PA8531401A1 - Inhibidores de espiropirimidin-2,4,6-triona metaloproteinasas - Google Patents

Inhibidores de espiropirimidin-2,4,6-triona metaloproteinasas

Info

Publication number: PA8531401A1
Authority: PA; Panama
Prior art keywords: spiropirimidin; triona; inhibitors; metaloproteinase inhibitors; metaloproteinase
Prior art date: 2000-10-26

Application number

PA20018531401A

Other languages

English (en)

Spanish (es)

Inventor

Mark Carl Noe

Brian Scott Bronk

Martin James Wythes

Original Assignee

Pfizer Prod Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-10-26

Filing date

2001-10-26

Publication date

2003-06-30

2001-10-26 Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc

2003-06-30 Publication of PA8531401A1 publication Critical patent/PA8531401A1/es

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/10—Spiro-condensed systems
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- C07D487/10—Spiro-condensed systems

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Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Physical Education & Sports Medicine (AREA)
Immunology (AREA)
Reproductive Health (AREA)
Endocrinology (AREA)
Oncology (AREA)
Rheumatology (AREA)
Dermatology (AREA)
Communicable Diseases (AREA)
Pain & Pain Management (AREA)
Orthopedic Medicine & Surgery (AREA)
Pulmonology (AREA)
Gynecology & Obstetrics (AREA)
Diabetes (AREA)
Virology (AREA)
Hematology (AREA)
Tropical Medicine & Parasitology (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Pregnancy & Childbirth (AREA)
Ophthalmology & Optometry (AREA)
Psychology (AREA)
Psychiatry (AREA)

PA20018531401A 2000-10-26 2001-10-26 Inhibidores de espiropirimidin-2,4,6-triona metaloproteinasas PA8531401A1 (es)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US24338900P	2000-10-26	2000-10-26

Publications (1)

Publication Number	Publication Date
PA8531401A1 true PA8531401A1 (es)	2003-06-30

Family

ID=22918584

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PA20018531401A PA8531401A1 (es)	2000-10-26	2001-10-26	Inhibidores de espiropirimidin-2,4,6-triona metaloproteinasas

Country Status (32)

Country	Link
EP (1)	EP1332146A2 (xx)
JP (1)	JP2004518635A (xx)
KR (1)	KR20040004412A (xx)
CN (1)	CN1501937A (xx)
AP (1)	AP2001002318A0 (xx)
AR (1)	AR035069A1 (xx)
AU (1)	AU2002210813A1 (xx)
BG (1)	BG107653A (xx)
BR (1)	BR0114913A (xx)
CA (1)	CA2425283A1 (xx)
CZ (1)	CZ20031083A3 (xx)
EA (1)	EA005762B1 (xx)
EC (1)	ECSP034567A (xx)
EE (1)	EE200300196A (xx)
GT (1)	GT200100213A (xx)
HN (1)	HN2001000244A (xx)
HR (1)	HRP20030332A2 (xx)
HU (1)	HUP0301577A3 (xx)
IL (1)	IL154948A0 (xx)
IS (1)	IS6762A (xx)
MA (1)	MA26957A1 (xx)
MX (1)	MXPA03003735A (xx)
NO (1)	NO20031853L (xx)
OA (1)	OA12529A (xx)
PA (1)	PA8531401A1 (xx)
PE (1)	PE20020589A1 (xx)
PL (1)	PL366201A1 (xx)
SK (1)	SK4972003A3 (xx)
SV (1)	SV2003000705A (xx)
TN (1)	TNSN01149A1 (xx)
WO (1)	WO2002034753A2 (xx)
ZA (1)	ZA200302190B (xx)

