SE8301408L - Mellanprodukter for framstellning av heterocyklopyrimidiner samt forfarande for framstellning derav - Google Patents

Mellanprodukter for framstellning av heterocyklopyrimidiner samt forfarande for framstellning derav

Info

Publication number
SE8301408L
SE8301408L SE8301408A SE8301408A SE8301408L SE 8301408 L SE8301408 L SE 8301408L SE 8301408 A SE8301408 A SE 8301408A SE 8301408 A SE8301408 A SE 8301408A SE 8301408 L SE8301408 L SE 8301408L
Authority
SE
Sweden
Prior art keywords
carbon atoms
intermediates
aralkyl
alkyl
aryloxyalkyl
Prior art date
Application number
SE8301408A
Other languages
English (en)
Other versions
SE8301408D0 (sv
Inventor
Jr D L Temple
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of SE8301408D0 publication Critical patent/SE8301408D0/sv
Publication of SE8301408L publication Critical patent/SE8301408L/sv

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/14Ortho-condensed systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)

Claims (1)

Patentkrav
1. Mellanprodukter med formeln III van i 88 betecknar vAte eller en grapp A, som Br 1Bgre alkyl eller 1Bgre alkenyl, vardera med upp till 8 kolatomer, pyridyametyl, aralkyl mod 7-12 kolatomer, subatituerad aralkyl med 7-12 kolatomer, aryloxialkyl med 8-12 kolatomer eller substituerad aryloxialkyl med 8-12 kolatomer, varvid var och en av nhmnda substituerade aralkyl- och substituerade aryloxialkylgrupper innehaller 1 eller 2 substituenter, som utgOrs av halogen, alkoxi eller alkyl, varvid alkoxi- och alkylgrupperna innehAller upp till 6 kolatomer; B betecknar vite, nitroso, amino eller formylamino; R6 och R7 betecknar kolbundna ringsubstituenter och utgOrs av vdte, metyl el en etyl; n Br he talet 1, 2 eller 3; och Z Br oxo eller amioh syraadditalter dBrav.
SE8301408A 1977-02-14 1983-03-15 Mellanprodukter for framstellning av heterocyklopyrimidiner samt forfarande for framstellning derav SE8301408L (sv)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US76829177A 1977-02-14 1977-02-14

Publications (2)

Publication Number Publication Date
SE8301408D0 SE8301408D0 (sv) 1983-03-15
SE8301408L true SE8301408L (sv) 1983-03-15

Family

ID=25082078

Family Applications (2)

Application Number Title Priority Date Filing Date
SE7801637A SE7801637L (sv) 1977-02-14 1978-02-13 Heterocyklopyrimidiner
SE8301408A SE8301408L (sv) 1977-02-14 1983-03-15 Mellanprodukter for framstellning av heterocyklopyrimidiner samt forfarande for framstellning derav

Family Applications Before (1)

Application Number Title Priority Date Filing Date
SE7801637A SE7801637L (sv) 1977-02-14 1978-02-13 Heterocyklopyrimidiner

Country Status (22)

Country Link
JP (1) JPS53103497A (sv)
AR (1) AR229078A1 (sv)
AT (1) AT363948B (sv)
AU (1) AU519271B2 (sv)
BE (1) BE863525A (sv)
CS (1) CS207499B2 (sv)
DD (1) DD138211A5 (sv)
DE (1) DE2806199A1 (sv)
DK (1) DK60578A (sv)
ES (1) ES466981A1 (sv)
FI (1) FI64598C (sv)
FR (1) FR2380282A1 (sv)
GB (1) GB1596320A (sv)
GR (1) GR72456B (sv)
HU (1) HU182460B (sv)
IE (1) IE46456B1 (sv)
IL (1) IL54037A (sv)
NO (1) NO780504L (sv)
PH (1) PH14777A (sv)
SE (2) SE7801637L (sv)
YU (4) YU40578A (sv)
ZA (1) ZA78870B (sv)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
YU45690B (sh) * 1984-12-22 1992-07-20 Krka Tovarna Zdraviln.Sol.O. Postopek za pripravo 9-(2-hidroksietoksimetil)-gvanina
JP2988711B2 (ja) * 1989-10-20 1999-12-13 協和醗酵工業株式会社 縮合プリン誘導体
ZA914727B (en) * 1990-06-21 1992-03-25 Schering Corp Polycyclic guanine derivatives
MY125533A (en) 1999-12-06 2006-08-30 Bristol Myers Squibb Co Heterocyclic dihydropyrimidine compounds
US7772232B2 (en) 2004-04-15 2010-08-10 Bristol-Myers Squibb Company Quinazolinyl compounds as inhibitors of potassium channel function
WO2007150025A2 (en) 2006-06-23 2007-12-27 Incyte Corporation Purinone derivatives as hm74a agonists

