NL187116B - Werkwijze voor het bereiden van delta15-steroiden, werkwijze voor het bereiden of vervaardigen van een geneesmiddel met gestagene werking en gevormd geneesmiddel. - Google Patents
Werkwijze voor het bereiden van delta15-steroiden, werkwijze voor het bereiden of vervaardigen van een geneesmiddel met gestagene werking en gevormd geneesmiddel.Info
- Publication number
- NL187116B NL187116B NLAANVRAGE7611073,A NL7611073A NL187116B NL 187116 B NL187116 B NL 187116B NL 7611073 A NL7611073 A NL 7611073A NL 187116 B NL187116 B NL 187116B
- Authority
- NL
- Netherlands
- Prior art keywords
- preparing
- medicinal product
- steroids
- manufacturing
- molded
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0051—Estrane derivatives
- C07J1/0081—Substituted in position 17 alfa and 17 beta
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0051—Estrane derivatives
- C07J1/0081—Substituted in position 17 alfa and 17 beta
- C07J1/0088—Substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being an unsaturated hydrocarbon group
- C07J1/0096—Alkynyl derivatives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
- C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
- C07J41/0016—Oximes
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J51/00—Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 - C07J43/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19752546062 DE2546062A1 (de) | 1975-10-10 | 1975-10-10 | Delta hoch 15 -steroide |
DE19762636404 DE2636404C2 (de) | 1976-08-12 | 1976-08-12 | Δ↑1↑↑5↑-17α-Äthinylsteroide der Östranreihe, Verfahren zu ihrer Herstellung sowie diese enthaltende pharmazeutische Präparate |
DE19762636407 DE2636407A1 (de) | 1976-08-12 | 1976-08-12 | Delta hoch 15 -steroide |
DE19762636405 DE2636405C2 (de) | 1976-08-12 | 1976-08-12 | Δ↑1↑↑5↑-17α-Chloräthinyl- und -Propinylsteroide der Östranreihe, Verfahren zu ihrer Herstellung sowie diese enthaltende pharmazeutische Präparate |
Publications (3)
Publication Number | Publication Date |
---|---|
NL7611073A NL7611073A (nl) | 1977-04-13 |
NL187116B true NL187116B (nl) | 1991-01-02 |
NL187116C NL187116C (nl) | 1991-06-03 |
Family
ID=27432034
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NLAANVRAGE7611073,A NL187116C (nl) | 1975-10-10 | 1976-10-07 | Werkwijze voor het bereiden van delta15-steroiden, werkwijze voor het bereiden of vervaardigen van een geneesmiddel met gestagene werking en gevormd geneesmiddel. |
NL930071C NL930071I2 (nl) | 1975-10-10 | 1993-06-14 | Werkwijze voor het bereiden van delta 15-steroiden, werkwijze voor het bereiden of vervaardigen van een geneesmiddel met gestagene werking en gevormd geneesmiddel. |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NL930071C NL930071I2 (nl) | 1975-10-10 | 1993-06-14 | Werkwijze voor het bereiden van delta 15-steroiden, werkwijze voor het bereiden of vervaardigen van een geneesmiddel met gestagene werking en gevormd geneesmiddel. |
Country Status (33)
Country | Link |
---|---|
US (1) | US4081537A (nl) |
JP (1) | JPS5246060A (nl) |
AT (1) | AT358199B (nl) |
AU (1) | AU500942B2 (nl) |
BE (1) | BE847090A (nl) |
BG (1) | BG34187A3 (nl) |
CA (1) | CA1069885A (nl) |
CH (2) | CH630392A5 (nl) |
CY (1) | CY1119A (nl) |
DD (1) | DD126925B3 (nl) |
DK (2) | DK138749C (nl) |
ES (1) | ES452226A1 (nl) |
FI (1) | FI56389C (nl) |
FR (1) | FR2326927A1 (nl) |
GB (1) | GB1569135A (nl) |
GR (1) | GR60835B (nl) |
HK (1) | HK41381A (nl) |
HU (1) | HU176164B (nl) |
IE (1) | IE43742B1 (nl) |
IT (1) | IT1070580B (nl) |
KE (1) | KE3153A (nl) |
LU (2) | LU75961A1 (nl) |
