MX2020003730A - Nueva sal y formas en estado solido de escitalopram. - Google Patents

Nueva sal y formas en estado solido de escitalopram.

Info

Publication number
MX2020003730A
MX2020003730A MX2020003730A MX2020003730A MX2020003730A MX 2020003730 A MX2020003730 A MX 2020003730A MX 2020003730 A MX2020003730 A MX 2020003730A MX 2020003730 A MX2020003730 A MX 2020003730A MX 2020003730 A MX2020003730 A MX 2020003730A
Authority
MX
Mexico
Prior art keywords
solid state
escitalopram
state forms
new salt
new
Prior art date
Application number
MX2020003730A
Other languages
English (en)
Inventor
Anton Frenkel
Raeann Ruiyun Wu
Original Assignee
Teva Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Teva Pharma filed Critical Teva Pharma
Publication of MX2020003730A publication Critical patent/MX2020003730A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87Benzo [c] furans; Hydrogenated benzo [c] furans
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/34Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • A61K31/343Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La presente descripción se refiere a una nueva sal de escitalopram y sus formas en estado sólido, procesos para la preparación de la misma, sus composiciones farmacéuticas y sus métodos de uso.
MX2020003730A 2017-10-09 2018-10-09 Nueva sal y formas en estado solido de escitalopram. MX2020003730A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201762569755P 2017-10-09 2017-10-09
PCT/IB2018/057824 WO2019073388A1 (en) 2017-10-09 2018-10-09 NEW SALT AND FORMS IN THE STRONG STATE OF ESCITALOPRAM

Publications (1)

Publication Number Publication Date
MX2020003730A true MX2020003730A (es) 2020-08-03

Family

ID=64100686

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2020003730A MX2020003730A (es) 2017-10-09 2018-10-09 Nueva sal y formas en estado solido de escitalopram.

Country Status (12)

Country Link
US (2) US11390597B2 (es)
EP (1) EP3694843B1 (es)
JP (1) JP7237269B2 (es)
KR (1) KR102505669B1 (es)
CN (1) CN111194312A (es)
AU (1) AU2018349284B2 (es)
CA (2) CA3215809A1 (es)
ES (1) ES2911894T3 (es)
MX (1) MX2020003730A (es)
PL (1) PL3694843T3 (es)
RU (1) RU2020111694A (es)
WO (1) WO2019073388A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11390597B2 (en) * 2017-10-09 2022-07-19 Mark Hasleton Salt and solid state forms of escitalopram
US20240100012A1 (en) * 2021-01-18 2024-03-28 Mark Hasleton Pharmaceutical dosage form
AU2022308198A1 (en) * 2021-07-06 2024-02-01 Mark Hasleton Treatment of serotonin reuptake inhibitor withdrawal syndrome

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8814057D0 (en) 1988-06-14 1988-07-20 Lundbeck & Co As H New enantiomers & their isolation
RS51092B (sr) * 2002-12-23 2010-10-31 H. Lundbeck A/S. Escitalopram bromhidrat i postupak za njegovo pripremanje
US20050154052A1 (en) * 2003-03-24 2005-07-14 Hetero Drugs Limited Novel crystalline forms of (s)-citalopram oxalate
KR100841409B1 (ko) * 2003-12-16 2008-06-25 에스케이케미칼주식회사 암로디핀 겐티세이트 염과 이의 제조방법
US7834201B2 (en) 2005-06-22 2010-11-16 H. Lundbeck A/S Crystalline base of escitalopram and orodispersible tablets comprising escitalopram base
KR101235116B1 (ko) * 2005-10-17 2013-02-20 에스케이케미칼주식회사 광학활성 암로디핀 겐티세이트 염의 제조방법
EP2231648A1 (en) * 2007-12-05 2010-09-29 BIAL - Portela & Ca., S.A. New salts and crystal forms
TW201729810A (zh) * 2015-10-26 2017-09-01 札爾科製藥公司 嘧啶組成物、其超純組成物及鹽類、製造彼之方法、及使用彼於治療組織胺h4受體(h 4 )仲介之疾病與病情之方法
US11390597B2 (en) * 2017-10-09 2022-07-19 Mark Hasleton Salt and solid state forms of escitalopram

Also Published As

Publication number Publication date
US20220363655A1 (en) 2022-11-17
EP3694843B1 (en) 2022-01-26
CA3215809A1 (en) 2019-04-18
KR20200067152A (ko) 2020-06-11
JP7237269B2 (ja) 2023-03-13
EP3694843A1 (en) 2020-08-19
ES2911894T3 (es) 2022-05-23
RU2020111694A (ru) 2021-11-12
KR102505669B1 (ko) 2023-03-03
CA3077506A1 (en) 2019-04-18
JP2020536961A (ja) 2020-12-17
WO2019073388A1 (en) 2019-04-18
CN111194312A (zh) 2020-05-22
AU2018349284B2 (en) 2023-11-16
AU2018349284A1 (en) 2020-04-30
US11390597B2 (en) 2022-07-19
US20210380550A1 (en) 2021-12-09
US11897858B2 (en) 2024-02-13
PL3694843T3 (pl) 2022-06-20
RU2020111694A3 (es) 2022-03-18

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