MX2014013315A - Nanoparticulas farmaceuticas que muestran la mejora del transporte de la mucosa. - Google Patents

Nanoparticulas farmaceuticas que muestran la mejora del transporte de la mucosa.

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Publication number
MX2014013315A
MX2014013315A MX2014013315A MX2014013315A MX2014013315A MX 2014013315 A MX2014013315 A MX 2014013315A MX 2014013315 A MX2014013315 A MX 2014013315A MX 2014013315 A MX2014013315 A MX 2014013315A MX 2014013315 A MX2014013315 A MX 2014013315A
Authority
MX
Mexico
Prior art keywords
particles
showing improved
improved mucosal
mucosal transport
nanoparticles showing
Prior art date
Application number
MX2014013315A
Other languages
English (en)
Inventor
Alexey Popov
Elizabeth M Enlow
Hongming Chen
Original Assignee
Kala Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=48464113&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX2014013315(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Kala Pharmaceuticals Inc filed Critical Kala Pharmaceuticals Inc
Publication of MX2014013315A publication Critical patent/MX2014013315A/es

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    • AHUMAN NECESSITIES
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • AHUMAN NECESSITIES
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/51Nanocapsules; Nanoparticles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
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    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/196Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
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    • A61K31/407Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
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    • A61K31/517Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
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    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
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    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
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    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/34Macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyesters, polyamino acids, polysiloxanes, polyphosphazines, copolymers of polyalkylene glycol or poloxamers
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    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
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    • A61P5/44Glucocorticosteroids; Drugs increasing or potentiating the activity of glucocorticosteroids
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10STECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S977/00Nanotechnology
    • Y10S977/70Nanostructure
    • Y10S977/773Nanoparticle, i.e. structure having three dimensions of 100 nm or less

Abstract

Se proporcionan partículas, composiciones, y métodos que ayudan al transporte de partículas en el moco. En algunas modalidades, las composiciones y los métodos pueden incluir modificar los revestimientos de superficie de las partículas, tales como las partículas de los agentes farmacéuticos que tienen una baja solubilidad acuosa. La composición farmacéutica que incluye tales partículas se adecua bien para las aplicaciones oftálmicas, y puede utilizarse para suministrar agentes farmacéuticos a la parte frontal del ojo y/o la parte posterior del ojo.
MX2014013315A 2012-05-03 2013-05-03 Nanoparticulas farmaceuticas que muestran la mejora del transporte de la mucosa. MX2014013315A (es)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201261642313P 2012-05-03 2012-05-03
US201261642261P 2012-05-03 2012-05-03
US201261738949P 2012-12-18 2012-12-18
US201361784701P 2013-03-14 2013-03-14
PCT/US2013/039540 WO2013166436A1 (en) 2012-05-03 2013-05-03 Pharmaceutical nanoparticles showing improved mucosal transport

Publications (1)

Publication Number Publication Date
MX2014013315A true MX2014013315A (es) 2015-09-10

Family

ID=48464113

Family Applications (2)

Application Number Title Priority Date Filing Date
MX2014013315A MX2014013315A (es) 2012-05-03 2013-05-03 Nanoparticulas farmaceuticas que muestran la mejora del transporte de la mucosa.
MX2020007227A MX2020007227A (es) 2012-05-03 2014-11-03 Nanoparticulas farmaceuticas que muestran la mejora del transporte de la mucosa.

Family Applications After (1)

Application Number Title Priority Date Filing Date
MX2020007227A MX2020007227A (es) 2012-05-03 2014-11-03 Nanoparticulas farmaceuticas que muestran la mejora del transporte de la mucosa.

Country Status (13)

Country Link
US (4) US20130316006A1 (es)
EP (1) EP2844223A1 (es)
JP (3) JP6720443B2 (es)
KR (2) KR102373259B1 (es)
CN (5) CN111700880A (es)
AU (3) AU2013256092B2 (es)
BR (1) BR112014027296B1 (es)
CA (1) CA2871748C (es)
CL (3) CL2014002956A1 (es)
HK (2) HK1208161A1 (es)
MX (2) MX2014013315A (es)
NZ (5) NZ741873A (es)
WO (1) WO2013166436A1 (es)

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