MX (1) | MX3847E (nl) |
MY (1) | MY8200128A (nl) |
NL (2) | NL187116C (nl) |
NO (2) | NO144490C (nl) |
NZ (1) | NZ182237A (nl) |
PH (1) | PH12941A (nl) |
PL (1) | PL103002B1 (nl) |
PT (1) | PT65697B (nl) |
SE (2) | SE415839B (nl) |
SU (1) | SU671733A3 (nl) |
YU (1) | YU39668B (nl) |
Families Citing this family (20)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3178784A (en) * | 1963-03-27 | 1965-04-20 | Krauthamer Charles | Magnetic pocket pencil holder |
DE3002746A1 (de) * | 1980-01-23 | 1981-07-30 | Schering Ag Berlin Und Bergkamen, 1000 Berlin | 1-hydroxysteroide, verfahren zu ihrer herstellung und pharmazeutische praeparate, die diese verbindungen enthalten |
DE3005374A1 (de) * | 1980-02-11 | 1981-08-20 | Schering Ag Berlin Und Bergkamen, 1000 Berlin | 3-desoxy-delta hoch 15 -steroide, verfahren zu ihrer herstellung sowie diese enthaltende pharmazeutische praeparate |
DE3042529A1 (de) * | 1980-11-07 | 1982-06-24 | Schering Ag, 1000 Berlin Und 4619 Bergkamen | 11-methylen- (delta)(pfeil hoch)1(pfeil hoch)(pfeil hoch)5(pfeil hoch) -steroide, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische praeparate |
DE3214690A1 (de) * | 1982-04-16 | 1983-10-27 | Schering AG, 1000 Berlin und 4709 Bergkamen | 11ss-chlor-(delta)(pfeil hoch)1(pfeil hoch)(pfeil hoch)5(pfeil hoch)-steroide, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische praeparate |
CN1008820B (zh) * | 1985-05-10 | 1990-07-18 | 施林工业产权保护股份公司 | 17α-乙炔基-17β-羟基-18-甲基-4,15-雌甾二烯-3-酮的制备方法 |
CA1317283C (en) * | 1986-11-05 | 1993-05-04 | Douglas Alan Livingston | Steroidal 17-silyl ethers and process to corticoids and progesterones |
DE3710728A1 (de) * | 1987-03-31 | 1988-10-13 | Schering Ag | Verfahren zur herstellung von 17(alpha)-ethinyl-17ss-hydroxy-18-methyl-4,15-estradien-3-on und die neuen zwischenprodukte fuer dieses verfahren |
PT99338A (pt) * | 1990-10-29 | 1992-10-30 | Alza Corp | Processo para a preparacao de composicoes de farmacos anticoncepcionais administradas transdermicamente contendo uma mistura dum estrogeno e gestodeno e dispositivos para a sua administracao transdermica |
US5512292A (en) * | 1990-10-29 | 1996-04-30 | Alza Corporation | Transdermal contraceptive formulations methods and devices |
CA2100514C (en) * | 1992-07-29 | 2005-03-29 | Johannes A. M. Hamersma | 17-spiromethylene steroids |
DE4329242A1 (de) * | 1993-08-26 | 1995-03-02 | Schering Ag | Mittel zur transdermalen Applikation enthaltend Gestodenester |
US5567830A (en) * | 1994-02-14 | 1996-10-22 | Cocensys, Inc. | Process for synthesis of acetylenic carbinols |
IT1271004B (it) * | 1994-09-09 | 1997-05-26 | Ind Chimica Srl | Processo per la preparazione del gestodene |
WO2002062391A2 (en) * | 2001-02-02 | 2002-08-15 | Pharmacia Corporation | Method of using a cyclooxygenase-2 inhibitor and sex steroids as a combination therapy for the treatment and prevention of dismenorrhea |
UA89766C2 (en) | 2003-12-12 | 2010-03-10 | Байер Шеринг Фарма Акциенгезельшафт | Transdermal delivery system of gestodene |
EP2354150A1 (en) | 2010-02-09 | 2011-08-10 | Laboratoire Theramex | Process for the preparation of gestodene |
HUE031326T2 (hu) | 2010-09-06 | 2017-07-28 | Bayer Ip Gmbh | Alacsony dózisú transzdermális tapaszok magas hatóanyagleadással |
CN105237605B (zh) * | 2014-07-11 | 2019-01-25 | 上海迪赛诺生物医药有限公司 | 一种用于合成孕二烯酮的中间体及其制备方法和应用 |
CN115850359B (zh) * | 2022-12-14 | 2024-06-11 | 梯尔希(南京)药物研发有限公司 | 一种孕二烯酮杂质i的制备方法 |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3433785A (en) * | 1966-07-11 | 1969-03-18 | Sterling Drug Inc | 15,16-disubstituted aromatic steroids,intermediates and processes |
