NO20082365L - Ny metode for fremstilling av 5-amino-3H-tiazolo[4,5-D]pyrimidin-2-on - Google Patents

Ny metode for fremstilling av 5-amino-3H-tiazolo[4,5-D]pyrimidin-2-on

Info

Publication number
NO20082365L
NO20082365L NO20082365A NO20082365A NO20082365L NO 20082365 L NO20082365 L NO 20082365L NO 20082365 A NO20082365 A NO 20082365A NO 20082365 A NO20082365 A NO 20082365A NO 20082365 L NO20082365 L NO 20082365L
Authority
NO
Norway
Prior art keywords
preparation
thiazolo
pyrimidin
amino
new method
Prior art date
Application number
NO20082365A
Other languages
English (en)
Inventor
Stephen E Webber
Tingmin Wang
John S Ng
Original Assignee
Anadys Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Anadys Pharmaceuticals Inc filed Critical Anadys Pharmaceuticals Inc
Publication of NO20082365L publication Critical patent/NO20082365L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

Foreliggende oppfinnelse angår en fremgangsmåte for fremstilling av tittelforbindelsen, 5-amino-3H-tiazolo[4,5-d]pyrimidin-2-on, som er et anvendelig mellomprodukt ved fremstilling av visse tiazolo[4,5-d]pyrimidin-nukleosider, som kan ha nytte som immunmodulerende midler.
NO20082365A 2005-11-21 2008-05-26 Ny metode for fremstilling av 5-amino-3H-tiazolo[4,5-D]pyrimidin-2-on NO20082365L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US73805505P 2005-11-21 2005-11-21
PCT/US2006/061111 WO2007062355A2 (en) 2005-11-21 2006-11-20 PROCESS FOR THE PREPARATION OF 5-AMINO-3H- THIAZOLO [4 , 5 -d] PYRIMIDIN- 2 -ONE

Publications (1)

Publication Number Publication Date
NO20082365L true NO20082365L (no) 2008-08-18

Family

ID=37908057

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20082365A NO20082365L (no) 2005-11-21 2008-05-26 Ny metode for fremstilling av 5-amino-3H-tiazolo[4,5-D]pyrimidin-2-on

Country Status (18)

Country Link
US (1) US7781581B2 (no)
EP (1) EP1973920B1 (no)
JP (1) JP5117391B2 (no)
KR (1) KR20080090400A (no)
CN (1) CN101365705A (no)
AR (1) AR058210A1 (no)
AT (1) ATE474842T1 (no)
AU (1) AU2006318260B2 (no)
BR (1) BRPI0618789A2 (no)
CA (1) CA2630463C (no)
DE (1) DE602006015700D1 (no)
EA (1) EA200801404A1 (no)
ES (1) ES2345904T3 (no)
IL (1) IL191568A0 (no)
NO (1) NO20082365L (no)
SG (1) SG152296A1 (no)
TW (1) TWI383987B (no)
WO (1) WO2007062355A2 (no)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE496924T1 (de) 2006-06-22 2011-02-15 Anadys Pharmaceuticals Inc Prodrugs von 5-amino-3-(3'-deoxy-beta-d- ribofuranosyl)-thiazolä4,5-düpyrimidin-2,7-dion
JPWO2012102366A1 (ja) * 2011-01-28 2014-06-30 日本たばこ産業株式会社 新規ピペラジン化合物の製造方法
CN103012284A (zh) * 2012-12-26 2013-04-03 无锡捷化医药科技有限公司 一种2-氨基-5-溴嘧啶类化合物的制备方法
JP6817217B2 (ja) 2014-12-08 2021-01-20 エフ．ホフマン−ラ ロシュ アーゲーＦ． Ｈｏｆｆｍａｎｎ−Ｌａ Ｒｏｃｈｅ Ａｋｔｉｅｎｇｅｓｅｌｌｓｃｈａｆｔ ウイルス感染症の治療および予防のための３−置換された５−アミノ−６Ｈ−チアゾロ［４，５−ｄ］ピリミジン−２，７−ジオン化合物
JP7201598B2 (ja) 2017-01-06 2023-01-10 エフ．ホフマン－ラ ロシュ アーゲー ３位置換５－アミノ－６Ｈ－チアゾロ［４，５－ｄ］ピリミジン－２，７－ジオン化合物の製造法
CN111635368B (zh) * 2020-06-12 2021-06-29 东莞市东阳光仿制药研发有限公司 一种胺化合物的制备方法

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Also Published As

Publication number Publication date
WO2007062355A2 (en) 2007-05-31
ATE474842T1 (de) 2010-08-15
AU2006318260B2 (en) 2012-05-17
AR058210A1 (es) 2008-01-23
AU2006318260A1 (en) 2007-05-31
US20070117979A1 (en) 2007-05-24
TW200736265A (en) 2007-10-01
EP1973920A2 (en) 2008-10-01
KR20080090400A (ko) 2008-10-08
DE602006015700D1 (de) 2010-09-02
JP5117391B2 (ja) 2013-01-16
CN101365705A (zh) 2009-02-11
ES2345904T3 (es) 2010-10-05
BRPI0618789A2 (pt) 2016-08-30
IL191568A0 (en) 2008-12-29
CA2630463A1 (en) 2007-05-31
EA200801404A1 (ru) 2008-10-30
JP2009516709A (ja) 2009-04-23
CA2630463C (en) 2015-01-06
EP1973920B1 (en) 2010-07-21
US7781581B2 (en) 2010-08-24
WO2007062355A3 (en) 2007-07-26
TWI383987B (zh) 2013-02-01
SG152296A1 (en) 2009-05-29

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