GB9926302D0 - Novel compounds - Google Patents
Novel compoundsInfo
- Publication number
- GB9926302D0 GB9926302D0 GBGB9926302.2A GB9926302A GB9926302D0 GB 9926302 D0 GB9926302 D0 GB 9926302D0 GB 9926302 A GB9926302 A GB 9926302A GB 9926302 D0 GB9926302 D0 GB 9926302D0
- Authority
- GB
- United Kingdom
- Prior art keywords
- novel compounds
- novel
- compounds
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Ceased
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/38—Nitrogen atoms
- C07D215/42—Nitrogen atoms attached in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Priority Applications (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB9926302.2A GB9926302D0 (en) | 1999-11-05 | 1999-11-05 | Novel compounds |
PCT/EP2000/010911 WO2001032646A2 (en) | 1999-11-05 | 2000-11-02 | Sulfonamide derivatives |
JP2001534797A JP2003513085A (en) | 1999-11-05 | 2000-11-02 | New compound |
AU12787/01A AU1278701A (en) | 1999-11-05 | 2000-11-02 | Novel compounds |
EP00974509A EP1228066A2 (en) | 1999-11-05 | 2000-11-02 | Sulfonamide derivatives |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB9926302.2A GB9926302D0 (en) | 1999-11-05 | 1999-11-05 | Novel compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
GB9926302D0 true GB9926302D0 (en) | 2000-01-12 |
Family
ID=10864071
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
GBGB9926302.2A Ceased GB9926302D0 (en) | 1999-11-05 | 1999-11-05 | Novel compounds |
Country Status (5)
Country | Link |
---|---|
EP (1) | EP1228066A2 (en) |
JP (1) | JP2003513085A (en) |
AU (1) | AU1278701A (en) |
GB (1) | GB9926302D0 (en) |
WO (1) | WO2001032646A2 (en) |
Families Citing this family (56)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR100888906B1 (en) | 2001-06-11 | 2009-03-16 | 바이오비트럼 에이비(피유비엘) | Substituted sulfonamide compounds, process for their use as medicament for the treatment of cns disorders, obesity and type ⅱ diabetes |
AU2002340804B2 (en) | 2001-08-10 | 2008-04-03 | F. Hoffmann-La Roche Ag | Arylsulfonyl derivatives with 5-HT6 receptor affinity |
SE0103644D0 (en) * | 2001-11-01 | 2001-11-01 | Astrazeneca Ab | Therapeutic isoquinoline compounds |
DE60232173D1 (en) | 2001-11-09 | 2009-06-10 | Biovitrum Ab Publ | USE OF SULFONAMIDE DERIVATIVES IN THE TREATMENT OF ADIPOSITAS OR TO REDUCE FOOD RECEPTION |
AU2002352878B2 (en) | 2001-11-27 | 2007-11-22 | Merck Sharp & Dohme Corp. | 2-Aminoquinoline compounds |
MXPA04007612A (en) * | 2002-02-05 | 2004-11-10 | Novo Nordisk As | Novel aryl- and heteroarylpiperazines. |
CN1630642A (en) * | 2002-02-13 | 2005-06-22 | 葛兰素集团有限公司 | Benzenesulfonamide derivatives |
WO2003068751A1 (en) * | 2002-02-13 | 2003-08-21 | Glaxo Group Limited | 7-arylsulfonamido-2,3,4,5-tetrahydro-1h-benzo'diazepine derivatives with 5-ht6 receptor affinity for the reatment of cns disorders |
AU2003218660A1 (en) * | 2002-02-13 | 2003-09-04 | Glaxo Group Limited | Benzenesulfonamide derivatives and their use as dopamine d3 and d2 receptor liga ds |
JP4455064B2 (en) | 2002-03-27 | 2010-04-21 | グラクソ グループ リミテッド | Quinoline derivatives and their use as 5-HT6 ligands |
