ME02314B - Derivati tieno[2,3-d] pirimidina i njihova primena u lečenju aritmije - Google Patents

Derivati tieno[2,3-d] pirimidina i njihova primena u lečenju aritmije

Info

Publication number
ME02314B
ME02314B MEP-2015-219A MEP2015219A ME02314B ME 02314 B ME02314 B ME 02314B ME P2015219 A MEP2015219 A ME P2015219A ME 02314 B ME02314 B ME 02314B
Authority
ME
Montenegro
Prior art keywords
thieno
pyrimidine derivatives
treat arrhythmia
arrhythmia
treat
Prior art date
Application number
MEP-2015-219A
Other languages
English (en)
Inventor
Derek Edward John
John Ford
Original Assignee
Xention Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=44071904&utm_source=***_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ME02314(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Xention Ltd filed Critical Xention Ltd
Publication of ME02314B publication Critical patent/ME02314B/me

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/06—Antiarrhythmics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Epidemiology (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
MEP-2015-219A 2011-04-01 2012-03-29 Derivati tieno[2,3-d] pirimidina i njihova primena u lečenju aritmije ME02314B (me)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB1105659.5A GB201105659D0 (en) 2011-04-01 2011-04-01 Compounds
PCT/GB2012/050710 WO2012131379A1 (en) 2011-04-01 2012-03-29 Thieno [2, 3 -d] pyrimidine derivatives and their use to treat arrhythmia
EP12718725.0A EP2694518B1 (en) 2011-04-01 2012-03-29 Thieno[2,3-d]pyrimidine derivatives and their use to treat arrhythmia

Publications (1)

Publication Number Publication Date
ME02314B true ME02314B (me) 2016-06-20

Family

ID=44071904

Family Applications (1)

Application Number Title Priority Date Filing Date
MEP-2015-219A ME02314B (me) 2011-04-01 2012-03-29 Derivati tieno[2,3-d] pirimidina i njihova primena u lečenju aritmije

Country Status (42)

Country Link
US (1) US9249155B2 (me)
EP (1) EP2694518B1 (me)
JP (1) JP5826374B2 (me)
KR (1) KR20140023332A (me)
CN (1) CN103492392B (me)
AP (1) AP2013007198A0 (me)
AR (1) AR088735A1 (me)
AU (1) AU2012235882B2 (me)
BR (1) BR112013025236A2 (me)
CA (1) CA2831493A1 (me)
CL (1) CL2013002789A1 (me)
CO (1) CO6801756A2 (me)
CR (1) CR20130488A (me)
CU (1) CU24173B1 (me)
CY (1) CY1117025T1 (me)
DK (1) DK2694518T3 (me)
EA (1) EA201301111A1 (me)
EC (1) ECSP13012988A (me)
ES (1) ES2558563T3 (me)
GB (1) GB201105659D0 (me)
GT (1) GT201300225A (me)
HK (2) HK1193096A1 (me)
HR (1) HRP20151340T1 (me)
HU (1) HUE028438T2 (me)
IL (1) IL228555A0 (me)
MA (1) MA35064B1 (me)
ME (1) ME02314B (me)
MX (1) MX335937B (me)
NI (1) NI201300100A (me)
PE (1) PE20141021A1 (me)
PL (1) PL2694518T3 (me)
PT (1) PT2694518E (me)
RS (1) RS54458B1 (me)
RU (1) RU2013148627A (me)
SG (1) SG193578A1 (me)
SI (1) SI2694518T1 (me)
SM (1) SMT201500322B (me)
TN (1) TN2013000377A1 (me)
TW (1) TWI516265B (me)
UA (1) UA110131C2 (me)
WO (1) WO2012131379A1 (me)
ZA (1) ZA201307085B (me)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20150307532A1 (en) * 2012-11-20 2015-10-29 The Royal Institution For The Advancement Of Learning/Mcgill University Thienopyrimidine inhibitors of farnesyl and/or geranylgeranyl pyrophosphate synthase
SG11201804901WA (en) 2015-12-22 2018-07-30 SHY Therapeutics LLC Compounds for the treatment of cancer and inflammatory disease
CN106727587A (zh) * 2016-11-28 2017-05-31 李娜 一种治疗心律失常的药物组合物
CN111032662A (zh) 2017-06-21 2020-04-17 尚医治疗有限责任公司 与ras超家族相互作用的用于治疗癌症、炎性疾病、ras蛋白病和纤维化疾病的化合物

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Also Published As

Publication number Publication date
JP2014509637A (ja) 2014-04-21
DK2694518T3 (en) 2015-11-09
AR088735A1 (es) 2014-07-02
AU2012235882B2 (en) 2015-08-06
SMT201500322B (it) 2016-02-25
EP2694518B1 (en) 2015-10-07
WO2012131379A1 (en) 2012-10-04
JP5826374B2 (ja) 2015-12-02
AU2012235882A1 (en) 2013-05-02
ZA201307085B (en) 2015-04-29
CN103492392A (zh) 2014-01-01
CR20130488A (es) 2013-12-06
HUE028438T2 (en) 2017-02-28
HRP20151340T1 (hr) 2016-02-26
RU2013148627A (ru) 2015-05-10
TN2013000377A1 (en) 2015-01-20
CU24173B1 (es) 2016-04-25
CL2013002789A1 (es) 2014-07-18
PE20141021A1 (es) 2014-08-30
NI201300100A (es) 2014-01-07
CU20130124A7 (es) 2014-01-29
AP2013007198A0 (en) 2013-10-31
HK1193806A1 (zh) 2014-10-03
CO6801756A2 (es) 2013-11-29
RS54458B1 (en) 2016-06-30
BR112013025236A2 (pt) 2019-09-24
UA110131C2 (ru) 2015-11-25
US20140206703A1 (en) 2014-07-24
EP2694518A1 (en) 2014-02-12
CA2831493A1 (en) 2012-10-04
CN103492392B (zh) 2015-11-25
GT201300225A (es) 2014-12-30
PT2694518E (pt) 2016-02-05
GB201105659D0 (en) 2011-05-18
EA201301111A1 (ru) 2014-02-28
TW201244720A (en) 2012-11-16
PL2694518T3 (pl) 2016-03-31
ES2558563T3 (es) 2016-02-05
HK1193096A1 (zh) 2014-09-12
NZ615621A (en) 2015-01-30
MX335937B (es) 2016-01-04
US9249155B2 (en) 2016-02-02
ECSP13012988A (es) 2013-12-31
KR20140023332A (ko) 2014-02-26
CY1117025T1 (el) 2017-04-05
SG193578A1 (en) 2013-10-30
IL228555A0 (en) 2013-12-31
MA35064B1 (fr) 2014-04-03
SI2694518T1 (sl) 2016-02-29
TWI516265B (zh) 2016-01-11
MX2013011301A (es) 2014-04-16

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