KR20030091946A
(ko)
|
2000-12-12 |
2003-12-03 |
쉐링 코포레이션 |
C형 간염 바이러스의 ns3-세린 프로테아제억제제로서의 디아릴 펩티드
|
MXPA04003954A
(es)
|
2001-10-26 |
2004-11-29 |
Aventis Pharma Inc |
Bencimidazoles.
|
ES2361011T3
(es)
|
2002-05-20 |
2011-06-13 |
Bristol-Myers Squibb Company |
Inhibidores del virus de la hepatitis c.
|
DE60334205D1
(en)
|
2002-05-20 |
2010-10-28 |
Bristol Myers Squibb Co |
Heterocyclische sulfonamid-hepatitis-c-virus-hemmer
|
PL213029B1
(pl)
|
2002-05-20 |
2012-12-31 |
Bristol Myers Squibb Co |
Podstawiona pochodna cykloalkilowa, zawierajaca ja kompozycja oraz ich zastosowanie
|
ES2320771T3
(es)
|
2003-04-16 |
2009-05-28 |
Bristol-Myers Squibb Company |
Inhibidores peptidicos de isoquinolina macrociclicos del virus de la hepatitis c.
|
US7176208B2
(en)
|
2003-04-18 |
2007-02-13 |
Enanta Pharmaceuticals, Inc. |
Quinoxalinyl macrocyclic hepatitis C serine protease inhibitors
|
PT1615613E
(pt)
|
2003-04-18 |
2010-02-09 |
Enanta Pharm Inc |
Inibidores da serina protease da hepatite c macrocíclicos de quinoxalinilo
|
JP4447603B2
(ja)
|
2003-05-21 |
2010-04-07 |
ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング |
C型肝炎インヒビター化合物
|
WO2005018330A1
(en)
*
|
2003-08-18 |
2005-03-03 |
Pharmasset, Inc. |
Dosing regimen for flaviviridae therapy
|
US7135462B2
(en)
|
2003-11-20 |
2006-11-14 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
AU2005274700B2
(en)
|
2004-07-16 |
2011-11-10 |
Gilead Sciences, Inc. |
Antiviral compounds
|
UY29016A1
(es)
|
2004-07-20 |
2006-02-24 |
Boehringer Ingelheim Int |
Analogos de dipeptidos inhibidores de la hepatitis c
|
WO2007001406A2
(en)
|
2004-10-05 |
2007-01-04 |
Chiron Corporation |
Aryl-containing macrocyclic compounds
|
WO2006119061A2
(en)
|
2005-05-02 |
2006-11-09 |
Merck & Co., Inc. |
Hcv ns3 protease inhibitors
|
US7470664B2
(en)
|
2005-07-20 |
2008-12-30 |
Merck & Co., Inc. |
HCV NS3 protease inhibitors
|
EA019888B1
(ru)
|
2005-07-25 |
2014-07-30 |
Интермьюн, Инк. |
Промежуточное соединение для получения макроциклических ингибиторов репликации вируса гепатита с и способ его синтеза
|
PE20070211A1
(es)
|
2005-07-29 |
2007-05-12 |
Medivir Ab |
Compuestos macrociclicos como inhibidores del virus de hepatitis c
|
EP1913016B1
(en)
|
2005-08-01 |
2013-01-16 |
Merck Sharp & Dohme Corp. |
Macrocyclic peptides as hcv ns3 protease inhibitors
|
DK1999129T3
(da)
|
2005-10-11 |
2011-02-07 |
Intermune Inc |
Forbindelser og fremgangsmåder til inhibering af replikationen af hepatitis C-virus
|
US7772183B2
(en)
|
2005-10-12 |
2010-08-10 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
GB0609492D0
(en)
*
|
2006-05-15 |
2006-06-21 |
Angeletti P Ist Richerche Bio |
Therapeutic agents
|
GB0612423D0
(en)
|
2006-06-23 |
2006-08-02 |
Angeletti P Ist Richerche Bio |
Therapeutic agents
|
KR20090024834A
(ko)
