35/00Antineoplastic agents
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    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/12Antidiuretics, e.g. drugs for diabetes insipidus
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08Bridged systems
SI200830807T 2007-06-07 2008-06-05 Derivati oskadizola in njihova uporaba kot ojačevalci -842 receptorja metabotropskega glutamata SI2167502T1 (sl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US94255307P 2007-06-07 2007-06-07
EP08779348.5A EP2167502B3 (en) 2007-06-07 2008-06-05 Oxadiazole derivatives and their use as metabotropic glutamate receptor potentiators - 842
PCT/SE2008/050666 WO2008150233A1 (en) 2007-06-07 2008-06-05 Oxadiazole derivatives and their use as metabotropic glutamate receptor potentiators - 842

Publications (1)

Publication Number Publication Date
SI2167502T1 true SI2167502T1 (sl) 2012-12-31

Family

ID=40093925

Family Applications (2)

Application Number Title Priority Date Filing Date
SI200830807T SI2167502T1 (sl) 2007-06-07 2008-06-05 Derivati oskadizola in njihova uporaba kot ojačevalci -842 receptorja metabotropskega glutamata
SI200831385T SI2444399T1 (sl) 2007-06-07 2008-06-05 Derivati oksadizola in njihova uporaba kot potenciator metabotropskega receptorja glutamata -842

Family Applications After (1)

Application Number Title Priority Date Filing Date
SI200831385T SI2444399T1 (sl) 2007-06-07 2008-06-05 Derivati oksadizola in njihova uporaba kot potenciator metabotropskega receptorja glutamata -842

Country Status (34)

Country Link
US (2) US8377940B2 (sl)
EP (2) EP2167502B3 (sl)
JP (2) JP5416696B2 (sl)
KR (2) KR20150116907A (sl)
CN (2) CN101679403B (sl)
AR (1) AR066882A1 (sl)
AU (1) AU2008260717B2 (sl)
BR (1) BRPI0812889A2 (sl)
CA (1) CA2690856C (sl)
CL (1) CL2008001667A1 (sl)
CO (1) CO6251287A2 (sl)
CY (2) CY1113422T1 (sl)
DK (2) DK2444399T3 (sl)
EC (1) ECSP109856A (sl)
ES (2) ES2393425T7 (sl)
HK (2) HK1142318A1 (sl)
HR (2) HRP20120909T4 (sl)
IL (1) IL202158A (sl)
ME (1) ME01488B (sl)
MX (1) MX2009013078A (sl)
MY (1) MY158066A (sl)
NZ (1) NZ582445A (sl)
PE (1) PE20090328A1 (sl)
PL (2) PL2444399T3 (sl)
PT (2) PT2167502E (sl)
RS (2) RS52526B2 (sl)
RU (2) RU2470931C2 (sl)
SA (1) SA08290344B1 (sl)
SI (2) SI2167502T1 (sl)
TW (1) TWI417100B (sl)
UA (1) UA99129C2 (sl)
UY (1) UY31124A1 (sl)
WO (1) WO2008150233A1 (sl)
ZA (1) ZA200908285B (sl)

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