NO20090811L - Fremgangsmate for fremstilling av 3(R)-(2-hydroksy-2,2-ditien-2-ylacetoksy)-1-(3-fenoksypropyl)-1-azoniabicyklo[2.2.2]oktanbromid - Google Patents

Fremgangsmate for fremstilling av 3(R)-(2-hydroksy-2,2-ditien-2-ylacetoksy)-1-(3-fenoksypropyl)-1-azoniabicyklo[2.2.2]oktanbromid

Info

Publication number
NO20090811L
NO20090811L NO20090811A NO20090811A NO20090811L NO 20090811 L NO20090811 L NO 20090811L NO 20090811 A NO20090811 A NO 20090811A NO 20090811 A NO20090811 A NO 20090811A NO 20090811 L NO20090811 L NO 20090811L
Authority
NO
Norway
Prior art keywords
dithien
hydroxy
phenoxypropyl
ylacetoxy
azoniabicyclo
Prior art date
Application number
NO20090811A
Other languages
English (en)
Norwegian (no)
Inventor
Nuria Busquets Baque
Francesca Pajuelo Lorenzo
Original Assignee
Almirall Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37808353&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20090811(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Almirall Lab filed Critical Almirall Lab
Publication of NO20090811L publication Critical patent/NO20090811L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/439Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
NO20090811A 2006-07-21 2009-02-20 Fremgangsmate for fremstilling av 3(R)-(2-hydroksy-2,2-ditien-2-ylacetoksy)-1-(3-fenoksypropyl)-1-azoniabicyklo[2.2.2]oktanbromid NO20090811L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
ES200601951A ES2298049B1 (es) 2006-07-21 2006-07-21 Procedimiento para fabricar bromuro de 3(r)-(2-hidroxi-2,2-ditien-2-ilacetoxi)-1-(3-fenoxipropil)-1-azoniabiciclo (2.2.2) octano.
PCT/EP2007/006278 WO2008009397A1 (en) 2006-07-21 2007-07-16 Process for manufacturing 3(r)-(2-hydroxy-2,2-dithien-2-ylacetoxy)-1-(3-phenoxypropyl)-1-azoniabicyclo[2.2.2]octane bromide

Publications (1)

Publication Number Publication Date
NO20090811L true NO20090811L (no) 2009-02-20

Family

ID=37808353

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20090811A NO20090811L (no) 2006-07-21 2009-02-20 Fremgangsmate for fremstilling av 3(R)-(2-hydroksy-2,2-ditien-2-ylacetoksy)-1-(3-fenoksypropyl)-1-azoniabicyklo[2.2.2]oktanbromid

Country Status (37)

Country Link
US (1) US8044205B2 (es)
EP (1) EP2044067B1 (es)
JP (1) JP5279708B2 (es)
KR (1) KR101410198B1 (es)
CN (1) CN101490048B (es)
AR (1) AR061933A1 (es)
AT (1) ATE449096T1 (es)
AU (1) AU2007276395B2 (es)
BR (1) BRPI0711500B1 (es)
CA (1) CA2657679C (es)
CL (1) CL2007002078A1 (es)
CO (1) CO6460740A2 (es)
CY (1) CY1109792T1 (es)
DE (1) DE602007003375D1 (es)
DK (1) DK2044067T3 (es)
EC (1) ECSP099033A (es)
EG (1) EG25727A (es)
ES (2) ES2298049B1 (es)
HK (1) HK1124051A1 (es)
HR (1) HRP20090652T1 (es)
IL (1) IL196324A (es)
ME (1) ME01773B (es)
MX (1) MX2009000573A (es)
MY (1) MY145285A (es)
NO (1) NO20090811L (es)
NZ (1) NZ573170A (es)
PE (1) PE20081307A1 (es)
PL (1) PL2044067T3 (es)
PT (1) PT2044067E (es)
RS (1) RS51264B (es)
RU (1) RU2439070C2 (es)
SI (1) SI2044067T1 (es)
TW (1) TWI363057B (es)
UA (1) UA96453C2 (es)
UY (1) UY30475A1 (es)
WO (1) WO2008009397A1 (es)
ZA (1) ZA200810051B (es)

