SE8501679L - Stereokontrollerat acetoxiazetidinon-forfarande - Google Patents

Stereokontrollerat acetoxiazetidinon-forfarande

Info

Publication number: SE8501679L
Authority: SE; Sweden
Prior art keywords: acetoxiazetidinon; stereo; procedure; controlled; dihaloanhydropenicillin
Prior art date: 1984-04-06

Application number

SE8501679A

Other languages

English (en)

Other versions

SE466201B (sv

SE8501679D0 (sv

Inventor

Alain Martel

Jean-Paul Daris

Original Assignee

Bristol Myers Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1984-04-06

Filing date

1985-04-03

Publication date

1985-10-07

1985-04-03 Application filed by Bristol Myers Co filed Critical Bristol Myers Co

1985-04-03 Publication of SE8501679D0 publication Critical patent/SE8501679D0/sv

1985-10-07 Publication of SE8501679L publication Critical patent/SE8501679L/sv

1992-01-13 Publication of SE466201B publication Critical patent/SE466201B/sv

Links

NGHVIOIJCVXTGV-ALEPSDHESA-N 6-aminopenicillanic acid Chemical compound [O-]C(=O)[C@H]1C(C)(C)S[C@@H]2[C@H]([NH3+])C(=O)N21 NGHVIOIJCVXTGV-ALEPSDHESA-N 0.000 abstract 1
NGHVIOIJCVXTGV-UHFFFAOYSA-N 6beta-amino-penicillanic acid Natural products OC(=O)C1C(C)(C)SC2C(N)C(=O)N21 NGHVIOIJCVXTGV-UHFFFAOYSA-N 0.000 abstract 1
MNFORVFSTILPAW-UHFFFAOYSA-N azetidin-2-one Chemical compound O=C1CCN1 MNFORVFSTILPAW-UHFFFAOYSA-N 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D499/88—Compounds with a double bond between positions 2 and 3 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D499/86—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with only atoms other than nitrogen atoms directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/18—Compounds having one or more C—Si linkages as well as one or more C—O—Si linkages
- C07F7/1804—Compounds having Si-O-C linkages
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)

SE8501679A 1984-04-06 1985-04-03 Foerfarande foer omvandling av 6-aminopenicillan-syra till en optiskt aktiv azetidinon SE466201B (sv)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US06/597,765 US4596677A (en)	1984-04-06	1984-04-06	Anhydropenicillin intermediates

Publications (3)

Publication Number	Publication Date
SE8501679D0 SE8501679D0 (sv)	1985-04-03
SE8501679L true SE8501679L (sv)	1985-10-07
SE466201B SE466201B (sv)	1992-01-13

Family

ID=24392838

Family Applications (3)

Application Number	Title	Priority Date	Filing Date
SE8501679A SE466201B (sv)	1984-04-06	1985-04-03	Foerfarande foer omvandling av 6-aminopenicillan-syra till en optiskt aktiv azetidinon
SE9000790A SE9000790L (sv)	1984-04-06	1990-03-06	Mellanprodukter vid stereokontrollerat acetoxi-azetidinon-foerfarande
SE9000791A SE9000791L (sv)	1984-04-06	1990-03-06	Mellanprodukter vid stereokontrollerat acetoxi-azetidinon-foerfarande

Family Applications After (2)

Application Number	Title	Priority Date	Filing Date
SE9000790A SE9000790L (sv)	1984-04-06	1990-03-06	Mellanprodukter vid stereokontrollerat acetoxi-azetidinon-foerfarande
SE9000791A SE9000791L (sv)	1984-04-06	1990-03-06	Mellanprodukter vid stereokontrollerat acetoxi-azetidinon-foerfarande

Country Status (36)

