MA48800A - Cycles 5-5 fusionnés utilisés en tant qu'inhibiteurs de c5a - Google Patents
Cycles 5-5 fusionnés utilisés en tant qu'inhibiteurs de c5aInfo
- Publication number
- MA48800A MA48800A MA048800A MA48800A MA48800A MA 48800 A MA48800 A MA 48800A MA 048800 A MA048800 A MA 048800A MA 48800 A MA48800 A MA 48800A MA 48800 A MA48800 A MA 48800A
- Authority
- MA
- Morocco
- Prior art keywords
- inhibitors
- fused cycles
- fused
- cycles
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
- A61K31/4162—1,2-Diazoles condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201762513025P | 2017-05-31 | 2017-05-31 |
Publications (1)
Publication Number | Publication Date |
---|---|
MA48800A true MA48800A (fr) | 2020-04-08 |
Family
ID=64455572
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MA048800A MA48800A (fr) | 2017-05-31 | 2018-05-29 | Cycles 5-5 fusionnés utilisés en tant qu'inhibiteurs de c5a |
Country Status (16)
Country | Link |
---|---|
US (2) | US10683294B2 (fr) |
EP (1) | EP3630774B1 (fr) |
JP (1) | JP7141129B2 (fr) |
KR (1) | KR102586710B1 (fr) |
CN (1) | CN111032658B (fr) |
AR (1) | AR111841A1 (fr) |
AU (1) | AU2018277523B2 (fr) |
BR (1) | BR112019025230A2 (fr) |
CA (1) | CA3064025A1 (fr) |
ES (1) | ES2934507T3 (fr) |
IL (1) | IL270842B2 (fr) |
MA (1) | MA48800A (fr) |
MX (1) | MX2019014292A (fr) |
TW (1) | TWI813570B (fr) |
WO (1) | WO2018222601A1 (fr) |
ZA (1) | ZA201907755B (fr) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR102586710B1 (ko) | 2017-05-31 | 2023-10-10 | 케모센트릭스, 인크. | C5a 억제제로서의 5-5 융합 고리 |
EP3630775B1 (fr) | 2017-05-31 | 2022-12-14 | ChemoCentryx, Inc. | Cycles 6-5 fusionnés utilisés en tant qu'inhibiteurs de c5a |
JP7254082B2 (ja) | 2017-12-22 | 2023-04-07 | ケモセントリックス,インコーポレイティド | C5aR阻害剤としてのジアリール置換6,5-縮合環化合物 |
WO2019126431A1 (fr) * | 2017-12-22 | 2019-06-27 | Chemocentryx, Inc. | Composés cycliques fusionnés en 5,5 à substitution diaryle, utilisés en tant qu'inhibiteurs du c5ar |
MX2020010390A (es) * | 2018-04-02 | 2021-01-15 | Chemocentryx Inc | Profarmacos de antagonistas de c5ar biciclicos fusionados. |
JP2022539830A (ja) | 2019-07-10 | 2022-09-13 | ケモセントリックス,インコーポレイティド | Pd-l1阻害剤としてのインダン |
CN112300169B (zh) * | 2019-07-26 | 2022-03-04 | 上海美迪西生物医药股份有限公司 | 吡咯并吡唑类衍生物、其制备方法及其在医药上的应用 |
US11844790B2 (en) | 2020-10-28 | 2023-12-19 | Chemocentryx, Inc. | Methods of treating hidradenitis suppurativa |
Family Cites Families (32)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EA006381B1 (ru) | 2000-08-10 | 2005-12-29 | Фармация Италия С.П.А. | Бициклопиразолы, активные в качестве ингибиторов киназы, способ их получения и включающие их фармацевтические композиции |
AU7622500A (en) | 2000-09-29 | 2002-07-01 | Neurogen Corp | High affinity small molecule c5a receptor modulators |
SE524438C2 (sv) | 2000-10-05 | 2004-08-10 | Magnus Georg Goertz | Fjärrstyrt dörrelaterat låsarrangemang, första och andra datorpogramprodukt, bärande medium och ett datorlösbart medium |