AU2003248549B2 (en) | 2002-05-24 | 2010-04-08 | Millennium Pharmaceuticals, Inc. | CCR9 inhibitors and methods of use thereof |
WO2004000828A1 (en) * | 2002-06-20 | 2003-12-31 | Biovitrum Ab | New compounds useful for the treatment of obesity, type ii diabetes and cns disorders |
US7943639B2 (en) | 2002-06-20 | 2011-05-17 | Proximagen Limited | Compounds |
EP1897881A3 (en) | 2002-06-20 | 2009-03-18 | Biovitrum AB (publ) | Compounds useful for the treatment of obesity, type II diabetes and CNS disorders |
ES2264003T3 (en) * | 2002-10-07 | 2006-12-16 | Glaxo Group Limited | DERIVATIVES OF SULFONAMIDE AS ANTIPSYTIC AGENTS. |
US7741519B2 (en) | 2007-04-23 | 2010-06-22 | Chemocentryx, Inc. | Bis-aryl sulfonamides |
US7227035B2 (en) | 2002-11-18 | 2007-06-05 | Chemocentryx | Bis-aryl sulfonamides |
US7420055B2 (en) | 2002-11-18 | 2008-09-02 | Chemocentryx, Inc. | Aryl sulfonamides |
CN100360526C (en) | 2002-11-18 | 2008-01-09 | 坎莫森特里克斯公司 | Aryl sulfonamides |
OA13050A (en) | 2003-04-29 | 2006-11-10 | Pfizer Ltd | 5,7-diaminopyrazolo [4,3-D] pyrimidines useful in the treatment of hypertension. |
EA009732B1 (en) | 2003-07-22 | 2008-02-28 | Арена Фармасьютикалз, Инк. | Diaryl and arylheteroaryl urea derivatives as modulators of the 5-htserotonin receptor useful for the prophylaxis and treatment of disorders related thereto |
ES2222832B1 (en) | 2003-07-30 | 2006-02-16 | Laboratorios Del Dr. Esteve, S.A. | DERIVATIVES OF 6-INDOLILSULFONAMIDS, ITS PREPARATION AND ITS APPLICATION AS MEDICINES. |
ES2222829B1 (en) | 2003-07-30 | 2006-03-01 | Laboratorios Del Dr. Esteve, S.A. | DERIVATIVES OF 4-INDOLILSULFONAMIDS, ITS PREPARATION AND ITS APPLICATION AS MEDICATIONS. |
GB0320320D0 (en) * | 2003-08-29 | 2003-10-01 | Glaxo Group Ltd | Novel compounds |
US7572799B2 (en) | 2003-11-24 | 2009-08-11 | Pfizer Inc | Pyrazolo[4,3-d]pyrimidines as Phosphodiesterase Inhibitors |
AU2004299438A1 (en) * | 2003-12-19 | 2005-06-30 | Biovitrum Ab | Novel benzofuran derivatives, which can be used in prophylaxis or treatment of 5-HT6 receptor-related disorder |
SE0303480D0 (en) * | 2003-12-19 | 2003-12-19 | Biovitrum Ab | Benzofuranes |
DK1742950T3 (en) | 2004-04-07 | 2009-03-16 | Pfizer Ltd | The pyrazolo [4,3-d] pyrimidines |
WO2006062481A1 (en) * | 2004-12-09 | 2006-06-15 | Biovitrum Ab | New benzofuran derivatives and their use in the treatment of obesity, type ii diabetes and cns disorders . |
EP1676841A1 (en) * | 2004-12-30 | 2006-07-05 | Esteve Laboratorios Dr. Esteve S.A. | Substitited indazolyl sulfonamide and 2,3-dihydro-indolyl sulfonamide compounds, their prepartion and use in medicaments |
AU2006264966B2 (en) | 2005-07-04 | 2013-02-21 | High Point Pharmaceuticals, Llc | Histamine H3 receptor antagonists |
WO2007004960A1 (en) * | 2005-07-05 | 2007-01-11 | Astrazeneca Ab | New compounds, process for their preparation, intermediates, pharmaceutical compositions and their use in the treatment of 5-ht6 mediated disorders such as alzheimer’s desease, cognitive disorders, cognitive impairment associated with schizophrenia, obesity and parkinson’s disease |
