NO20055624L - Tropanderivater og deres anvendelse som Ace-inhibitorer - Google Patents
Tropanderivater og deres anvendelse som Ace-inhibitorerInfo
- Publication number
- NO20055624L NO20055624L NO20055624A NO20055624A NO20055624L NO 20055624 L NO20055624 L NO 20055624L NO 20055624 A NO20055624 A NO 20055624A NO 20055624 A NO20055624 A NO 20055624A NO 20055624 L NO20055624 L NO 20055624L
- Authority
- NO
- Norway
- Prior art keywords
- ace inhibitors
- compounds
- tropane derivatives
- derivatives
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Urology & Nephrology (AREA)
- Ophthalmology & Optometry (AREA)
- Hospice & Palliative Care (AREA)
- Vascular Medicine (AREA)
- Gynecology & Obstetrics (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
Oppfmnelsen angår nye fropan-derivater og beslektede forbindelser og deres anvendelse som aktive bestanddeler ved fremstilling av farmasøytiske preparater. Oppfirmelsen angår også relaterte aspekter, inkludert fremgangsmåter for fremstilling av forbindelsene, farmasøytiske preparater som irmeholder en eller flere av disse forbindelsene, og spesielt deres anvendelse som inhibitorer av renin.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP0304490 | 2003-04-30 | ||
PCT/EP2004/004375 WO2004096799A1 (en) | 2003-04-30 | 2004-04-26 | Tropane derivatives and their use as ace inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20055624L true NO20055624L (no) | 2005-11-29 |
Family
ID=33395688
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20055624A NO20055624L (no) | 2003-04-30 | 2005-11-29 | Tropanderivater og deres anvendelse som Ace-inhibitorer |
Country Status (13)
Country | Link |
---|---|
US (1) | US20060205768A1 (no) |
EP (1) | EP1622901A1 (no) |
JP (1) | JP2006524657A (no) |
KR (1) | KR20060015546A (no) |
CN (1) | CN1780833A (no) |
AU (1) | AU2004234042A1 (no) |
BR (1) | BRPI0409878A (no) |
CA (1) | CA2521957A1 (no) |
MX (1) | MXPA05011497A (no) |
NO (1) | NO20055624L (no) |
RU (1) | RU2005137184A (no) |
WO (1) | WO2004096799A1 (no) |
ZA (1) | ZA200509663B (no) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN1930170A (zh) * | 2003-10-23 | 2007-03-14 | 埃科特莱茵药品有限公司 | 二氮杂二环壬烯及四氢吡啶衍生物用作肾素抑制剂 |
JP2007513107A (ja) * | 2003-12-05 | 2007-05-24 | アクテリオン ファマシューティカルズ リミテッド | ジアザビシクロノネンおよび新側鎖を有するテトラヒドロピリジン誘導体 |
ATE462703T1 (de) | 2004-08-25 | 2010-04-15 | Actelion Pharmaceuticals Ltd | Bicyclononen-derivate als renin-inhibitoren |
GB0428526D0 (en) | 2004-12-30 | 2005-02-09 | Novartis Ag | Organic compounds |
WO2006092268A1 (en) * | 2005-03-02 | 2006-09-08 | Actelion Pharmaceuticals Ltd | Bicyclic five-membered heteroaryl derivatives and their use as renin inhibitors |
GB0514203D0 (en) | 2005-07-11 | 2005-08-17 | Novartis Ag | Organic compounds |
WO2007049224A1 (en) * | 2005-10-25 | 2007-05-03 | Actelion Pharmaceuticals Ltd | Novel hexahydro- or octahydro-cyclopenta[c]pyrrole derivatives |
US8129411B2 (en) | 2005-12-30 | 2012-03-06 | Novartis Ag | Organic compounds |
US7968720B2 (en) | 2006-02-02 | 2011-06-28 | Actelion Pharmaceuticals Ltd. | Secondary amines as renin inhibitors |
US20100166839A1 (en) * | 2006-03-16 | 2010-07-01 | Nicox S.A | Non peptidic renin inhibitors nitroderivatives |
AU2008253519A1 (en) | 2007-05-24 | 2008-11-27 | Merck Frosst Canada Ltd | Novel case of renin inhibitors |
BRPI0813900A2 (pt) | 2007-06-25 | 2014-12-30 | Novartis Ag | Derivados de n5-(2-etoxietil)-n3-(2-piridinil)-3,5-piperidinodicarboxa mida para uso como inibidores de renina |
US8334308B2 (en) | 2007-08-20 | 2012-12-18 | Merck Sharp & Dohme Corp. | Renin inhibitors |
CA2722734C (en) | 2008-05-05 | 2013-11-05 | Merck Frosst Canada Ltd. | 3,4-substituted piperidine derivatives as renin inhibitors |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3509161A (en) * | 1967-07-10 | 1970-04-28 | Boehringer & Soehne Gmbh | 3-phenyl-granatene-(2)-derivatives |
US6329520B1 (en) * | 1990-08-09 | 2001-12-11 | Research Triangle Institute | Cocaine receptor binding ligands |
US7011813B2 (en) * | 1990-08-09 | 2006-03-14 | Research Triangle Institute | Cocaine receptor binding ligands |
US5380758A (en) * | 1991-03-29 | 1995-01-10 | Brigham And Women's Hospital | S-nitrosothiols as smooth muscle relaxants and therapeutic uses thereof |
PL294866A1 (en) * | 1991-06-21 | 1993-05-31 | Hoechst Ag | Method of obtaining novel rennin redtarding heterocyclic compounds |