Country	Link
US (2)	US4596677A (sv)
JP (2)	JPS6117586A (sv)
KR (1)	KR920006919B1 (sv)
AR (1)	AR241139A1 (sv)
AT (1)	AT388556B (sv)
AU (1)	AU580043B2 (sv)
BE (1)	BE902133A (sv)
CA (1)	CA1261318A (sv)
CH (1)	CH665420A5 (sv)
CS (1)	CS253724B2 (sv)
CY (1)	CY1572A (sv)
DD (1)	DD232132A5 (sv)
DE (1)	DE3512250A1 (sv)
DK (1)	DK156085A (sv)
ES (1)	ES8702422A1 (sv)
FI (1)	FI86852C (sv)
FR (1)	FR2562541B1 (sv)
GB (1)	GB2156814B (sv)
GR (1)	GR850879B (sv)
HK (1)	HK106090A (sv)
HU (2)	HU193959B (sv)
IE (1)	IE58409B1 (sv)
IL (1)	IL74799A (sv)
IT (1)	IT1190351B (sv)
LU (1)	LU85841A1 (sv)
NL (1)	NL8500986A (sv)
NO (2)	NO164902C (sv)
NZ (1)	NZ211457A (sv)
OA (1)	OA07984A (sv)
PT (1)	PT80235B (sv)
SE (3)	SE466201B (sv)
SG (1)	SG91090G (sv)
SU (2)	SU1400504A3 (sv)
YU (3)	YU45918B (sv)
ZA (1)	ZA852237B (sv)
ZW (1)	ZW5585A1 (sv)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CA1256444A (en) *	1986-04-30	1989-06-27	Kazunori Kan	Process for preparing 4-acetoxy-3- hydroxyethylazetidin-2-one derivatives
US5053502A (en) *	1986-07-21	1991-10-01	Schering Corporation	Anhydro penicillin derivatives
US4767853A (en) *	1986-07-21	1988-08-30	Schering Corporation	Synthesis of 1-(allyloxycarbonyl)-methyl-3-(hydroxyethyl)-4-beta-naphthoxythiocarbonylthio-2-azetidinones and hydroxy protected analogs thereof
US5075438A (en) *	1986-07-21	1991-12-24	Schering Corporation	Synthesis of azetidinones
US4876338A (en) *	1986-07-21	1989-10-24	Schering Corporation	Synthesis of azetidinones using CuCl
US4948885A (en) *	1986-07-21	1990-08-14	Schering-Plough Corp.	Synthesis of azetidinones
US5274188A (en) *	1987-05-04	1993-12-28	Ciba-Geigy Corporation	Process for the manufacture of 4-acyloxy-3-hydroxyethyl-azetidinones
EP0290385B1 (de) *	1987-05-04	1992-10-21	Ciba-Geigy Ag	Neues Verfahren zur Herstellung von 4-Acyloxy-3-hydroxyethyl-azetidinonen
US4876365A (en) *	1988-12-05	1989-10-24	Schering Corporation	Intermediate compounds for preparing penems and carbapenems
CA2537406C (en) *	2003-09-03	2010-09-14	Otsuka Chemical Co., Ltd.	Process for producing penicillanic acid compound
US8293893B2 (en) *	2007-03-09	2012-10-23	Otsuka Chemical Co., Ltd.	Method for producing 6-hydroxyethylpenam compound

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3311638A (en) *	1961-08-16	1967-03-28	Bristol Myers Co	Anhydropenicillins
US3950352A (en) *	1972-04-10	1976-04-13	Queen's University	2,2-Dimethyl-3R-carboxy-6S-phenyl(or phenoxy)acetamido-1-oxa-4-aza-5R-bicyclo[3,2,0]heptan-7-one and processes for their production
SE449103B (sv) *	1979-03-05	1987-04-06	Pfizer	Sett att framstella penicillansyra-1,1-dioxid samt estrar derav
US4356120A (en) *	1979-07-23	1982-10-26	Merck & Co., Inc.	3-(1-Hydroxyethyl)-4-(but-2-ene)-azetidin-2-one and derivatives
US4468351A (en) *	1983-06-06	1984-08-28	Pfizer Inc.	Process for debromination of dibromopenicillanic acid and derivatives

