NO20015362L - Heterocyklisk substituerte benzimidazoler, deres fremstilling og anvendelse derav - Google Patents
Heterocyklisk substituerte benzimidazoler, deres fremstilling og anvendelse deravInfo
- Publication number
- NO20015362L NO20015362L NO20015362A NO20015362A NO20015362L NO 20015362 L NO20015362 L NO 20015362L NO 20015362 A NO20015362 A NO 20015362A NO 20015362 A NO20015362 A NO 20015362A NO 20015362 L NO20015362 L NO 20015362L
- Authority
- NO
- Norway
- Prior art keywords
- preparation
- heterocyclic substituted
- substituted benzimidazoles
- benzimidazoles
- heterocyclic
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A61P25/10—Antiepileptics; Anticonvulsants for petit-mal
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/18—Benzimidazoles; Hydrogenated benzimidazoles with aryl radicals directly attached in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19920936A DE19920936A1 (de) | 1999-05-07 | 1999-05-07 | Heterozyklisch substituierte Benzimidazole, deren Herstellung und Anwendung |
PCT/EP2000/003813 WO2000068206A1 (de) | 1999-05-07 | 2000-04-27 | Heterozyklisch substituierte benzimidazole, deren herstellung und anwendung |
Publications (2)
Publication Number | Publication Date |
---|---|
NO20015362L true NO20015362L (no) | 2001-11-02 |
NO20015362D0 NO20015362D0 (no) | 2001-11-02 |
Family
ID=7907219
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20015362A NO20015362D0 (no) | 1999-05-07 | 2001-11-02 | Heterocyklisk substituerte benzimidazoler, deres fremstilling og anvendelse derav |
Country Status (27)
Country | Link |
---|---|
US (1) | US6696437B1 (no) |
EP (1) | EP1177178B1 (no) |
JP (1) | JP4004737B2 (no) |
KR (1) | KR20010112477A (no) |
CN (1) | CN1353695A (no) |
AR (1) | AR029161A1 (no) |
AT (1) | ATE286029T1 (no) |
AU (1) | AU4558400A (no) |
BG (1) | BG106035A (no) |
BR (1) | BR0010342A (no) |
CA (1) | CA2371645C (no) |
CO (1) | CO5170517A1 (no) |
DE (2) | DE19920936A1 (no) |
DK (1) | DK1177178T3 (no) |
ES (1) | ES2235869T3 (no) |
HK (1) | HK1046281A1 (no) |
HU (1) | HUP0202970A2 (no) |
IL (1) | IL146147A0 (no) |
MY (1) | MY122771A (no) |
NO (1) | NO20015362D0 (no) |
PL (1) | PL351558A1 (no) |
PT (1) | PT1177178E (no) |
SK (1) | SK15962001A3 (no) |
TR (1) | TR200103221T2 (no) |
UA (1) | UA68436C2 (no) |
WO (1) | WO2000068206A1 (no) |
ZA (1) | ZA200108609B (no) |
Families Citing this family (78)
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DE59911249D1 (de) | 1998-11-03 | 2005-01-13 | Abbott Gmbh & Co Kg | Substituierte 2-phenylbenzimidazole, deren herstellung und anwendung |
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RU2003127367A (ru) | 2001-03-12 | 2005-03-20 | Аванир Фармасьютиклз (Us) | Бензимидазоловые соединения для модулирования ige и ингибирования клеточной пролиферации |
US6716866B2 (en) | 2001-06-13 | 2004-04-06 | Genesoft Pharmaceuticals, Inc. | Aryl-benzimidazole compounds having antiinfective activity |
US7642278B2 (en) | 2001-07-03 | 2010-01-05 | Novartis Vaccines And Diagnostics, Inc. | Indazole benzimidazole compounds |
JP2004536113A (ja) | 2001-07-03 | 2004-12-02 | カイロン コーポレイション | チロシンキナーゼおよびセリン/スレオニンキナーゼのインヒビターとしてのインダゾールベンズイミダゾール化合物 |
AU2003215087B2 (en) * | 2002-02-06 | 2009-07-16 | Vertex Pharmaceuticals Incorporated | Heteroaryl compounds useful as inhibitors of GSK-3 |
DE10227668A1 (de) * | 2002-06-20 | 2004-01-08 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Arzneimittel zur Behandlung des systemic inflammatory response syndrome |
US7786344B2 (en) | 2002-07-26 | 2010-08-31 | Basf Plant Science Gmbh | Selection method |
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WO2004024655A2 (en) | 2002-09-12 | 2004-03-25 | Avanir Pharmaceuticals | Phenyl-indole compounds for modulating ige and inhibiting cellular proliferation |
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WO2004039318A2 (en) | 2002-10-25 | 2004-05-13 | Genesoft Pharmaceuticals, Inc. | Anti-infective biaryl compounds |
TW200412959A (en) | 2002-11-22 | 2004-08-01 | Mitsubishi Pharma Corp | Isoquinoline compounds and medicinal use thereof |
JP2006509027A (ja) | 2002-12-10 | 2006-03-16 | オーシェント ファーマシューティカルズ コーポレーション | (ピロールカルボキサミド)−(ベンズアミド)−(イミダゾールカルボキサミド)モチーフを有する抗菌化合物 |
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BRPI0414918A (pt) * | 2003-09-30 | 2006-11-07 | Janssen Pharmaceutica Nv | compostos de benzoimidazola |
