FR2380282A1 - Imidazopyrimidinones et autres diazaheterocyclo-pyrimidinones, leur application comme medicaments et leur procede de fabrication - Google Patents
Imidazopyrimidinones et autres diazaheterocyclo-pyrimidinones, leur application comme medicaments et leur procede de fabricationInfo
- Publication number
- FR2380282A1 FR2380282A1 FR7804165A FR7804165A FR2380282A1 FR 2380282 A1 FR2380282 A1 FR 2380282A1 FR 7804165 A FR7804165 A FR 7804165A FR 7804165 A FR7804165 A FR 7804165A FR 2380282 A1 FR2380282 A1 FR 2380282A1
- Authority
- FR
- France
- Prior art keywords
- imidazopyrimidinones
- diazaheterocyclo
- pyrimidinones
- manufacturing
- application
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
- C07D487/14—Ortho-condensed systems
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Pulmonology (AREA)
- Immunology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
L'invention concerne des imidazopyrimidinones et autres diazahétérocyclopyrimidinones ayant un noyau condensé imidazole ou triazole convenant comme bronchodilatateur inhibiteur de phosphodiestérase et vasodilatateur périphérique. Ils sont appliqués par voie orale pour la prophylaxie et le traitement de l'asthme, un des composés préférés étant la 4-Ø(4-chlorophényl)méthylõ-6,7-dihydro-3H-imidazo Ø1,2-aõ - purin-9(4H)-one.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US76829177A | 1977-02-14 | 1977-02-14 |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2380282A1 true FR2380282A1 (fr) | 1978-09-08 |
FR2380282B1 FR2380282B1 (fr) | 1982-03-05 |
Family
ID=25082078
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR7804165A Granted FR2380282A1 (fr) | 1977-02-14 | 1978-02-14 | Imidazopyrimidinones et autres diazaheterocyclo-pyrimidinones, leur application comme medicaments et leur procede de fabrication |
Country Status (22)
Country | Link |
---|---|
JP (1) | JPS53103497A (fr) |
AR (1) | AR229078A1 (fr) |
AT (1) | AT363948B (fr) |
AU (1) | AU519271B2 (fr) |
BE (1) | BE863525A (fr) |
CS (1) | CS207499B2 (fr) |
DD (1) | DD138211A5 (fr) |
DE (1) | DE2806199A1 (fr) |
DK (1) | DK60578A (fr) |
ES (1) | ES466981A1 (fr) |
FI (1) | FI64598C (fr) |
FR (1) | FR2380282A1 (fr) |
GB (1) | GB1596320A (fr) |
GR (1) | GR72456B (fr) |
HU (1) | HU182460B (fr) |
IE (1) | IE46456B1 (fr) |
IL (1) | IL54037A (fr) |
NO (1) | NO780504L (fr) |
PH (1) | PH14777A (fr) |
SE (2) | SE7801637L (fr) |
YU (4) | YU40578A (fr) |
ZA (1) | ZA78870B (fr) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0423805A3 (en) * | 1989-10-20 | 1992-01-02 | Kyowa Hakko Kogyo Kabushiki Kaisha | Condensed purine derivatives |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
YU45690B (sh) * | 1984-12-22 | 1992-07-20 | Krka Tovarna Zdraviln.Sol.O. | Postopek za pripravo 9-(2-hidroksietoksimetil)-gvanina |
ZA914727B (en) * | 1990-06-21 | 1992-03-25 | Schering Corp | Polycyclic guanine derivatives |
MY125533A (en) | 1999-12-06 | 2006-08-30 | Bristol Myers Squibb Co | Heterocyclic dihydropyrimidine compounds |
US7772232B2 (en) | 2004-04-15 | 2010-08-10 | Bristol-Myers Squibb Company | Quinazolinyl compounds as inhibitors of potassium channel function |