Families Citing this family (36)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
PA8539501A1 (es)	2001-02-14	2002-09-30	Warner Lambert Co	Compuestos triazolo como inhibidores de mmp
DOP2002000333A (es)	2001-02-14	2002-09-30	Warner Lambert Co	Derivados de acido isoftalico como inhibidores de metaloproteinasas de la matriz
WO2002064578A1 (en)	2001-02-14	2002-08-22	Warner-Lambert Company Llc	Benzo thiadiazine matrix metalloproteinase inhibitors
DOP2002000332A (es)	2001-02-14	2002-08-30	Warner Lambert Co	Inhibidores de piridina de metaloproteinasas de la matriz
MXPA03004920A (es)	2001-02-14	2003-09-05	Warner Lambert Co	Pirimidinas inhibidoras de metaloproteinasas de matriz.
US6924276B2 (en)	2001-09-10	2005-08-02	Warner-Lambert Company	Diacid-substituted heteroaryl derivatives as matrix metalloproteinase inhibitors
MXPA04002537A (es)	2001-10-12	2004-05-31	Warner Lambert Co	Alquinos como inhibidores de metaloproteinasa de matriz.
US6962922B2 (en)	2001-10-12	2005-11-08	Warner-Lambert Company Llc	Alkynylated quinazoline compounds
US6894057B2 (en)	2002-03-08	2005-05-17	Warner-Lambert Company	Oxo-azabicyclic compounds
WO2003091252A1 (en) *	2002-04-25	2003-11-06	Bristol-Myers Squibb Company	Spirobarbituric acid derivatives useful as inhibitors of matrix metalloproteases
BR0308787A (pt) *	2002-04-26	2005-01-11	Pfizer Prod Inc	Inibidores de metaloproteinase de n-substituìdos-heteroarilóxi-aril-espiro-pirimidina- 2,4,6-triona
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2001
- 2001-10-23 AU AU2002210813A patent/AU2002210813A1/en not_active Abandoned
- 2001-10-23 IL IL15494801A patent/IL154948A0/xx unknown
- 2001-10-23 CA CA002425283A patent/CA2425283A1/en not_active Abandoned
- 2001-10-23 HU HU0301577A patent/HUP0301577A3/hu unknown
- 2001-10-23 WO PCT/IB2001/001986 patent/WO2002034753A2/en not_active Application Discontinuation
- 2001-10-23 AP APAP/P/2001/002318A patent/AP2001002318A0/en unknown
- 2001-10-23 KR KR10-2003-7005753A patent/KR20040004412A/ko not_active Application Discontinuation
- 2001-10-23 JP JP2002537743A patent/JP2004518635A/ja not_active Withdrawn
- 2001-10-23 CN CNA018179231A patent/CN1501937A/zh active Pending
- 2001-10-23 EA EA200300306A patent/EA005762B1/ru not_active IP Right Cessation
- 2001-10-23 OA OA1200300123A patent/OA12529A/en unknown
- 2001-10-23 PL PL01366201A patent/PL366201A1/xx not_active Application Discontinuation
- 2001-10-23 SK SK497-2003A patent/SK4972003A3/sk unknown
- 2001-10-23 MX MXPA03003735A patent/MXPA03003735A/es unknown
- 2001-10-23 EP EP01978721A patent/EP1332146A2/en not_active Withdrawn
- 2001-10-23 CZ CZ20031083A patent/CZ20031083A3/cs unknown
- 2001-10-23 EE EEP200300196A patent/EE200300196A/xx unknown
- 2001-10-23 BR BR0114913-0A patent/BR0114913A/pt not_active IP Right Cessation
- 2001-10-24 HN HN2001000244A patent/HN2001000244A/es unknown
- 2001-10-24 AR ARP010104977A patent/AR035069A1/es unknown
- 2001-10-25 PE PE2001001060A patent/PE20020589A1/es not_active Application Discontinuation
- 2001-10-25 GT GT200100213A patent/GT200100213A/es unknown
- 2001-10-25 SV SV2001000705A patent/SV2003000705A/es unknown
- 2001-10-25 TN TNTNSN01149A patent/TNSN01149A1/fr unknown
- 2001-10-26 PA PA20018531401A patent/PA8531401A1/es unknown
2003
- 2003-03-19 ZA ZA200302190A patent/ZA200302190B/en unknown
- 2003-03-20 BG BG107653A patent/BG107653A/bg unknown
- 2003-03-27 IS IS6762A patent/IS6762A/is unknown
- 2003-04-22 MA MA27117A patent/MA26957A1/fr unknown
- 2003-04-24 NO NO20031853A patent/NO20031853L/no not_active Application Discontinuation
- 2003-04-25 EC EC2003004567A patent/ECSP034567A/es unknown
- 2003-04-28 HR HR20030332A patent/HRP20030332A2/hr not_active Application Discontinuation

Also Published As

Publication number	Publication date
AR035069A1 (es)	2004-04-14
WO2002034753A2 (en)	2002-05-02
EA005762B1 (ru)	2005-06-30
CA2425283A1 (en)	2002-05-02
SV2003000705A (es)	2003-01-13
BG107653A (bg)	2003-12-31
HUP0301577A2 (hu)	2003-11-28
OA12529A (en)	2006-06-02
WO2002034753A3 (en)	2002-08-15
PE20020589A1 (es)	2002-07-06
HUP0301577A3 (en)	2006-02-28
IS6762A (is)	2003-03-27
KR20040004412A (ko)	2004-01-13
CN1501937A (zh)	2004-06-02
AU2002210813A1 (en)	2002-05-06
TNSN01149A1 (fr)	2005-11-10
GT200100213A (es)	2002-07-03
HRP20030332A2 (en)	2003-06-30
MXPA03003735A (es)	2003-07-28
CZ20031083A3 (cs)	2004-03-17
EA200300306A1 (ru)	2003-08-28
NO20031853L (no)	2003-06-23
PL366201A1 (en)	2005-01-24
EP1332146A2 (en)	2003-08-06
ECSP034567A (es)	2003-06-25
NO20031853D0 (no)	2003-04-24
MA26957A1 (fr)	2004-12-20
HN2001000244A (es)	2003-11-07
JP2004518635A (ja)	2004-06-24
AP2001002318A0 (en)	2001-12-31
IL154948A0 (en)	2003-10-31
ZA200302190B (en)	2004-04-28
EE200300196A (et)	2003-10-15
SK4972003A3 (en)	2004-05-04
BR0114913A (pt)	2003-07-01

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