MXPA03003246A - Derivados de indolina y su uso como ligandos del receptor 5-ht2. - Google Patents

Derivados de indolina y su uso como ligandos del receptor 5-ht2.

Info

Publication number
MXPA03003246A
MXPA03003246A MXPA03003246A MXPA03003246A MXPA03003246A MX PA03003246 A MXPA03003246 A MX PA03003246A MX PA03003246 A MXPA03003246 A MX PA03003246A MX PA03003246 A MXPA03003246 A MX PA03003246A MX PA03003246 A MXPA03003246 A MX PA03003246A
Authority
MX
Mexico
Prior art keywords
receptor ligands
indoline derivatives
indoline
derivatives
ligands
Prior art date
Application number
MXPA03003246A
Other languages
English (en)
Inventor
Edward Paul Davidson James
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of MXPA03003246A publication Critical patent/MXPA03003246A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56—Ring systems containing three or more rings
    • C07D209/80—[b, c]- or [b, d]-condensed
    • C07D209/94—[b, c]- or [b, d]-condensed containing carbocyclic rings other than six-membered
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Endocrinology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
MXPA03003246A 2000-10-16 2001-10-12 Derivados de indolina y su uso como ligandos del receptor 5-ht2. MXPA03003246A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP00122539 2000-10-16
PCT/EP2001/011814 WO2002044152A1 (en) 2000-10-16 2001-10-12 Indoline derivatives and their use as 5-ht2 receptor ligands

Publications (1)

Publication Number Publication Date
MXPA03003246A true MXPA03003246A (es) 2003-06-06

Family

ID=8170101

Family Applications (1)

Application Number Title Priority Date Filing Date
MXPA03003246A MXPA03003246A (es) 2000-10-16 2001-10-12 Derivados de indolina y su uso como ligandos del receptor 5-ht2.

Country Status (15)

Country Link
US (1) US6479534B1 (es)
EP (1) EP1328515B1 (es)
JP (1) JP4047723B2 (es)
KR (1) KR100545435B1 (es)
CN (1) CN100334076C (es)
AR (1) AR038762A1 (es)
AT (1) ATE403647T1 (es)
AU (2) AU2002221670B2 (es)
BR (1) BR0114708A (es)
CA (1) CA2422698C (es)
DE (1) DE60135239D1 (es)
ES (1) ES2311563T3 (es)
MX (1) MXPA03003246A (es)
WO (1) WO2002044152A1 (es)
ZA (1) ZA200302516B (es)

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Also Published As

Publication number Publication date
JP2004527467A (ja) 2004-09-09
BR0114708A (pt) 2003-07-01
US6479534B1 (en) 2002-11-12
KR20030048437A (ko) 2003-06-19
US20020183349A1 (en) 2002-12-05
DE60135239D1 (de) 2008-09-18
JP4047723B2 (ja) 2008-02-13
WO2002044152A1 (en) 2002-06-06
ES2311563T3 (es) 2009-02-16
AU2167002A (en) 2002-06-11
CN1630636A (zh) 2005-06-22
CA2422698A1 (en) 2002-06-06
AU2002221670B2 (en) 2006-11-02
EP1328515B1 (en) 2008-08-06
ATE403647T1 (de) 2008-08-15
ZA200302516B (en) 2004-06-30
CA2422698C (en) 2009-12-15
AR038762A1 (es) 2005-01-26
EP1328515A1 (en) 2003-07-23
CN100334076C (zh) 2007-08-29
KR100545435B1 (ko) 2006-01-24

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