NO326497B1 - Arylsulfonylderivater med 5-HT6 reseptor affinitet, farmasoytisk medikament omfattende slike, fremgangsmate for fremstilling av slike samt anvendelse av slike for fremstilling av medikament for behandling av sykdom - Google Patents

Arylsulfonylderivater med 5-HT6 reseptor affinitet, farmasoytisk medikament omfattende slike, fremgangsmate for fremstilling av slike samt anvendelse av slike for fremstilling av medikament for behandling av sykdom Download PDF

Info

Publication number: NO326497B1
Authority: NO; Norway
Prior art keywords: methoxy; phenyl; compound; piperazine; benzenesulfonyl
Prior art date: 2001-08-10

Application number

NO20040589A

Other languages

English (en)

Norwegian (no)

Other versions

NO20040589L (no

Inventor

Jacob Berger

Shu-Hai Zhao

Robin Douglas Clark

Original Assignee

Hoffmann La Roche

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-08-10

Filing date

2004-02-09

Publication date

2008-12-15

2004-02-09 Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche

2004-03-19 Publication of NO20040589L publication Critical patent/NO20040589L/no

2008-12-15 Publication of NO326497B1 publication Critical patent/NO326497B1/no

Links

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NO20040589A 2001-08-10 2004-02-09 Arylsulfonylderivater med 5-HT6 reseptor affinitet, farmasoytisk medikament omfattende slike, fremgangsmate for fremstilling av slike samt anvendelse av slike for fremstilling av medikament for behandling av sykdom NO326497B1 (no)

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US31150401P	2001-08-10	2001-08-10
US38471102P	2002-05-31	2002-05-31
PCT/EP2002/008696 WO2003014097A1 (en)	2001-08-10	2002-08-05	Arylsulfonyl derivatives with 5-ht6 receptor affinity

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US (1)	US6825202B2 (ja)
EP (1)	EP1423106B1 (ja)
JP (1)	JP4187650B2 (ja)
KR (1)	KR100608417B1 (ja)
CN (1)	CN1254469C (ja)
AT (1)	ATE417838T1 (ja)
AU (1)	AU2002340804B2 (ja)
CA (1)	CA2456250A1 (ja)
CO (1)	CO5550439A2 (ja)
DE (1)	DE60230424D1 (ja)
ES (1)	ES2316619T3 (ja)
HK (1)	HK1070054A1 (ja)
HR (1)	HRP20040090A2 (ja)
HU (1)	HUP0401235A2 (ja)
IL (1)	IL159880A0 (ja)
MX (1)	MXPA04001250A (ja)
NO (1)	NO326497B1 (ja)
NZ (1)	NZ530742A (ja)
PL (1)	PL373397A1 (ja)
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US7452888B2 (en)	2002-03-27	2008-11-18	Glaxo Group Limited	Quinoline derivatives and their use as 5-ht6 ligands
ATE384054T1 (de) *	2002-11-08	2008-02-15	Hoffmann La Roche	Substituierte benzoxazinones und ihre verwendung
GB0305575D0 (en) *	2003-03-11	2003-04-16	Glaxo Group Ltd	Novel compounds
TWI289141B (en) *	2003-03-11	2007-11-01	Hoffmann La Roche F. Ag.	Quinolinone derivatives and uses thereof
TW200523253A (en)	2003-07-22	2005-07-16	Arena Pharm Inc	Diaryl and arylheteroaryl urea derivatives as modulators of the 5-ht2a serotonin receptor useful for the prophylaxis and treatment of disorders related thereto
WO2006062481A1 (en) *	2004-12-09	2006-06-15	Biovitrum Ab	New benzofuran derivatives and their use in the treatment of obesity, type ii diabetes and cns disorders .
PL1831159T3 (pl) *	2004-12-21	2010-06-30	Hoffmann La Roche	Pochodne tetraliny i indanu oraz ich zastosowania
EP1695971A1 (en) *	2004-12-30	2006-08-30	Laboratorios Del Dr. Esteve, S.A.	Substituted phenyl-piperazine compounds, their preparation and use in medicaments
WO2009074607A1 (en)	2007-12-12	2009-06-18	Glaxo Group Limited	Combinations comprising 3-phenylsulfonyl-8-piperazinyl-1yl-quinoline
US20110021538A1 (en)	2008-04-02	2011-01-27	Arena Pharmaceuticals, Inc.	Processes for the preparation of pyrazole derivatives useful as modulators of the 5-ht2a serotonin receptor
US9126946B2 (en)	2008-10-28	2015-09-08	Arena Pharmaceuticals, Inc.	Processes useful for the preparation of 1-[3-(4-bromo-2-methyl-2H-pyrazol-3-yl)-4-methoxy-phenyl]-3-(2,4-difluoro-phenyl)urea and crystalline forms related thereto
US8183237B2 (en)	2009-04-30	2012-05-22	Abbott Laboratories	Benzenesulfonanilide compounds suitable for treating disorders that respond to modulation of the serotonin 5-HT6 receptor
ES2536779T3 (es) *	2009-04-30	2015-05-28	Abbvie Deutschland Gmbh & Co Kg	Compuestos de N-fenil-(piperazinil u homopiperazinil)-bencensulfonamida o bencensulfonil-fenil-(piperazina u homopiperazina) adecuados para tratar trastornos que responden a la modulación del receptor de serotonina 5-HT6
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AU2002340804B2 (en)	2008-04-03
MXPA04001250A (es)	2004-05-27
WO2003014097A1 (en)	2003-02-20
JP2005502649A (ja)	2005-01-27
NZ530742A (en)	2007-07-27
KR20040023738A (ko)	2004-03-18
CN1541210A (zh)	2004-10-27
IL159880A0 (en)	2004-06-20
HRP20040090A2 (en)	2004-12-31
RU2004107261A (ru)	2005-09-10
ES2316619T3 (es)	2009-04-16
HK1070054A1 (en)	2005-06-10
CN1254469C (zh)	2006-05-03
EP1423106A1 (en)	2004-06-02
US6825202B2 (en)	2004-11-30
CO5550439A2 (es)	2005-08-31
US20030069254A1 (en)	2003-04-10
EP1423106B1 (en)	2008-12-17
JP4187650B2 (ja)	2008-11-26
HUP0401235A2 (hu)	2004-10-28
DE60230424D1 (en)	2009-01-29
NO20040589L (no)	2004-03-19
KR100608417B1 (ko)	2006-08-02
ATE417838T1 (de)	2009-01-15
CA2456250A1 (en)	2003-02-20
PL373397A1 (en)	2005-08-22
RU2268884C2 (ru)	2006-01-27

