MXPA05007857A - Moduladores derivados de indol de receptores nucleares de hormonas esteroideas. - Google Patents

Moduladores derivados de indol de receptores nucleares de hormonas esteroideas.

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Publication number
MXPA05007857A
MXPA05007857A MXPA05007857A MXPA05007857A MXPA05007857A MX PA05007857 A MXPA05007857 A MX PA05007857A MX PA05007857 A MXPA05007857 A MX PA05007857A MX PA05007857 A MXPA05007857 A MX PA05007857A MX PA05007857 A MXPA05007857 A MX PA05007857A
Authority
MX
Mexico
Prior art keywords
indole
steroid hormone
nuclear receptors
hormone nuclear
compound
Prior art date
Application number
MXPA05007857A
Other languages
English (en)
Inventor
Irvin Steinberg Mitchell
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of MXPA05007857A publication Critical patent/MXPA05007857A/es

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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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Abstract

La presente invencion se refiere a un compuesto de la formula I o una sal farmaceuticamente aceptable de la misma, a composiciones farmaceuticas que incluyen una cantidad eficaz del compuesto de la Formula I en combinacion con un vehiculo, diluyente o excipiente adecuado y a procedimientos de tratamiento de trastornos fisiologicos, en especial, insuficiencia cardiaca congestiva, que incluyen la administracion a un paciente de una cantidad efectiva de un compuesto de la Formula I (ver Formula I).
MXPA05007857A 2003-01-22 2004-01-20 Moduladores derivados de indol de receptores nucleares de hormonas esteroideas. MXPA05007857A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US44194703P 2003-01-22 2003-01-22
PCT/US2004/000017 WO2004067529A1 (en) 2003-01-22 2004-01-20 Indole-derivative modulators of steroid hormone nuclear receptors

Publications (1)

Publication Number Publication Date
MXPA05007857A true MXPA05007857A (es) 2005-10-18

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MXPA05007857A MXPA05007857A (es) 2003-01-22 2004-01-20 Moduladores derivados de indol de receptores nucleares de hormonas esteroideas.

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Country Link
US (1) US20060235222A1 (es)
EP (1) EP1597254A1 (es)
JP (1) JP2007500253A (es)
CN (1) CN1742007A (es)
AU (1) AU2004207740A1 (es)
BR (1) BRPI0406883A (es)
CA (1) CA2511806A1 (es)
MX (1) MXPA05007857A (es)
WO (1) WO2004067529A1 (es)

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EP1723105B1 (en) * 2004-03-03 2013-05-15 Eli Lilly And Company Bicyclic substituted indole-derivative steroid hormone nuclear receptor modulators
DE102004021637A1 (de) * 2004-05-03 2005-12-01 Merck Patent Gmbh Dihydrobenzothiophene
EP1632491A1 (en) * 2004-08-30 2006-03-08 Laboratorios Del Dr. Esteve, S.A. Substituted indole compounds and their use as 5-HT6 receptor modulators
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