|
2006-07-05 |
2009-03-09 |
인터뮨, 인크. |
C형 간염 바이러스 복제의 신규 억제제
|
CA2667165A1
(en)
|
2006-10-24 |
2008-05-02 |
Merck & Co., Inc. |
Hcv ns3 protease inhibitors
|
CN101583372A
(zh)
|
2006-10-24 |
2009-11-18 |
默克公司 |
Hcv ns3蛋白酶抑制剂
|
WO2008051475A2
(en)
|
2006-10-24 |
2008-05-02 |
Merck & Co., Inc. |
Hcv ns3 protease inhibitors
|
AU2007318165B2
(en)
|
2006-10-27 |
2011-11-17 |
Msd Italia S.R.L. |
HCV NS3 protease inhibitors
|
ES2444575T3
(es)
|
2006-10-27 |
2014-02-25 |
Merck Sharp & Dohme Corp. |
Inhibidores de la proteasa NS3 del VHC
|
US7888464B2
(en)
|
2006-11-16 |
2011-02-15 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
WO2008134397A1
(en)
|
2007-04-26 |
2008-11-06 |
Enanta Pharmaceuticals, Inc. |
Aza-tripeptide hepatitis c serine protease inhibitors
|
BRPI0811020A2
(pt)
|
2007-05-03 |
2015-07-21 |
Intermune Inc |
Composto, composição farmacêutica e métodos de inibição da atividade da protease ns3/ns4, de tratamento da fibrose hepática, de intensificação da função hepática em indivíduo com infecção do vírus da hepatite c e métodos de síntese de compostos, de administração de inibidor da infecção do vírus da hepatite c (hcv) e de distribuição de forma de dosagem oral.
|
CA2686546A1
(en)
|
2007-05-10 |
2008-11-20 |
Intermune, Inc. |
Novel peptide inhibitors of hepatitis c virus replication
|
US20090005387A1
(en)
|
2007-06-26 |
2009-01-01 |
Deqiang Niu |
Quinoxalinyl macrocyclic hepatitis c virus serine protease inhibitors
|
EP2162431B1
(en)
*
|
2007-06-29 |
2017-06-07 |
Gilead Sciences, Inc. |
Antiviral compounds
|
JP5465667B2
(ja)
|
2007-06-29 |
2014-04-09 |
ギリアード サイエンシーズ, インコーポレイテッド |
抗ウイルス化合物
|
JP5433573B2
(ja)
|
2007-07-19 |
2014-03-05 |
イステイチユート・デイ・リチエルケ・デイ・ビオロジア・モレコラーレ・ピ・アンジエレツテイ・エツセ・エルレ・エルレ |
抗ウイルス剤としての大環状化合物
|
JP2010540549A
(ja)
|
2007-09-24 |
2010-12-24 |
アキリオン ファーマシューティカルズ,インコーポレーテッド |
ウイルス複製阻害剤としての尿素含有ペプチド
|
EP2215076A4
(en)
|
2007-10-24 |
2012-05-02 |
Virobay Inc |
COMPOUNDS CAPABLE OF INHIBITING CATHEPSIN S PROTEASE AND HCV REPLICATION
|
US20090111757A1
(en)
|
2007-10-25 |
2009-04-30 |
Taigen Biotechnology Co., Ltd. |
Hcv protease inhibitors
|
CL2008003384A1
(es)
|
2007-11-14 |
2009-12-11 |
Enanta Pharm Inc |
Compuestos derivados de quinoxalina macrocíclica, inhibidores de serina proteasa; composicion farmaceutica que los comprende; y su uso en el tratamiento de la hepatitis c.
|
WO2009070689A1
(en)
|
2007-11-29 |
2009-06-04 |
Enanta Pharmaceuticals, Inc. |
Bicyclic, c5-substituted proline derivatives as inhibitors of the hepatitis c virus ns3 protease
|
WO2009070692A1
(en)
|
2007-11-29 |
2009-06-04 |
Enanta Pharmaceuticals, Inc. |
C5-substituted, proline-derived, macrocyclic hepatitis c serine protease inhibitors
|
MX2010006209A
(es)
|
2007-12-05 |
2010-08-10 |
Enanta Pharm Inc |
Derivados de quinoxalinilo.