US5703073A (en) * | 1995-04-19 | 1997-12-30 | Nitromed, Inc. | Compositions and methods to prevent toxicity induced by nonsteroidal antiinflammatory drugs |
WO1997009311A1 (de) * | 1995-09-07 | 1997-03-13 | F. Hoffmann-La Roche Ag | Neue 4-(oxyalkoxyphenyl)-3-oxy-piperidine zur behandlung von herz- und niereninsuffizienz |
US20030013883A1 (en) * | 2000-06-16 | 2003-01-16 | Tamagnan Gilles D. | Tropane analogs binding to monoamine transporters |
US20060079533A1 (en) * | 2001-03-23 | 2006-04-13 | Nieman James A | Methods of treating alzheimer's disease |
AU2003233963B2 (en) * | 2002-04-29 | 2008-09-11 | Actelion Pharmaceuticals Ltd | 7-aryl-3,9-diazabicyclo(3.3.1)non-6-ene derivatives and their use as renin inhibitors in the treatment of hypertension, cardiovascular or renal diseases |
-
2004
- 2004-04-26 RU RU2005137184/04A patent/RU2005137184A/ru not_active Application Discontinuation
- 2004-04-26 WO PCT/EP2004/004375 patent/WO2004096799A1/en not_active Application Discontinuation
- 2004-04-26 CN CNA2004800114420A patent/CN1780833A/zh active Pending
- 2004-04-26 MX MXPA05011497A patent/MXPA05011497A/es not_active Application Discontinuation
- 2004-04-26 JP JP2006505264A patent/JP2006524657A/ja active Pending
- 2004-04-26 CA CA002521957A patent/CA2521957A1/en not_active Abandoned
- 2004-04-26 BR BRPI0409878-1A patent/BRPI0409878A/pt not_active Application Discontinuation
- 2004-04-26 AU AU2004234042A patent/AU2004234042A1/en not_active Abandoned
- 2004-04-26 US US10/554,704 patent/US20060205768A1/en not_active Abandoned
- 2004-04-26 EP EP04729423A patent/EP1622901A1/en not_active Withdrawn
- 2004-04-26 KR KR1020057020498A patent/KR20060015546A/ko not_active Application Discontinuation
-
2005
- 2005-11-29 ZA ZA200509663A patent/ZA200509663B/en unknown
- 2005-11-29 NO NO20055624A patent/NO20055624L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
RU2005137184A (ru) | 2006-03-20 |
CA2521957A1 (en) | 2004-11-11 |
CN1780833A (zh) | 2006-05-31 |
KR20060015546A (ko) | 2006-02-17 |
BRPI0409878A (pt) | 2006-05-23 |
MXPA05011497A (es) | 2005-12-15 |
ZA200509663B (en) | 2006-09-27 |
AU2004234042A1 (en) | 2004-11-11 |
US20060205768A1 (en) | 2006-09-14 |
JP2006524657A (ja) | 2006-11-02 |
EP1622901A1 (en) | 2006-02-08 |
WO2004096799A1 (en) | 2004-11-11 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
NO20055624L (no) | Tropanderivater og deres anvendelse som Ace-inhibitorer | |
NO20050290L (no) | Nye tetrahydropyridin-derivater som renin-inhibitorer | |
NO20055623L (no) | Azabicyklononenderivater | |
NO20064347L (no) | Substituerte 1,2,3,4-tetrahydroisokinolinderivater | |
NO20064584L (no) | Tetrahydropyridoindolderivater | |
NO20054974L (no) | 9-azabicyklo(3.3.1)non-6-en derivater med et heteroatom i 3-posisjonen som renin inhibitorer | |
NO20050932L (no) | 1-pyridin-4-yl-ureaderivater | |
NO20061395L (no) | Nye pyridinderivater | |
NO20090628L (no) | Pyridizinon derivativater | |
NO20045042L (no) | 7-aryl -3,9-diazabicyklo (3.1.1)non-6-en-derivater og deres anvendelse som renin. inhibitorer ved behandling av hypertensjon, kardiovaskulaere og nyresykdommer | |
BRPI0508579A (pt) | composto, composição farmacêutica, e, uso de um composto | |
NO20066055L (no) | Pyridinderivater | |
ECSP067076A (es) | Derivados de pirimidina urea como inhibidores de la quinasa | |
ATE532781T1 (de) | 5-(acylamino)indazol-derivate als kinase- inhibitoren | |
NO20084186L (no) | Nye aminer | |
NO20082530L (no) | Imidazopyraziner som proteinkinaseinhibitorer | |
NO20082269L (no) | Nye piperaziner som antimalariamidler | |
ATE462703T1 (de) | Bicyclononen-derivate als renin-inhibitoren | |
NO20083738L (no) | Sekundaere aminer som renininhibitorer | |
NO20085212L (no) | Nye pyridinanaloger | |
NO20076448L (no) | Novel piperidine carboxylic acid amide derivatives | |
NO20084055L (no) | Nye primaere aminer | |
TW200628468A (en) | Bicyclononene derivatives | |
WO2006042478A8 (fr) | Inhibiteurs de petites molecules de la protease principale des coronavirus, leur preparation et utilisation | |
WO2005054244A3 (en) | Azabicyclooctene and other tetrahydropyridine derivatives with a new side-chain |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
FC2A | Withdrawal, rejection or dismissal of laid open patent application |