SG11201700703XA - Salt of monocyclic pyridine derivative and crystal thereof - Google Patents
Salt of monocyclic pyridine derivative and crystal thereofInfo
- Publication number
- SG11201700703XA SG11201700703XA SG11201700703XA SG11201700703XA SG11201700703XA SG 11201700703X A SG11201700703X A SG 11201700703XA SG 11201700703X A SG11201700703X A SG 11201700703XA SG 11201700703X A SG11201700703X A SG 11201700703XA SG 11201700703X A SG11201700703X A SG 11201700703XA
- Authority
- SG
- Singapore
- Prior art keywords
- salt
- crystal
- pyridine derivative
- monocyclic pyridine
- monocyclic
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/4545—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C55/00—Saturated compounds having more than one carboxyl group bound to acyclic carbon atoms
- C07C55/02—Dicarboxylic acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C55/00—Saturated compounds having more than one carboxyl group bound to acyclic carbon atoms
- C07C55/02—Dicarboxylic acids
- C07C55/10—Succinic acid
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2014166118 | 2014-08-18 | ||
| PCT/JP2015/073047 WO2016027781A1 (ja) | 2014-08-18 | 2015-08-17 | 単環ピリジン誘導体の塩およびその結晶 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SG11201700703XA true SG11201700703XA (en) | 2017-03-30 |
Family
ID=55350725
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SG11201700703XA SG11201700703XA (en) | 2014-08-18 | 2015-08-17 | Salt of monocyclic pyridine derivative and crystal thereof |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US9951047B2 (ru) |
| EP (1) | EP3184520B1 (ru) |
| JP (1) | JP5925978B1 (ru) |
| KR (1) | KR102344105B1 (ru) |
| CN (1) | CN106660997B (ru) |
| AU (1) | AU2015304465B2 (ru) |
| BR (1) | BR112017002268B1 (ru) |
| CA (1) | CA2956270C (ru) |
| ES (1) | ES2914072T3 (ru) |
| IL (1) | IL250290B (ru) |
| MX (1) | MX369646B (ru) |
| RU (1) | RU2658821C1 (ru) |
| SG (1) | SG11201700703XA (ru) |
| WO (1) | WO2016027781A1 (ru) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN115177619A (zh) * | 2015-12-17 | 2022-10-14 | 卫材R&D管理有限公司 | 用于乳腺癌的治疗剂 |
| WO2019073998A1 (en) * | 2017-10-12 | 2019-04-18 | Eisai R&D Management Co., Ltd. | PHARMACEUTICAL COMPOSITION COMPRISING A TYPICAL KINASE FGFR SELECTIVE INHIBITOR |
| SG11202007591RA (en) | 2018-03-28 | 2020-09-29 | Eisai R&D Man Co Ltd | Therapeutic agent for hepatocellular carcinoma |
| CA3180128A1 (en) | 2020-04-17 | 2021-10-21 | Eisai R&D Management Co., Ltd. | Breast cancer therapeutic agent |
| KR20230047056A (ko) | 2020-07-31 | 2023-04-06 | 에자이 알앤드디 매니지먼트 가부시키가이샤 | 유방암 치료제 |
| US20230330081A1 (en) | 2020-10-28 | 2023-10-19 | Eisai R&D Management Co., Ltd. | Pharmaceutical composition for treating tumors |
| IL310339A (en) | 2021-08-31 | 2024-03-01 | Eisai R&D Man Co Ltd | A method for the production of a monocyclic pyridine derivative |
| IL310338A (en) | 2021-08-31 | 2024-03-01 | Eisai R&D Man Co Ltd | Production method for a synthetic intermediate of a monocyclic pyridine derivative |
| CN116768856A (zh) * | 2022-03-18 | 2023-09-19 | 上海润石医药科技有限公司 | 一种取代的氨基六元氮杂环类化合物的盐及其晶型、制备方法和应用 |
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| CL2008003675A1 (es) | 2007-12-13 | 2009-03-20 | Wyeth Corp | Compuestos derivados de 5-alquil o alquenil 3-cianopiridinas, procedimiento de preparacion, composicion farmaceutica, util para reducir la actividad incrementada de una enzima en un mamifero, en donde dicha enzima es una proteina quinasa, destinado al tratamiento de la inflamacion, asma, colitis, esclerosis multiple, soriasis, artritis reumatoide. |
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| JP5739820B2 (ja) | 2008-12-30 | 2015-06-24 | アークル インコーポレイテッド | 置換５，６−ジヒドロ−６−フェニルベンゾ［ｆ］イソキノリン−２−アミン化合物 |
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| AR094812A1 (es) * | 2013-02-20 | 2015-08-26 | Eisai R&D Man Co Ltd | Derivado de piridina monocíclico como inhibidor del fgfr |
| TWI628176B (zh) | 2013-04-04 | 2018-07-01 | 奧利安公司 | 蛋白質激酶抑制劑 |
-
2015
- 2015-08-17 SG SG11201700703XA patent/SG11201700703XA/en unknown
- 2015-08-17 US US15/500,429 patent/US9951047B2/en active Active
- 2015-08-17 ES ES15834302T patent/ES2914072T3/es active Active
- 2015-08-17 CN CN201580042132.3A patent/CN106660997B/zh active Active
- 2015-08-17 AU AU2015304465A patent/AU2015304465B2/en active Active
- 2015-08-17 MX MX2017001624A patent/MX369646B/es active IP Right Grant
- 2015-08-17 WO PCT/JP2015/073047 patent/WO2016027781A1/ja active Application Filing
- 2015-08-17 CA CA2956270A patent/CA2956270C/en active Active
- 2015-08-17 BR BR112017002268-0A patent/BR112017002268B1/pt active IP Right Grant
- 2015-08-17 EP EP15834302.0A patent/EP3184520B1/en active Active
- 2015-08-17 JP JP2015560425A patent/JP5925978B1/ja active Active
- 2015-08-17 KR KR1020177002791A patent/KR102344105B1/ko active IP Right Grant
- 2015-08-17 RU RU2017103439A patent/RU2658821C1/ru active
-
2017
- 2017-01-25 IL IL250290A patent/IL250290B/en active IP Right Grant
Also Published As
| Publication number | Publication date |
|---|---|
| JPWO2016027781A1 (ja) | 2017-04-27 |
| CA2956270A1 (en) | 2016-02-25 |
| AU2015304465B2 (en) | 2019-05-09 |
| JP5925978B1 (ja) | 2016-05-25 |
| IL250290B (en) | 2020-06-30 |
| CN106660997A (zh) | 2017-05-10 |
| KR20170035927A (ko) | 2017-03-31 |
| ES2914072T3 (es) | 2022-06-07 |
| IL250290A0 (en) | 2017-03-30 |
| MX369646B (es) | 2019-11-15 |
| RU2658821C1 (ru) | 2018-06-25 |
| CA2956270C (en) | 2022-08-09 |
| US20170217935A1 (en) | 2017-08-03 |
| KR102344105B1 (ko) | 2021-12-29 |
| BR112017002268B1 (pt) | 2022-11-08 |
| EP3184520A4 (en) | 2018-04-18 |
| WO2016027781A1 (ja) | 2016-02-25 |
| US9951047B2 (en) | 2018-04-24 |
| BR112017002268A2 (pt) | 2017-11-21 |
| EP3184520B1 (en) | 2022-03-23 |
| CN106660997B (zh) | 2019-05-21 |
| MX2017001624A (es) | 2017-04-27 |
| AU2015304465A1 (en) | 2017-02-23 |
| EP3184520A1 (en) | 2017-06-28 |
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