US3475463A (en) * | 1966-07-11 | 1969-10-28 | Sterling Drug Inc | 15,16-unsaturated 19-norsteroids and their preparation |
DE2439082A1 (de) * | 1974-08-12 | 1976-02-26 | Schering Ag | 17 alpha-hydroxy-1,3,5(10),15-oestratetraene und verfahren zu ihrer herstellung |
-
1976
- 1976-10-04 US US05/728,896 patent/US4081537A/en not_active Expired - Lifetime
- 1976-10-05 IT IT27981/76A patent/IT1070580B/it active
- 1976-10-05 BG BG7634359A patent/BG34187A3/xx unknown
- 1976-10-05 NZ NZ182237A patent/NZ182237A/xx unknown
- 1976-10-06 MX MX764963U patent/MX3847E/es unknown
- 1976-10-06 DD DD76195196A patent/DD126925B3/de unknown
- 1976-10-06 YU YU2452/76A patent/YU39668B/xx unknown
- 1976-10-07 SE SE7611145A patent/SE415839B/xx not_active IP Right Cessation
- 1976-10-07 NL NLAANVRAGE7611073,A patent/NL187116C/nl not_active IP Right Cessation
- 1976-10-07 CH CH1272376A patent/CH630392A5/de active Protection Beyond IP Right Term
- 1976-10-08 CA CA263,032A patent/CA1069885A/en not_active Expired
- 1976-10-08 BE BE171353A patent/BE847090A/xx active Protection Beyond IP Right Term
- 1976-10-08 SU SU762407731A patent/SU671733A3/ru active
- 1976-10-08 NO NO763434A patent/NO144490C/no unknown
- 1976-10-08 DK DK454376A patent/DK138749C/da not_active IP Right Cessation
- 1976-10-08 LU LU75961A patent/LU75961A1/xx unknown
- 1976-10-08 FI FI762876A patent/FI56389C/fi not_active IP Right Cessation
- 1976-10-08 PH PH18991A patent/PH12941A/en unknown
- 1976-10-08 AT AT748776A patent/AT358199B/de not_active IP Right Cessation
- 1976-10-08 IE IE2225/76A patent/IE43742B1/en not_active IP Right Cessation
- 1976-10-08 ES ES452226A patent/ES452226A1/es not_active Expired
- 1976-10-08 PT PT65697A patent/PT65697B/pt unknown
- 1976-10-08 AU AU18510/76A patent/AU500942B2/en not_active Expired
- 1976-10-08 PL PL1976192908A patent/PL103002B1/pl unknown
- 1976-10-08 HU HU76SCHE580A patent/HU176164B/hu unknown
- 1976-10-09 GR GR51898A patent/GR60835B/el unknown
- 1976-10-11 GB GB42124/76A patent/GB1569135A/en not_active Expired
- 1976-10-11 CY CY1119A patent/CY1119A/xx unknown
- 1976-10-11 FR FR7630492A patent/FR2326927A1/fr active Granted
- 1976-10-12 JP JP51122203A patent/JPS5246060A/ja active Granted
-
1978
- 1978-02-21 DK DK77678A patent/DK143604C/da not_active IP Right Cessation
-
1979
- 1979-08-30 SE SE7907224A patent/SE428929B/sv not_active IP Right Cessation
-
1980
- 1980-04-09 NO NO801013A patent/NO144967C/no unknown
- 1980-12-03 CH CH894080A patent/CH626636A5/de not_active IP Right Cessation
-
1981
- 1981-08-12 KE KE3153A patent/KE3153A/xx unknown
- 1981-08-20 HK HK413/81A patent/HK41381A/xx unknown
-
1982
- 1982-12-30 MY MY128/82A patent/MY8200128A/xx unknown
-
1993
- 1993-06-09 LU LU88290C patent/LU88290I2/de unknown
- 1993-06-14 NL NL930071C patent/NL930071I2/nl unknown
Also Published As
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
BA | A request for search or an international-type search has been filed | ||
BB | A search report has been drawn up | ||
BC | A request for examination has been filed | ||
A85 | Still pending on 85-01-01 | ||
BK | Erratum |
Free format text: CORRECTION TO PAMPHLET |
|
AC1 | Application for a supplementary protection certificate |
Free format text: 930071, 930614 |
|
KC1 | Grant of a supplementary protection certificate |
Free format text: 930071, 961007, EXPIRES:20010721 |
|
AC1 | Application for a supplementary protection certificate |
Free format text: 930071, 930614 |
|
V4 | Discontinued because of reaching the maximum lifetime of a patent |
Free format text: 961007 |