|
WO2009079353A1
(en)
|
2007-12-14 |
2009-06-25 |
Enanta Pharmaceuticals, Inc. |
Triazole-containing macrocyclic hcv serine protease inhibitors
|
US8293705B2
(en)
|
2007-12-21 |
2012-10-23 |
Avila Therapeutics, Inc. |
HCV protease inhibitors and uses thereof
|
US8202996B2
(en)
|
2007-12-21 |
2012-06-19 |
Bristol-Myers Squibb Company |
Crystalline forms of N-(tert-butoxycarbonyl)-3-methyl-L-valyl-(4R)-4-((7-chloro-4-methoxy-1-isoquinolinyl)oxy)-N- ((1R,2S)-1-((cyclopropylsulfonyl)carbamoyl)-2-vinylcyclopropyl)-L-prolinamide
|
US8309685B2
(en)
|
2007-12-21 |
2012-11-13 |
Celgene Avilomics Research, Inc. |
HCV protease inhibitors and uses thereof
|
JP5755449B2
(ja)
|
2007-12-21 |
2015-07-29 |
セルジーン アビロミクス リサーチ, インコーポレイテッド |
Hcvプロテアーゼ阻害剤およびその使用
|
JP2011510927A
(ja)
|
2008-01-24 |
2011-04-07 |
エナンタ ファーマシューティカルズ インコーポレイテッド |
Hcvセリンプロテアーゼ阻害剤としての二フッ素化トリペプチド
|
JP5574982B2
(ja)
|
2008-02-04 |
2014-08-20 |
イデニク プハルマセウティカルス,インコーポレイテッド |
大環状セリンプロテアーゼ阻害剤
|
WO2009108507A1
(en)
|
2008-02-25 |
2009-09-03 |
Merck & Co., Inc. |
Therapeutic compounds
|
WO2009114633A1
(en)
|
2008-03-12 |
2009-09-17 |
Virobay, Inc. |
Process for the preparation of (3s)-3-amino-n-cyclopropyl-2-hydroxyalkanamide derivatives
|
CN102015652A
(zh)
|
2008-03-20 |
2011-04-13 |
益安药业 |
作为丙型肝炎病毒抑制剂的氟化大环化合物
|
AP2010005416A0
(en)
|
2008-04-15 |
2010-10-31 |
Intermune Inc |
Novel macrocyclic inhibitors of hepatitis c virus replication.
|
US8163921B2
(en)
|
2008-04-16 |
2012-04-24 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
AU2009241445A1
(en)
|
2008-04-28 |
2009-11-05 |
Merck Sharp & Dohme Corp. |
HCV NS3 protease inhibitors
|
US8211891B2
(en)
|
2008-04-30 |
2012-07-03 |
Enanta Pharmaceuticals, Inc. |
Difluoromethyl-containing macrocyclic compounds as hepatitis C virus inhibitors
|
KR101313675B1
(ko)
|
2008-07-22 |
2013-10-02 |
이스티투토 디 리세르쉐 디 비올로지아 몰레콜라레 피. 안젤레티 에스.알.엘. |
Hcv ns3 프로테아제 억제제로서의 마크로사이클릭 퀴녹살린 화합물
|
KR101647520B1
(ko)
|
2008-08-07 |
2016-08-10 |
에프. 호프만-라 로슈 아게 |
거대환식 화합물의 제조 방법
|
EP2334680A2
(en)
|
2008-08-20 |
2011-06-22 |
Sequoia Pharmaceuticals, Inc. |
Hcv protease inhibitors
|
UY32099A
(es)
|
2008-09-11 |
2010-04-30 |
Enanta Pharm Inc |
Inhibidores macrocíclicos de serina proteasas de hepatitis c
|
WO2010033466A1
(en)
|
2008-09-16 |
2010-03-25 |
Phenomix Corporation |
Macrocyclic inhibitors of hepatitis c protease
|
EP2687526A1
(en)
|
2008-09-16 |
2014-01-22 |
Boehringer Ingelheim International Gmbh |
Crystalline forms of a 2-thiazolyl- 4-quinolinyl-oxy derivative, a potent HCV inhibitor
|
US8563505B2
(en)
|
2008-09-29 |
2013-10-22 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
US20100080770A1
(en)
|
2008-09-29 |
2010-04-01 |
Bristol-Myers Squibb Company |
Hepatitis C Virus Inhibitors
|
US8044087B2
(en)
|
2008-09-29 |
2011-10-25 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
AP2011005695A0
(en)
|
2008-10-15 |
2011-06-30 |
Intermune Inc |
Therapeutic antiviral poptides.
