PT79890B - Process for preparing tetrahydro-methylimidazolylcarbazolones - Google Patents

Process for preparing tetrahydro-methylimidazolylcarbazolones

Info

Publication number
PT79890B
PT79890B PT79890A PT7989085A PT79890B PT 79890 B PT79890 B PT 79890B PT 79890 A PT79890 A PT 79890A PT 7989085 A PT7989085 A PT 7989085A PT 79890 B PT79890 B PT 79890B
Authority
PT
Portugal
Prior art keywords
methylimidazolylcarbazolones
preparing tetrahydro
tetrahydro
preparing
Prior art date
Application number
PT79890A
Other languages
Portuguese (pt)
Other versions
PT79890A (en
Inventor
Ian Harold Coates
Angus Bell S James
David Cedric Humber
Georg Blanch Ewan
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB848401888A external-priority patent/GB8401888D0/en
Priority claimed from GB848425959A external-priority patent/GB8425959D0/en
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of PT79890A publication Critical patent/PT79890A/en
Publication of PT79890B publication Critical patent/PT79890B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56Ring systems containing three or more rings
    • C07D209/80[b, c]- or [b, d]-condensed
    • C07D209/82Carbazoles; Hydrogenated carbazoles
    • C07D209/88Carbazoles; Hydrogenated carbazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the ring system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
PT79890A 1984-01-25 1985-01-25 Process for preparing tetrahydro-methylimidazolylcarbazolones PT79890B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB848401888A GB8401888D0 (en) 1984-01-25 1984-01-25 Heterocyclic compounds
GB848425959A GB8425959D0 (en) 1984-10-15 1984-10-15 Heterocyclic compounds

Publications (2)

Publication Number Publication Date
PT79890A PT79890A (en) 1985-02-01
PT79890B true PT79890B (en) 1987-02-03

Family

ID=26287221

Family Applications (1)

Application Number Title Priority Date Filing Date
PT79890A PT79890B (en) 1984-01-25 1985-01-25 Process for preparing tetrahydro-methylimidazolylcarbazolones

Country Status (29)

Country Link
KR (1) KR920003064B1 (en)
AT (1) AT392276B (en)
AU (1) AU579132B2 (en)
BE (1) BE901576A (en)
CA (1) CA1252793A (en)
CH (1) CH664152A5 (en)
CY (1) CY1479A (en)
CZ (1) CZ404391A3 (en)
DE (2) DE19375046I2 (en)
DK (1) DK169521B1 (en)
ES (3) ES8609309A1 (en)
FI (1) FI84349C (en)
FR (1) FR2561244B1 (en)
GB (1) GB2153821B (en)
GR (1) GR850219B (en)
HK (1) HK33189A (en)
HU (1) HU193592B (en)
IE (1) IE57809B1 (en)
IL (1) IL74165A (en)
IT (1) IT1182150B (en)
LU (2) LU85743A1 (en)
NL (2) NL190373C (en)
NO (2) NO164025C (en)
NZ (1) NZ210940A (en)
PH (1) PH22672A (en)
PT (1) PT79890B (en)
SE (1) SE460359B (en)
SG (1) SG7089G (en)
SK (1) SK277923B6 (en)

