DK454376A - Delta 15-steroider - Google Patents

Delta 15-steroider

Info

Publication number: DK454376A
Authority: DK; Denmark
Prior art keywords: steroider; delta
Prior art date: 1975-10-10

Application number

DK454376A

Other languages

English (en)

Other versions

DK138749C (da

DK138749B (da

Inventor

H Hofmeister

R Wiechert

K Annen

H Laurent

H Steinbeck

Original Assignee

Schering Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1975-10-10

Filing date

1976-10-08

Publication date

1977-04-11

1975-10-10 Priority claimed from DE19752546062 external-priority patent/DE2546062A1/de

1976-08-12 Priority claimed from DE19762636405 external-priority patent/DE2636405C2/de

1976-08-12 Priority claimed from DE19762636407 external-priority patent/DE2636407A1/de

1976-08-12 Priority claimed from DE19762636404 external-priority patent/DE2636404C2/de

1976-10-08 Application filed by Schering Ag filed Critical Schering Ag

1977-04-11 Publication of DK454376A publication Critical patent/DK454376A/da

1978-02-21 Priority to DK77678A priority Critical patent/DK143604C/da

1978-10-23 Publication of DK138749B publication Critical patent/DK138749B/da

1979-04-02 Application granted granted Critical

1979-04-02 Publication of DK138749C publication Critical patent/DK138749C/da

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0051—Estrane derivatives
- C07J1/0081—Substituted in position 17 alfa and 17 beta
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0051—Estrane derivatives
- C07J1/0081—Substituted in position 17 alfa and 17 beta
- C07J1/0088—Substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being an unsaturated hydrocarbon group
- C07J1/0096—Alkynyl derivatives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
- C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
- C07J41/0016—Oximes
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J51/00—Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 - C07J43/00

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Steroid Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

DK454376A 1975-10-10 1976-10-08 Analogifremgangsmaade til fremstilling af 18-methyl-4,15-oestradiener DK138749C (da)

Priority Applications (1)

Application Number	Priority Date	Filing Date	Title
DK77678A DK143604C (da)	1975-10-10	1978-02-21	18-methyl-4,15-oestradiener til anvendelse i svangerskabsforebyggende midler

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
DE19752546062 DE2546062A1 (de)	1975-10-10	1975-10-10	Delta hoch 15 -steroide
DE19762636405 DE2636405C2 (de)	1976-08-12	1976-08-12	Δ↑1↑↑5↑-17α-Chloräthinyl- und -Propinylsteroide der Östranreihe, Verfahren zu ihrer Herstellung sowie diese enthaltende pharmazeutische Präparate
DE19762636407 DE2636407A1 (de)	1976-08-12	1976-08-12	Delta hoch 15 -steroide
DE19762636404 DE2636404C2 (de)	1976-08-12	1976-08-12	Δ↑1↑↑5↑-17α-Äthinylsteroide der Östranreihe, Verfahren zu ihrer Herstellung sowie diese enthaltende pharmazeutische Präparate

Publications (3)

Publication Number	Publication Date
DK454376A true DK454376A (da)	1977-04-11
DK138749B DK138749B (da)	1978-10-23
DK138749C DK138749C (da)	1979-04-02

Family

ID=27432034

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
DK454376A DK138749C (da)	1975-10-10	1976-10-08	Analogifremgangsmaade til fremstilling af 18-methyl-4,15-oestradiener
DK77678A DK143604C (da)	1975-10-10	1978-02-21	18-methyl-4,15-oestradiener til anvendelse i svangerskabsforebyggende midler

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
DK77678A DK143604C (da)	1975-10-10	1978-02-21	18-methyl-4,15-oestradiener til anvendelse i svangerskabsforebyggende midler

Country Status (33)