JP4196678B2 (ja) | 2001-04-26 | 2008-12-17 | 味の素株式会社 | 複素環化合物 |
ITMI20012025A1 (it) | 2001-09-28 | 2003-03-28 | Dompe Spa | Sali di ammonio quaternari di omega-amminoalchilammidi di acidi r 2-aril-propionici e composizioni farmaceutiche che li contengono |
AU2003218374A1 (en) | 2002-03-28 | 2003-10-13 | Neurogen Corporation | Substituted tetrahydroisoquinolines as c5a receptor modulators |
EP1487796A4 (fr) | 2002-03-28 | 2005-11-16 | Neurogen Corp | Biarylamides substitues en tant que modulateurs du recepteur c5a |
US20040014782A1 (en) | 2002-03-29 | 2004-01-22 | Krause James E. | Combination therapy for the treatment of diseases involving inflammatory components |
US7166619B2 (en) | 2002-08-14 | 2007-01-23 | Ppd Discovery , Inc. | Prenylation inhibitors and methods of their synthesis and use |
US7169775B2 (en) | 2002-08-21 | 2007-01-30 | Neurogen Corporation | Amino methyl imidazoles as C5a receptor modulators |
WO2004043925A2 (fr) | 2002-11-08 | 2004-05-27 | Neurogen Corporation | 6-aryl pyridines substituees en 3 |
US20040214856A1 (en) | 2003-04-23 | 2004-10-28 | Pfizer Inc | Cannabinoid receptor ligands and uses thereof |
US7145012B2 (en) | 2003-04-23 | 2006-12-05 | Pfizer Inc. | Cannabinoid receptor ligands and uses thereof |
AU2003902354A0 (en) | 2003-05-15 | 2003-05-29 | Harkin, Denis W. | Treatment of haemorrhagic shock |
WO2005007087A2 (fr) | 2003-07-03 | 2005-01-27 | Neurogen Corporation | Derives (heterocycloalkyl)methyle substitues de type azole utilises comme modulateurs des recepteurs c5a |
US7906528B2 (en) * | 2004-10-05 | 2011-03-15 | Novartis International Pharmaceutical Ltd. | Pyrrolo-pyridine, pyrrolo-pyrimidine and related heterocyclic compounds |
US7598255B2 (en) | 2005-08-04 | 2009-10-06 | Janssen Pharmaceutica Nv | Pyrimidine compounds as serotonin receptor modulators |
US20070112015A1 (en) | 2005-10-28 | 2007-05-17 | Chemocentryx, Inc. | Substituted dihydropyridines and methods of use |
JP5595389B2 (ja) | 2008-06-20 | 2014-09-24 | ジェネンテック, インコーポレイテッド | トリアゾロピリジンjak阻害剤化合物と方法 |
US20110275639A1 (en) | 2008-12-22 | 2011-11-10 | Chemocentryx, Inc. | C5aR ANTAGONISTS |
WO2010075257A1 (fr) | 2008-12-22 | 2010-07-01 | Chemocentryx, Inc. | Antagonistes de c5ar |
PL2585064T3 (pl) | 2010-06-24 | 2017-09-29 | Chemocentryx, Inc. | Antagoniści C5AR |
US8846656B2 (en) | 2011-07-22 | 2014-09-30 | Novartis Ag | Tetrahydropyrido-pyridine and tetrahydropyrido-pyrimidine compounds and use thereof as C5a receptor modulators |
AU2013302473B2 (en) | 2012-08-16 | 2017-08-10 | Janssen Pharmaceutica Nv | Pyrrolopyrazoles as N-type calcium channel blockers |
CN103421006B (zh) | 2013-08-18 | 2016-06-22 | 上海师范大学 | 2,3,5,7-四取代二氢吡唑并六氢吡啶衍生物及其制备方法和应用 |
GB201321746D0 (en) | 2013-12-09 | 2014-01-22 | Ucb Pharma Sa | Therapeutic agents |