1984
- 1984-04-06 US US06/597,765 patent/US4596677A/en not_active Expired - Fee Related
1985
- 1985-03-15 NZ NZ211457A patent/NZ211457A/xx unknown
- 1985-03-22 CA CA000477210A patent/CA1261318A/en not_active Expired
- 1985-03-22 FR FR8504289A patent/FR2562541B1/fr not_active Expired
- 1985-03-25 ZW ZW55/85A patent/ZW5585A1/xx unknown
- 1985-03-25 AR AR299861A patent/AR241139A1/es active
- 1985-03-25 ZA ZA852237A patent/ZA852237B/xx unknown
- 1985-04-01 NO NO851310A patent/NO164902C/no unknown
- 1985-04-02 ES ES541866A patent/ES8702422A1/es not_active Expired
- 1985-04-02 FI FI851324A patent/FI86852C/sv not_active IP Right Cessation
- 1985-04-02 DD DD85274771A patent/DD232132A5/de not_active IP Right Cessation
- 1985-04-03 DE DE19853512250 patent/DE3512250A1/de not_active Ceased
- 1985-04-03 IL IL74799A patent/IL74799A/xx unknown
- 1985-04-03 NL NL8500986A patent/NL8500986A/nl not_active Application Discontinuation
- 1985-04-03 DK DK156085A patent/DK156085A/da not_active IP Right Cessation
- 1985-04-03 SE SE8501679A patent/SE466201B/sv not_active IP Right Cessation
- 1985-04-04 PT PT80235A patent/PT80235B/pt not_active IP Right Cessation
- 1985-04-04 OA OA58560A patent/OA07984A/xx unknown
- 1985-04-04 GB GB08508847A patent/GB2156814B/en not_active Expired
- 1985-04-04 IE IE86785A patent/IE58409B1/en not_active IP Right Cessation
- 1985-04-04 AU AU40864/85A patent/AU580043B2/en not_active Ceased
- 1985-04-04 JP JP60071880A patent/JPS6117586A/ja active Granted
- 1985-04-04 CS CS852529A patent/CS253724B2/cs unknown
- 1985-04-04 KR KR1019850002256A patent/KR920006919B1/ko not_active IP Right Cessation
- 1985-04-04 CH CH1496/85A patent/CH665420A5/de not_active IP Right Cessation
- 1985-04-05 IT IT20246/85A patent/IT1190351B/it active
- 1985-04-05 HU HU851289A patent/HU193959B/hu not_active IP Right Cessation
- 1985-04-05 HU HU86107A patent/HU194250B/hu not_active IP Right Cessation
- 1985-04-05 AT AT0104285A patent/AT388556B/de not_active IP Right Cessation
- 1985-04-05 SU SU853873602A patent/SU1400504A3/ru active
- 1985-04-05 BE BE0/214802A patent/BE902133A/fr not_active IP Right Cessation
- 1985-04-05 LU LU85841A patent/LU85841A1/fr unknown
- 1985-04-05 YU YU57185A patent/YU45918B/sh unknown
- 1985-04-08 GR GR850879A patent/GR850879B/el unknown
- 1985-10-04 JP JP60221720A patent/JPS61171485A/ja active Granted
1986
- 1986-01-13 US US06/818,145 patent/US4639335A/en not_active Expired - Fee Related
- 1986-01-30 NO NO86860326A patent/NO166132C/no unknown
- 1986-06-13 SU SU864027635A patent/SU1435154A3/ru active
1987
- 1987-07-17 YU YU134587A patent/YU46060B/sh unknown
- 1987-07-17 YU YU134487A patent/YU46059B/sh unknown
1990
- 1990-03-06 SE SE9000790A patent/SE9000790L/sv not_active Application Discontinuation
- 1990-03-06 SE SE9000791A patent/SE9000791L/sv not_active Application Discontinuation
- 1990-11-09 SG SG910/90A patent/SG91090G/en unknown
- 1990-12-13 HK HK1060/90A patent/HK106090A/xx unknown
1991
- 1991-12-20 CY CY1572A patent/CY1572A/xx unknown

Also Published As

Publication number	Publication date
BE902133A (fr)	1985-10-07
SE9000790D0 (sv)	1990-03-06
ZW5585A1 (en)	1985-11-06
NZ211457A (en)	1989-03-29
HU194250B (en)	1988-01-28
JPH0312072B2 (sv)	1991-02-19
FR2562541B1 (fr)	1986-12-26
DK156085D0 (da)	1985-04-03
FR2562541A1 (fr)	1985-10-11
YU134487A (en)	1988-02-29
ZA852237B (en)	1985-11-27
GR850879B (sv)	1985-11-25
DD232132A5 (de)	1986-01-15
SE9000791D0 (sv)	1990-03-06
NO851310L (no)	1985-10-07
NO166132B (no)	1991-02-25
CY1572A (en)	1991-12-20
ATA104285A (de)	1988-12-15
SE9000790L (sv)	1991-09-07
ES8702422A1 (es)	1987-01-01
NL8500986A (nl)	1985-11-01
KR850007585A (ko)	1985-12-07
SE9000791L (sv)	1991-09-07
FI851324L (fi)	1985-10-07
GB2156814B (en)	1987-12-31
IT1190351B (it)	1988-02-16
JPS61171485A (ja)	1986-08-02
IE58409B1 (en)	1993-09-22
AT388556B (de)	1989-07-25
SU1435154A3 (ru)	1988-10-30
SE466201B (sv)	1992-01-13
SU1400504A3 (ru)	1988-05-30
US4639335A (en)	1987-01-27
YU46059B (sh)	1992-12-21
IL74799A0 (en)	1985-07-31
IE850867L (en)	1985-10-06
YU57185A (en)	1988-02-29
FI86852B (fi)	1992-07-15
JPS6117586A (ja)	1986-01-25
SE8501679D0 (sv)	1985-04-03
NO164902B (no)	1990-08-20
CS253724B2 (en)	1987-12-17
IT8520246A0 (it)	1985-04-05
HUT40442A (en)	1986-12-28
AR241139A2 (es)	1991-11-29
AU580043B2 (en)	1988-12-22
NO166132C (no)	1991-06-05
NO164902C (no)	1990-11-28
HK106090A (en)	1990-12-21
DE3512250A1 (de)	1985-10-17
OA07984A (fr)	1987-01-31
FI851324A0 (fi)	1985-04-02
HUT38349A (en)	1986-05-28
SG91090G (en)	1991-01-18
KR920006919B1 (ko)	1992-08-22
PT80235B (pt)	1987-10-20
FI86852C (sv)	1992-10-26
DK156085A (da)	1985-10-07
GB8508847D0 (en)	1985-05-09
LU85841A1 (fr)	1985-12-16
YU134587A (en)	1988-02-29
PT80235A (en)	1985-05-01
IL74799A (en)	1988-11-15
CA1261318A (en)	1989-09-26
HU193959B (en)	1987-12-28
NO860326L (no)	1985-10-07
AR241139A1 (es)	1991-11-29
CH665420A5 (de)	1988-05-13
YU46060B (sh)	1992-12-21
US4596677A (en)	1986-06-24
GB2156814A (en)	1985-10-16
AU4086485A (en)	1985-10-10
YU45918B (sh)	1992-09-07
JPH032157B2 (sv)	1991-01-14
ES541866A0 (es)	1987-01-01