Country	Link
US (1)	US4081537A (da)
JP (1)	JPS5246060A (da)
AT (1)	AT358199B (da)
AU (1)	AU500942B2 (da)
BE (1)	BE847090A (da)
BG (1)	BG34187A3 (da)
CA (1)	CA1069885A (da)
CH (2)	CH630392A5 (da)
CY (1)	CY1119A (da)
DD (1)	DD126925B3 (da)
DK (2)	DK138749C (da)
ES (1)	ES452226A1 (da)
FI (1)	FI56389C (da)
FR (1)	FR2326927A1 (da)
GB (1)	GB1569135A (da)
GR (1)	GR60835B (da)
HK (1)	HK41381A (da)
HU (1)	HU176164B (da)
IE (1)	IE43742B1 (da)
IT (1)	IT1070580B (da)
KE (1)	KE3153A (da)
LU (2)	LU75961A1 (da)
MX (1)	MX3847E (da)
MY (1)	MY8200128A (da)
NL (2)	NL187116C (da)
NO (2)	NO144490C (da)
NZ (1)	NZ182237A (da)
PH (1)	PH12941A (da)
PL (1)	PL103002B1 (da)
PT (1)	PT65697B (da)
SE (2)	SE415839B (da)
SU (1)	SU671733A3 (da)
YU (1)	YU39668B (da)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3178784A (en) *	1963-03-27	1965-04-20	Krauthamer Charles	Magnetic pocket pencil holder
DE3002746A1 (de) *	1980-01-23	1981-07-30	Schering Ag Berlin Und Bergkamen, 1000 Berlin	1-hydroxysteroide, verfahren zu ihrer herstellung und pharmazeutische praeparate, die diese verbindungen enthalten
DE3005374A1 (de) *	1980-02-11	1981-08-20	Schering Ag Berlin Und Bergkamen, 1000 Berlin	3-desoxy-delta hoch 15 -steroide, verfahren zu ihrer herstellung sowie diese enthaltende pharmazeutische praeparate
DE3042529A1 (de) *	1980-11-07	1982-06-24	Schering Ag, 1000 Berlin Und 4619 Bergkamen	11-methylen- (delta)(pfeil hoch)1(pfeil hoch)(pfeil hoch)5(pfeil hoch) -steroide, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische praeparate
DE3214690A1 (de) *	1982-04-16	1983-10-27	Schering AG, 1000 Berlin und 4709 Bergkamen	11ss-chlor-(delta)(pfeil hoch)1(pfeil hoch)(pfeil hoch)5(pfeil hoch)-steroide, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische praeparate
CN1008820B (zh) *	1985-05-10	1990-07-18	施林工业产权保护股份公司	17α-乙炔基-17β-羟基-18-甲基-4，15-雌甾二烯-3-酮的制备方法
CA1317283C (en) *	1986-11-05	1993-05-04	Douglas Alan Livingston	Steroidal 17-silyl ethers and process to corticoids and progesterones
DE3710728A1 (de) *	1987-03-31	1988-10-13	Schering Ag	Verfahren zur herstellung von 17(alpha)-ethinyl-17ss-hydroxy-18-methyl-4,15-estradien-3-on und die neuen zwischenprodukte fuer dieses verfahren
CA2091883A1 (en) *	1990-10-29	1992-04-30	Robert M. Gale	Transdermal contraceptive formulations, methods and devices
US5512292A (en) *	1990-10-29	1996-04-30	Alza Corporation	Transdermal contraceptive formulations methods and devices
CA2100514C (en) *	1992-07-29	2005-03-29	Johannes A. M. Hamersma	17-spiromethylene steroids
DE4329242A1 (de) *	1993-08-26	1995-03-02	Schering Ag	Mittel zur transdermalen Applikation enthaltend Gestodenester
US5567830A (en) *	1994-02-14	1996-10-22	Cocensys, Inc.	Process for synthesis of acetylenic carbinols
IT1271004B (it) *	1994-09-09	1997-05-26	Ind Chimica Srl	Processo per la preparazione del gestodene
US20050143360A1 (en) *	2001-02-02	2005-06-30	Joel Krasnow	Method of using a cyclooxygenase-2 inhibitor and sex steroids as a combination therapy for the treatment and prevention of dismenorrhea
UA89766C2 (en)	2003-12-12	2010-03-10	Байер Шеринг Фарма Акциенгезельшафт	Transdermal delivery system of gestodene
EP2354150A1 (en)	2010-02-09	2011-08-10	Laboratoire Theramex	Process for the preparation of gestodene
ME02618B (me)	2010-09-06	2017-06-20	Bayer Ip Gmbh	Transdermalni flasteri sa malom dozom i velikim oslobađanjem leka
CN105237605B (zh) *	2014-07-11	2019-01-25	上海迪赛诺生物医药有限公司	一种用于合成孕二烯酮的中间体及其制备方法和应用
CN115850359B (zh) *	2022-12-14	2024-06-11	梯尔希（南京）药物研发有限公司	一种孕二烯酮杂质i的制备方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3433785A (en) *	1966-07-11	1969-03-18	Sterling Drug Inc	15,16-disubstituted aromatic steroids,intermediates and processes
US3475463A (en) *	1966-07-11	1969-10-28	Sterling Drug Inc	15,16-unsaturated 19-norsteroids and their preparation
DE2439082A1 (de) *	1974-08-12	1976-02-26	Schering Ag	17 alpha-hydroxy-1,3,5(10),15-oestratetraene und verfahren zu ihrer herstellung

