NO327182B1 - Glukopyranosyloksybenzylbenzen-derivater og medisinske sammensetninger inneholdende det samme - Google Patents
Glukopyranosyloksybenzylbenzen-derivater og medisinske sammensetninger inneholdende det samme Download PDFInfo
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- NO327182B1 NO327182B1 NO20031407A NO20031407A NO327182B1 NO 327182 B1 NO327182 B1 NO 327182B1 NO 20031407 A NO20031407 A NO 20031407A NO 20031407 A NO20031407 A NO 20031407A NO 327182 B1 NO327182 B1 NO 327182B1
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/20—Carbocyclic rings
- C07H15/203—Monocyclic carbocyclic rings other than cyclohexane rings; Bicyclic carbocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7028—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages
- A61K31/7034—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2000301523 | 2000-09-29 | ||
| PCT/JP2001/008239 WO2002028872A1 (fr) | 2000-09-29 | 2001-09-21 | Derives de glucopyranosiloxybenzylbenzene et compositions therapeutiques contenant ces composes |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO20031407D0 NO20031407D0 (no) | 2003-03-27 |
| NO20031407L NO20031407L (no) | 2003-04-30 |
| NO327182B1 true NO327182B1 (no) | 2009-05-04 |
Family
ID=18783054
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20031407A NO327182B1 (no) | 2000-09-29 | 2003-03-27 | Glukopyranosyloksybenzylbenzen-derivater og medisinske sammensetninger inneholdende det samme |
Country Status (33)
| Country | Link |
|---|---|
| US (2) | US6872706B2 (cs) |
| EP (1) | EP1329456B1 (cs) |
| JP (1) | JP3798375B2 (cs) |
| KR (1) | KR100647204B1 (cs) |
| CN (1) | CN1293087C (cs) |
| AR (1) | AR030816A1 (cs) |
| AT (1) | ATE335753T1 (cs) |
| AU (2) | AU9025701A (cs) |
| BG (1) | BG66015B1 (cs) |
| BR (1) | BR0114310A (cs) |
| CA (1) | CA2423568C (cs) |
| CY (1) | CY1106076T1 (cs) |
| CZ (1) | CZ303544B6 (cs) |
| DE (1) | DE60122193T2 (cs) |
| DK (1) | DK1329456T3 (cs) |
| EA (1) | EA005994B1 (cs) |
| ES (1) | ES2269456T3 (cs) |
| HK (1) | HK1061037A1 (cs) |
| HU (1) | HUP0301178A3 (cs) |
| IL (2) | IL155071A0 (cs) |
| MX (1) | MXPA03002779A (cs) |
| MY (1) | MY129023A (cs) |
| NO (1) | NO327182B1 (cs) |
| NZ (1) | NZ524917A (cs) |
| PE (1) | PE20020476A1 (cs) |
| PL (1) | PL205607B1 (cs) |
| PT (1) | PT1329456E (cs) |
| SI (1) | SI1329456T1 (cs) |
| SK (1) | SK287811B6 (cs) |
| TW (1) | TWI284641B (cs) |
| UA (1) | UA73606C2 (cs) |
| WO (1) | WO2002028872A1 (cs) |
| ZA (1) | ZA200302283B (cs) |
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|---|---|---|---|---|
| CN1020944C (zh) | 1990-01-30 | 1993-05-26 | 阿图尔-费希尔股份公司费希尔厂 | 紧固件 |
| SI1329456T1 (sl) | 2000-09-29 | 2006-12-31 | Kissei Pharmaceutical | Glukopiranoziloksibenzilbenzenski derivati in zdravilni sestavki, ki vsebujejo te spojine |
| AU2002223127A1 (en) * | 2000-11-30 | 2002-06-11 | Kissei Pharmaceutical Co., Ltd. Intellectual Property | Glucopyranosyloxybenzyl benzene derivatives, medicinal compositions containing the same and intermediates in the production thereof |
