PL2289872T3 - Medyczne zastosowania selektywnego modulatora receptora androgenowego - Google Patents

Medyczne zastosowania selektywnego modulatora receptora androgenowego

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Publication number
PL2289872T3
PL2289872T3 PL10075691T PL10075691T PL2289872T3 PL 2289872 T3 PL2289872 T3 PL 2289872T3 PL 10075691 T PL10075691 T PL 10075691T PL 10075691 T PL10075691 T PL 10075691T PL 2289872 T3 PL2289872 T3 PL 2289872T3
Authority
PL
Poland
Prior art keywords
bone
disorder
androgen receptor
receptor modulator
selective androgen
Prior art date
Application number
PL10075691T
Other languages
English (en)
Inventor
James T. Dalton
Duane D. Miller
Karen A. Veverka
Juhyun Kim
Original Assignee
University Of Tennessee Research Foundation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US10/861,923 external-priority patent/US8008348B2/en
Priority claimed from US10/863,524 external-priority patent/US20050038110A1/en
Priority claimed from US10/961,380 external-priority patent/US20060019931A1/en
Application filed by University Of Tennessee Research Foundation filed Critical University Of Tennessee Research Foundation
Publication of PL2289872T3 publication Critical patent/PL2289872T3/pl

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    • C07C255/00Carboxylic acid nitriles
    • C07C255/49Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C255/58Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the carbon skeleton
    • C07C255/60Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the carbon skeleton at least one of the singly-bound nitrogen atoms being acylated
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    • A61K31/17Amides, e.g. hydroxamic acids having the group >N—C(O)—N< or >N—C(S)—N<, e.g. urea, thiourea, carmustine
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    • C07C235/04Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton the carbon skeleton being acyclic and saturated
    • C07C235/18Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton the carbon skeleton being acyclic and saturated having at least one of the singly-bound oxygen atoms further bound to a carbon atom of a six-membered aromatic ring, e.g. phenoxyacetamides
    • C07C235/24Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton the carbon skeleton being acyclic and saturated having at least one of the singly-bound oxygen atoms further bound to a carbon atom of a six-membered aromatic ring, e.g. phenoxyacetamides having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a six-membered aromatic ring
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PL10075691T 2004-06-07 2005-06-07 Medyczne zastosowania selektywnego modulatora receptora androgenowego PL2289872T3 (pl)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US10/861,923 US8008348B2 (en) 2001-12-06 2004-06-07 Treating muscle wasting with selective androgen receptor modulators
US10/863,524 US20050038110A1 (en) 2000-08-24 2004-06-09 Selective androgen receptor modulators and methods of use thereof
US10/961,380 US20060019931A1 (en) 2003-10-14 2004-10-12 Treating bone-related disorders with selective androgen receptor modulators
EP10075691.5A EP2289872B1 (en) 2004-06-07 2005-06-07 Medical uses of a selective androgen receptor modulator
EP05758756A EP1753417B1 (en) 2004-06-07 2005-06-07 A selective androgen receptor modulator and medical uses thereof

Publications (1)

Publication Number Publication Date
PL2289872T3 true PL2289872T3 (pl) 2017-12-29

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Family Applications (2)

Application Number Title Priority Date Filing Date
PL10075691T PL2289872T3 (pl) 2004-06-07 2005-06-07 Medyczne zastosowania selektywnego modulatora receptora androgenowego
PL05758756T PL1753417T3 (pl) 2004-06-07 2005-06-07 Selektywny modulator receptora androgenowego i jego zastosowania medyczne

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Application Number Title Priority Date Filing Date
PL05758756T PL1753417T3 (pl) 2004-06-07 2005-06-07 Selektywny modulator receptora androgenowego i jego zastosowania medyczne

Country Status (14)

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EP (2) EP2289872B1 (pl)
JP (2) JP4201818B2 (pl)
AT (1) ATE552235T1 (pl)
AU (1) AU2005251781C1 (pl)
BR (1) BRPI0511308B8 (pl)
CA (1) CA2543827C (pl)
CY (1) CY1120469T1 (pl)
DK (1) DK2289872T3 (pl)
EA (2) EA018699B1 (pl)
GE (1) GEP20094851B (pl)
IL (1) IL178716A (pl)
MX (1) MXPA06013958A (pl)
PL (2) PL2289872T3 (pl)
WO (1) WO2005120483A2 (pl)

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US8853266B2 (en) * 2001-12-06 2014-10-07 University Of Tennessee Research Foundation Selective androgen receptor modulators for treating diabetes
US8309603B2 (en) 2004-06-07 2012-11-13 University Of Tennessee Research Foundation SARMs and method of use thereof
US9884038B2 (en) 2004-06-07 2018-02-06 University Of Tennessee Research Foundation Selective androgen receptor modulator and methods of use thereof
US9889110B2 (en) 2004-06-07 2018-02-13 University Of Tennessee Research Foundation Selective androgen receptor modulator for treating hormone-related conditions
MXPA06013958A (es) * 2004-06-07 2007-03-15 Univ Tennessee Res Foundation Moduladores del receptor de androgenos selectivo metodos para utilizar los mismos.
US7709516B2 (en) 2005-06-17 2010-05-04 Endorecherche, Inc. Helix 12 directed non-steroidal antiandrogens
EP2425715B1 (en) * 2005-08-31 2014-03-05 University of Tennessee Research Foundation Treating symptoms of renal disease with selective androgen receptor modulators (SARM)
EP2040694A2 (en) * 2006-07-14 2009-04-01 VIB vzw Use of ppar-alpha agonists to treat skeletal muscle wasting disorders
US9844528B2 (en) 2006-08-24 2017-12-19 University Of Tennessee Research Foundation SARMs and method of use thereof
PL2054049T3 (pl) * 2006-08-24 2016-11-30 Podstawione acyloanilidy i sposoby ich stosowania
US10010521B2 (en) 2006-08-24 2018-07-03 University Of Tennessee Research Foundation SARMs and method of use thereof
US9730908B2 (en) 2006-08-24 2017-08-15 University Of Tennessee Research Foundation SARMs and method of use thereof
US9284345B2 (en) 2007-04-12 2016-03-15 Endorecherche, Inc. 17alpha-substituted steroids as systemic antiandrogens and selective androgen receptor modulators
DK2176220T3 (da) 2007-08-07 2013-06-10 Takeda Pharmaceutical Pyrrolidin-2-on-derivater som androgenreceptormodulatorer.
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