Also Published As

Publication number Publication date
ES466981A1 (es) 1979-08-16
JPS53103497A (en) 1978-09-08
AR229078A1 (es) 1983-06-15
PH14777A (en) 1981-12-09
FR2380282B1 (sv) 1982-03-05
IE780310L (en) 1978-08-14
AU3322178A (en) 1979-08-23
DE2806199A1 (de) 1978-08-17
YU198882A (en) 1983-04-30
ATA106778A (de) 1981-02-15
IL54037A (en) 1982-02-28
AU519271B2 (en) 1981-11-19
FI64598C (fi) 1983-12-12
IL54037A0 (en) 1978-04-30
GR72456B (sv) 1983-11-09
SE7801637L (sv) 1978-08-15
ZA78870B (en) 1979-01-31
FI64598B (fi) 1983-08-31
SE8301408D0 (sv) 1983-03-15
IE46456B1 (en) 1983-06-15
CS207499B2 (en) 1981-07-31
YU198682A (en) 1983-04-30
NO780504L (no) 1978-08-15
YU198782A (en) 1983-04-30
FR2380282A1 (fr) 1978-09-08
AT363948B (de) 1981-09-10
DK60578A (da) 1978-08-15
HU182460B (en) 1984-01-30
BE863525A (fr) 1978-07-31
FI780427A (fi) 1978-08-15
DD138211A5 (de) 1979-10-17
GB1596320A (en) 1981-08-26
YU40578A (en) 1983-04-30

Similar Documents

Publication Publication Date Title
ES469953A1 (es) Un procedimiento para la preparacion de nuevos derivados de aminoalquilbenceno
SE7601207L (sv) Acetylenderivat av acetyleniska aminosyror
ES474215A1 (es) Procedimiento para la preparacion de derivados imidazolile- tiloxialcoxilicos y sus analogos con agrupacion tio
FI800502A (fi) Difenylhydantoinderivat dessa innehaollande farmaceutiska kompositioner samt foerfarande foer framstaellning av dessa derivat
AR018014A1 (es) Compuestos derivados de 3,6-hemicetales de la clase de los 9a-azalidos, un procedimiento para prepararlos y composiciones farmaceuticas que los comprenden.
SE7906472L (sv) Nya 3-(aminoetyl)-fenol-derivat och salter derav, sett for framstellning och anvendning derav sasom lekemedel samt farmaceutiska kompositioner innehallande dessa foreningar
SE8301408L (sv) Mellanprodukter for framstellning av heterocyklopyrimidiner samt forfarande for framstellning derav
GB9215844D0 (en) Novel compounds
SE8003821L (sv) Nya 3-aminovinylcefalosporiner och forfarande for framstellning derav
SE7501365L (sv)
ES8106903A1 (es) Procedimiento de preparar compuestos de acido benzo(ij)qui- nolicin-2-carboxilico
ES484255A1 (es) Un procedimiento para la preparacion de derivados de n-ben- cilnalocetamida.
NZ182556A (en) Tricylick azacyloalkanones
ES8207538A1 (es) Un procedimiento para la preparacion de acidos 1-carbadetiapen-2-em-3-carboxilicos 6-, 1- y 2-sustituidos.
ES442057A1 (es) Procedimiento para la obtencion de penicilinas.
ES467948A1 (es) Un procedimiento para la preparacion de un derivado de fe- nilpiperazina.
JPS5297934A (en) N#-arylsulfonyl-l-argininamides and their salts acceptable as medicine s
ES438102A1 (es) Un procedimiento para la preparacion de derivados de amidino-hidrazona.
CA1268183A (en) INTERMEDIATES OF PHOSPHORANE USED IN THE PREPARATION OF ANTIBIOTIC PENEMS
SE7905865L (sv) Nya acetylenderivat av androsten-4-en, sett for framstellning och anvendning derav sasom lekemedel samt farmaceutiska kompositioner innehallande dessa foreningar
SE7908439L (sv) Nya beta-laktonderivat av 2-hydroxicyklopentankarboxylsyra, sett for framstellning och anvendning derav som lekemedel samt farmaceutiska kompositioner innehallande dessa foreningar
ES428673A1 (es) Procedimiento para la obtencion de derivados de nitrobenzo-fenona sustituidos.
ES8705379A1 (es) Procedimiento para la obtencion de derivados de benzaldoxim-carbamato
SE8603798L (sv) Karbapenem-antibiotika
ES422753A1 (es) Procedimiento de preparacion de nuevos derivados cefalospo-ranicos.

Legal Events

Date Code Title Description
NAV Patent application has lapsed

Ref document number: 8301408-4

Effective date: 19851011

Format of ref document f/p: F