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CN104140426B (zh) * | 2013-05-07 | 2017-02-01 | 上海汇伦生命科技有限公司 | 嘧啶并咪唑类化合物、其药物组合物及其制备方法和用途 |
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ZA885929B (en) * | 1987-08-25 | 1989-04-26 | Oxi Gene Inc | Agents for use in tumor or cancer cell killing therapy |
ES2183004T3 (es) * | 1995-08-02 | 2003-03-16 | Univ Newcastle Ventures Ltd | Compuestos de benzimidazol. |
AU3102697A (en) * | 1996-06-19 | 1998-01-07 | Rhone-Poulenc Rorer Limited | Substituted azabicylic compounds and their use as inhibitors of the production of tnf and cyclic amp phosphodiesterase |
DE59911249D1 (de) * | 1998-11-03 | 2005-01-13 | Abbott Gmbh & Co Kg | Substituierte 2-phenylbenzimidazole, deren herstellung und anwendung |
SK6742001A3 (en) * | 1998-11-17 | 2001-12-03 | Basf Ag | 2-phenylbenzimidazoles and 2-phenylindoles, and production and use thereof |
PT1133477E (pt) * | 1998-11-27 | 2004-06-30 | Abbott Gmbh & Co Kg | Benzimidazois substituidos e a utilizacao dos mesmos como inibidores da parp |
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1999
- 1999-05-07 DE DE19920936A patent/DE19920936A1/de not_active Withdrawn
-
2000
- 2000-04-27 HU HU0202970A patent/HUP0202970A2/hu unknown
- 2000-04-27 IL IL14614700A patent/IL146147A0/xx unknown
- 2000-04-27 EP EP00927088A patent/EP1177178B1/de not_active Expired - Lifetime
- 2000-04-27 BR BR0010342-0A patent/BR0010342A/pt not_active IP Right Cessation
- 2000-04-27 AT AT00927088T patent/ATE286029T1/de active
- 2000-04-27 WO PCT/EP2000/003813 patent/WO2000068206A1/de not_active Application Discontinuation
- 2000-04-27 ES ES00927088T patent/ES2235869T3/es not_active Expired - Lifetime
- 2000-04-27 KR KR1020017014145A patent/KR20010112477A/ko not_active Application Discontinuation
- 2000-04-27 DE DE50009118T patent/DE50009118D1/de not_active Expired - Lifetime
- 2000-04-27 DK DK00927088T patent/DK1177178T3/da active
- 2000-04-27 PL PL00351558A patent/PL351558A1/xx not_active Application Discontinuation
- 2000-04-27 US US09/959,632 patent/US6696437B1/en not_active Expired - Lifetime
- 2000-04-27 TR TR2001/03221T patent/TR200103221T2/xx unknown
- 2000-04-27 CA CA002371645A patent/CA2371645C/en not_active Expired - Fee Related
- 2000-04-27 PT PT00927088T patent/PT1177178E/pt unknown
- 2000-04-27 JP JP2000617186A patent/JP4004737B2/ja not_active Expired - Fee Related
- 2000-04-27 SK SK1596-2001A patent/SK15962001A3/sk unknown
- 2000-04-27 AU AU45584/00A patent/AU4558400A/en not_active Abandoned
- 2000-04-27 UA UA2001128419A patent/UA68436C2/uk unknown
- 2000-04-27 CN CN00808364A patent/CN1353695A/zh active Pending
- 2000-05-05 MY MYPI20001934A patent/MY122771A/en unknown
- 2000-05-05 AR ARP000102178A patent/AR029161A1/es unknown
- 2000-05-05 CO CO00032472A patent/CO5170517A1/es not_active Application Discontinuation
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2001
- 2001-10-19 ZA ZA200108609A patent/ZA200108609B/en unknown
- 2001-10-22 BG BG106035A patent/BG106035A/xx unknown
- 2001-11-02 NO NO20015362A patent/NO20015362D0/no not_active Application Discontinuation
-
2002
- 2002-10-30 HK HK02107871.7A patent/HK1046281A1/zh unknown
Also Published As
Publication number | Publication date |
---|---|
HK1046281A1 (zh) | 2003-01-03 |
WO2000068206A1 (de) | 2000-11-16 |
AR029161A1 (es) | 2003-06-18 |
UA68436C2 (en) | 2004-08-16 |
HUP0202970A2 (hu) | 2002-12-28 |
PL351558A1 (en) | 2003-05-05 |
ATE286029T1 (de) | 2005-01-15 |
JP2002544199A (ja) | 2002-12-24 |
AU4558400A (en) | 2000-11-21 |
JP4004737B2 (ja) | 2007-11-07 |
CN1353695A (zh) | 2002-06-12 |
BR0010342A (pt) | 2002-05-28 |
KR20010112477A (ko) | 2001-12-20 |
DK1177178T3 (da) | 2005-05-02 |
CA2371645A1 (en) | 2000-11-16 |
CO5170517A1 (es) | 2002-06-27 |
MY122771A (en) | 2006-05-31 |
TR200103221T2 (tr) | 2002-04-22 |
NO20015362D0 (no) | 2001-11-02 |
DE50009118D1 (de) | 2005-02-03 |
SK15962001A3 (sk) | 2002-06-04 |
ES2235869T3 (es) | 2005-07-16 |
EP1177178A1 (de) | 2002-02-06 |
DE19920936A1 (de) | 2000-11-09 |
CA2371645C (en) | 2007-04-17 |
IL146147A0 (en) | 2002-07-25 |
US6696437B1 (en) | 2004-02-24 |
EP1177178B1 (de) | 2004-12-29 |
ZA200108609B (en) | 2002-10-21 |
PT1177178E (pt) | 2005-05-31 |
BG106035A (en) | 2002-06-28 |
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