WO2007150025A2 (fr) | 2006-06-23 | 2007-12-27 | Incyte Corporation | Dérivés de purinone en tant qu'agonistes du hm74a |
-
1978
- 1978-01-31 BE BE184799A patent/BE863525A/fr not_active IP Right Cessation
- 1978-02-08 GR GR55383A patent/GR72456B/el unknown
- 1978-02-09 FI FI780427A patent/FI64598C/fi not_active IP Right Cessation
- 1978-02-10 DK DK60578A patent/DK60578A/da not_active Application Discontinuation
- 1978-02-13 SE SE7801637A patent/SE7801637L/xx unknown
- 1978-02-13 GB GB5629/78A patent/GB1596320A/en not_active Expired
- 1978-02-13 HU HU78BI561A patent/HU182460B/hu unknown
- 1978-02-13 IE IE310/78A patent/IE46456B1/en unknown
- 1978-02-13 AU AU33221/78A patent/AU519271B2/en not_active Expired
- 1978-02-13 IL IL54037A patent/IL54037A/xx unknown
- 1978-02-13 AR AR271079A patent/AR229078A1/es active
- 1978-02-13 DD DD78203684A patent/DD138211A5/xx unknown
- 1978-02-14 FR FR7804165A patent/FR2380282A1/fr active Granted
- 1978-02-14 JP JP1505778A patent/JPS53103497A/ja active Pending
- 1978-02-14 AT AT0106778A patent/AT363948B/de not_active IP Right Cessation
- 1978-02-14 ES ES466981A patent/ES466981A1/es not_active Expired
- 1978-02-14 DE DE19782806199 patent/DE2806199A1/de not_active Withdrawn
- 1978-02-14 NO NO780504A patent/NO780504L/no unknown
- 1978-02-14 CS CS78959A patent/CS207499B2/cs unknown
- 1978-02-14 ZA ZA00780870A patent/ZA78870B/xx unknown
- 1978-02-15 PH PH20777A patent/PH14777A/en unknown
- 1978-02-22 YU YU00405/78A patent/YU40578A/xx unknown
-
1982
- 1982-09-02 YU YU01987/82A patent/YU198782A/xx unknown
- 1982-09-02 YU YU01988/82A patent/YU198882A/xx unknown
- 1982-09-02 YU YU01986/82A patent/YU198682A/xx unknown
-
1983
- 1983-03-15 SE SE8301408A patent/SE8301408L/sv not_active Application Discontinuation
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0423805A3 (en) * | 1989-10-20 | 1992-01-02 | Kyowa Hakko Kogyo Kabushiki Kaisha | Condensed purine derivatives |
Also Published As
Publication number | Publication date |
---|---|
ES466981A1 (es) | 1979-08-16 |
JPS53103497A (en) | 1978-09-08 |
AR229078A1 (es) | 1983-06-15 |
PH14777A (en) | 1981-12-09 |
FR2380282B1 (fr) | 1982-03-05 |
IE780310L (en) | 1978-08-14 |
AU3322178A (en) | 1979-08-23 |
DE2806199A1 (de) | 1978-08-17 |
YU198882A (en) | 1983-04-30 |
ATA106778A (de) | 1981-02-15 |
IL54037A (en) | 1982-02-28 |
AU519271B2 (en) | 1981-11-19 |
FI64598C (fi) | 1983-12-12 |
IL54037A0 (en) | 1978-04-30 |
GR72456B (fr) | 1983-11-09 |
SE7801637L (sv) | 1978-08-15 |
ZA78870B (en) | 1979-01-31 |
FI64598B (fi) | 1983-08-31 |
SE8301408D0 (sv) | 1983-03-15 |
IE46456B1 (en) | 1983-06-15 |
CS207499B2 (en) | 1981-07-31 |
YU198682A (en) | 1983-04-30 |
NO780504L (no) | 1978-08-15 |
SE8301408L (sv) | 1983-03-15 |
YU198782A (en) | 1983-04-30 |
AT363948B (de) | 1981-09-10 |
DK60578A (da) | 1978-08-15 |
HU182460B (en) | 1984-01-30 |
BE863525A (fr) | 1978-07-31 |
FI780427A (fi) | 1978-08-15 |
DD138211A5 (de) | 1979-10-17 |
GB1596320A (en) | 1981-08-26 |
YU40578A (en) | 1983-04-30 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
ST | Notification of lapse |