MX2009010363A - Compuestos de 1,3-tiazol-2(3h)-ilideno como ligandos del receptor canabinoide. - Google Patents
Compuestos de 1,3-tiazol-2(3h)-ilideno como ligandos del receptor canabinoide.Info
- Publication number
- MX2009010363A MX2009010363A MX2009010363A MX2009010363A MX2009010363A MX 2009010363 A MX2009010363 A MX 2009010363A MX 2009010363 A MX2009010363 A MX 2009010363A MX 2009010363 A MX2009010363 A MX 2009010363A MX 2009010363 A MX2009010363 A MX 2009010363A
- Authority
- MX
- Mexico
- Prior art keywords
- thiazol
- receptor ligands
- cannabinoid receptor
- compounds
- ylidene compounds
- Prior art date
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/44—Acylated amino or imino radicals
- C07D277/46—Acylated amino or imino radicals by carboxylic acids, or sulfur or nitrogen analogues thereof
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/582—Recycling of unreacted starting or intermediate materials
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Immunology (AREA)
- Neurology (AREA)
- Pulmonology (AREA)
- Physical Education & Sports Medicine (AREA)
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- Orthopedic Medicine & Surgery (AREA)
- Neurosurgery (AREA)
- Diabetes (AREA)
- Dermatology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pain & Pain Management (AREA)
- Emergency Medicine (AREA)
- Hematology (AREA)
- Obesity (AREA)
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- Hospice & Palliative Care (AREA)
- Vascular Medicine (AREA)
- Urology & Nephrology (AREA)
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- Endocrinology (AREA)
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente solicitud se refiere a compuestos que contienen tiazolilideno de la fórmula (I), en donde R1, R2, R3, R4, L2 y A son como se definen en la especificación. También se describen composiciones que comprenden dichos compuestos, y métodos para tratar condiciones y trastornos utilizando tales compuestos y composiciones.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US90845507P | 2007-03-28 | 2007-03-28 | |
PCT/US2008/057460 WO2008121558A1 (en) | 2007-03-28 | 2008-03-19 | 1, 3-thiazol-2 (3h) -ylidene compounds as cannabinoid receptor ligands |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2009010363A true MX2009010363A (es) | 2009-12-04 |
Family
ID=39671674
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2009010363A MX2009010363A (es) | 2007-03-28 | 2008-03-19 | Compuestos de 1,3-tiazol-2(3h)-ilideno como ligandos del receptor canabinoide. |
Country Status (7)
Country | Link |
---|---|
US (2) | US7875640B2 (es) |
EP (1) | EP2142522A1 (es) |
JP (1) | JP2010522760A (es) |
CN (1) | CN101765594A (es) |
CA (1) | CA2681586A1 (es) |
MX (1) | MX2009010363A (es) |
WO (1) | WO2008121558A1 (es) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8841334B2 (en) | 2006-05-31 | 2014-09-23 | Abbvie Inc. | Compounds as cannabinoid receptor ligands and uses thereof |
US7875639B2 (en) | 2006-05-31 | 2011-01-25 | Abbott Laboratories | Compounds as cannabinoid receptor ligands and uses thereof |
CA2647597A1 (en) * | 2006-05-31 | 2007-12-06 | Abbott Laboratories | Thiazole compounds as cannabinoid receptor ligands and uses thereof |
EP2142522A1 (en) | 2007-03-28 | 2010-01-13 | Abbott Laboratories | 1, 3-thiazol-2 (3h) -ylidene compounds as cannabinoid receptor ligands |
US7872033B2 (en) * | 2007-04-17 | 2011-01-18 | Abbott Laboratories | Compounds as cannabinoid receptor ligands |
MX2009012374A (es) * | 2007-05-18 | 2009-12-01 | Abbott Lab | Compuestos novedosos como ligandos del receptor de canabinoides. |
US9193713B2 (en) * | 2007-10-12 | 2015-11-24 | Abbvie Inc. | Compounds as cannabinoid receptor ligands |
US8044071B2 (en) * | 2007-10-18 | 2011-10-25 | Abbott Laboratories | Method for reducing side effects of CB2 receptor agonist therapy using a combination of a selective CB2 receptor agonist and a selective CB1 receptor antagonist |
CA2716857A1 (en) * | 2008-03-11 | 2009-09-17 | Teodozyi Kolasa | Novel compounds as cannabinoid receptor ligands |
JP2012500198A (ja) * | 2008-08-15 | 2012-01-05 | アボット・ラボラトリーズ | カンナビノイド受容体リガンドとしてのイミン誘導体 |
US8846730B2 (en) | 2008-09-08 | 2014-09-30 | Abbvie Inc. | Compounds as cannabinoid receptor ligands |
TW201016692A (en) * | 2008-09-16 | 2010-05-01 | Abbott Lab | Novel compounds as cannabinoid receptor ligands |
PA8854001A1 (es) | 2008-12-16 | 2010-07-27 | Abbott Lab | Compuestos novedosos como ligandos de receptores de canabinoides |
WO2013129692A2 (en) * | 2012-02-29 | 2013-09-06 | Meiji Seika Pharma Co., Ltd. | Nitrogen-containing heterocyclic derivative having 2-imino group and pest control agent including the same |
GB202216324D0 (en) * | 2022-11-02 | 2022-12-14 | Cerevance Ltd | Novel compounds |
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-
2008
- 2008-03-19 EP EP08732454A patent/EP2142522A1/en not_active Withdrawn
- 2008-03-19 US US12/051,538 patent/US7875640B2/en not_active Expired - Fee Related
- 2008-03-19 MX MX2009010363A patent/MX2009010363A/es not_active Application Discontinuation
- 2008-03-19 JP JP2010501085A patent/JP2010522760A/ja active Pending
- 2008-03-19 WO PCT/US2008/057460 patent/WO2008121558A1/en active Application Filing
- 2008-03-19 CA CA002681586A patent/CA2681586A1/en not_active Abandoned
- 2008-03-19 CN CN200880017654A patent/CN101765594A/zh active Pending
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2010
- 2010-12-16 US US12/970,435 patent/US8865753B2/en not_active Expired - Fee Related
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US20110086832A1 (en) | 2011-04-14 |
US8865753B2 (en) | 2014-10-21 |
EP2142522A1 (en) | 2010-01-13 |
JP2010522760A (ja) | 2010-07-08 |
US7875640B2 (en) | 2011-01-25 |
CA2681586A1 (en) | 2008-10-09 |
CN101765594A (zh) | 2010-06-30 |
WO2008121558A1 (en) | 2008-10-09 |
US20080242654A1 (en) | 2008-10-02 |
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