MX9708611A - Compuestos de dialquiltiacumicina. - Google Patents

Compuestos de dialquiltiacumicina.

Info

Publication number
MX9708611A
MX9708611A MX9708611A MX9708611A MX9708611A MX 9708611 A MX9708611 A MX 9708611A MX 9708611 A MX9708611 A MX 9708611A MX 9708611 A MX9708611 A MX 9708611A MX 9708611 A MX9708611 A MX 9708611A
Authority
MX
Mexico
Prior art keywords
compounds
dialkyltiacumicin
colitis
administration
formula
Prior art date
Application number
MX9708611A
Other languages
English (en)
Other versions
MXPA97008611A (es
Inventor
James B Mcalpine
Jill E Hochlowski
Original Assignee
Abbott Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbott Lab filed Critical Abbott Lab
Publication of MXPA97008611A publication Critical patent/MXPA97008611A/es
Publication of MX9708611A publication Critical patent/MX9708611A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Molecular Biology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Polymerisation Methods In General (AREA)

Abstract

Se describen compuestos que tienen la formula (I) así como composiciones farmacéuticas que comprenden dichos compuestos y métodos para el tratamiento de infeccion causada por bacterias y colitis, a través de la administracion de los mismos.
MX9708611A 1995-05-09 1996-05-02 Compuestos de dialquiltiacumicina. MX9708611A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US08/437,761 US5583115A (en) 1995-05-09 1995-05-09 Dialkyltiacumicin compounds
US08437761 1995-05-09
PCT/US1996/006204 WO1996035702A1 (en) 1995-05-09 1996-05-02 Dialkyltiacumicin compounds

Publications (2)

Publication Number Publication Date
MXPA97008611A MXPA97008611A (es) 1998-02-01
MX9708611A true MX9708611A (es) 1998-02-28

Family

ID=23737769

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9708611A MX9708611A (es) 1995-05-09 1996-05-02 Compuestos de dialquiltiacumicina.

Country Status (12)

Country Link
US (1) US5583115A (es)
EP (1) EP0824539B1 (es)
JP (1) JPH11504937A (es)
AT (1) ATE203246T1 (es)
CA (1) CA2218916A1 (es)
DE (1) DE69613975T2 (es)
DK (1) DK0824539T3 (es)
ES (1) ES2159733T3 (es)
GR (1) GR3036873T3 (es)
MX (1) MX9708611A (es)
PT (1) PT824539E (es)
WO (1) WO1996035702A1 (es)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20070105791A1 (en) * 2002-07-29 2007-05-10 Optimer Pharmaceuticals, Inc. Method of treating clostridium difficile-associated diarrhea
US7906489B2 (en) * 2004-05-14 2011-03-15 Optimer Pharmaceuticals, Inc. 18-membered macrocycles and analogs thereof
BRPI0511119A (pt) * 2004-05-14 2007-11-27 Optimer Pharmaceuticals Inc tratamento de doenças associadas com o uso de antibióticos
CN101128114B (zh) * 2005-01-31 2012-03-28 浩鼎生技公司 18元环大环化合物及其类似物
US7378508B2 (en) * 2007-01-22 2008-05-27 Optimer Pharmaceuticals, Inc. Polymorphic crystalline forms of tiacumicin B
EP1940417A4 (en) * 2005-10-21 2010-07-07 Optimer Pharmaceuticals Inc METHOD FOR TREATING DIARRHOE IN CONNECTION WITH CLOSTRIDIUM DIFFICILE
US20080176927A1 (en) * 2007-01-19 2008-07-24 Optimer Pharmaceuticals, Inc. Compositions of stable tiacumicins
ZA200905337B (en) * 2007-01-22 2010-10-27 Optimer Pharmaceuticals Inc Macrocyclic polymorphs, compositions comprising such polymorphs, and methods of use and manufacture thereof
TWI523654B (zh) * 2007-11-27 2016-03-01 默沙東藥廠 抗生素巨環化合物以及其製造及使用之方法
JP5825217B2 (ja) * 2012-07-27 2015-12-02 メルク シャープ アンド ドーム コーポレーションMerck Sharp & Dohme Corp. 18員大環状化合物及びその類似化合物
JO3464B1 (ar) 2013-01-15 2020-07-05 Astellas Pharma Europe Ltd التركيبات الخاصة بمركبات التياكوميسين
TR201815891T4 (tr) 2014-05-09 2018-11-21 Astellas Pharma Europe Ltd Tiakumisin bileşiği için tedavi rejimi.
JP2018519344A (ja) 2015-07-03 2018-07-19 アステラス ファーマ ユーロープ リミテッド チアクマイシン化合物の新規の投薬レジメン
EP3508492A1 (en) * 2018-01-08 2019-07-10 Universität Zürich Tiacumicin derivatives and their use as antibiotics

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4918174A (en) * 1986-09-26 1990-04-17 Abbott Laboratories Tiacumicin compounds

Also Published As

Publication number Publication date
PT824539E (pt) 2002-01-30
DE69613975T2 (de) 2002-04-04
EP0824539B1 (en) 2001-07-18
JPH11504937A (ja) 1999-05-11
CA2218916A1 (en) 1996-11-14
GR3036873T3 (en) 2002-01-31
ATE203246T1 (de) 2001-08-15
DE69613975D1 (de) 2001-08-23
EP0824539A1 (en) 1998-02-25
WO1996035702A1 (en) 1996-11-14
US5583115A (en) 1996-12-10
ES2159733T3 (es) 2001-10-16
DK0824539T3 (da) 2001-09-24

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Legal Events

Date Code Title Description
FG Grant or registration
MM Annulment or lapse due to non-payment of fees