|
EP2364159A4
(en)
|
2008-10-23 |
2012-06-13 |
Concert Pharmaceuticals Inc |
DETERIORIC MACROCYCLIC INHIBITORS OF NS3 VIRAL PROTEASE
|
CA2743912A1
(en)
|
2008-11-20 |
2010-05-27 |
Achillion Pharmaceuticals, Inc. |
Cyclic carboxamide compounds and analogues thereof as of hepatitis c virus
|
CA2738732A1
(en)
|
2008-11-21 |
2010-05-27 |
Boehringer Ingelheim International Gmbh |
Pharmaceutical composition of a potent hcv inhibitor for oral administration
|
US20100272674A1
(en)
|
2008-12-04 |
2010-10-28 |
Bristol-Myers Squibb Company |
Hepatitis C Virus Inhibitors
|
AU2009324644B2
(en)
|
2008-12-10 |
2013-12-05 |
Achillion Pharmaceuticals, Inc. |
4-amino-4-oxobutanoyl peptide cyclic analogues, inhibitors of viral replication
|
US8283310B2
(en)
|
2008-12-15 |
2012-10-09 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
CA2747636A1
(en)
|
2008-12-19 |
2010-07-15 |
Gilead Sciences, Inc. |
Hcv ns3 protease inhibitors
|
AU2009331530B2
(en)
|
2008-12-23 |
2015-04-09 |
Ortho-Mcneil-Janssen Pharmaceuticals, Inc |
Processes and intermediates for preparing a macrocyclic protease inhibitor of HCV
|
WO2010132163A1
(en)
|
2009-05-13 |
2010-11-18 |
Enanta Pharmaceuticals, Inc. |
Macrocyclic compounds as hepatitis c virus inhibitors
|
US8703700B2
(en)
|
2009-05-22 |
2014-04-22 |
Sequoia Pharmaceuticals, Inc. |
Bimacrocylic HCV NS3 protease inhibitors
|
WO2011014487A1
(en)
|
2009-07-30 |
2011-02-03 |
Merck Sharp & Dohme Corp. |
Hepatitis c virus ns3 protease inhibitors
|
JP5789260B2
(ja)
|
2009-08-27 |
2015-10-07 |
メルク・シャープ・エンド・ドーム・コーポレイション |
C型肝炎ウイルスのプロテアーゼ阻害薬の調製方法
|
EP2483290A4
(en)
|
2009-09-28 |
2013-05-01 |
Intermune Inc |
CYCLIC PEPTIC INHIBITORS FOR REPLICATION OF HEPATITIS C VIRUS
|
WO2011041551A1
(en)
|
2009-10-01 |
2011-04-07 |
Intermune, Inc. |
Therapeutic antiviral peptides
|
US9193740B2
(en)
|
2009-10-19 |
2015-11-24 |
Enanta Pharmaceuticals, Inc. |
Bismacrocyclic compounds as hepatitis C virus inhibitors
|
ES2613608T3
(es)
|
2010-03-10 |
2017-05-24 |
Abbvie Ireland Unlimited Company |
Composiciones sólidas
|
US8530497B2
(en)
|
2010-03-11 |
2013-09-10 |
Boehringer Ingelheim International Gmbh |
Crystalline salts of a potent HCV inhibitor
|
EP2576564A4
(en)
|
2010-06-07 |
2014-01-22 |
Abbvie Inc |
MACROCYCLIC HEPATITIS C SERIN PROTEASE INHIBITORS
|