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Publication	Publication Date	Title
NO326497B1 (no)	2008-12-15	Arylsulfonylderivater med 5-HT6 reseptor affinitet, farmasoytisk medikament omfattende slike, fremgangsmate for fremstilling av slike samt anvendelse av slike for fremstilling av medikament for behandling av sykdom
EP1401812B1 (en)	2006-06-28	4-piperazinylindole derivatives with 5-ht6 receptor affinity
US6774241B2 (en)	2004-08-10	1-sulfonyl-4-aminoalkoxy indole derivatives and uses thereof
JP2008524277A (ja)	2008-07-10	テトラリン及びインダン誘導体、並びにそれらの５−ｈｔ拮抗薬としての使用
HRP20050457A2 (en)	2005-10-31	Aminoalkoxyindoles as 5-ht6-receptor ligands for the treatment of cns-disorders
AU2002340804A1 (en)	2003-06-19	Arylsulfonyl derivatives with 5-HT6 receptor affinity
MX2011011520A (es)	2012-06-19	Compuestos de n-fenil-(piperazinil u homopiperazinil)-bencensulfon amida o bencensulfonil-fenil-(piperazina u homopiperazina) adecuados para tratar trastornos que responden a la modulacion del receptor de serotonina 5-ht6.
EP1910296B1 (en)	2010-04-21	4-aryloxy quinoline derivatives as 5-ht6 modulators
ZA200309258B (en)	2005-02-28	4-Piperazinylindole derivatives with 5-HT6 receptor affinity.
JP2008524274A (ja)	2008-07-10	テトラリン及びインダン誘導体、並びにそれらの使用
SK137597A3 (en)	1998-05-06	1-£'omega'-(3,4-dihydro-2-naphthalenyl)alkyl\| cyclic amine derivatives, process for producing the same, and medicinal composition containing the same
ZA200400749B (en)	2005-04-29	Arylsulfonyl derivatives with 5-HT6 receptor affinity.
KR100922486B1 (ko)	2009-10-20	비만, 제 ⅱ 형 당뇨병 및 ｃｎｓ 장애의 치료를 위한신규한 아릴술폰아미드 화합물
AU2002345587A1 (en)	2003-01-02	4-Piperazinylindole derivatives with 5-HT6 receptor affinity
MXPA06005840A (en)	2006-10-17	Benzoxazine derivatives and uses thereof