1976
- 1976-10-04 US US05/728,896 patent/US4081537A/en not_active Expired - Lifetime
- 1976-10-05 IT IT27981/76A patent/IT1070580B/it active
- 1976-10-05 NZ NZ182237A patent/NZ182237A/xx unknown
- 1976-10-05 BG BG7634359A patent/BG34187A3/xx unknown
- 1976-10-06 MX MX764963U patent/MX3847E/es unknown
- 1976-10-06 DD DD76195196A patent/DD126925B3/de unknown
- 1976-10-06 YU YU2452/76A patent/YU39668B/xx unknown
- 1976-10-07 CH CH1272376A patent/CH630392A5/de active Protection Beyond IP Right Term
- 1976-10-07 SE SE7611145A patent/SE415839B/xx not_active IP Right Cessation
- 1976-10-07 NL NLAANVRAGE7611073,A patent/NL187116C/xx not_active IP Right Cessation
- 1976-10-08 PL PL1976192908A patent/PL103002B1/pl unknown
- 1976-10-08 NO NO763434A patent/NO144490C/no unknown
- 1976-10-08 PT PT65697A patent/PT65697B/pt unknown
- 1976-10-08 IE IE2225/76A patent/IE43742B1/en not_active IP Right Cessation
- 1976-10-08 HU HU76SCHE580A patent/HU176164B/hu unknown
- 1976-10-08 PH PH18991A patent/PH12941A/en unknown
- 1976-10-08 SU SU762407731A patent/SU671733A3/ru active
- 1976-10-08 AT AT748776A patent/AT358199B/de not_active IP Right Cessation
- 1976-10-08 BE BE171353A patent/BE847090A/xx active Protection Beyond IP Right Term
- 1976-10-08 FI FI762876A patent/FI56389C/fi not_active IP Right Cessation
- 1976-10-08 AU AU18510/76A patent/AU500942B2/en not_active Expired
- 1976-10-08 DK DK454376A patent/DK138749C/da not_active IP Right Cessation
- 1976-10-08 CA CA263,032A patent/CA1069885A/en not_active Expired
- 1976-10-08 ES ES452226A patent/ES452226A1/es not_active Expired
- 1976-10-08 LU LU75961A patent/LU75961A1/xx unknown
- 1976-10-09 GR GR51898A patent/GR60835B/el unknown
- 1976-10-11 CY CY1119A patent/CY1119A/xx unknown
- 1976-10-11 FR FR7630492A patent/FR2326927A1/fr active Granted
- 1976-10-11 GB GB42124/76A patent/GB1569135A/en not_active Expired
- 1976-10-12 JP JP51122203A patent/JPS5246060A/ja active Granted
1978
- 1978-02-21 DK DK77678A patent/DK143604C/da not_active IP Right Cessation
1979
- 1979-08-30 SE SE7907224A patent/SE428929B/sv not_active IP Right Cessation
1980
- 1980-04-09 NO NO801013A patent/NO144967C/no unknown
- 1980-12-03 CH CH894080A patent/CH626636A5/de not_active IP Right Cessation
1981
- 1981-08-12 KE KE3153A patent/KE3153A/xx unknown
- 1981-08-20 HK HK413/81A patent/HK41381A/xx unknown
1982
- 1982-12-30 MY MY128/82A patent/MY8200128A/xx unknown
1993
- 1993-06-09 LU LU88290C patent/LU88290I2/de unknown
- 1993-06-14 NL NL930071C patent/NL930071I2/nl unknown