WO2012019299A1
(en)
|
2010-08-11 |
2012-02-16 |
Boehringer Ingelheim International Gmbh |
Hepatitis c inhibitor compounds
|
US20120094897A1
(en)
|
2010-09-15 |
2012-04-19 |
Intermune, Inc. |
Novel inhibitors of hepatitis c virus replication
|
US20130178413A1
(en)
|
2010-09-21 |
2013-07-11 |
John A. McCauley |
Hcv ns3 protease inhibitors
|
JP5857053B2
(ja)
|
2010-09-21 |
2016-02-10 |
エナンタ ファーマシューティカルズ インコーポレイテッド |
大環式プロリン由来hcvセリンプロテアーゼ阻害剤
|
US20120095211A1
(en)
|
2010-09-22 |
2012-04-19 |
Intermune, Inc. |
Substituted proline inhibitors of hepatitis c virus replication
|
WO2012047764A1
(en)
|
2010-10-04 |
2012-04-12 |
Intermune, Inc. |
Therapeutic antiviral peptides
|
WO2012054874A1
(en)
|
2010-10-22 |
2012-04-26 |
Intermune, Inc. |
Novel macrocyclic inhibitors of hepatitis c virus replication
|
CA2815855C
(en)
|
2010-11-01 |
2016-02-02 |
Rfs Pharma, Llc |
Novel specific hcv ns3 protease inhibitors
|
CN103717067A
(zh)
|
2010-12-14 |
2014-04-09 |
默沙东公司 |
制备大环内酰胺的方法与中间体
|
EP2658859A4
(en)
|
2010-12-30 |
2014-07-30 |
Enanta Pharm Inc |
MACROCYCLIC HEPATITIS C SERIN PROTEASE INHIBITORS
|
AU2011352145A1
(en)
|
2010-12-30 |
2013-07-18 |
Abbvie Inc. |
Phenanthridine macrocyclic hepatitis C serine protease inhibitors
|
US8957203B2
(en)
|
2011-05-05 |
2015-02-17 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
CN103562199B
(zh)
|
2011-05-27 |
2016-03-30 |
百时美施贵宝公司 |
作为丙型肝炎病毒抑制剂的掺入氘的三肽
|
US8691757B2
(en)
|
2011-06-15 |
2014-04-08 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
AU2012269643A1
(en)
|
2011-06-16 |
2014-02-06 |
AB Pharma Ltd. |
Macrocyclic heterocyclic compound for inhibiting hepatitis C virus and preparation and use thereof
|
EP2723337A1
(en)
|
2011-06-23 |
2014-04-30 |
Panmed Ltd. |
Treatment of hepatitis c virus
|
JP2014521750A
(ja)
|
2011-08-19 |
2014-08-28 |
メルク・シャープ・アンド・ドーム・コーポレーション |
マクロラクタムを調製するための方法および中間体
|
RU2014122154A
(ru)
|
2011-10-31 |
2015-12-10 |
Мерк Шарп И Доум Корп. |
Композиции, пригодные для лечения вирусных заболеваний
|
US9328138B2
(en)
|
2011-11-15 |
2016-05-03 |
Msd Italia S.R.L. |
HCV NS3 protease inhibitors
|
KR20140109433A
(ko)
|
2012-01-12 |
2014-09-15 |
베링거 인겔하임 인터내셔날 게엠베하 |
강력한 hcv 억제제의 안정화된 약제학적 제형
|
UA119315C2
(uk)
|
2012-07-03 |
2019-06-10 |
Гіліад Фармассет Елелсі |
Інгібітори вірусу гепатиту с
|