WO2007004959A1 (en) * | 2005-07-05 | 2007-01-11 | Astrazeneca Ab | New compounds, process for their preparation, intermediates, pharmaceutical compositions and their use in the treatment of 5-ht6 mediated disorders such as alzheimer's disease, cognitive disorders, cognitive impairment associated with schizophrenia, obesity and parkinson's disease |
EP1919896B1 (en) | 2005-08-12 | 2009-12-23 | Suven Life Sciences Limited | Aminoaryl sulphonamide derivatives as functional 5-ht6 ligands. |
US7923566B2 (en) | 2005-08-16 | 2011-04-12 | Suven Life Sciences Limited | Alternative process for the preparation of losartan |
WO2007108744A2 (en) * | 2006-03-17 | 2007-09-27 | Astrazeneca Ab | Novel quinazolines as 5-ht6 modulators |
WO2007108743A2 (en) * | 2006-03-17 | 2007-09-27 | Astrazeneca Ab | Novel quinazolines as 5-ht6 modulators ii |
EP1837332A1 (en) * | 2006-03-23 | 2007-09-26 | Laboratorios Del Dr. Esteve, S.A. | Substituted tetrahydroisoquinoline compounds, their preparation and use in medicaments |
SI2079732T1 (en) | 2006-05-29 | 2012-03-30 | High Point Pharmaceuticals Llc | 3- (1, 3-benz0di0x0l-5-yl) -6- (4-cyclopropylpiperazin-1-yl) -pyridazine, its salts and solvates and its use as histamine h3 receptor antagonist |
EA016456B1 (en) | 2006-10-30 | 2012-05-30 | Биовитрум Аб (Пабл) | 8-sulfonyl-1,3,4,8-tetrahydro-2h-[1,4]oxazepino[6,7-e]indole derivatives and their use as 5-htreceptor ligands |
CA2670717C (en) | 2007-01-08 | 2012-01-10 | Suven Life Sciences Limited | 5-(heterocyclyl)alkyl-n-(arylsulfonyl)indole compounds and their use as 5-ht6 ligands |
DK2155674T3 (en) | 2007-05-03 | 2011-09-26 | Suven Life Sciences Ltd | Aminoalkoxy-aryl-sulfonamide compounds and their use as 5-HT6 ligands |
EP2014656A3 (en) | 2007-06-11 | 2011-08-24 | High Point Pharmaceuticals, LLC | New heteocyclic h3 antagonists |
DE102007042154A1 (en) * | 2007-09-05 | 2009-03-12 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Arylsulfonylaminomethyphosphonsäure derivatives, their preparation and their use as medicaments |
BRPI0816571A2 (en) | 2007-10-26 | 2015-12-22 | Suven Life Sciences Ltd | "compound, process for preparing the compound, pharmaceutical composition, agent and method for treating a disease or disorder of the central nervous system related to or affected by the 5-ht6 receptor" |
WO2009074607A1 (en) | 2007-12-12 | 2009-06-18 | Glaxo Group Limited | Combinations comprising 3-phenylsulfonyl-8-piperazinyl-1yl-quinoline |
JP2011512340A (en) * | 2008-02-15 | 2011-04-21 | エフ.ホフマン−ラ ロシュ アーゲー | 3-alkylpiperazine derivatives and uses thereof |
WO2009123714A2 (en) | 2008-04-02 | 2009-10-08 | Arena Pharmaceuticals, Inc. | Processes for the preparation of pyrazole derivatives useful as modulators of the 5-ht2a serotonin receptor |
EP2116547A1 (en) * | 2008-05-09 | 2009-11-11 | Laboratorios Del. Dr. Esteve, S.A. | Substituted N-imidazo(2, 1-b) thiazole-5-sulfonamide derivatives as 5-TH6 ligands |
KR101308819B1 (en) | 2008-09-17 | 2013-09-13 | 수벤 라이프 사이언시스 리미티드 | Aryl sulfonamide amine compounds and their use as 5-ht6 ligands |