Also Published As

Publication number	Publication date
CH626636A5 (en)	1981-11-30
HK41381A (en)	1981-08-28
PT65697B (pt)	1978-04-17
NZ182237A (en)	1978-09-20
NL187116B (nl)	1991-01-02
KE3153A (en)	1981-09-18
MX3847E (es)	1981-08-18
ES452226A1 (es)	1977-11-01
DD126925B3 (de)	1990-06-06
JPS6119640B2 (da)	1986-05-17
PH12941A (en)	1979-10-18
FI56389B (fi)	1979-09-28
FR2326927A1 (fr)	1977-05-06
LU75961A1 (da)	1977-05-09
AT358199B (de)	1980-08-25
DK77678A (da)	1978-02-21
DK138749C (da)	1979-04-02
LU88290I2 (de)	1994-05-04
DD126925A5 (da)	1977-08-24
SE415839B (sv)	1980-11-03
AU500942B2 (en)	1979-06-07
DK138749B (da)	1978-10-23
CY1119A (en)	1981-12-04
MY8200128A (en)	1982-12-31
JPS5246060A (en)	1977-04-12
ATA748776A (de)	1980-01-15
NO144490C (no)	1981-09-09
GB1569135A (en)	1980-06-11
NO801013L (no)	1977-04-13
FR2326927B1 (da)	1979-09-28
GR60835B (en)	1978-08-31
NO763434L (da)	1977-04-13
DK143604B (da)	1981-09-14
NL187116C (nl)	1991-06-03
SE7611145L (sv)	1977-04-11
PT65697A (en)	1976-11-01
CH630392A5 (de)	1982-06-15
IE43742L (en)	1977-04-10
BG34187A3 (en)	1983-07-15
PL103002B1 (pl)	1979-05-31
NO144967B (no)	1981-09-07
BE847090A (fr)	1977-04-08
YU245276A (en)	1982-08-31
SU671733A3 (ru)	1979-06-30
CA1069885A (en)	1980-01-15
AU1851076A (en)	1978-04-13
US4081537A (en)	1978-03-28
IT1070580B (it)	1985-03-29
NL930071I2 (nl)	1994-02-16
FI56389C (fi)	1980-01-10
FI762876A (da)	1977-04-11
SE7907224L (sv)	1979-08-30
SE428929B (sv)	1983-08-01
NL930071I1 (nl)	1993-09-01
DK143604C (da)	1982-02-22
NL7611073A (nl)	1977-04-13
NO144967C (no)	1981-12-16
IE43742B1 (en)	1981-05-20
YU39668B (en)	1985-03-20
HU176164B (en)	1980-12-28
NO144490B (no)	1981-06-01

Legal Events

Date	Code	Title	Description
1996-11-11	PUP	Patent expired

Publication	Publication Date	Title
AR214181A1 (es)	1979-05-15	Hemodializador
DK454376A (da)	1977-04-11	Delta 15-steroider
AT344259B (de)	1978-07-10	Ablenkjoch
AT361361B (de)	1981-03-10	Skiroller
AT349233B (de)	1979-03-26	Mikroskopokular
JPS51106458A (ja)	1976-09-21	Futatsunotaishobutsunoaitaiichiosokuteishitari*aruihachoseishitarisurutamenosokuchosochi
AT359544B (de)	1980-11-10	Randstreifenfertiger
AT341259B (de)	1978-01-25	Schmiegeegge
JPS51100054A (ja)	1976-09-03	Shokubaisansakanju1*55jimechirutetorarinyorikaisansaojokyosuruhoho
AT362274B (de)	1981-04-27	Skistock
AT346618B (de)	1978-11-27	Mikroskopokular
AT351347B (de)	1979-07-25	Siliermittel
AT348103B (de)	1979-01-25	Dentallot
JPS51102157A (ja)	1976-09-09	Tasunotairanabutsutai*tokunitateitokanshibanobunruisurutamenohohooyobidohohoojitsushisurutamenokeiretsu
JPS51110544A (ja)	1976-09-30	Eoyobifretsunoshinkino111deokishiichikanpurosutaguranjinruikagobutsusonorasemikagobutsukyozotaioyobisonoen
JPS51105331A (ja)	1976-09-17	Azosenryosonoseizohohooyobigoseihorimaazairyoosenshokusuruhoho
JPS51105026A (ja)	1976-09-17	22aminoonnbbhidorokishiifuenechiru*asetoamidoojudotainarabinisonoennoseiho
AT360216B (de)	1980-12-29	Rostmatte
JPS51100390A (ja)	1976-09-04	Setsudantoishi
JPS51102860A (ja)	1976-09-10	Hinjishikihishigatakozonorifuto*jatsuki
JPS51102190A (ja)	1976-09-09	Hannoseisenryo*sonoseizohooyobiseruroosusenizairyonosenshokuho
JPS5186433A (ja)	1976-07-29	Hokozokukarubonsanruioyobi * matahasoreranomechiruesuterunoseiho
JPS51101026A (ja)	1976-09-07	Shinkienkiseiazosenryo*sonoseihooyobisonoshoho
JPS51108851A (ja)	1976-09-27	Hikaridensoyogarasusenino setsudangu
JPS51100721A (ja)	1976-09-06	Shashinkankozaishakopatsuku