EA200802181A1 - Избирательные модуляторы андрогеновых рецепторов и способы их применения - Google Patents

Избирательные модуляторы андрогеновых рецепторов и способы их применения

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Publication number
EA200802181A1
EA200802181A1 EA200802181A EA200802181A EA200802181A1 EA 200802181 A1 EA200802181 A1 EA 200802181A1 EA 200802181 A EA200802181 A EA 200802181A EA 200802181 A EA200802181 A EA 200802181A EA 200802181 A1 EA200802181 A1 EA 200802181A1
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EA
Eurasian Patent Office
Prior art keywords
bone
disorder
promoting
compounds
electional
Prior art date
Application number
EA200802181A
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English (en)
Other versions
EA018699B1 (ru
Inventor
Джеймс Т. Далтон
Дуэйн Д. Миллер
Карен А. Веверка
Original Assignee
Юниверсити Оф Теннесси Рисерч Фаундейшн
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Priority claimed from US10/861,923 external-priority patent/US8008348B2/en
Priority claimed from US10/863,524 external-priority patent/US20050038110A1/en
Priority claimed from US10/961,380 external-priority patent/US20060019931A1/en
Application filed by Юниверсити Оф Теннесси Рисерч Фаундейшн filed Critical Юниверсити Оф Теннесси Рисерч Фаундейшн
Publication of EA200802181A1 publication Critical patent/EA200802181A1/ru
Publication of EA018699B1 publication Critical patent/EA018699B1/ru

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    • C07C255/49Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C255/58Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the carbon skeleton
    • C07C255/60Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the carbon skeleton at least one of the singly-bound nitrogen atoms being acylated
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Abstract

Изобретение относится к соединениям SARM и к их применению для лечения различных заболеваний или состояний у индивидуума, включая наряду с прочим истощающее мышцы заболевание и/или расстройство или связанное с костями заболевание и/или расстройство.
EA200802181A 2004-06-07 2005-06-07 Применение соединения селективного модулятора андрогеновых рецепторов EA018699B1 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US10/861,923 US8008348B2 (en) 2001-12-06 2004-06-07 Treating muscle wasting with selective androgen receptor modulators
US10/863,524 US20050038110A1 (en) 2000-08-24 2004-06-09 Selective androgen receptor modulators and methods of use thereof
US10/961,380 US20060019931A1 (en) 2003-10-14 2004-10-12 Treating bone-related disorders with selective androgen receptor modulators

Publications (2)

Publication Number Publication Date
EA200802181A1 true EA200802181A1 (ru) 2009-02-27
EA018699B1 EA018699B1 (ru) 2013-10-30

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Application Number Title Priority Date Filing Date
EA200602278A EA011306B8 (ru) 2004-06-07 2005-06-07 Избирательные модуляторы андрогеновых рецепторов и способы их применения
EA200802181A EA018699B1 (ru) 2004-06-07 2005-06-07 Применение соединения селективного модулятора андрогеновых рецепторов

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EA200602278A EA011306B8 (ru) 2004-06-07 2005-06-07 Избирательные модуляторы андрогеновых рецепторов и способы их применения

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EP (2) EP1753417B1 (ru)
JP (2) JP4201818B2 (ru)
AT (1) ATE552235T1 (ru)
AU (1) AU2005251781C1 (ru)
BR (1) BRPI0511308B8 (ru)
CA (1) CA2543827C (ru)
CY (1) CY1120469T1 (ru)
DK (1) DK2289872T3 (ru)
EA (2) EA011306B8 (ru)
GE (1) GEP20094851B (ru)
IL (1) IL178716A (ru)
MX (1) MXPA06013958A (ru)
PL (2) PL2289872T3 (ru)
WO (1) WO2005120483A2 (ru)

Families Citing this family (34)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8853266B2 (en) * 2001-12-06 2014-10-07 University Of Tennessee Research Foundation Selective androgen receptor modulators for treating diabetes
US8309603B2 (en) 2004-06-07 2012-11-13 University Of Tennessee Research Foundation SARMs and method of use thereof
EA011306B8 (ru) * 2004-06-07 2012-10-30 Юниверсити Оф Теннесси Рисерч Фаундейшн Избирательные модуляторы андрогеновых рецепторов и способы их применения
US9889110B2 (en) 2004-06-07 2018-02-13 University Of Tennessee Research Foundation Selective androgen receptor modulator for treating hormone-related conditions
US9884038B2 (en) 2004-06-07 2018-02-06 University Of Tennessee Research Foundation Selective androgen receptor modulator and methods of use thereof
US7709516B2 (en) 2005-06-17 2010-05-04 Endorecherche, Inc. Helix 12 directed non-steroidal antiandrogens
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