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EP2510928A1 (en) 2011-04-15 2012-10-17 Almirall, S.A. Aclidinium for use in improving the quality of sleep in respiratory patients
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CZ306791B6 (cs) * 2013-10-29 2017-07-12 Zentiva, K.S. Průmyslově využitelný způsob přípravy aklidinium bromidu o vysoké čistotě
CN103755699A (zh) * 2014-01-06 2014-04-30 万特制药(海南)有限公司 一种2-羟基-2,2-二噻吩-2-基乙酸-1-氮杂二环[2,2,2]辛-3(r)-基酯制备方法
CN103755698A (zh) * 2014-01-06 2014-04-30 万特制药(海南)有限公司 一锅法制备阿地溴铵的工艺
CZ2014188A3 (cs) 2014-03-26 2015-10-07 Zentiva, K.S. Nové formy aclidinium chloridu a způsob jejich přípravy
CN104478871B (zh) * 2014-12-26 2016-09-07 东华大学 一种胆碱m受体拮抗剂阿地溴铵及其制备方法
PT108370B (pt) 2015-03-30 2018-10-25 Hovione Farm S A Processo de preparação de brometo de aclidínio
WO2016162878A1 (en) * 2015-04-04 2016-10-13 Harman Finochem Limited An advantageous process for preparing 1-azoniabicyclo[2.2.2]octane,3-[(hydroxydi-2-thienylacetyl)oxy]-1-(3¬phenoxypropyl)-, bromide, (3r)- and its novel crystalline form-i
CZ2015257A3 (cs) 2015-04-16 2016-10-26 Zentiva, K.S. Způsob pro zmenšování velikosti částic bromidu [(3R)-1-(3-fenoxypropyl)chinuklidin-1-ium-3-yl] 2-hydroxy-2,2-bis(2-thienyl)acetátu

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Also Published As

Publication number Publication date
US8044205B2 (en) 2011-10-25
UA96453C2 (uk) 2011-11-10
KR20090031578A (ko) 2009-03-26
AU2007276395B2 (en) 2012-03-08
IL196324A (en) 2012-12-31
ZA200810051B (en) 2009-11-25
PT2044067E (pt) 2009-12-21
UY30475A1 (es) 2008-01-02
PL2044067T3 (pl) 2010-04-30
BRPI0711500B1 (pt) 2014-09-16
AR061933A1 (es) 2008-10-01
ECSP099033A (es) 2009-02-27
RS51264B (sr) 2010-12-31
CY1109792T1 (el) 2014-09-10
BRPI0711500A2 (pt) 2011-11-01
RU2009105827A (ru) 2010-08-27
MY145285A (en) 2012-01-13
CN101490048A (zh) 2009-07-22
CO6460740A2 (es) 2012-06-15
JP5279708B2 (ja) 2013-09-04
MX2009000573A (es) 2009-01-29
JP2009544591A (ja) 2009-12-17
CA2657679A1 (en) 2008-01-24
SI2044067T1 (sl) 2010-03-31
RU2439070C2 (ru) 2012-01-10
ES2298049B1 (es) 2009-10-20
ME01773B (me) 2010-12-31
DK2044067T3 (da) 2010-02-01
IL196324A0 (en) 2009-09-22
WO2008009397A1 (en) 2008-01-24
ATE449096T1 (de) 2009-12-15
ES2298049A1 (es) 2008-05-01
HK1124051A1 (en) 2009-07-03
CN101490048B (zh) 2011-06-29
EP2044067A1 (en) 2009-04-08
EP2044067B1 (en) 2009-11-18
DE602007003375D1 (de) 2009-12-31
TW200821307A (en) 2008-05-16
KR101410198B1 (ko) 2014-06-19
WO2008009397A8 (en) 2009-01-22
NZ573170A (en) 2010-12-24
CA2657679C (en) 2014-10-21
AU2007276395A1 (en) 2008-01-24
TWI363057B (en) 2012-05-01
ES2336045T3 (es) 2010-04-07
US20090299042A1 (en) 2009-12-03
EG25727A (en) 2012-06-11
HRP20090652T1 (hr) 2010-01-31
PE20081307A1 (es) 2008-09-17
CL2007002078A1 (es) 2008-01-25

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