| TWI255817B (en) | 2001-02-14 | 2006-06-01 | Kissei Pharmaceutical | Glucopyranosyloxybenzylbenzene derivatives and medicinal use thereof |
| EP1489089A4 (en) * | 2002-03-22 | 2009-10-28 | Kissei Pharmaceutical | CRYSTALS OF GLUCOPYRANOSYLOXYBENZYLBENZEN DERIVATE |
| BR0310006A (pt) * | 2002-08-09 | 2005-02-15 | Taisho Pharmaceutical Co Ltd | Derivados de 5-tio-beta-d-glicopiranosìdeo de arila e agentes terapêuticos para diabetes contendo os mesmos |
| CN1744916A (zh) * | 2002-12-04 | 2006-03-08 | 橘生药品工业株式会社 | 预防和治疗高血糖所导致的疾病 |
| JP4651934B2 (ja) * | 2002-12-04 | 2011-03-16 | キッセイ薬品工業株式会社 | ベンジルフェノール誘導体、それを含有する医薬組成物およびその医薬用途 |
| DE10258008B4 (de) * | 2002-12-12 | 2006-02-02 | Sanofi-Aventis Deutschland Gmbh | Heterocyclische Fluorglycosidderivate, diese Verbindungen enthaltende Arzneimittel und Verfahren zur Herstellung dieser Arzneimittel |
| DE10258007B4 (de) | 2002-12-12 | 2006-02-09 | Sanofi-Aventis Deutschland Gmbh | Aromatische Fluorglycosidderivate, diese Verbindungen enthaltende Arzneimittel und Verfahren zur Herstellung dieser Arzneimittel |
| UA86042C2 (en) * | 2003-08-01 | 2009-03-25 | Янссен Фармацевтика Н.В. | Substituted indazole-o-glucosides |
| EA011158B1 (ru) * | 2004-03-16 | 2009-02-27 | Бёрингер Ингельхайм Интернациональ Гмбх | Замещённые глюкопиранозилом бензольные производные, содержащие эти соединения лекарственные средства, их применение и способ их получения |
| EP1731524A4 (en) * | 2004-03-31 | 2009-05-20 | Kissei Pharmaceutical | PHENOLE DERIVATIVE, MEDICINAL COMPOSITION CONTAINING THE DERIVATIVE, AND ITS MEDICINAL USE |
| JP5010918B2 (ja) * | 2004-07-21 | 2012-08-29 | キッセイ薬品工業株式会社 | 肝臓脂肪の異常蓄積に起因する疾患の進展抑制剤 |
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| CA2903770C (en) | 2013-03-14 | 2022-07-12 | Mars, Incorporated | Flavor composition containing 3-hydroxy-3-methylglutaric acid (hmg) glucosides |
| US11813275B2 (en) | 2013-04-05 | 2023-11-14 | Boehringer Ingelheim International Gmbh | Pharmaceutical composition, methods for treating and uses thereof |
| US20140303097A1 (en) | 2013-04-05 | 2014-10-09 | Boehringer Ingelheim International Gmbh | Pharmaceutical composition, methods for treating and uses thereof |
| PT2981271T (pt) | 2013-04-05 | 2019-02-19 | Boehringer Ingelheim Int | Utilizações terapêuticas de empagliflozina |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2549476B1 (fr) | 1983-07-20 | 1986-04-25 | Rech Ind | Benzyl-phenyl-osides, procede de preparation et utilisation en therapeutique |
| CA2102591C (en) | 1992-11-12 | 2000-12-26 | Kenji Tsujihara | Hypoglycemic agent |
| US5731292A (en) | 1992-11-12 | 1998-03-24 | Tanabe Seiyaku Co., Ltd. | Dihydrochalcone derivatives which are hypoglycemic agents |
| BR0109323A (pt) | 2000-03-17 | 2002-12-24 | Kissei Pharmaceutical | Derivados de gluco piranosiloxi benzil benzeno, composições medicinais contendo os mesmos e intermediários para a preparação dos derivados |