MX2018011831A (es) | 2016-04-04 | 2019-02-13 | Chemocentryx Inc | Antagonistas solubles de receptor de c5aa(c5ar). |
EP3630775B1 (fr) | 2017-05-31 | 2022-12-14 | ChemoCentryx, Inc. | Cycles 6-5 fusionnés utilisés en tant qu'inhibiteurs de c5a |
KR102586710B1 (ko) | 2017-05-31 | 2023-10-10 | 케모센트릭스, 인크. | C5a 억제제로서의 5-5 융합 고리 |
WO2019126431A1 (fr) | 2017-12-22 | 2019-06-27 | Chemocentryx, Inc. | Composés cycliques fusionnés en 5,5 à substitution diaryle, utilisés en tant qu'inhibiteurs du c5ar |
JP7254082B2 (ja) | 2017-12-22 | 2023-04-07 | ケモセントリックス,インコーポレイティド | C5aR阻害剤としてのジアリール置換6,5-縮合環化合物 |
MX2020010390A (es) | 2018-04-02 | 2021-01-15 | Chemocentryx Inc | Profarmacos de antagonistas de c5ar biciclicos fusionados. |
-
2018
- 2018-05-29 KR KR1020197038670A patent/KR102586710B1/ko active IP Right Grant
- 2018-05-29 EP EP18809125.0A patent/EP3630774B1/fr active Active
- 2018-05-29 JP JP2019565826A patent/JP7141129B2/ja active Active
- 2018-05-29 ES ES18809125T patent/ES2934507T3/es active Active
- 2018-05-29 MX MX2019014292A patent/MX2019014292A/es unknown
- 2018-05-29 AU AU2018277523A patent/AU2018277523B2/en active Active
- 2018-05-29 MA MA048800A patent/MA48800A/fr unknown
- 2018-05-29 CA CA3064025A patent/CA3064025A1/fr active Pending
- 2018-05-29 BR BR112019025230-4A patent/BR112019025230A2/pt unknown
- 2018-05-29 CN CN201880036650.8A patent/CN111032658B/zh active Active
- 2018-05-29 WO PCT/US2018/034908 patent/WO2018222601A1/fr active Application Filing
- 2018-05-29 US US15/991,747 patent/US10683294B2/en active Active
- 2018-05-31 TW TW107118603A patent/TWI813570B/zh active
- 2018-05-31 AR ARP180101445A patent/AR111841A1/es unknown
-
2019
- 2019-11-21 IL IL270842A patent/IL270842B2/en unknown
- 2019-11-22 ZA ZA2019/07755A patent/ZA201907755B/en unknown
-
2020
- 2020-05-04 US US16/865,648 patent/US11479553B2/en active Active
Also Published As
Publication number | Publication date |
---|---|
CN111032658A (zh) | 2020-04-17 |
CA3064025A1 (fr) | 2018-12-06 |
ZA201907755B (en) | 2023-05-31 |
MX2019014292A (es) | 2022-04-07 |
EP3630774A1 (fr) | 2020-04-08 |
AR111841A1 (es) | 2019-08-21 |
EP3630774B1 (fr) | 2022-11-23 |
RU2019142985A3 (fr) | 2021-09-03 |
IL270842B1 (en) | 2023-01-01 |
KR20200013720A (ko) | 2020-02-07 |
IL270842A (en) | 2020-01-30 |
US20210009594A1 (en) | 2021-01-14 |
AU2018277523A1 (en) | 2019-12-05 |
IL270842B2 (en) | 2023-05-01 |
CN111032658B (zh) | 2022-12-20 |
TWI813570B (zh) | 2023-09-01 |
RU2019142985A (ru) | 2021-06-30 |
BR112019025230A2 (pt) | 2020-06-16 |
JP7141129B2 (ja) | 2022-09-22 |
US11479553B2 (en) | 2022-10-25 |
ES2934507T3 (es) | 2023-02-22 |
AU2018277523B2 (en) | 2022-06-23 |
TW201902897A (zh) | 2019-01-16 |
US10683294B2 (en) | 2020-06-16 |
US20180346471A1 (en) | 2018-12-06 |
JP2020522483A (ja) | 2020-07-30 |
KR102586710B1 (ko) | 2023-10-10 |
EP3630774A4 (fr) | 2020-10-07 |
WO2018222601A1 (fr) | 2018-12-06 |
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