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GB8812636D0 (en) * 1988-05-27 1988-06-29 Glaxo Group Ltd Chemical compounds
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US5290785A (en) * 1988-09-27 1994-03-01 Fujisawa Pharmaceutical Co., Ltd. Therapeutic agent for ischemic diseases
AU627221B2 (en) * 1988-09-27 1992-08-20 Fujisawa Pharmaceutical Co., Ltd. Pyridoindole derivatives and processes for preparation thereof
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GB8917557D0 (en) * 1989-08-01 1989-09-13 Glaxo Group Ltd Medicaments
US5276050A (en) * 1989-08-01 1994-01-04 Glaxo Group Limited Medicaments
US5126343A (en) * 1989-09-11 1992-06-30 G. D. Searle & Co. N-azabicyclo [3.3.0]octane amides of aromatic acids
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ES2043535B1 (en) * 1992-03-13 1994-08-01 Vita Invest Sa PROCEDURE FOR OBTAINING 1,2,3,9-TETRAHYDRO-9-METHYL-3- (2-METHYL-1H-IMIDAZOL-1-IL) METHYL * -4H-CARBAZOL-4-ONA.
HU212934B (en) 1992-10-14 1996-12-30 Richter Gedeon Vegyeszet Process for producing novel alkoxalylated carbazolone derivatives
CA2106642C (en) * 1992-10-14 2005-08-16 Peter Bod Carbazolone derivatives and process for preparing the same
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US5969137A (en) * 1996-09-19 1999-10-19 Virginia Commonwealth University Benzylamidine derivatives with serotonin receptor binding activity
EP1181015A2 (en) 1999-03-01 2002-02-27 Sepracor Inc. Methods for treating apnea and apnea disorders using optically pure r(+)ondansetron
EP1207160A1 (en) * 2000-11-20 2002-05-22 Hanmi Pharm. Co., Ltd. Process for the preparation of 1,2,3,9-tetrahydro-9-methyl-3-((2-methyl-1H-imidazol-1-yl)-methyl)-4H-carbazol-4-one
JP2005529142A (en) 2002-04-29 2005-09-29 テバ ジョジセルジャール レースベニュタールシャシャーグ Process for producing 1,2,3,9-tetrahydro-9-methyl-3-[(2-methyl-1H-imidazol-1-yl) methyl] -4H-carbazol-4-one
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US7288660B2 (en) 2004-05-07 2007-10-30 Taro Pharmaceutical Industries Limited Process for preparing ondansetron hydrochloride dihydrate having a defined particle size
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PT2432467T (en) 2009-05-20 2018-04-04 Inst Nat Sante Rech Med Serotonin 5-ht3 receptor antagonists for use in the treatment of lesional vestibular disorders
ES2432618T3 (en) 2009-05-20 2013-12-04 Inserm (Institut National De La Santé Et De La Recherche Medicale) Serotonin 5-HT3 receptor antagonists for use in the treatment or prevention of a pathology of the inner ear with vestibular deficit
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Also Published As

Publication number Publication date
KR850005439A (en) 1985-08-26
DE3502508C2 (en) 1990-05-03
SE460359B (en) 1989-10-02
CH664152A5 (en) 1988-02-15
BE901576A (en) 1985-07-25
ES556101A0 (en) 1987-12-16
SK404391A3 (en) 1995-08-09
PT79890A (en) 1985-02-01
NL8500202A (en) 1985-08-16
NL190373B (en) 1993-09-01
HUT37784A (en) 1986-02-28
GB8501889D0 (en) 1985-02-27
DK169521B1 (en) 1994-11-21
ES548430A0 (en) 1987-10-01
NZ210940A (en) 1989-08-29
IL74165A (en) 1988-11-15
ES8801247A1 (en) 1987-12-16
NO164025B (en) 1990-05-14
ATA20485A (en) 1990-08-15
SE8500368D0 (en) 1985-01-25
HU193592B (en) 1987-11-30
CZ404391A3 (en) 1993-04-14
CY1479A (en) 1989-07-21
IT8547600A0 (en) 1985-01-25
DK35785D0 (en) 1985-01-25
KR920003064B1 (en) 1992-04-13
ES539852A0 (en) 1986-07-16
SG7089G (en) 1989-06-09
NL940009I1 (en) 1994-07-18
FR2561244B1 (en) 1988-03-04
FR2561244A1 (en) 1985-09-20
DE19375046I2 (en) 2002-10-10
SK277923B6 (en) 1995-08-09
DE3502508A1 (en) 1985-08-14
AT392276B (en) 1991-02-25
GB2153821B (en) 1988-01-20
FI84349C (en) 1991-11-25
AU579132B2 (en) 1988-11-17
PH22672A (en) 1988-11-14
ES8708224A1 (en) 1987-10-01
DK35785A (en) 1985-07-26
GB2153821A (en) 1985-08-29
HK33189A (en) 1989-04-28
FI84349B (en) 1991-08-15
NL940009I2 (en) 1999-05-03
SE8500368L (en) 1985-07-26
LU88268I2 (en) 1994-02-03
FI850323A0 (en) 1985-01-25
FI850323L (en) 1985-07-26
IE57809B1 (en) 1993-04-21
NO164025C (en) 1990-08-22
IT1182150B (en) 1987-09-30
NO850300L (en) 1985-07-26
LU85743A1 (en) 1986-08-04
NO1994022I1 (en) 1994-11-09
ES8609309A1 (en) 1986-07-16
IE850187L (en) 1985-07-25
GR850219B (en) 1985-05-23
NL190373C (en) 1994-02-01
AU3809785A (en) 1985-08-01
CA1252793A (en) 1989-04-18

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