| US6683056B2 (en) * | 2000-03-30 | 2004-01-27 | Bristol-Myers Squibb Company | O-aryl glucoside SGLT2 inhibitors and method |
| SI1329456T1 (sl) | 2000-09-29 | 2006-12-31 | Kissei Pharmaceutical | Glukopiranoziloksibenzilbenzenski derivati in zdravilni sestavki, ki vsebujejo te spojine |
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2001
- 2001-09-21 SI SI200130638T patent/SI1329456T1/sl unknown
- 2001-09-21 JP JP2002532454A patent/JP3798375B2/ja not_active Expired - Fee Related
- 2001-09-21 US US10/381,846 patent/US6872706B2/en not_active Expired - Lifetime
- 2001-09-21 DK DK01970186T patent/DK1329456T3/da active
- 2001-09-21 MX MXPA03002779A patent/MXPA03002779A/es active IP Right Grant
- 2001-09-21 NZ NZ524917A patent/NZ524917A/en not_active IP Right Cessation
- 2001-09-21 ES ES01970186T patent/ES2269456T3/es not_active Expired - Lifetime
- 2001-09-21 WO PCT/JP2001/008239 patent/WO2002028872A1/ja active IP Right Grant
- 2001-09-21 EA EA200300316A patent/EA005994B1/ru not_active IP Right Cessation
- 2001-09-21 AT AT01970186T patent/ATE335753T1/de active
- 2001-09-21 EP EP01970186A patent/EP1329456B1/en not_active Expired - Lifetime
- 2001-09-21 HU HU0301178A patent/HUP0301178A3/hu unknown
- 2001-09-21 SK SK334-2003A patent/SK287811B6/sk not_active IP Right Cessation
- 2001-09-21 PL PL362177A patent/PL205607B1/pl not_active IP Right Cessation
- 2001-09-21 AU AU9025701A patent/AU9025701A/xx active Pending
- 2001-09-21 DE DE60122193T patent/DE60122193T2/de not_active Expired - Lifetime
- 2001-09-21 CA CA2423568A patent/CA2423568C/en not_active Expired - Fee Related
- 2001-09-21 KR KR1020037004588A patent/KR100647204B1/ko not_active IP Right Cessation
- 2001-09-21 AU AU2001290257A patent/AU2001290257B2/en not_active Ceased
- 2001-09-21 IL IL15507101A patent/IL155071A0/xx unknown
- 2001-09-21 PT PT01970186T patent/PT1329456E/pt unknown
- 2001-09-21 CN CNB018165605A patent/CN1293087C/zh not_active Expired - Fee Related
- 2001-09-21 CZ CZ20030777A patent/CZ303544B6/cs not_active IP Right Cessation
- 2001-09-21 UA UA2003032735A patent/UA73606C2/uk unknown
- 2001-09-21 BR BR0114310-7A patent/BR0114310A/pt not_active Application Discontinuation
- 2001-09-26 MY MYPI20014500A patent/MY129023A/en unknown
- 2001-09-28 AR ARP010104589A patent/AR030816A1/es unknown
- 2001-09-28 TW TW090124049A patent/TWI284641B/zh not_active IP Right Cessation
- 2001-09-28 PE PE2001000975A patent/PE20020476A1/es not_active Application Discontinuation
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- 2003-03-25 IL IL155071A patent/IL155071A/en not_active IP Right Cessation
- 2003-03-26 BG BG107674A patent/BG66015B1/bg unknown
- 2003-03-27 NO NO20031407A patent/NO327182B1/no not_active IP Right Cessation
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2004
- 2004-06-09 HK HK04104109A patent/HK1061037A1/xx not_active IP Right Cessation
- 2004-08-12 US US10/916,548 patent/US20050065098A1/en not_active Abandoned
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