SG11201700703XA - Salt of monocyclic pyridine derivative and crystal thereof - Google Patents

Salt of monocyclic pyridine derivative and crystal thereof

Info

Publication number
SG11201700703XA
SG11201700703XA SG11201700703XA SG11201700703XA SG11201700703XA SG 11201700703X A SG11201700703X A SG 11201700703XA SG 11201700703X A SG11201700703X A SG 11201700703XA SG 11201700703X A SG11201700703X A SG 11201700703XA SG 11201700703X A SG11201700703X A SG 11201700703XA
Authority
SG
Singapore
Prior art keywords
salt
crystal
pyridine derivative
monocyclic pyridine
monocyclic
Prior art date
Application number
SG11201700703XA
Other languages
English (en)
Inventor
Shunsuke Ozaki
Kenshi Yoshida
Original Assignee
Eisai R&D Man Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eisai R&D Man Co Ltd filed Critical Eisai R&D Man Co Ltd
Publication of SG11201700703XA publication Critical patent/SG11201700703XA/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4545Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C55/00Saturated compounds having more than one carboxyl group bound to acyclic carbon atoms
    • C07C55/02Dicarboxylic acids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C55/00Saturated compounds having more than one carboxyl group bound to acyclic carbon atoms
    • C07C55/02Dicarboxylic acids
    • C07C55/10Succinic acid
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs
SG11201700703XA 2014-08-18 2015-08-17 Salt of monocyclic pyridine derivative and crystal thereof SG11201700703XA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2014166118 2014-08-18
PCT/JP2015/073047 WO2016027781A1 (ja) 2014-08-18 2015-08-17 単環ピリジン誘導体の塩およびその結晶

Publications (1)

Publication Number Publication Date
SG11201700703XA true SG11201700703XA (en) 2017-03-30

Family

ID=55350725

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11201700703XA SG11201700703XA (en) 2014-08-18 2015-08-17 Salt of monocyclic pyridine derivative and crystal thereof

Country Status (14)

Country Link
US (1) US9951047B2 (ru)
EP (1) EP3184520B1 (ru)
JP (1) JP5925978B1 (ru)
KR (1) KR102344105B1 (ru)
CN (1) CN106660997B (ru)
AU (1) AU2015304465B2 (ru)
BR (1) BR112017002268B1 (ru)
CA (1) CA2956270C (ru)
ES (1) ES2914072T3 (ru)
IL (1) IL250290B (ru)
MX (1) MX369646B (ru)
RU (1) RU2658821C1 (ru)
SG (1) SG11201700703XA (ru)
WO (1) WO2016027781A1 (ru)

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EP3694513A4 (en) * 2017-10-12 2021-06-30 Eisai R&D Management Co., Ltd. PHARMACEUTICAL COMPOSITION WITH FGFR-SELECTIVE TYROSINKINAS INHIBITOR
EP3777860A4 (en) * 2018-03-28 2021-12-15 Eisai R&D Management Co., Ltd. THERAPEUTIC FOR HEPATOCELLULAR CARCINOMA
BR112022020786A2 (pt) 2020-04-17 2022-11-29 Eisai R&D Man Co Ltd Agente terapêutico de câncer de mama
AU2021315234A1 (en) 2020-07-31 2023-01-19 Eisai R&D Management Co., Ltd. Therapeutic agent for breast cancer
WO2022092085A1 (ja) 2020-10-28 2022-05-05 エーザイ・アール・アンド・ディー・マネジメント株式会社 腫瘍治療用医薬組成物
EP4361143A1 (en) 2021-08-31 2024-05-01 Eisai R&D Management Co., Ltd. Method for producing monocyclic pyridine derivative
CA3227445A1 (en) 2021-08-31 2023-03-09 Eisai R&D Management Co., Ltd. Production method for synthetic intermediate of monocyclic pyridine derivative
WO2023174400A1 (zh) * 2022-03-18 2023-09-21 上海润石医药科技有限公司 一种取代的氨基六元氮杂环类化合物的盐及其晶型、制备方法和应用

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Also Published As

Publication number Publication date
MX2017001624A (es) 2017-04-27
US9951047B2 (en) 2018-04-24
BR112017002268A2 (pt) 2017-11-21
RU2658821C1 (ru) 2018-06-25
BR112017002268B1 (pt) 2022-11-08
CA2956270A1 (en) 2016-02-25
IL250290B (en) 2020-06-30
MX369646B (es) 2019-11-15
EP3184520A1 (en) 2017-06-28
IL250290A0 (en) 2017-03-30
CN106660997A (zh) 2017-05-10
AU2015304465B2 (en) 2019-05-09
JPWO2016027781A1 (ja) 2017-04-27
EP3184520A4 (en) 2018-04-18
ES2914072T3 (es) 2022-06-07
JP5925978B1 (ja) 2016-05-25
CA2956270C (en) 2022-08-09
KR102344105B1 (ko) 2021-12-29
EP3184520B1 (en) 2022-03-23
WO2016027781A1 (ja) 2016-02-25
AU2015304465A1 (en) 2017-02-23
US20170217935A1 (en) 2017-08-03
CN106660997B (zh) 2019-05-21
KR20170035927A (ko) 2017-03-31

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