LU79949A1 - Nouveaux derives solubles de 2,4-diamino-pyrimidines,leur preparation et leur utilisation en tant que medicaments - Google Patents

Nouveaux derives solubles de 2,4-diamino-pyrimidines,leur preparation et leur utilisation en tant que medicaments

Info

Publication number
LU79949A1
LU79949A1 LU79949A LU79949A LU79949A1 LU 79949 A1 LU79949 A1 LU 79949A1 LU 79949 A LU79949 A LU 79949A LU 79949 A LU79949 A LU 79949A LU 79949 A1 LU79949 A1 LU 79949A1
Authority
LU
Luxembourg
Prior art keywords
diamino
preparation
pyrimidine derivatives
medicinal products
new soluble
Prior art date
Application number
LU79949A
Other languages
English (en)
Original Assignee
Dick P
Rombi M
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dick P, Rombi M filed Critical Dick P
Publication of LU79949A1 publication Critical patent/LU79949A1/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • C07D239/49Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/02Heterocyclic radicals containing only nitrogen as ring hetero atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
LU79949A 1977-07-11 1978-07-10 Nouveaux derives solubles de 2,4-diamino-pyrimidines,leur preparation et leur utilisation en tant que medicaments LU79949A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7722323A FR2397407A2 (fr) 1977-07-11 1977-07-11 Derives de 2,4-diamino pyrimidines et leur mise en solution en association avec des sulfamides

Publications (1)

Publication Number Publication Date
LU79949A1 true LU79949A1 (fr) 1979-04-09

Family

ID=9193583

Family Applications (1)

Application Number Title Priority Date Filing Date
LU79949A LU79949A1 (fr) 1977-07-11 1978-07-10 Nouveaux derives solubles de 2,4-diamino-pyrimidines,leur preparation et leur utilisation en tant que medicaments

Country Status (13)

Country Link
US (1) US4232023A (fr)
JP (1) JPS5448776A (fr)
AT (1) AT362381B (fr)
AU (1) AU3793378A (fr)
BE (1) BE868893A (fr)
DE (1) DE2829820A1 (fr)
FR (1) FR2397407A2 (fr)
GB (1) GB2001965B (fr)
IE (1) IE47232B1 (fr)
IT (1) IT1096690B (fr)
LU (1) LU79949A1 (fr)
NL (1) NL7807440A (fr)
ZA (1) ZA783957B (fr)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2502152A1 (fr) 1981-03-20 1982-09-24 Panmedica Laboratoires Nouveaux derives solubles n2 substitues de la diamino-2,4-benzyl-5-pyrimidines, leur procede de preparation et medicaments les contenant
US6583148B1 (en) 1999-04-08 2003-06-24 Krenitsky Pharmaceuticals, Inc. Neurotrophic substituted pyrimidines
JP5154728B2 (ja) 2000-07-24 2013-02-27 クレニツキー・ファーマシューティカルズ,インコーポレイテッド 神経栄養活性を有する置換5−アルキニルピリミジン
AU2005229331B2 (en) * 2004-03-05 2011-10-13 F. Hoffmann-La Roche Ag Diaminopyrimidines as P2X3 and P2X2/3 antagonists
EP1924566B1 (fr) * 2005-09-01 2016-01-13 F.Hoffmann-La Roche Ag Diaminopyrimidines comme modulateurs p2x3 et p2x2/3
JP4850911B2 (ja) * 2005-09-01 2012-01-11 エフ.ホフマン−ラ ロシュ アーゲー P2x3およびp2x2/3モジュレーターとしてのジアミノピリミジン
CN101253159B (zh) * 2005-09-01 2011-12-07 弗·哈夫曼-拉罗切有限公司 作为p2x3和p2x2/3调节剂的二氨基嘧啶类化合物
CA2700880C (fr) * 2007-10-08 2016-03-08 Bongkoch Tarnchompoo Composes antimalariens a chaine laterales flexibles
US9000003B2 (en) * 2011-03-10 2015-04-07 National Science And Technology Development Agency Anti-folate antimalarials with dual-binding modes and their preparation

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2287071A (en) * 1938-08-08 1942-06-23 Parke Davis & Co Organic amine derivatives and method of obtaining same
US2374791A (en) * 1942-06-22 1945-05-01 Parke Davis & Co Organic amine derivatives and method of obtaining same
US3111521A (en) * 1962-04-25 1963-11-19 Parke Davis & Co 2-aryl-nu-(polyamino-5-pyrimidinyl)-glycinonitriles
GB1375162A (fr) * 1970-10-22 1974-11-27
BE791627A (fr) * 1971-11-20 1973-05-21 Knapsack Ag Procede pour l'oxydation du monoxyde de carbone et des hydrocarbures

Also Published As

Publication number Publication date
GB2001965B (en) 1982-03-10
ATA496978A (de) 1980-10-15
IT1096690B (it) 1985-08-26
NL7807440A (nl) 1979-01-15
FR2397407B2 (fr) 1980-01-04
ZA783957B (en) 1979-09-26
IE781377L (en) 1979-01-11
JPS5448776A (en) 1979-04-17
IT7825569A0 (it) 1978-07-11
AU3793378A (en) 1980-01-17
DE2829820A1 (de) 1979-02-01
GB2001965A (en) 1979-02-14
IE47232B1 (en) 1984-01-25
AT362381B (de) 1981-05-11
US4232023A (en) 1980-11-04
BE868893A (fr) 1979-01-11
FR2397407A2 (fr) 1979-02-09

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