Legal Events

Date

Code

Title

Description

1995-01-31

NUG

Patent has lapsed

Ref document number: 8501679-8

Effective date: 19941110

Format of ref document f/p: F

Publication	Publication Date	Title
ATE158798T1 (de)	1997-10-15	Verfahren zur herstellung von optisch aktiven zyklobutannukleosiden
SE7900952L (sv)	1979-08-07	Metronidazolfosfat och salter derav
PT99509A (pt)	1992-10-30	Processo para a preparacao de derivados de fenoxi-pirimidinas e de benzofuranonas
SE8501679L (sv)	1985-10-07	Stereokontrollerat acetoxiazetidinon-forfarande
ES8800138A1 (es)	1987-10-16	Un procedimiento para la preparacion de derivados de aciluretano polimerizables.
FI875596A (fi)	1988-06-24	Foerfarande foer framstaellning av tienyletylaminer och aeven ditienyletylaminer.
JPS5517386A (en)	1980-02-06	Novel oxadiazolopyrimidine derivative
FR2394514A1 (fr)	1979-01-12	Nouvel acide cyclohexanecarboxylique et ses derives
DE3379904D1 (en)	1989-06-29	Process for preparing optically active derivatives of hydroquinone and d-alpha-tocopherol
PT80791B (pt)	1987-09-18	Processo para a preparacao de novas fenil-naftiridinas uteis nomeadamente como medicamentos anti-ulcerosos
BR8207274A (pt)	1983-10-18	Processo para preparacao de um 2-exo-hidroxi-7-octabiciclo-(2,2,1)-heptano, e composto.
PT88355A (pt)	1989-06-30	Processo para a conversao da estrutura cristalina polimorfica do cloridrato de buspirona
AU568064B2 (en)	1987-12-17	4-acylamino-1-aza-adamantanes
ATE82291T1 (de)	1992-11-15	Clavamderivate, herstellung und zwischenprodukte.
ATE63119T1 (de)	1991-05-15	5- oder 6-substituierte-beta-carbolin-3carbons\|ureester.
ES2051767T3 (es)	1994-07-01	Cetorreduccion estereoespecifica de esteres de acido carboxilico-biciclooctanodiona por microorganismos.
DK464985D0 (da)	1985-10-10	Fremgangsmaade til fremstilling af optisk aktive forbindelser
FR2377387A1 (fr)	1978-08-11	Procede de preparation de 2,4,5-trichloropyrimidine
BR8202816A (pt)	1983-04-26	Processo de preparacao de imidas n-benzil
FR2453160A1 (fr)	1980-10-31	Procede de preparation de quinazolinones
FR2396739A1 (fr)	1979-02-02	1-aminomethyltricyclo(4.3.1.12,5)undecane et ses sels d'addition d'acide
PT84067B (pt)	1989-02-28	Processo de preparacao de novos derivados de pregnano
FI863897A (fi)	1988-03-27	Kemiskt foerfarande.
FR2446818A1 (fr)	1980-08-14	Tetrahydro-2h-benzo(c)pyrroles utiles comme intermediaires