US8318725B2 (en) | 2008-09-17 | 2012-11-27 | Suven Life Sciences Limited | Aryl indolyl sulfonamide compounds and their use as 5-HT6 ligands |
US9126946B2 (en) | 2008-10-28 | 2015-09-08 | Arena Pharmaceuticals, Inc. | Processes useful for the preparation of 1-[3-(4-bromo-2-methyl-2H-pyrazol-3-yl)-4-methoxy-phenyl]-3-(2,4-difluoro-phenyl)urea and crystalline forms related thereto |
SG181992A1 (en) | 2010-01-05 | 2012-08-30 | Suven Life Sciences Ltd | Sulfone compounds as 5-ht6 receptor ligands |
WO2015158313A1 (en) | 2014-04-19 | 2015-10-22 | Sunshine Lake Pharma Co., Ltd. | Sulfonamide derivatives and pharmaceutical applications thereof |
EP4119141A1 (en) | 2015-06-12 | 2023-01-18 | Axovant Sciences GmbH | Nelotanserin for the prophylaxis and treatment of rem sleep behavior disorder |
BR112018000728A2 (en) | 2015-07-15 | 2018-09-04 | Axovant Sciences Gmbh | method for the prophylaxis and / or treatment of visual hallucinations in a subject in need |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
PT689536E (en) * | 1993-03-16 | 2001-11-30 | Pfizer | NAFTALENE DERIVATIVES |
DZ2376A1 (en) * | 1996-12-19 | 2002-12-28 | Smithkline Beecham Plc | New sulfonamide derivatives process for their preparation and pharmaceutical compositions containing them. |
-
1999
- 1999-11-05 GB GBGB9926302.2A patent/GB9926302D0/en not_active Ceased
-
2000
- 2000-11-02 WO PCT/EP2000/010911 patent/WO2001032646A2/en not_active Application Discontinuation
- 2000-11-02 JP JP2001534797A patent/JP2003513085A/en not_active Withdrawn
- 2000-11-02 EP EP00974509A patent/EP1228066A2/en not_active Withdrawn
- 2000-11-02 AU AU12787/01A patent/AU1278701A/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
WO2001032646A3 (en) | 2001-12-27 |
EP1228066A2 (en) | 2002-08-07 |
WO2001032646A2 (en) | 2001-05-10 |
JP2003513085A (en) | 2003-04-08 |
AU1278701A (en) | 2001-05-14 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
EP1140083A4 (en) | Novel compounds | |
GB9902084D0 (en) | Novel compounds | |
GB9902697D0 (en) | Novel compounds | |
EG24063A (en) | Novel compounds | |
GB9901256D0 (en) | Novel compounds | |
GB9902937D0 (en) | Novel compounds | |
GB9902070D0 (en) | Novel compounds | |
GB9902880D0 (en) | Novel compounds | |
GB9901948D0 (en) | Novel compounds | |
GB9902078D0 (en) | Novel compounds | |
GB9900952D0 (en) | Novel compounds | |
GB9900959D0 (en) | Novel compounds | |
GB9901078D0 (en) | Novel compounds | |
GB9901209D0 (en) | Novel compounds | |
GB9901368D0 (en) | Novel compounds | |
GB9903402D0 (en) | Novel compounds | |
GB9901463D0 (en) | Novel compounds | |
GB9901465D0 (en) | Novel compounds | |
GB9901602D0 (en) | Novel compounds | |
GB9901903D0 (en) | Novel compounds | |
GB9901944D0 (en) | Novel compounds | |
GB9901945D0 (en) | Novel compounds | |
GB9901946D0 (en) | Novel compounds | |
GB9901947D0 (en) | Novel compounds | |
GB9900090D0 (en) | Novel compounds |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
AT | Applications terminated before publication under section 16(1) |